JP2010527915A5 - - Google Patents

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Publication number
JP2010527915A5
JP2010527915A5 JP2010506273A JP2010506273A JP2010527915A5 JP 2010527915 A5 JP2010527915 A5 JP 2010527915A5 JP 2010506273 A JP2010506273 A JP 2010506273A JP 2010506273 A JP2010506273 A JP 2010506273A JP 2010527915 A5 JP2010527915 A5 JP 2010527915A5
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JP
Japan
Prior art keywords
alkyl
ring atom
ring
aryl
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2010506273A
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English (en)
Japanese (ja)
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JP2010527915A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/005331 external-priority patent/WO2008133975A1/en
Publication of JP2010527915A publication Critical patent/JP2010527915A/ja
Publication of JP2010527915A5 publication Critical patent/JP2010527915A5/ja
Withdrawn legal-status Critical Current

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JP2010506273A 2007-04-26 2008-04-25 多重環化合物及びその用途 Withdrawn JP2010527915A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US92628907P 2007-04-26 2007-04-26
PCT/US2008/005331 WO2008133975A1 (en) 2007-04-26 2008-04-25 Multi-ring compounds and uses thereof

Publications (2)

Publication Number Publication Date
JP2010527915A JP2010527915A (ja) 2010-08-19
JP2010527915A5 true JP2010527915A5 (enExample) 2012-07-05

Family

ID=39925991

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010506273A Withdrawn JP2010527915A (ja) 2007-04-26 2008-04-25 多重環化合物及びその用途

Country Status (5)

Country Link
US (1) US20100249111A1 (enExample)
EP (1) EP2141994A4 (enExample)
JP (1) JP2010527915A (enExample)
CA (1) CA2685029A1 (enExample)
WO (1) WO2008133975A1 (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008083124A1 (en) 2006-12-28 2008-07-10 Rigel Pharmaceuticals, Inc. N-substituted-heterocycloalkyloxybenzamide compounds and methods of use
JP5544296B2 (ja) * 2007-11-16 2014-07-09 ライジェル ファーマシューティカルズ， インコーポレイテッド 代謝障害のためのカルボキサミド、スルホンアミド、およびアミン化合物
ES2553340T3 (es) 2007-12-12 2015-12-07 Rigel Pharmaceuticals, Inc. Compuestos de carboxamida, sulfonamida y amina para trastornos metabólicos
CA2719784A1 (en) * 2008-04-17 2009-10-22 Pfizer Inc. Ether benzylidene piperidine 5-membered aryl carboxamide compounds
WO2009127946A1 (en) * 2008-04-17 2009-10-22 Pfizer Inc. 4-benzylidene-3-methylpiperidine aryl carboxamide compounds useful as faah inhibitors
US20110060012A1 (en) * 2008-04-17 2011-03-10 Pfizer Inc. 4-[3-(aryloxy)benzylidene]-3-methyl piperidine 5-membered aryl carboxamide compounds useful as faah inhibitors
JP2011518146A (ja) * 2008-04-17 2011-06-23 ファイザー・インク Ｆａａｈ阻害剤として有用な４−［３−（アリールオキシ）ベンジリデン］−３−メチルピペリジンアリールカルボキサミド化合物
CA2719785A1 (en) * 2008-04-17 2009-10-22 Pfizer Inc. Ether benzylidene piperidine aryl carboxamide compounds
JP5658138B2 (ja) * 2008-04-23 2015-01-21 ライジェル ファーマシューティカルズ， インコーポレイテッド 代謝障害の処置のためのカルボキサミド化合物
WO2012033069A1 (ja) * 2010-09-07 2012-03-15 大鵬薬品工業株式会社 プロスタグランジンd合成酵素を阻害するピペリジン化合物
UY36391A (es) * 2014-11-05 2016-06-01 Flexus Biosciences Inc Compuestos moduladores de la enzima indolamina 2,3-dioxigenasa (ido1), sus métodos de síntesis y composiciones farmacèuticas que las contienen
EP3886854A4 (en) 2018-11-30 2022-07-06 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof

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US3577415A (en) * 1968-12-23 1971-05-04 Robins Co Inc A H 1-substituted-3-substituted phenoxypyrrolidines
US4263438A (en) * 1977-09-13 1981-04-21 Pfizer Inc. 3-[2,4-(Disubstituted)-phenyl]azacycloalkanones as analgesics
US4452809A (en) * 1980-03-10 1984-06-05 A. H. Robins Company, Inc. Trans-4-(2-chlorophenoxy)-1-ethyl-3-pyrrolidinol and anti-depressant use thereof
ATE201669T1 (de) * 1991-04-17 2001-06-15 Upjohn Co Substituierte (s)-3-phenylpiperidin derivate, deren herstellung und deren verwendung als dopamin autorezeptor antagonisten
US5519134A (en) * 1994-01-11 1996-05-21 Isis Pharmaceuticals, Inc. Pyrrolidine-containing monomers and oligomers
EP0880501A1 (en) * 1996-02-02 1998-12-02 Zeneca Limited Heterocyclic compounds useful as pharmaceutical agents
HRP970371A2 (en) * 1996-07-13 1998-08-31 Kathryn Jane Smith Heterocyclic compounds
US6022884A (en) * 1997-11-07 2000-02-08 Amgen Inc. Substituted pyridine compounds and methods of use
AR033517A1 (es) * 2000-04-08 2003-12-26 Astrazeneca Ab Derivados de piperidina, proceso para su preparacion y uso de estos derivados en la fabricacion de medicamentos
AUPR362001A0 (en) * 2001-03-08 2001-04-05 Fujisawa Pharmaceutical Co., Ltd. New compound
DE10217006A1 (de) * 2002-04-16 2003-11-06 Merck Patent Gmbh Substituierte Indole
WO2004009603A1 (en) * 2002-07-24 2004-01-29 Eli Lilly And Company Dihydro-dibenzo[b,e]oxepine based selective estrogen receptor modulators, compositions and methods
SE0300456D0 (sv) * 2003-02-19 2003-02-19 Astrazeneca Ab Novel compounds
SE0301368D0 (sv) * 2003-05-09 2003-05-09 Astrazeneca Ab Chemical compounds
CA2528669A1 (en) * 2003-06-09 2005-01-20 The Regents Of The University Of Michigan Compositions and methods for treating and diagnosing cancer
US7094791B2 (en) * 2003-07-31 2006-08-22 Avalon Pharmaceuticals, Inc. Derivatives of 3-hydroxy-pyrrole-2,4-dicarboxylic acid and uses thereof
AU2004273658A1 (en) * 2003-09-19 2005-03-31 Wisconsin Alumni Research Foundation (Warf) Pharmaceutical compositions and methods comprising combinations of 2-alkylidene-19-nor-vitamin D derivatives and an estrogen agonist/antagonist
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JPWO2005073210A1 (ja) * 2004-01-28 2007-09-06 キッセイ薬品工業株式会社 新規なベンゾフラン誘導体、それを含有する医薬組成物およびそれらの用途
US20070232659A1 (en) * 2004-06-18 2007-10-04 Dan Peters Novel Alkyl Substituted Piperidine Derivatives as Monoamine Neurotransmitter Re-Uptake Inhibitors
MY179032A (en) * 2004-10-25 2020-10-26 Cancer Research Tech Ltd Ortho-condensed pyridine and pyrimidine derivatives (e.g.purines) as protein kinase inhibitors
DE602005019316D1 (en) * 2004-11-24 2010-03-25 Lilly Co Eli Aromatische etherderivate als thrombin-hemmer
AP2007004047A0 (en) * 2005-01-20 2007-06-30 Pfizer Ltd Substituted triazole derivatives as oxtocin antagonists
FR2884516B1 (fr) * 2005-04-15 2007-06-22 Cerep Sa Antagonistes npy, preparation et utilisations
JP2008546784A (ja) * 2005-06-20 2008-12-25 シェーリング コーポレイション ヒスタミンｈ３アンタゴニストとして有用なピペリジン誘導体
US20090036429A1 (en) * 2006-02-17 2009-02-05 Ohler Norman E Hydroxypiperidine Derivatives and Uses Thereof

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