JP2008512477A - 新規化合物およびその標的に関連する組成物ならびに方法 - Google Patents

新規化合物およびその標的に関連する組成物ならびに方法 Download PDF

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JP2008512477A
JP2008512477A JP2007531319A JP2007531319A JP2008512477A JP 2008512477 A JP2008512477 A JP 2008512477A JP 2007531319 A JP2007531319 A JP 2007531319A JP 2007531319 A JP2007531319 A JP 2007531319A JP 2008512477 A JP2008512477 A JP 2008512477A
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ゲイリー ディー. グリック
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University of Michigan
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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  • Diabetes (AREA)
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  • Cardiology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
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  • Obesity (AREA)
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  • Pulmonology (AREA)
  • Psychiatry (AREA)
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  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Vascular Medicine (AREA)
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  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
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JP2007531319A 2004-09-07 2005-09-07 新規化合物およびその標的に関連する組成物ならびに方法 Pending JP2008512477A (ja)

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US10/935,333 US20050113460A1 (en) 1999-04-30 2004-09-07 Compositions and methods relating to novel compounds and targets thereof
PCT/US2005/031942 WO2006029245A2 (en) 2004-09-07 2005-09-07 Compositions and methods relating to novel compounds and targets thereof

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JP (2) JP2008512477A (US20050113460A1-20050526-C00003.png)
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JP2012197305A (ja) * 2004-09-07 2012-10-18 Regents Of The Univ Of Michigan 新規化合物およびその標的に関連する組成物ならびに方法
US8759340B2 (en) 2007-11-06 2014-06-24 The Regents Of The University Of Michigan Benzodiazepinone compounds useful in the treatment of skin conditions
US8791104B2 (en) 2005-11-01 2014-07-29 The Regents Of The University Of Michigan 1,4-benzodiazepine-2,5-diones with therapeutic properties
US8809323B2 (en) 1999-04-30 2014-08-19 The Regents Of The University Of Michigan Therapeutic applications of pro-apoptotic benzodiazepines

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US20040176358A1 (en) * 1999-04-30 2004-09-09 The Regents Of The University Of Michigan Compositions and methods relating to novel compounds and targets thereof
US7276348B2 (en) * 1999-04-30 2007-10-02 Regents Of The University Of Michigan Compositions and methods relating to F1F0-ATPase inhibitors and targets thereof
US20060025388A1 (en) 1999-04-30 2006-02-02 Glick Gary D Compositions and methods relating to novel compounds and targets thereof
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US9011329B2 (en) 2004-04-19 2015-04-21 Searete Llc Lumenally-active device
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JP2007533753A (ja) * 2004-04-23 2007-11-22 タケダ サン ディエゴ インコーポレイテッド インドール誘導体及びキナーゼ阻害剤としてのその使用
US20050272723A1 (en) * 2004-04-27 2005-12-08 The Regents Of The University Of Michigan Methods and compositions for treating diseases and conditions associated with mitochondrial function
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US7638624B2 (en) * 2005-01-03 2009-12-29 The Regents Of The University Of Michigan Compositions and methods relating to novel benzodiazepine compounds and derivatives
US20070043033A1 (en) * 2005-06-01 2007-02-22 The Regents Of The University Of Michigan Unsolvated benzodiazepine compositions and methods
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US20070105844A1 (en) * 2005-10-26 2007-05-10 Regents Of The University Of Michigan Therapeutic compositions and methods
JP2009513644A (ja) * 2005-10-26 2009-04-02 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン 治療組成物および方法
US20120035437A1 (en) 2006-04-12 2012-02-09 Searete Llc, A Limited Liability Corporation Of The State Of Delaware Navigation of a lumen traveling device toward a target
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JP2010505961A (ja) * 2006-10-09 2010-02-25 タケダ サン ディエゴ インコーポレイテッド キナーゼ阻害剤
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AU2008298870C1 (en) 2007-09-14 2014-10-09 The Regents Of The University Of Michigan F1F0-ATPase inhibitors and related methods
US8598150B1 (en) 2008-04-02 2013-12-03 Jonathan R. Brestoff Composition and method for affecting obesity and related conditions
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JP5856063B2 (ja) 2009-11-17 2016-02-09 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン 治療特性を有する1,4−ベンゾジアゼピン−2,5−ジオンおよび関連化合物
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