JP2007532593A - Ｍｃｈ拮抗作用を有する新規アルキン化合物及び前記化合物を含有する薬物 - Google Patents

Ｍｃｈ拮抗作用を有する新規アルキン化合物及び前記化合物を含有する薬物 Download PDF

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JP2007532593A
JP2007532593A JP2007507706A JP2007507706A JP2007532593A JP 2007532593 A JP2007532593 A JP 2007532593A JP 2007507706 A JP2007507706 A JP 2007507706A JP 2007507706 A JP2007507706 A JP 2007507706A JP 2007532593 A JP2007532593 A JP 2007532593A
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alkyl
group
phenyl
cycloalkyl
hydroxy
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JP2007532593A5 (cg-RX-API-DMAC7.html
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ディルク シュテンカンプ
シュテファン ゲオルク ミューラー
フィリップ ルシュテンベルガー
リンツ トルシュテン レーマン
レオ トーマス
マルクス シンドラー
ゲラルト ユールゲン ロート
クラウス ルドルフ
ラルフ エル ハー ロッツ
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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Application filed by ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング filed Critical ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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  • Health & Medical Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Rheumatology (AREA)
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  • Vascular Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Child & Adolescent Psychology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
JP2007507706A 2004-04-14 2005-04-08 Ｍｃｈ拮抗作用を有する新規アルキン化合物及び前記化合物を含有する薬物 Pending JP2007532593A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004017935A DE102004017935A1 (de) 2004-04-14 2004-04-14 Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel
PCT/EP2005/003683 WO2005103031A1 (de) 2004-04-14 2005-04-08 Neue alkin-verbindungen mit mch-antagonistischer wirkung und diese verbindungen enthaltende arzneimittel

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JP2007532593A true JP2007532593A (ja) 2007-11-15
JP2007532593A5 JP2007532593A5 (cg-RX-API-DMAC7.html) 2008-05-29

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JP2007507706A Pending JP2007532593A (ja) 2004-04-14 2005-04-08 Ｍｃｈ拮抗作用を有する新規アルキン化合物及び前記化合物を含有する薬物

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EP (1) EP1740572A1 (cg-RX-API-DMAC7.html)
JP (1) JP2007532593A (cg-RX-API-DMAC7.html)
AR (1) AR048692A1 (cg-RX-API-DMAC7.html)
CA (1) CA2559021A1 (cg-RX-API-DMAC7.html)
DE (1) DE102004017935A1 (cg-RX-API-DMAC7.html)
PE (1) PE20060333A1 (cg-RX-API-DMAC7.html)
TW (1) TW200602025A (cg-RX-API-DMAC7.html)
UY (1) UY28853A1 (cg-RX-API-DMAC7.html)
WO (1) WO2005103031A1 (cg-RX-API-DMAC7.html)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007532596A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗効果を有する新規アルキン化合物及び前記化合物を含有する薬物
JP2007532595A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗作用を有する新規アルキン化合物及び該化合物を含む医薬

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7452911B2 (en) 2002-10-31 2008-11-18 Boehringer Ingelheim Pharma Gmbh & Co. Kg Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds
JP5073746B2 (ja) 2006-08-25 2012-11-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗作用を有する新規ピリドン誘導体及びこの化合物を含む薬物
CA2671984A1 (en) 2006-12-11 2008-06-19 Boehringer Ingelheim International Gmbh New pyridazine derivatives with mch antagonistic activity and medicaments comprising these compounds
CN118878822B (zh) * 2024-07-05 2025-09-16 江苏师范大学 一种阳离子自由基型三嗪基聚乙炔及其制备方法与光催化应用

Citations (5)

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Publication number Priority date Publication date Assignee Title
US5856510A (en) * 1996-12-16 1999-01-05 Allelix Biopharmaceuticals Inc. 5-alkenyl and 5-alkynyl indole compounds
JP2001509504A (ja) * 1997-07-11 2001-07-24 ノバルティス アクチエンゲゼルシャフト ピリジン誘導体
JP2006511492A (ja) * 2002-10-31 2006-04-06 ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト Ｍｃｈ拮抗活性を有する新規アルキン化合物及びこれらの化合物を含む薬物
JP2007532595A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗作用を有する新規アルキン化合物及び該化合物を含む医薬
JP2007532596A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗効果を有する新規アルキン化合物及び前記化合物を含有する薬物

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7115750B1 (en) * 1999-09-20 2006-10-03 Takeda Pharmaceutical Company Limited Melanin concentrating hormone antagonist

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5856510A (en) * 1996-12-16 1999-01-05 Allelix Biopharmaceuticals Inc. 5-alkenyl and 5-alkynyl indole compounds
JP2001509504A (ja) * 1997-07-11 2001-07-24 ノバルティス アクチエンゲゼルシャフト ピリジン誘導体
JP2006511492A (ja) * 2002-10-31 2006-04-06 ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト Ｍｃｈ拮抗活性を有する新規アルキン化合物及びこれらの化合物を含む薬物
JP2007532595A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗作用を有する新規アルキン化合物及び該化合物を含む医薬
JP2007532596A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗効果を有する新規アルキン化合物及び前記化合物を含有する薬物

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007532596A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗効果を有する新規アルキン化合物及び前記化合物を含有する薬物
JP2007532595A (ja) * 2004-04-14 2007-11-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｍｃｈ拮抗作用を有する新規アルキン化合物及び該化合物を含む医薬

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AR048692A1 (es) 2006-05-17
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EP1740572A1 (de) 2007-01-10
UY28853A1 (es) 2005-11-30
DE102004017935A1 (de) 2005-11-03
CA2559021A1 (en) 2005-11-03
TW200602025A (en) 2006-01-16

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