JP2008513427A5 - - Google Patents

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Publication number
JP2008513427A5
JP2008513427A5 JP2007531832A JP2007531832A JP2008513427A5 JP 2008513427 A5 JP2008513427 A5 JP 2008513427A5 JP 2007531832 A JP2007531832 A JP 2007531832A JP 2007531832 A JP2007531832 A JP 2007531832A JP 2008513427 A5 JP2008513427 A5 JP 2008513427A5
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JP
Japan
Prior art keywords
pharmacology
medicament
inhibition
diseases
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007531832A
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English (en)
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JP2008513427A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/GB2005/003584 external-priority patent/WO2006032852A1/en
Publication of JP2008513427A publication Critical patent/JP2008513427A/ja
Publication of JP2008513427A5 publication Critical patent/JP2008513427A5/ja
Withdrawn legal-status Critical Current

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Claims (1)

  1. リポキシゲナーゼの活性阻害が所望される及び／又は必要とされる疾患の治療のための医薬において、但し書きを含まない、請求項１ないし２１のいずれか１項に記載の式Ｉの化合物、又はその薬学的に許容可能な塩を含有することを特徴とする医薬。
JP2007531832A 2004-09-20 2005-09-19 炎症の治療に有用なピラゾール化合物 Withdrawn JP2008513427A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61095204P 2004-09-20 2004-09-20
PCT/GB2005/003584 WO2006032852A1 (en) 2004-09-20 2005-09-19 Pyrazole compounds useful uin the treatment of inflammation

Publications (2)

Publication Number Publication Date
JP2008513427A JP2008513427A (ja) 2008-05-01
JP2008513427A5 true JP2008513427A5 (ja) 2008-11-20

Family

ID=34956280

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007531832A Withdrawn JP2008513427A (ja) 2004-09-20 2005-09-19 炎症の治療に有用なピラゾール化合物

Country Status (4)

Country Link
US (1) US20080090836A1 (ja)
EP (1) EP1794130A1 (ja)
JP (1) JP2008513427A (ja)
WO (1) WO2006032852A1 (ja)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008513426A (ja) * 2004-09-20 2008-05-01 バイオリポックス エービー 炎症の治療に有用なピラゾール化合物
TW200800911A (en) * 2005-10-20 2008-01-01 Biolipox Ab Pyrazoles useful in the treatment of inflammation
TW200732320A (en) * 2005-10-31 2007-09-01 Biolipox Ab Pyrazoles useful in the treatment of inflammation
AU2006310367A1 (en) * 2005-10-31 2007-05-10 Biolipox Ab Triazole compounds as lipoxygenase inhibitors
WO2007052000A1 (en) * 2005-11-01 2007-05-10 Biolipox Ab Pyrazoles useful in the treatment of inflammation
BR122013027950A2 (pt) * 2008-12-24 2019-12-10 BIAL PORTELA & Cª S A compostos farmacêuticos
US9238643B2 (en) 2010-09-06 2016-01-19 Guangzhou Institutes Of Biomedicine And Health, Chinese Academy Of Sciences Amide compounds
JP6520588B2 (ja) * 2015-09-10 2019-05-29 日本軽金属株式会社 スルホニルブロマイド化合物類の製造方法

Family Cites Families (26)

* Cited by examiner, † Cited by third party
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US5464860A (en) * 1988-11-30 1995-11-07 Novapharme N(pyrazol-3-yl) benzamides and pharmaceutical compositions
FR2639636B1 (fr) * 1988-11-30 1994-03-04 Novapharme Nouveaux composes heterocycliques a activite anticonvulsivante, procede de preparation et compositions therapeutiques les contenant
FR2662692B1 (fr) * 1990-05-30 1995-04-28 Novapharme Derives heterocycliques doues d'activite anticonvulsivante, procede de preparation et composition pharmaceutique.
US5258397A (en) * 1988-11-30 1993-11-02 Novapharme 3-Isoxazoyl derivatives endowed with anticonvulsant activity, procedure for their preparation and their pharmaceutical compositions
DE69329240D1 (de) * 1992-05-20 2000-09-21 Merck & Co Inc 17-ether und thioether von 4-aza-steroiden
ATE198601T1 (de) * 1992-05-20 2001-01-15 Merck & Co Inc Ester derivate von 4-aza-steroiden
US6372770B1 (en) * 1994-10-12 2002-04-16 Euro-Celtique, S.A. Benzoxazoles
US5665737B1 (en) * 1994-10-12 1999-02-16 Euro Celtique Sa Substituted benzoxazoles
US5663357A (en) * 1995-11-22 1997-09-02 Allergan Substituted heteroarylamides having retinoid-like biological activity
AUPP042397A0 (en) * 1997-11-18 1997-12-11 Fujisawa Pharmaceutical Co., Ltd. 5-arylpyrazole compounds
WO2001019788A2 (en) * 1999-09-17 2001-03-22 Cor Therapeutics, Inc. BENZAMIDES AND RELATED INHIBITORS OF FACTOR Xa
US7393842B2 (en) * 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
GB0002666D0 (en) * 2000-02-04 2000-03-29 Univ London Blockade of voltage dependent sodium channels
JP2004502642A (ja) * 2000-02-11 2004-01-29 ブリストル−マイヤーズ　スクイブ　カンパニー カンナビノイドレセプターモジュレーター、それらの製造方法、および呼吸系および非呼吸系疾患の処置のためのカンナビノイドレセプターモジュレーターの使用
US20040043904A1 (en) * 2000-09-22 2004-03-04 Hiroshi Yamaguchi N-(4-pyrazolyl) amide derivatives, chemicals for agricultural and horticultural use, and usage of the same
JP4465133B2 (ja) * 2001-02-08 2010-05-19 クミアイ化学工業株式会社 イソオキサゾリン誘導体及びこれを有効成分とする除草剤
EP1451160B1 (en) * 2001-11-01 2010-01-13 Icagen, Inc. Pyrazole-amides for use in the treatment of pain
US7016421B2 (en) * 2001-11-15 2006-03-21 Hrl Laboratories, Llc Time-interleaved delta sigma analog to digital modulator
TWI263497B (en) * 2002-03-29 2006-10-11 Lilly Co Eli Pyridinoylpiperidines as 5-HT1F agonists
WO2004039795A2 (en) * 2002-10-29 2004-05-13 Fujisawa Pharmaceutical Co., Ltd. Amide compounds for the treatment of hyperlipidemia
JP2006512314A (ja) * 2002-11-01 2006-04-13 バーテックス ファーマシューティカルズ インコーポレイテッド Ｊａｋインヒビターおよび他のプロテインキナーゼインヒビターとしての組成物の使用
EP1571671A4 (en) * 2002-12-13 2008-04-02 Matsushita Electric Ind Co Ltd OPTICAL DISK DEVICE
US7429581B2 (en) * 2002-12-23 2008-09-30 Sanofi-Aventis Deutschland Gmbh Pyrazole-derivatives as factor Xa inhibitors
JP2006520373A (ja) * 2003-03-14 2006-09-07 バイオリポックス エービー 炎症の治療に有用なピラゾール化合物
SE0300705D0 (sv) * 2003-03-14 2003-03-14 Biolipox Ab New compounds
JP2007525460A (ja) * 2003-04-25 2007-09-06 オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド ｃ−ｆｍｓキナーゼ阻害剤

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