JP2010031006A

JP2010031006A - 有機化合物の使用

有機化合物の使用 Download PDF

Info

Publication number: JP2010031006A
Authority: JP; Japan
Prior art keywords: salt; type; diabetes; pharmaceutically acceptable; group
Prior art date: 2008-07-17
Legal status : Pending

Application number

JP2009165467A

Other languages

English (en)

Japanese (ja)

Other versions

JP2010031006A5 (cg-RX-API-DMAC7.html

Inventor

Baker Kenneth

ケネス・ベーカー

Kumar Rajesh

ラジェシュ・クマール

Singh Vivek

ヴィヴェク・シン

Current Assignee

Novartis AG

Original Assignee

Novartis AG

Priority date

2008-07-17

Filing date

2009-07-14

Publication date

2010-02-12

2009-07-14 Application filed by Novartis AG filed Critical Novartis AG

2010-02-12 Publication of JP2010031006A publication Critical patent/JP2010031006A/ja

2012-08-02 Publication of JP2010031006A5 publication Critical patent/JP2010031006A5/ja

Status Pending legal-status Critical Current

Links

150000002894 organic compounds Chemical class 0.000 title 1
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NOESYZHRGYRDHS-UHFFFAOYSA-N insulin Chemical compound N1C(=O)C(NC(=O)C(CCC(N)=O)NC(=O)C(CCC(O)=O)NC(=O)C(C(C)C)NC(=O)C(NC(=O)CN)C(C)CC)CSSCC(C(NC(CO)C(=O)NC(CC(C)C)C(=O)NC(CC=2C=CC(O)=CC=2)C(=O)NC(CCC(N)=O)C(=O)NC(CC(C)C)C(=O)NC(CCC(O)=O)C(=O)NC(CC(N)=O)C(=O)NC(CC=2C=CC(O)=CC=2)C(=O)NC(CSSCC(NC(=O)C(C(C)C)NC(=O)C(CC(C)C)NC(=O)C(CC=2C=CC(O)=CC=2)NC(=O)C(CC(C)C)NC(=O)C(C)NC(=O)C(CCC(O)=O)NC(=O)C(C(C)C)NC(=O)C(CC(C)C)NC(=O)C(CC=2NC=NC=2)NC(=O)C(CO)NC(=O)CNC2=O)C(=O)NCC(=O)NC(CCC(O)=O)C(=O)NC(CCCNC(N)=N)C(=O)NCC(=O)NC(CC=3C=CC=CC=3)C(=O)NC(CC=3C=CC=CC=3)C(=O)NC(CC=3C=CC(O)=CC=3)C(=O)NC(C(C)O)C(=O)N3C(CCC3)C(=O)NC(CCCCN)C(=O)NC(C)C(O)=O)C(=O)NC(CC(N)=O)C(O)=O)=O)NC(=O)C(C(C)CC)NC(=O)C(CO)NC(=O)C(C(C)O)NC(=O)C1CSSCC2NC(=O)C(CC(C)C)NC(=O)C(NC(=O)C(CCC(N)=O)NC(=O)C(CC(N)=O)NC(=O)C(NC(=O)C(N)CC=1C=CC=CC=1)C(C)C)CC1=CN=CN1 NOESYZHRGYRDHS-UHFFFAOYSA-N 0.000 claims abstract description 57
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