JP2006501215A5 - - Google Patents

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Publication number
JP2006501215A5
JP2006501215A5 JP2004527226A JP2004527226A JP2006501215A5 JP 2006501215 A5 JP2006501215 A5 JP 2006501215A5 JP 2004527226 A JP2004527226 A JP 2004527226A JP 2004527226 A JP2004527226 A JP 2004527226A JP 2006501215 A5 JP2006501215 A5 JP 2006501215A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
composition according
treating
rheumatoid arthritis
osteoarthritis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2004527226A
Other languages
English (en)
Japanese (ja)
Other versions
JP2006501215A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2003/003613 external-priority patent/WO2004014892A1/en
Publication of JP2006501215A publication Critical patent/JP2006501215A/ja
Publication of JP2006501215A5 publication Critical patent/JP2006501215A5/ja
Pending legal-status Critical Current

Links

JP2004527226A 2002-08-13 2003-08-03 マトリックスメタロプロテイナーゼ阻害剤としての単環式誘導体 Pending JP2006501215A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40304002P 2002-08-13 2002-08-13
PCT/IB2003/003613 WO2004014892A1 (en) 2002-08-13 2003-08-03 Monocyclic derivatives as matrix metalloproteinase inhibitors

Publications (2)

Publication Number Publication Date
JP2006501215A JP2006501215A (ja) 2006-01-12
JP2006501215A5 true JP2006501215A5 (enExample) 2006-09-14

Family

ID=31715927

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004527226A Pending JP2006501215A (ja) 2002-08-13 2003-08-03 マトリックスメタロプロテイナーゼ阻害剤としての単環式誘導体

Country Status (8)

Country Link
US (1) US7132424B2 (enExample)
EP (1) EP1537098A1 (enExample)
JP (1) JP2006501215A (enExample)
AU (1) AU2003253176A1 (enExample)
BR (1) BR0313459A (enExample)
CA (1) CA2494014A1 (enExample)
MX (1) MXPA05001603A (enExample)
WO (1) WO2004014892A1 (enExample)

Families Citing this family (22)

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MXPA04002537A (es) 2001-10-12 2004-05-31 Warner Lambert Co Alquinos como inhibidores de metaloproteinasa de matriz.
AU2003237532B2 (en) 2002-06-12 2009-07-30 Symphony Evolution, Inc. Human ADAM-10 inhibitors
PA8578101A1 (es) * 2002-08-13 2004-05-07 Warner Lambert Co Derivados de heterobiarilo como inhibidores de metaloproteinasa de la matriz
EP1394159A1 (fr) * 2002-08-13 2004-03-03 Warner-Lambert Company LLC Nouveaux dérivés de thiophène, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
US20040142950A1 (en) * 2003-01-17 2004-07-22 Bunker Amy Mae Amide and ester matrix metalloproteinase inhibitors
US20060247231A1 (en) * 2003-12-18 2006-11-02 Warner-Lambert Company Llc Amide and ester matrix metalloproteinase inhibitors
AP2007004244A0 (en) 2005-05-10 2007-12-31 Intermune Inc Method of modulating stress-activated protein kinase system
EP2296653B1 (en) 2008-06-03 2016-01-27 Intermune, Inc. Compounds and methods for treating inflammatory and fibrotic disorders
WO2013097052A1 (en) 2011-12-30 2013-07-04 Abbott Laboratories Bromodomain inhibitors
AR092742A1 (es) 2012-10-02 2015-04-29 Intermune Inc Piridinonas antifibroticas
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US9580396B2 (en) 2012-12-21 2017-02-28 Merck Sharp & Dohme Corp. C6-spiro iminothiadiazine dioxides as BACE inhibitors, compositions, and their use
RU2692485C2 (ru) 2014-04-02 2019-06-25 Интермьюн, Инк. Противофиброзные пиридиноны
AU2017251537B2 (en) 2016-04-15 2020-10-08 Abbvie Inc. Bromodomain inhibitors
EP3529245A4 (en) 2016-10-24 2020-12-23 Yumanity Therapeutics, Inc. COMPOUNDS AND USES OF THE LATEST
MA47212A (fr) 2017-01-06 2019-11-13 Yumanity Therapeutics Inc Méthodes de traitement de troubles neurologiques
WO2019084157A1 (en) 2017-10-24 2019-05-02 Yumanity Therapeutics, Inc. COMPOUNDS AND USES THEREOF
ES3043183T3 (en) 2018-03-23 2025-11-25 Janssen Pharmaceutica Nv Compounds and uses thereof
AU2019387370A1 (en) 2018-11-30 2021-06-10 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
MA54829A (fr) 2019-01-24 2021-12-01 Yumanity Therapeutics Inc Composés et leurs utilisations
EA202192047A1 (ru) 2019-11-13 2021-12-08 Юманити Терапьютикс, Инк. Соединения и их применение
EP4685143A1 (en) * 2023-03-21 2026-01-28 Vivozon,Inc. Double regulator for mglur5 and hdac6 and use thereof

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