JP2005126418A - Substituted benzanilide and pest control agent - Google Patents

Abstract

<P>PROBLEM TO BE SOLVED: To provide a new agrochemical, particularly insecticidal and acaricidal agent. <P>SOLUTION: The pest control agent includes a substituted benzanilide represented by general formula (1) [wherein W<SP>1</SP>and W<SP>2</SP>are each O or S atom; X is a halogen atom or the like; Y is a 1-6C alkyl or the like; R<SP>1</SP>is a 1-6C alkylthio(a 1-6C)alkyl; R<SP>2</SP>and R<SP>3</SP>are each H or the like; R<SP>4</SP>is a 1-6C haloalkyl; R<SP>5</SP>is a phenoxy(1-6C)haloalkyl, or L or the like; R<SP>6</SP>is H atom or a 1-6C alkylcarbonyl; L represents an aromatic heterocyclic ring, for example, L-1 through L-4, L-8 through L-13, L-15 through L-23, L-45 through L-52 or L-53 and the like; Z is a halogen atom or a 1-6C haloalkoxy(1-6C)haloalkoxy; m and n are each independently an integer of 0 through 4 and p1 is an integer of 1 through 5]. <P>COPYRIGHT: (C)2005,JPO&NCIPI

Description

  The present invention relates to a novel substituted benzanilide compound and a salt thereof, and a pest control agent comprising the compound as an active ingredient. The pest control agent in the present invention means a pest control agent for harmful arthropods in the fields of agriculture, horticulture, animal husbandry, and hygiene (animal medicine, household use, commercial insecticide). The agrochemical in the present invention means an insecticide / acaricide, nematicide, herbicide and fungicide in the field of agriculture and horticulture.

Conventionally, it is known that a specific substituted benzanilide derivative has a cytokine production inhibitory activity, a vasopressin antagonistic activity, and the like, and is used as a pharmaceutical product (see, for example, Patent Documents 1 to 3). Moreover, it is known that a specific substituted benzanilide derivative has insecticidal activity (for example, refer patent documents 4-12). However, there is no disclosure regarding the substituted benzanilide compound according to the present invention.
International Publication No. 98/024771 Pamphlet WO99 / 051580 pamphlet JP 2002-249473 A European Patent Application No. 0919542 European Patent Application No. 1006107 International Publication No. 01/021576 pamphlet International Publication No. 01/046124 Pamphlet JP 2001-335559 A International Publication No. 02/062807 Pamphlet International Publication No. 02/094765 Pamphlet International Publication No. 2004/000796 Pamphlet International Publication No. 2004/018415 Pamphlet

  Pest control agents such as insecticides and fungicides have been used for many years, and in recent years, pests have acquired resistance, making it difficult to control them with conventionally used insecticides and fungicides. Also, some of the existing pest control agents are highly toxic or some are disrupting the ecosystem due to long-term persistence. Under such circumstances, development of a novel pesticide with low toxicity and low persistence is always expected.

  As a result of intensive research aimed at solving the above problems, the present inventors have found that the novel substituted benzanilide compound represented by the following general formula (1) according to the present invention has excellent pest control activity, particularly insecticide The present invention was completed by discovering that it is a very useful compound that exhibits acaricidal activity and has almost no adverse effect on non-target organisms such as mammals, fish and beneficial insects.

  That is, the present invention relates to the following [1] to [8].

  [1] General formula (1):

[Wherein, W ¹ and W ² each independently represent an oxygen atom or a sulfur atom,
X is a halogen atom, cyano, nitro, _{azido, -SCN, -SF 5, C 1} ~C 6 alkyl, optionally substituted by R ⁷ (C ₁ ~C ₆₎ alkyl, C ₃ -C ₈ cycloalkyl , optionally substituted by R ⁷ (C ₃ ~C ₈₎ cycloalkyl, C ₂ -C ₆ alkenyl, optionally substituted by R ⁷ (C ₂ ~C ₆₎ alkenyl, C ₃ -C ₈ cycloalkenyl , C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₂ -C ₆ alkynyl, optionally substituted by R ⁷ (C ₂ ~C ₆₎ ^{alkynyl, -OH, -OR 8, -OS (} O) 2 R 8, -SH, -S (O) _r R ⁸ , -CHO, -C (O) R ⁹ , -C (O) OR ⁹ , -C (O) SR ⁹ , -C (O) NHR ¹⁰ , -C ( O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , -CH = NOR ¹¹ , -C (R ⁹ ) = NOR ¹¹ , -S (O) ₂ OR ⁹ , -S (O) ₂ NHR ¹⁰ , -S (O) ₂ N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴⁾ R ^12, phenyl, (Z) phenyl substituted by _p1, represents L or M, when m represents 2, 3 or 4, each X May be the or different from each other the same as each other,
Further, when two Xs are adjacent to each other, the two adjacent Xs are -CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ O-, -CH ₂ OCH _2- , -OCH ₂ O-, -CH ₂ CH ₂ S-, -CH ₂ SCH _2- , -CH ₂ CH ₂ N (R ¹⁵ )-, -CH ₂ N (R ¹⁵ ) CH _2- , -CH ₂ CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ CH ₂ O-, -CH ₂ CH ₂ OCH _2- , -CH ₂ OCH ₂ O-, -OCH ₂ CH ₂ O-, -OCH ₂ CH ₂ S-, -CH ₂ CH = CH-,- OCH = CH-, -SCH = CH-, -N (R ¹⁵ ) CH = CH-, -OCH = N-, -SCH = N-, -N (R ¹⁵ ) CH = N-, -N (R ¹⁵ By forming N = CH-, -CH = CHCH = CH-, -OCH ₂ CH = CH-, -N = CHCH = CH-, -N = CHCH = N- or -N = CHN = CH- A 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each of two Xs is bonded. At this time, the hydrogen atom bonded to each carbon atom forming the ring is optionally substituted by Z. In addition, when simultaneously substituted with two or more Z, each Z may be the same as or different from each other,
Y is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, optionally substituted by R ⁷ (C ₁ ~C ₆₎ alkyl, C ₃ -C ₈ cycloalkyl, -OR ^8, -S (O ) _r R ⁸ , —NH ₂ , C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino or —Si (R ¹³ ) (R ¹⁴ ) R ¹² , n is 2, 3 or 4 Each Y may be the same as or different from each other;
Further, when two Ys are adjacent to each other, the two adjacent Ys are —CH ₂ CH ₂ CH ₂ —, —CH ₂ CH ₂ O—, —CH ₂ OCH ₂ —, —OCH ₂ O—, —CH ₂ CH ₂ S-, -CH ₂ SCH _2- , -SCH ₂ S-, -CH ₂ CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ CH ₂ O-, -CH ₂ CH ₂ OCH ₂ -,- By forming CH ₂ OCH ₂ O-, -OCH ₂ CH ₂ O-, -OCH ₂ CH ₂ S-, -SCH ₂ CH ₂ S-, -OCH = N- or -SCH = N- A 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each Y is bonded, and at this time, the hydrogen atom bonded to each carbon atom forming the ring may be optionally substituted by Z Furthermore, when two or more Z are substituted at the same time, each Z may be the same as or different from each other,
R ¹ is hydrogen atom, cyano, optionally substituted by C ₁ -C ₁₂ alkyl, optionally substituted by R ¹⁶ (C ₁ ~C ₁₂₎ alkyl, C ₃ -C ₁₂ cycloalkyl, R ¹⁶ ( C ₃ -C ₁₂₎ cycloalkyl, C ₃ -C ₁₂ alkenyl, optionally substituted by R ¹⁶ (C ₃ ~C ₁₂₎ alkenyl, C ₃ -C ₁₂ cycloalkenyl, C ₃ -C ₁₂ halo cycloalkenyl, C ₃ -C ₁₂ alkynyl, optionally substituted by R ¹⁶ (C ₃ ~C ₁₂₎ alkynyl, -OH, C ₁ -C ₈ alkoxy, C ₃ -C ₈ alkenyloxy, C ₃ -C ₈ haloalkenyloxy , phenoxy, (Z) _p1 phenoxy substituted by phenyl (C ₁ ~C ₄₎ alkoxy, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ ^{alkoxy, -N (R 20) R 19} , Phenyl, (Z) represents phenyl, L or M substituted by _p1 ,
R ² and R ³ are each independently a hydrogen atom, cyano, C ₁ -C ₁₂ alkyl, (C ₁ -C ₁₂ ) alkyl optionally substituted with R ¹⁶ , C ₃ -C ₁₂ alkenyl, C _3- C ₁₂ haloalkenyl, C ₃ -C ₁₂ alkynyl, C ₃ -C ₁₂ haloalkynyl, -OH, C ₁ -C ₈ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z) phenylthio substituted by _{p1, -S (O) 2 R} 9, -SN (R 18) R 17, -S (O) 2 N (R 10) R 9, -N (R 20) R 19, -C (O) R ⁹ , -C (O) OR ⁹ , -C (O) SR ⁹ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) N (R 10) R 9, or represents phenyl which is substituted by phenyl or (Z) _p1, or, R ² is formed a C ₂ -C ₆ alkylene chain together with R ¹ This represents that a 3- to 7-membered ring may be formed together with the nitrogen atom to be bonded. At this time, the alkylene chain has an oxygen atom, a sulfur atom or a nitrogen atom. Pieces comprise may, and halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ haloalkyl group, C ₁ -C ₆ alkoxy group, C ₁ -C ₆ alkylcarbonyl group or a C ₁ -C ₆ alkoxycarbonyl group Optionally substituted by
R ⁴ is optionally substituted by C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, R ²¹ (C ₁ ~C ₆₎ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, optionally substituted by R ²¹ (C ₃ ~C ₈₎ cycloalkyl, optionally substituted by R ²¹ (C ₃ ~C ₈₎ halocycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, phenyl, phenyl substituted by (Z) _p1, L or Represents M,
R ⁵ is cyano, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, R ²¹ (C ₃ -C ₈₎ cycloalkyl, optionally substituted optionally substituted by R ²¹ (C _{3 ~C 8)} halocycloalkyl, the R ²¹ (C ₂ ~C ₆₎ alkenyl, C ₃ -C ₈ cycloalkyl alkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ ^{alkynyl, -OR 8, -S (O)} r R 8, -N (R 10) R 9, -CHO, -C (O) R ⁹ , -CH = NOR ¹¹ , -C (R ⁹ ) = NOR ¹¹ , -C (O) OR ⁹ , -C (O) SR ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , phenyl, (Z) phenyl substituted by _p1, biphenyl, biphenyl substituted by (Z) _p1, phenoxyphenyl, phenoxyphenyl substituted by (Z) _p1, Pirijiruo Shifeniru, (Z) pyridyloxy phenyl substituted by _p1, phenylthiophenyl, (Z) phenylthio phenyl substituted by _p1, phenylsulfinyl phenyl, phenylsulfinyl phenyl substituted by (Z) _p1, phenylsulfonyl phenyl, (Z) phenylsulfonyl phenyl substituted by _p1, or represents L or M, or by forming a C ₂ -C ₃ alkylene chain together with Y being present on the adjacent position, it is condensed with a benzene ring Represents that a 5- to 6-membered ring may be formed, in which case the alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and optionally by a halogen atom or a C ₁ -C ₆ haloalkyl group May be replaced,
R ⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~ C ₆ ) haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, phenyl (C ₃ -C ₆ ) alkenyl, (Z) phenyl substituted by _p1 (C ₃ -C ₆₎ alkenyl, C ₃ -C ₈ cycloalkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, phenyl (C ₃ ~C ₆₎ alkynyl, phenyl substituted by (Z) _p1 (C ₃ -C _{6) ^{alkynyl, -S (O) 2 R 9}} , -C (O) R 9, -C (O) OR 9, -C (O) SR 9, -C (S) OR 9, -C (S) SR ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ or M,
L represents an aromatic heterocycle represented by any one of formulas L-1 to L-58,

  M represents a saturated heterocyclic ring represented by any one of formulas M-1 to M-28;

Z is a halogen atom, cyano, nitro, _{azido, -SCN, -SF 5, C 1} ~C 6 alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkoxy (C ₁ ~C ₃₎ alkyl, cyano (C ₁ ~C ₆₎ alkyl, hydroxy (C ₁ ~C ₃₎ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ ~C ₃₎ haloalkyl, C ₁ -C ₃ haloalkoxy (C _{1 ~C 3)} haloalkyl, C ₁ -C ₃ alkylthio (C _{1 ~C 3)} alkyl, C ₁ -C ₃ haloalkylthio (C _{1 ~C 3)} alkyl, C ₁ -C ₃ alkylsulfinyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₃ haloalkylsulfinyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₃ alkylsulfonyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₃ haloalkyl sulfonyl (C ₁ ~C ₃₎ alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₂ -C ₆ alkenyl, C ₂ -C ₆ haloalkenyl, C ₃ -C ₈ Cycloalkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₂ -C ₆ alkynyl, C ₂ -C ₆ haloalkynyl, -OH, C ₁ ~C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₃ haloalkoxy (C ₁ ~C ₃₎ haloalkoxy, C ₂ -C ₆ alkenyloxy, C ₂ -C ₆ haloalkenyloxy, C ₃ -C ₆ alkynyloxy, C ₃ -C ₆ haloalkynyloxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, -SH, C ₁ ~C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, -NH _2, C ₁ ~C ₆ alkyl amino, di (C ₁ -C ₆ alkyl) amino, C ₁ -C ₆ alkylsulfonylamino, C ₁ -C ₆ haloalkylsulfonyl amino, C ₁ -C ₆ an alkoxycarbonyl Boniru, C ₁ -C _{6 haloalkoxycarbonyl, -C (O) NH 2,} C 1 ~C 6 alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) _{aminocarbonyl, -C (S) NH 2,} C 1 -C ₆ alkylaminosulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl or a tri (C ₁ -C ₆ alkyl) a silyl, when p1, p2, p3 or p4 represents an integer of 2 or more, each of the Z may be the same as or different from each other,
Further, when two Zs are adjacent to each other, the two adjacent Zs are -CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ O-, -CH ₂ OCH _2- , -OCH ₂ O-, -CH ₂ CH ₂ S-, -CH ₂ SCH _2- , -CH ₂ CH ₂ CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ CH ₂ O-, -CH ₂ CH ₂ OCH _2- , -CH ₂ OCH ₂ O- , -OCH ₂ CH ₂ O-, -OCH ₂ CH ₂ S- or -CH = CHCH = CH- to form a 5-membered or 6-membered ring with the carbon atom to which each of the two Z bonds may be, at this time, the hydrogen atoms bonded to each carbon atom forming the ring may be optionally substituted by halogen atom or C ₁ -C ₆ alkyl group,
R ⁷ is a halogen atom, cyano, C _{3 to} C ₈ cycloalkyl, C _{3 to} C ₈ halocycloalkyl, —OH, —OR ⁸ , —SH, —S (O) _r R ⁸ , —N (R ¹⁰ ) R ⁹ , -N (R ¹⁰ ) CHO, -N (R ¹⁰ ) C (O) R ⁹ , -N (R ¹⁰ ) C (O) OR ⁹ , -N (R ¹⁰ ) C (O) SR ⁹ , -N (R ¹⁰ ) C (S) OR ⁹ , -N (R ¹⁰ ) C (S) SR ⁹ , -N (R ¹⁰ ) S (O) ₂ R ⁹ , -C (O) OR ⁹ ,- C (O) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , phenyl, (Z) represents phenyl, L or M substituted by _p1 ;
R ⁸ is optionally substituted by C ₁ -C ₆ alkyl, optionally substituted by R ²⁵ (C ₁ ~C ₆₎ alkyl, C ₃ -C ₈ cycloalkyl, R ²⁵ (C ₃ ~C ₈ ) cycloalkyl, C ₂ -C ₆ alkenyl, optionally substituted by R ²⁵ (C ₂ ~C ₆₎ alkenyl, C ₃ -C ₈ cycloalkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₃ -C ₆ It represents alkynyl, optionally substituted by R ²⁵ (C ₃ ~C ₆₎ alkynyl, phenyl, phenyl, L or M, which is substituted by (Z) _p1,
R ⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ cycloalkyl (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylthio (C _{1 ~C 4)} alkyl, cyano (C _{1 ~C 6)} alkyl, phenyl (C _{1 ~C 4)} alkyl, (Z) phenyl substituted by _p1 (C _{1 ~C 4)} Alkyl, L- (C ₁ -C ₄ ) alkyl, M- (C ₁ -C ₄ ) alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ represents haloalkenyl, C ₃ -C ₆ alkynyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁰ represents a hydrogen atom or C ₁ -C ₆ alkyl, or R ⁹ and R ¹⁰ together form a C ₂ -C ₆ alkylene chain to form 3-7 together with the atoms to be bonded. indicates that the members may form a ring, this time the alkylene chain an oxygen atom, may contain one sulfur atom or a nitrogen atom, and a halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ alkoxy group, a formyl group, may be optionally substituted by C ₁ -C ₆ alkylcarbonyl group or a C ₁ -C ₆ alkoxycarbonyl group,
R ¹¹ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, or represents C ₃ -C ₆ alkynyl or C ₃ -C ₆ haloalkynyl, or, R ¹¹ is C ₂ -C ₄ alkylene together with R ⁹ By forming a chain, it represents that a 5- to 7-membered ring may be formed together with the atoms to be bonded. At this time, the alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and a halogen atom. or it may be optionally substituted by C ₁ -C ₆ alkyl group,
R ¹² represents C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ alkenyl, phenyl or phenyl substituted by (Z) _p1 ;
R ¹³ and R ¹⁴ each independently represent C ₁ -C ₆ alkyl or C ₁ -C ₆ haloalkyl,
R ¹⁵ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxycarbonyl (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ haloalkoxycarbonyl (C ₁ -C ₄₎ alkyl, phenyl (C ₁ -C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ -C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ ~ C ₆ represents alkynyl, C ₃ -C ₆ haloalkynyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁶ is a halogen atom, cyano, nitro, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, -OR ²⁶ , -N (R ²⁷ ) R ²⁶ , -SH, -S (O) _r R ²⁸ , -SO ₂ NHR ³⁰ , -SO ₂ N (R ³⁰ ) R ²⁹ , -CHO, -C (O) R ²⁹ , -C (O) OH, -C (O) OR ²⁹ , -C (O ) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) OR ²⁹ , -C (R ³² ) = NOH, -C (R ³² ) = NOR ³¹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , -P (phenyl) ₂ , -P (O) (phenyl) ₂ , phenyl, (Z) represents phenyl, L or M substituted by _p1 ,
R ¹⁷ is C ₁ -C ₁₂ alkyl, C ₁ -C ₁₂ haloalkyl, C ₁ -C ₁₂ alkoxy (C ₁ -C ₁₂ ) alkyl, cyano (C ₁ -C ₁₂ ) alkyl, C ₁ -C ₁₂ alkoxycarbonyl (C ₁ ~C ₁₂₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₁₂ alkenyl, C ₃ -C ₁₂ halo represents alkenyl, C ₃ -C ₁₂ alkynyl, C ₃ -C ₁₂ haloalkynyl, C ₁ -C ₁₂ alkylcarbonyl, C ₁ -C ₁₂ alkoxycarbonyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁸ is C ₁ -C ₁₂ alkyl, C ₁ -C ₁₂ haloalkyl, C ₁ -C ₁₂ alkoxy (C ₁ -C ₁₂ ) alkyl, cyano (C ₁ -C ₁₂ ) alkyl, C ₁ -C ₁₂ alkoxycarbonyl (C ₁ ~C ₁₂₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₁₂ alkenyl, C ₃ -C ₁₂ halo alkenyl, C ₃ -C ₁₂ alkynyl, C ₃ -C ₁₂ haloalkynyl, or represents phenyl which is substituted by phenyl or (Z) _p1, or, C ₄ -C ₇ and R ¹⁷ and R ¹⁸ together By forming an alkylene chain, it represents that a 5- to 8-membered ring may be formed together with the nitrogen atom to be bonded. At this time, the alkylene chain may contain one oxygen atom or sulfur atom, and C _1- It may be optionally substituted by C ₄ alkyl group or a C ₁ -C ₄ alkoxy group,
R ¹⁹ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₆ alkynyl, -CHO, C ₁ ~C ₆ alkyl carbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenyl (C ₁ ~C ₄₎ alkoxycarbonyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkoxycarbonyl, phenoxycarbonyl, phenoxycarbonyl substituted by (Z) _p1 , Phenylcarbonyl, phenylcarbonyl substituted by (Z) _p1 , phenyl or phenyl substituted by (Z) _p1 ,
R ²⁰ represents a hydrogen atom, C ₁ -C ₆ alkyl, -CHO, C ₁ -C ₆ alkylcarbonyl, a C ₁ -C ₆ haloalkylcarbonyl or C ₁ -C ₆ alkoxycarbonyl,
R ²¹ is cyano, C _{3 to} C ₈ cycloalkyl, C _{3 to} C ₈ halocycloalkyl, —OH, —OR ⁸ , —SH, —S (O) _r R ⁸ , —N (R ¹⁰ ) R ⁹ , -N (R ¹⁰ ) CHO, -N (R ¹⁰ ) C (O) R ⁹ , -N (R ¹⁰ ) C (O) OR ⁹ , -N (R ¹⁰ ) C (O) SR ⁹ , -N (R ¹⁰ ) C (S) OR ⁹ , -N (R ¹⁰ ) C (S) SR ⁹ , -N (R ¹⁰ ) S (O) ₂ R ⁹ , -C (O) OR ⁹ , -C (O ) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , phenyl, (Z) represents phenyl, L or M substituted by _p1 ;
R ²² represents C ₁ -C ₆ alkyl or C ₁ -C ₆ haloalkyl,
R ²³ is a halogen atom, cyano, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, hydroxy (C ₁ -C ₆ ) alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkoxycarbonyl (C ₁ ~C ₄₎ represents alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkoxycarbonyl, phenyl substituted by phenyl or _{(Z) p1, q1, q2} , q3 or q4 When each represents an integer of 2 or more, each R ²³ may be the same as or different from each other;
R ²⁴ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, -CHO, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ haloalkylcarbonyl, phenyl (C ₁ ~C ₄₎ alkylcarbonyl (Z) phenyl (C ₁ -C ₄ ) alkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenyl (C ₁ -C ₄ ) alkoxycarbonyl, substituted by _p1 (Z ) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkoxycarbonyl, C ₁ -C ₆ alkylthiocarbonyl, C ₁ -C ₆ alkoxythiocarbonyl, C ₁ -C ₆ alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl, C ₁ -C ₆ alkylamino thiocarbonyl, di (C ₁ -C ₆ alkyl) aminothiocarbonyl, phenylcarbonyl, (Z) phenylcarbonyl substituted by _p1, C ₁ -C ₆ alkyl sulfonyl Represents C ₁ -C ₆ haloalkylsulfonyl, phenylsulfonyl, and (Z) phenylsulfonyl substituted by _{p1, -P (O) (OR} 22) 2 or ^{-P (S) (OR 22)} 2,
R ²⁵ is a halogen atom, cyano, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino, -CHO, C ₁ -C ₆ alkyl carbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ ^{haloalkoxycarbonyl, -CH = NOR 11, -C (} R 9) = NOR 11, phenyl, the (Z) _p1 Represents substituted phenyl, L or M;
R ²⁶ is a hydrogen atom, C ₁ -C ₈ alkyl, optionally substituted by R ³³ (C ₁ ~C ₈₎ alkyl, C ₃ -C ₈ cycloalkyl, optionally substituted by R ³³ (C ₃ -C ₈₎ cycloalkyl, C ₃ -C ₈ alkenyl, optionally substituted by R ³³ (C ₃ ~C ₈₎ alkenyl, optionally substituted by C ₃ -C ₈ alkynyl, R ³³ (C ₃ ~ C ₈ ) alkynyl, -CHO, -C (O) R ²⁹ , -C (O) OR ²⁹ , -C (O) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) R ²⁹ , -C (O) C (O) OR ²⁹ , -C (S) R ²⁹ , -C (S) OR ²⁹ , -C (S) SR ²⁹ , -C (S) NHR ³⁰ , -C (S) N (R ³⁰ ) R ²⁹ , -S (O) ₂ R ²⁹ , -S (O) ₂ N (R ³⁰ ) R ²⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , phenyl, (Z) represents phenyl, L or M substituted by _p1 ;
R ²⁷ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ cycloalkyl or C ₁ -C ₆ alkoxy, or R ²⁶ and R ²⁷ together by now it forms a C ₂ -C ₅ alkylene chain, represents that may form a 3-6 membered ring together with the nitrogen atom to which they are attached this case the alkylene chain may contain one oxygen atom or a sulfur atom But often, and halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ alkoxy group, a phenyl group or (Z) _p1 may be substituted by a phenyl group substituted by,
R ²⁸ is, C ₁ -C ₈ alkyl, optionally substituted by R ³³ (C ₁ ~C ₈₎ alkyl, optionally substituted by C ₃ -C ₈ cycloalkyl, R ³³ (C ₃ ~C ₈ ) cycloalkyl, optionally substituted by C ₃ -C _{8 ^{alkenyl, R 33 (C 3 ~C 8}} ) alkenyl, optionally substituted by C ₃ -C _{8 ^{alkynyl, R 33 (C 3 ~C 8}} ) alkynyl, -SH, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, phenylthio substituted by _{(Z) p1, -CHO, -C} (O) R 29, -C (O) OR 29 , -C (O) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) R ²⁹ , -C (O) C (O ) OR ²⁹ , -C (S) R ²⁹ , -C (S) OR ²⁹ , -C (S) SR ²⁹ , -C (S) NHR ³⁰ , -C (S) N (R ³⁰ ) R ²⁹ ,- P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , phenyl, phenyl substituted by (Z ¹ ) _p1 , L-18, L-21, L-25, L-30 ~ Represents L-35, L-45, L-48, L-49 or M;
R ²⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ haloalkoxy (C _{1 ~C 4)} alkyl, C ₁ -C ₆ alkylthio (C _{1 ~C 4)} alkyl, C ₁ -C ₆ haloalkylthio (C _{1 ~C 4)} alkyl, C ₁ -C ₆ alkylsulfonyl (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ haloalkylsulfonyl (C ₁ ~C ₄₎ alkyl, cyano (C ₁ -C ₆₎ alkyl, C ₁ -C ₆ alkylcarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₆ haloalkylcarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₆ alkoxycarbonyl (C ₁ -C ₄₎ alkyl, di (C ₁ -C ₆ alkyl) aminocarbonyl (C ₁ -C ₄₎ alkyl, tri (C ₁ -C ₄ alkyl) silyl (C ₁ -C ₄₎ alkyl, phenyl (C ₁ -C ₄₎ alkyl, phenyl substituted by _{(Z) p1 (C 1 ~C} 4 ) alkyl, L- (C ₁ C ₄₎ alkyl, M- (C ₁ ~C ₄₎ alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₂ -C ₆ alkenyl, C ₂ -C ₆ haloalkenyl, C ₂ -C ₆ alkynyl, C ₂ -C ₆ haloalkynyl, represents phenyl, phenyl, L or M, which is substituted by (Z) _p1,
R ³⁰ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl or phenyl substituted by (Z) _{p 1} , or R ²⁹ and R ³⁰ together represent C By forming a _{2 to} C ₅ alkylene chain, it represents that a 3 to 6 membered ring may be formed together with the nitrogen atom to be bonded. At this time, this alkylene chain contains one oxygen atom, sulfur atom or nitrogen atom. But often, and halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ alkoxy group, a formyl group, C ₁ -C ₆ alkylcarbonyl group, C ₁ -C ₆ alkoxycarbonyl group, a phenyl group or (Z) optionally substituted by a phenyl group substituted by _p1 ,
R ³¹ is hydrogen atom, C ₁ -C ₈ alkyl, (C ₁ -C ₈ ) alkyl optionally substituted by R ³³ , C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ alkenyl, optional by R ³³ substituted a (C ₃ ~C ₈₎ alkenyl, optionally substituted by C ₃ -C ₈ alkynyl, or R ³³ (C ₃ ~C ₈₎ alkynyl,
R ³² is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkoxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ haloalkoxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkylthio (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ haloalkylthio (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkylsulfonyl (C _{1 ~C 4)} alkyl, C ₁ -C ₆ haloalkylsulfonyl (C _{1 ~C 4)} alkyl, phenyl (C _{1 ~C 4)} alkyl, phenyl substituted by (Z) _p1 (C ₁ ~C ₄₎ represents alkyl, phenyl substituted by phenyl or (Z) _p1,
R ³³ is a halogen atom, cyano, nitro, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, —OH, —OR ³⁴ , —SH, —S (O) _r R ³⁴ , —NHR ³⁵ , -N (R ³⁵ ) R ³⁴ , -CHO, -C (O) R ²⁹ , -C (O) OR ²⁹ , -C (O) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) OR ²⁹ , -CH = NOR ¹¹ , -C (R ⁹ ) = NOR ¹¹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² ,- P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , -P (phenyl) ₂ , -P (O) (phenyl) ₂ , phenyl, phenyl substituted by (Z) _p1 , L or M represents
R ³⁴ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylthio (C ₁ -C ₄ ) alkyl, phenyl ( C ₁ -C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₈ cycloalkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, -CHO, C ₁ ~C ₆ alkyl carbonyl , C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, C ₁ -C ₆ alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl, phenylcarbonyl, (Z) phenylcarbonyl substituted by _p1, C _{1 ~C 6} alkylaminothiocarbonyl It represents di (C ₁ -C ₆ alkyl) aminothiocarbonyl, phenyl, phenyl, L or M, which is substituted by (Z) _p1,
R ³⁵ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, C ₁ -C ₆ alkylcarbonyl , C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenoxycarbonyl, phenoxycarbonyl substituted by (Z) _p1, phenylcarbonyl, substituted by (Z) _p1 phenylcarbonyl, C ₁ -C ₆ alkylsulfonyl and, C ₁ -C ₆ haloalkylsulfonyl, phenyl, phenyl substituted by (Z) _p1, or represents L or M, or the R ³⁴ and R ³⁵ together form by now it forms a C ₂ -C ₅ alkylene chain, represents that may form a 3-6 membered ring together with the nitrogen atom to which they are attached this case the alkylene chain may contain one oxygen atom or a sulfur atom so May, be substituted and the halogen atom or a methyl group,
m represents an integer of 0 to 4,
n represents an integer of 0 to 4,
p1 represents an integer of 1 to 5,
p2 represents an integer of 0 to 4,
p3 represents an integer of 0 to 3,
p4 represents an integer of 0 to 2,
p5 represents an integer of 0 or 1,
q1 represents an integer of 0 to 3,
q2 represents an integer of 0 to 5,
q3 represents an integer of 0 to 7,
q4 represents an integer of 0 to 9,
r represents an integer of 0 to 2;
t represents an integer of 0 or 1. ]
The substituted benzanilide compound or its salt represented by these.

[2] W ¹ and W ² represent oxygen atoms,
X is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl or C ₁ -C ₆ represents haloalkylsulfonyl, and when m represents 2 or 3, each X may be the same as or different from each other;
Further, when two Xs are adjacent to each other, the two adjacent Xs form —OCH ₂ O— or —OCH ₂ CH ₂ O— to form a 5-membered ring or 6-membered together with the carbon atom to which each is bonded. may form a ring, this time, the hydrogen atoms bonded to each carbon atom forming the ring is optionally substituted by halogen atom, C ₁ -C ₄ alkyl or C ₁ -C ₄ haloalkyl group Well,
Y is a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, hydroxy (C ₁ ~C ₆₎ alkyl, C ₁ -C ₃ alkoxy (C ₁ ~C ₃₎ alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ represents haloalkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, a C ₁ -C ₆ alkylamino or di (C ₁ -C ₆ alkyl) amino, n is 2 or 3 may be the same as or different from each other,
R ¹ is C ₁ -C ₈ alkyl, (C ₁ -C ₈ ) alkyl optionally substituted by R ¹⁶ , C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ alkenyl, C ₃ -C ₈ alkynyl, C ₁ -C ₈ -alkoxy, a M-4, M-5, M-8, M-9, M-13~M-19, M-21 or M-22,
R ² and R ³ are each independently a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl. , C ₁ -C ₄ alkylsulfonyl (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z ) represents phenylthio substituted by _p1 or —SN (R ¹⁸ ) R ¹⁷ , or R ² together with R ¹ forms a C ₂ -C ₆ alkylene chain, together with the nitrogen atom to which it is attached. Represents that a 3- to 7-membered ring may be formed, in which case this alkylene chain may contain one oxygen or sulfur atom,
R ⁴ is optionally substituted by C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, R ²¹ (C ₁ ~C ₆₎ represents haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₆ haloalkynyl, phenyl substituted by phenyl or (Z) _p1,
R ⁵ is cyano, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ alkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ ^{alkynyl, -C (O) OR 9,} - C (O) SR ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) NHR ^{10, -C (S) N (} R 10) R 9, phenyl, (Z) phenyl substituted by _p1, (Z) phenoxyphenyl phenyl substituted by _p1, pyridyloxy phenyl substituted by (Z) _p1, L-1 ~ L-4, L-8 ~ L-13, L-15 ~ L-23, L-25 ~ L-35, L-37, L-38, L-40, L-43 ~ L- 58, M-4, M-5, M-8, M-9, M-14 to M-18 or M-19, or C ₂ to C together with Y present in the adjacent position by forming a ₃ alkylene chain, condensed with a benzene ring 5 Membered indicates that may form a ring, this time the alkylene chain an oxygen atom, may contain one sulfur atom or a nitrogen atom, optionally substituted and the halogen atom or a C ₁ -C ₆ haloalkyl group You can,
R ⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl , cyano (C ₁ ~C ₆₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ substituted by (Z) _p1 alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, phenyl (C ₃ -C ₆₎ alkenyl, (Z) phenyl substituted by _p1 (C ₃ -C ₆₎ alkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, phenyl (C ₃ -C ₆ ) alkynyl, phenyl (C ₃ -C ₆ ) alkynyl substituted by (Z) _p1 , -S (O) ₂ R ⁹ , -C (O) R ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P ( O) (OR ²² ) ₂ or -P (S) (OR ²² ) ₂
Z is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkylthio (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylthio (C ₁ ~ C ₃₎ alkyl, C ₁ -C ₃ alkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ alkylsulfonyl (C ₁ -C ₃ ) alkyl, C ₁ -C ₃ haloalkylsulfonyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₃ haloalkoxy (C ₁ -C ₃₎ haloalkoxy , C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, -C (O) NH ₂ or - Represents C (S) NH _2, and when p1, p2, p3 or p4 represents an integer of 2 or more, each Z may be the same as or different from each other;
Further, when _two Zs are adjacent, the two adjacent Zs are -CF ₂ CF ₂ O-, -CF ₂ OCF _2- , -OCF ₂ O-, -OCF ₂ CHFO-, -OCF ₂ CF ₂ By forming O- or -CH = CHCH = CH-, a 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each of two Zs is bonded,
R ⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ cycloalkyl (C ₁ -C ₄ ) alkyl, phenyl (C ₁ -C ₄ ) alkyl, (Z) substituted by _p1 phenyl (C ₁ ~C ₄₎ represents alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁰ represents a hydrogen atom or C ₁ -C ₆ alkyl, or R ⁹ and R ¹⁰ together form a C ₄ -C ₅ alkylene chain to form a 5-membered atom together with the nitrogen atom to which it is attached. Represents that a ring or a 6-membered ring may be formed, in which case the alkylene chain may contain one oxygen atom or sulfur atom,
R ¹² represents C ₁ -C ₆ alkyl, phenyl or phenyl substituted by (Z) _{p 1}
R ¹³ and R ¹⁴ each independently represent C ₁ -C ₆ alkyl;
R ¹⁵ is, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ substituted by (Z) _p1 alkyl, phenyl or (Z ) represents phenyl substituted by _p1 ,
R ¹⁶ is a halogen atom, cyano, C ₃ -C ₆ cycloalkyl, -OR ²⁶ , -N (R ²⁷ ) R ²⁶ , -S (O) _r R ²⁸ , -SO ₂ N (R ³⁰ ) R ²⁹ , C ₁ -C ₆ alkoxycarbonyl, -C (O) N (R 30) R 29, -C (R 32) = NOH, -C (R 32) = NOR 31, -Si (R 13) (R 14) R ^{12 represents} phenyl, phenyl substituted by (Z) _p1 , L-1, L-2, L-3, L-4, L-45, L-46, L-47 or M;
R ¹⁷ represents C ₁ -C ₆ alkyl, C ₁ -C ₆ alkoxycarbonyl (C ₁ -C ₄ ) alkyl or C ₁ -C ₆ alkoxycarbonyl,
R ¹⁸ represents C ₁ -C ₆ alkyl, or R ¹⁷ and R ¹⁸ together form a C ₄ -C ₅ alkylene chain to form a 5-membered ring or 6 together with the nitrogen atom to which R ¹⁸ is bonded. The alkylene chain may contain one oxygen atom or one sulfur atom, and may be optionally substituted with a methyl group or a methoxy group,
R ²¹ is cyano, C ₃ -C ₆ cycloalkyl, C ₃ -C ₆ halocycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z) phenoxy substituted by _{p 1} , C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z) phenylthio substituted by _p1, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl , C ₁ -C ₆ haloalkylsulfonyl, phenylsulfonyl, phenylsulfonyl substituted by _{(Z) p1, C 1 ~C} 6 alkyl amino, di (C ₁ -C ₆ alkyl) amino, phenylamino, by (Z) _p1 substituted phenylamino, C ₁ -C ₆ alkoxycarbonyl, phenyl, (Z) phenyl substituted by _{p1, L-1~L-5,} L-8~L-24, L-36, L-39, Represents L-45 to L-52 or L-53,
R ²² represents C ₁ -C ₆ alkyl;
R ²³ represents C ₁ -C ₄ alkyl, and when q1, q2, q3 or q4 represents an integer of 2 or more, each R ²³ may be the same as or different from each other;
R ²⁴ represents -CHO, C ₁ -C ₆ alkylcarbonyl, a C ₁ -C ₆ alkoxycarbonyl or C ₁ -C ₆ alkylsulfonyl,
R ²⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl , phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₃ -C ₆ cycloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, -C (O) N (R 30) R 29, C 1 ~C 6 alkyl sulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl, phenylsulfonyl, (Z ) phenylsulfonyl substituted by _p1, di (C ₁ -C ₆ alkyl) phosphoryl, di (C ₁ -C ₆ alkyl) thiophosphoryl, tri (C ₁ -C ₄ alkyl) silyl, by phenyl or (Z) _p1 Represents substituted phenyl,
R ²⁷ represents a hydrogen atom or a C ₁ -C ₆ alkyl,
R ²⁸ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, hydroxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio ( C ₁ -C ₄₎ alkyl, C ₁ -C ₄ alkylcarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₄ alkoxycarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₄ alkylaminocarbonyl (C ₁ -C ₄₎ alkyl, di (C ₁ -C ₄ alkyl) aminocarbonyl (C ₁ -C ₄₎ alkyl, tri (C ₁ -C ₄ alkyl) silyl (C ₁ -C ₄₎ alkyl, phenyl (C ₁ -C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, C ₁ -C ₆ alkylthio, phenyl, (Z) _represents phenyl, L-21, L-35, L-45 or L-48 substituted by _p1 ,
R ²⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl, phenyl (C ₁ -C ₄ ) alkyl. It is replaced by (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ cycloalkyl, C ₃ -C ₆ alkenyl, C ₂ -C ₆ alkynyl, phenyl or (Z) _p1 Represents phenyl,
R ³⁰ represents a hydrogen atom or C _{1 to} C ₆ alkyl, or R ²⁹ and R ³⁰ together form a C _{2 to} C ₅ alkylene chain to form a 3- Represents that a 6-membered ring may be formed, in which case the alkylene chain may contain one oxygen or sulfur atom,
R ³¹ is, C ₁ -C ₆ alkyl, phenyl (C ₁ ~C ₄₎ phenyl substituted by alkyl or _{(Z) p1 (C 1 ~C} 4) alkyl,
R ³² represents a hydrogen atom or C ₁ -C ₆ alkyl,
m represents an integer of 0 to 3,
n represents an integer of 0 to 3,
q2, q3 and q4 each independently represents an integer of 0 to 2, and the substituted benzanilide compound or a salt thereof according to the above [1].

[3] X is a halogen atom, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ alkylthio, represent C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl or C ₁ -C ₆ haloalkylsulfonyl, m is 2 represents each X may be the same as or different from each other;
Y is a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy or C ₁ -C ₆ alkylthio, when n is 2, each Y is identical to each other May be different from each other,
R ¹ represents C ₁ -C ₈ alkyl, (C ₁ -C ₈ ) alkyl, C ₃ -C ₈ alkenyl or C ₃ -C ₈ alkynyl optionally substituted by R ¹⁶ ,
R ² represents a hydrogen atom or C ₁ -C ₆ alkyl,
R ³ represents a hydrogen atom,
R ⁴ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ -C ₃ ) haloalkyl, C ₁ -C ₃ alkylthio (C ₁ -C ₃ ) haloalkyl, C ₃ -C ₆ cycloalkyl or C ₃ -C ₆ halocycloalkyl,
R ⁵ is optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, optionally substituted by R ²¹ (C ₂ ~ C ₆₎ alkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ alkynyl, C ₁ -C ₆ alkoxycarbonyl, phenyl, phenyl substituted by (Z) _p1, substituted by (Z) _p1 Phenoxyphenyl, pyridyloxyphenyl substituted by (Z) _p1 , L-1 to L-4, L-8 to L-13, L-15 to L-23, L-45 to L-52 or L-53 or it represents, or indicates that by forming a C ₂ -C ₃ alkylene chain together with Y being present on the adjacent positions, may form a 5- or 6-membered ring fused with a benzene ring, In this case, the alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and may be optionally substituted with a halogen atom. ,
R ⁶ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylcarbonyl or tri (C ₁ -C ₄ alkyl) silyl;
R ¹⁶ is -OR ²⁶ , -N (R ²⁷ ) R ²⁶ , -S (O) _r R ²⁸ , -SO ₂ N (R ³⁰ ) R ²⁹ , -C (R ³² ) = NOH or -C (R ³² ) = NOR ³¹
R ²¹ is, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z) _p1 phenoxy substituted by, phenylthio, phenylthio substituted by (Z) _p1, phenylsulfonyl, (Z) _p1 phenylsulfonyl substituted by, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino, phenylamino, (Z) phenylamino substituted by _p1, C ₁ -C ₆ alkoxycarbonyl, phenyl, (Z) represents phenyl substituted by _p1 , L-1 to L-5, L-8 to L-24, L-36, L-39, L-45 to L-52 or L-53;
R ²⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl or represents C ₁ -C ₆ alkylsulfonyl,
R ²⁸ represents C ₁ -C ₆ alkyl,
R ²⁹ represents C ₁ -C ₆ alkyl;
R ³⁰ represents a hydrogen atom or C ₁ -C ₆ alkyl,
R ³¹ represents C ₁ -C ₆ alkyl;
R ³² represents a hydrogen atom,
m represents an integer of 0 to 2,
n is a substituted benzanilide compound or a salt thereof according to the above [2], wherein n represents an integer of 0 to 2.

[4] X represents a halogen atom, nitro, C ₁ -C ₄ alkyl, C ₁ -C ₄ haloalkyl, C ₁ -C ₄ alkylthio, a C ₁ -C ₄ alkylsulfinyl or C ₁ -C ₄ alkylsulfonyl, when m represents 2, each X may be the same as or different from each other;
Y represents a halogen atom or a C ₁ -C ₄ alkyl, when n is 2, each Y may be the even or different from each other the same as each other,
R ¹ is C ₁ -C ₈ alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylsulfinyl (C ₁ -C ₄ ) alkyl or C ₁ -C ₄ alkylsulfonyl ( C ₁ -C ₄₎ alkyl,
R ² represents a hydrogen atom,
R ⁴ represents C ₁ -C ₆ alkyl or C ₁ -C ₆ haloalkyl,
R ⁵ is phenyl, (Z) phenyl substituted by _p1, (Z) phenoxyphenyl phenyl substituted by _p1, (Z) pyridyloxy phenyl substituted by _{p1, L-1~L-4,} L-8 ~ L-13, L-15 ~ L-23, L-45 ~ L-52 or L-53,
R ⁶ represents a substituted benzanilide compound or a salt thereof according to the above [3], which represents a hydrogen atom.

  [5] General formula (2) or general formula (3):

[Wherein Y ¹ represents a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy or C ₁ -C ₆ alkylthio,
Y ² and Y ³ each independently represent a hydrogen atom, or, together with R ⁵ , form a C ₂ -C ₃ alkylene chain to form a 5- to 6-membered ring condensed with a benzene ring. The alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and may be optionally substituted with a halogen atom,
R ⁴ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ -C ₃ ) haloalkyl, C ₁ -C ₃ alkylthio (C ₁ -C ₃ ) haloalkyl, C ₃ -C ₆ cycloalkyl or C ₃ -C ₆ halocycloalkyl,
R ⁵ is optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, optionally substituted by R ²¹ (C ₂ ~ C ₆₎ alkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ alkynyl, C ₁ -C ₆ alkoxycarbonyl, phenyl, phenyl substituted by (Z) _p1, substituted by (Z) _p1 Phenoxyphenyl, pyridyloxyphenyl substituted by (Z) _p1 , L-1 to L-4, L-8 to L-13, L-15 to L-23, L-45 to L-52 or L-53 Represents
R ⁶ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylcarbonyl or tri (C ₁ -C ₄ alkyl) silyl;
R ²¹ is, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z) _p1 phenoxy substituted by, phenylthio, phenylthio substituted by (Z) _p1, phenylsulfonyl, (Z) _p1 phenylsulfonyl substituted by, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino, phenylamino, (Z) phenylamino substituted by _p1, C ₁ -C ₆ alkoxycarbonyl, phenyl, (Z) represents phenyl substituted by _p1 , L-1 to L-5, L-8 to L-24, L-36, L-39, L-45 to L-52 or L-53;
L-1 to L-5, L-8 to L-24, L-36, L-39, L-45 to L-52 or L-53 each represents the following aromatic heterocycle:

Z is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkylthio (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylthio (C ₁ ~ C ₃₎ alkyl, C ₁ -C ₃ alkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ alkylsulfonyl (C ₁ -C ₃ ) alkyl, C ₁ -C ₃ haloalkylsulfonyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₃ haloalkoxy (C ₁ -C ₃₎ haloalkoxy , C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, -C (O) NH ₂ or - Represents C (S) NH _2, and when p1, p2, p3 or p4 represents an integer of 2 or more, each Z may be the same as or different from each other;
Further, when _two Zs are adjacent, the two adjacent Zs are -CF ₂ CF ₂ O-, -CF ₂ OCF _2- , -OCF ₂ O-, -OCF ₂ CHFO-, -OCF ₂ CF ₂ By forming O- or -CH = CHCH = CH-, a 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each of two Zs is bonded,
R ¹⁵ represents C ₁ -C ₆ alkyl, phenyl or phenyl substituted by (Z) _p1 ,
p1 represents an integer of 1 to 5,
p2 represents an integer of 0 to 4,
p3 represents an integer of 0 to 3,
p4 represents an integer of 0 to 2,
p5 represents an integer of 0 or 1,
r represents an integer of 0 to 2;
t represents an integer of 0 or 1. ]
N-substituted phenyl-3-nitrophthalimide or substituted aniline represented by the formula:

  [6] A pest control agent comprising one or more selected from the substituted benzanilide compound according to any one of [1] to [4] above and a salt thereof as an active ingredient.

  [7] An agrochemical comprising one or more selected from the substituted benzanilide compound according to any one of [1] to [4] above and a salt thereof as an active ingredient.

  [8] An insecticide or acaricide characterized by containing, as an active ingredient, one or more selected from the substituted benzanilide compound according to any one of [1] to [4] above and a salt thereof.

  With the long-term use of insecticides and fungicides, pests have recently gained resistance, making it difficult to control with conventional insecticides and fungicides. In addition, some insecticides are highly toxic and those that remain in the environment for a long time. On the other hand, the compound of the present invention has excellent insecticidal and acaricidal activity against many agricultural pests and spider mites, and also exhibits a sufficient control effect against pests that have acquired resistance to existing insecticides. To do. Furthermore, it has little adverse effect on mammals, fish and beneficial insects, has low persistence, and has a light environmental impact.

  Therefore, the present invention can provide a useful novel pest control agent.

The compounds encompassed by the present invention may have geometrical isomers of E-form and Z-form depending on the type of substituent, but the present invention is not limited to these E-form, Z-form or E-form. And a mixture containing the Z-form in an arbitrary ratio. In addition, the compounds included in the present invention include optically active substances resulting from the presence of one or more asymmetric carbon atoms, but the present invention includes all optically active substances or racemates. Furthermore, in the compound of the present invention represented by the general formula (1), when R ² or R ³ is a hydrogen atom, the presence of a tautomer represented by the following formula is considered in some cases. The present invention includes these structures.

  Among the compounds included in the present invention, those that can be converted into acid addition salts according to a conventional method include, for example, hydrohalic acids such as hydrofluoric acid, hydrochloric acid, hydrobromic acid, hydroiodic acid, and the like. Salt of inorganic acid such as salt, nitric acid, sulfuric acid, phosphoric acid, chloric acid, perchloric acid, salt of sulfonic acid such as methanesulfonic acid, ethanesulfonic acid, trifluoromethanesulfonic acid, benzenesulfonic acid, p-toluenesulfonic acid, Salts of carboxylic acids such as formic acid, acetic acid, propionic acid, trifluoroacetic acid, fumaric acid, tartaric acid, succinic acid, maleic acid, malic acid, succinic acid, benzoic acid, mandelic acid, ascorbic acid, lactic acid, gluconic acid, citric acid, etc. A salt of an amino acid such as glutamic acid or aspartic acid can be used.

  Alternatively, among the compounds included in the present invention, those that can be converted into a metal salt according to a conventional method include, for example, alkali metal salts such as lithium, sodium, and potassium, and alkaline earth metals such as calcium, barium, and magnesium. It can be a salt or a salt of aluminum.

  Next, specific examples of each substituent shown in the present specification are shown below. Here, n- represents normal, i- represents iso, s- represents secondary, and t- represents tertiary, and Ph represents phenyl.

  As a halogen atom in this invention compound, a fluorine atom, a chlorine atom, a bromine atom, and an iodine atom are mentioned. In the present specification, the notation “halo” also represents these halogen atoms.

The notation of C _{a to} C _b alkyl in the present specification represents a linear or branched hydrocarbon group having a carbon number of _a to _b , for example, methyl group, ethyl group, n-propyl group, i-propyl group, n-butyl group, s-butyl group, i-butyl group, t-butyl group, n-pentyl group, 1-methylbutyl group, 2-methylbutyl group, 3-methylbutyl group, 1-ethylpropyl group 1,1-dimethylpropyl group, 1,2-dimethylpropyl group, neopentyl group, n-hexyl group, 1-methylpentyl group, 2-methylpentyl group, 3-methylpentyl group, 4-methylpentyl group, 1 -Ethylbutyl group, 2-ethylbutyl group, 1,1-dimethylbutyl group, 1,2-dimethylbutyl group, 1,3-dimethylbutyl group, 2,2-dimethylbutyl group, 2,3-dimethylbutyl group, 3 1,3-dimethylbutyl group, 1,1,2-trimethylpropyl group, 1,2,2-trimethylpropyl group, 1-ethyl-1-methylpropyl group Propyl group, 1-ethyl-2-methylpropyl group, heptyl group, 1-methylhexyl group, 1,1-dimethylpentyl group, octyl group, 1-methylheptyl group, 1,1-dimethylhexyl group, nonyl group, Specific examples include 1-methyloctyl group, 1,1-dimethylheptyl group, decyl group, 1-methylnonyl group, undecyl group, 1-methyldecyl group, dodecyl group, 1-methylundecyl group, etc. In the range of the number of carbon atoms.

In the present specification, C _a -C _b haloalkyl is represented by a linear or branched chain consisting of _a to _b carbon atoms in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. Represents a hydrocarbon group, and when substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, fluoromethyl group, chloromethyl group, bromomethyl group, difluoromethyl group, dichloromethyl group, trifluoromethyl group, chlorodifluoromethyl group, trichloromethyl group, bromodifluoromethyl group, 2-fluoroethyl group, 1-chloroethyl group, 2-chloroethyl group, 1-bromoethyl group, 2-bromoethyl group, 2,2-difluoroethyl group, 1,2-dichloroethyl group, 2,2-dichloroethyl group, 2-bromo-2-chloroethyl group, 2, 2,2-trifluoroethyl group, 2,2,2-trichloroethyl group, 1,1,2,2-tetrafluoroethyl group, 2-chloro-1,1,2-trifluoroethyl group, 2-bromo -1,1,2-trifluoroethyl group, pentafluoroethyl group, 2-chloro-1,1,2,2-tetrafluoroethyl group, 1-chloro-1,2,2,2-tetrafluoroethyl group 2-bromo-1,1,2,2-tetrafluoroethyl group, 2,2-dichloro-1,1,2-to Lifluoroethyl group, 2,2,2-trichloro-1,1-difluoroethyl group, 1-chloropropyl group, 2-chloropropyl group, 3-chloropropyl group, 3-bromopropyl group, 2-fluoro-1 -Methylethyl group, 2-chloro-1-methylethyl group, 2-bromo-1-methylethyl group, 2,2,3,3,3-pentafluoropropyl group, 1,1,2,3,3, 3-hexafluoropropyl group, 2,2,2-trifluoro-1-trifluoromethylethyl group, heptafluoropropyl group, 1,2,2,2-tetrafluoro-1-trifluoromethylethyl group, 2- Bromo-1,1,2,3,3,3-hexafluoropropyl group, 4-chlorobutyl group, 2-chloro-1,1-dimethylethyl group, 2-bromo-1,1-dimethylethyl group, 3, 3,3-trifluoro-1-methylpropyl group, nonafluorobutyl group, 5-chloropentyl group, 2,3-dibromo-1,1-dimethylpropyl group, 6-chlorohexyl group, tridecafluorohe Specific examples include syl group, 7-bromoheptyl group, 8-chlorooctyl group, 9-bromononyl group, 10-chlorodecyl group, 11-bromoundecyl group, 12-bromododecyl group, etc. It is selected in the range of the number of atoms.

The notation of hydroxy (C _a -C _b ) alkyl in the present specification is a linear or branched chain consisting of _a to _b carbon atoms, wherein a hydrogen atom bonded to a carbon atom is optionally substituted with a hydroxyl group And represents, for example, a hydroxymethyl group, 1-hydroxyethyl group, 2-hydroxyethyl group, 3-hydroxypropyl group, 2-hydroxy-1-methylethyl group, 4-hydroxybutyl group, 2-hydroxy- Specific examples include a 1,1-dimethylethyl group, a 3-hydroxy-1-methylpropyl group, a 6-hydroxyhexyl group, and the like, and each is selected within the specified number of carbon atoms.

The notation of cyano (C _a -C _b ) alkyl in the present specification is linear or branched having a carbon number of _a to _b , wherein a hydrogen atom bonded to a carbon atom is optionally substituted with a cyano group Represents a chain alkyl group, for example, cyanomethyl group, 1-cyanoethyl group, 2-cyanoethyl group, 3-cyanopropyl group, 1-cyano-1-methylethyl group, 4-cyanobutyl group, 2-cyano-1,1 Specific examples include -dimethylethyl group, 1-cyano-1-methylpropyl group, 6-cyanohexyl group and the like, and each is selected within the range of the designated number of carbon atoms.

In the present specification, C _a -C _b cycloalkyl represents a cyclic hydrocarbon group having _a to _b carbon atoms, and forms a monocyclic or complex ring structure having 3 to 6 members. I can do it. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms. For example, cyclopropyl group, 1-methylcyclopropyl group, 2-methylcyclopropyl group, 2,2-dimethylcyclopropyl group, 2,2,3,3-tetramethylcyclopropyl group, cyclobutyl group, cyclopentyl group, 1- Methylcyclopentyl group, 2-methylcyclopentyl group, 3-methylcyclopentyl group, cyclohexyl group, 1-methylcyclohexyl group, 2-methylcyclohexyl group, 3-methylcyclohexyl group, 4-methylcyclohexyl group, bicyclo [2.2.1] heptane Specific examples include -2-yl groups and the like, and each is selected within the range of the designated number of carbon atoms.

In the present specification, C _a -C _b halocycloalkyl represents a cyclic hydrocarbon group having _a to _b carbon atoms in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. And can form monocyclic or complex ring structures from 3 to 6-membered rings. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the substitution with a halogen atom may be a ring structure part, a side chain part, They may be both, and when substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, 1-bromocyclopropyl group, 2,2-dichlorocyclopropyl group, 2,2-dibromocyclopropyl group, 2,2-difluoro-1-methylcyclopropyl group, 2,2-dichloro-1-methylcyclopropyl Group, 2,2-dibromo-1-methylcyclopropyl group, 2,2-dichloro-3,3-dimethylcyclopropyl group, 2,2,3,3-tetrafluorocyclobutyl group, 2-fluorocyclohexyl group, Specific examples include 2-chlorocyclohexyl group, 3-chlorocyclohexyl group, 4-chlorocyclohexyl group, 2-trifluoromethylcyclohexyl group, 3-trifluoromethylcyclohexyl group, 4-trifluoromethylcyclohexyl group, etc. Is selected within the range of the specified number of carbon atoms.

In the present specification, C _a -C _b alkenyl is a linear or branched chain composed of _a to _b carbon atoms and has one or more double bonds in the molecule. Represents a saturated hydrocarbon group, for example, vinyl group, 1-propenyl group, 1-methylethenyl group, 2-propenyl group, 1-butenyl group, 1-methyl-1-propenyl group, 2-methyl-1-propenyl group, 2 -Butenyl group, 1-methyl-2-propenyl group, 2-methyl-2-propenyl group, 3-butenyl group, 1,3-butadienyl group, 1-methyl-2-butenyl group, 2-methyl-2-butenyl group Group, 3-methyl-2-butenyl group, 1,1-dimethyl-2-propenyl group, 2-hexenyl group, 2-methyl-2-pentenyl group, 1,3-dimethyl-2-butenyl group, 1,1 , 2-trimethyl-2-propenyl group, 1,1-dimethyl-3-butenyl group, 2,4-hexadienyl group, 2-heptenyl group, 1,1-dimethyl-4-pentenyl group, 2-octenyl group, 1 - Chill-2-heptenyl group, 2-undecenyl group, 10-undecenyl group, 2-dodecenyl group, 11-dodecenyl group, etc. As a specific example, may be selected from the range of the specified number of carbon atoms.

In the present specification, C _a -C _b haloalkenyl is a linear or branched chain consisting of _a to _b carbon atoms in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. And an unsaturated hydrocarbon group having one or more double bonds in the molecule. At this time, when substituted with two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, 2-chlorovinyl group, 2-bromovinyl group, 2,2-dichlorovinyl group, 2,2-dibromovinyl group, 3-bromo-2-propenyl group, 1-chloromethylvinyl group, 2-bromo-1- Methyl vinyl group, 1-trifluoromethyl vinyl group, 2-chloro-3,3,3-trifluoro-1-propenyl group, 1-trifluoromethyl-2,2-difluorovinyl group, 2-chloro-2- Propenyl group, 3,3-difluoro-2-propenyl group, 3,3-dichloro-2-propenyl group, 2,3,3-trifluoro-2-propenyl group, 2,3,3-trichloro-2-propenyl group Group, 4,4-difluoro-3-butenyl group, 3,3,4-trifluoro-3-butenyl group, 3-chloro-4,4,4-trifluoro-2-butenyl group, 3,3,3 -Trifluoro-1-methyl-1-propenyl group, 3,3,3-trifluoro-2-trifluoromethyl-1-propenyl group, 1,3,3,3-tetrafluoro-2-trifluoromethyl- 1-propenyl group, 3,3,4,4,5,5,5-heptaf Oro-1-pentenyl group, 5,5-difluoro-4-pentenyl group, 4,5,5-trifluoro-4-pentenyl group, 3,4,4,4-tetrafluoro-3-trifluoromethyl-1 -Butenyl group, 4,4,5,5,6,6,6-heptafluoro-2-hexenyl group, 3,4,4,5,5,5-hexafluoro-3-trifluoromethyl-1-pentenyl Specific examples include a group, a 2-perfluorohexylethenyl group, and the like, and each is selected within the range of the designated number of carbon atoms.

In the present specification, C _a -C _b cycloalkenyl represents a cyclic unsaturated hydrocarbon group having 1 to 2 carbon atoms and having 1 to 2 carbon atoms. A monocyclic or complex ring structure from a member ring to a 6-member ring can be formed. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the double bond may be either endo- or exo-. For example, cyclopenten-1-yl group, 2-cyclopenten-1-yl group, 3-cyclopenten-1-yl group, cyclohexen-1-yl group, 2-cyclohexen-1-yl group, 3-cyclohexen-1-yl group Specific examples include 2-methyl-2-cyclohexen-1-yl group, 3-methyl-2-cyclohexen-1-yl group, bicyclo [2.2.1] -5-hepten-2-yl group, Each selected range of carbon atoms is selected.

In the present specification, C _a -C _b halocycloalkenyl has the following meaning: a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom, a cyclic one having 1 to b carbon atoms, and one Alternatively, it represents an unsaturated hydrocarbon group having two or more double bonds, and can form a monocyclic or complex ring structure having 3 to 6 members. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the double bond may be either endo- or exo-. In addition, the substitution by a halogen atom may be a ring structure part, a side chain part or both of them, and when substituted by two or more halogen atoms, those halogen atoms May be the same as or different from each other. For example, a 2-chlorobicyclo [2.2.1] -5-hepten-2-yl group and the like are given as specific examples, and each group is selected within the range of the designated number of carbon atoms.

In the present specification, C _a -C _b alkynyl is a linear or branched chain having a carbon number of _a to _b , and is unsaturated having one or more triple bonds in the molecule. Represents a hydrocarbon group, such as ethynyl, 1-propynyl, 2-propynyl, 1-methyl-2-propynyl, 2-butynyl, 3-butynyl, 2-pentynyl, 1-methyl-2- Butynyl group, 1-methyl-3-butynyl group, 1,1-dimethyl-2-propynyl group, 1-hexynyl group, 3,3-dimethyl-1-butynyl group, 2-hexynyl group, 1-methyl-2- Pentynyl group, 1,1-dimethyl-2-butynyl group, 2-heptynyl group, 1,1-dimethyl-2-pentynyl group, 2-octynyl group, 2-noninyl group, 2-decynyl group, 2-undecynyl group, etc. Are given as specific examples and are selected within the range of each designated number of carbon atoms.

In the present specification, C _a -C _b haloalkynyl represents a linear or branched chain having _a to _b carbon atoms in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. And an unsaturated hydrocarbon group having one or more triple bonds in the molecule. At this time, when substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, 2-chloroethynyl group, 2-bromoethynyl group, 2-iodoethynyl group, 3-chloro-2-propynyl group, 3-bromo-2-propynyl group, 3-iodo-2-propynyl group, 3,3, 3-trifluoro-1-propynyl group, 3-chloro-1-methyl-2-propynyl group, 3-bromo-1-methyl-2-propynyl group, 3-iodo-1-methyl-2-propynyl group, 3 Specific examples include -chloro-1,1-dimethyl-2-propynyl group, 3-bromo-1,1-dimethyl-2-propynyl group, 3-iodo-1,1-dimethyl-2-propynyl group and the like. , Each selected range of carbon atoms.

The notation of C _a -C _b alkoxy in the present specification represents an alkyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methoxy group, ethoxy group, n-propyloxy group, i-propyloxy group, n-butyloxy group, s-butyloxy group, i-butyloxy group, t-butyloxy group, n-pentyloxy group, 1-methylbutyloxy group, 2-methylbutyloxy group, 3-methylbutyl Specific examples include oxy, 1-ethylpropyloxy, 1,1-dimethylpropyloxy, 1,2-dimethylpropyloxy, neopentyloxy, n-hexyloxy, 1,1-dimethylbutyloxy As an example, each selected range of carbon atoms is selected.

The notation of C _a -C _b haloalkoxy in the present specification represents a haloalkyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, difluoromethoxy group, trifluoromethoxy group, chlorodifluoro Methoxy group, bromodifluoromethoxy group, 2-fluoroethoxy group, 2-chloroethoxy group, 2,2,2-trifluoroethoxy group, 1,1,2,2, -tetrafluoroethoxy group, 2-chloro-1 1,2-trifluoroethoxy group, 2-bromo-1,1,2-trifluoroethoxy group, pentafluoroethoxy group, 2-bromo-1,1,2,2-tetrafluoroethoxy group, 2,2 -Dichloro-1,1,2-trifluoroethoxy group, 2,2,2-trichloro-1,1-difluoroethoxy group, 2-chloropropyloxy group, 3-chloropropyloxy group, heptafluoropropyloxy group, 2,2,2-trifluoro-1-trifluoromethylethoxy group 2,2,3,3-tetrafluoropropyloxy group, 1,1,2,3,3,3-hexafluoropropyloxy group, 2-bromo-1,1,2,3,3,3-hexafluoro Specific examples include a propyloxy group and the like, and each is selected within the range of the designated number of carbon atoms.

The notation of C _a -C _b alkenyloxy in the present specification represents an alkenyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as 2-propenyloxy group, 2-butenyloxy group, Specific examples include 2-methyl-2-propenyloxy group, 3-methyl-2-butenyloxy group and the like, and each is selected within the range of the designated number of carbon atoms.

The notation of C _a -C _b haloalkenyloxy in the present specification represents a haloalkenyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as a 2-chloro-2-propenyl group, Specific examples include 3-chloro-2-propenyl group, 3,3-difluoro-2-propenyl group, 3,3-dichloro-2-propenyl group, 2,3,3-trifluoro-2-propenyl group and the like. Selected within the range of each specified number of carbon atoms.

The notation of C _a -C _b alkylthio in the present specification represents an alkyl-S-group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylthio group, ethylthio group, n-propylthio group, i -Propylthio group, n-butylthio group, s-butylthio group, i-butylthio group, t-butylthio group, n-pentylthio group, 1-methylbutylthio group, 2-methylbutylthio group, 3-methylbutylthio group, Specific examples include 1-ethylpropylthio group, 1,1-dimethylpropylthio group, 1,2-dimethylpropylthio group, neopentylthio group, n-hexylthio group, and the like. Selected by range.

The notation of C _a -C _b haloalkylthio in the present specification represents a haloalkyl-S-group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, difluoromethylthio group, trifluoromethylthio group, bromodifluoro Methylthio group, 2,2,2-trifluoroethylthio group, 1,1,2,2-tetrafluoroethylthio group, 1,1,2-trifluoro-2-chloroethylthio group, pentafluoroethylthio group 2-bromo-1,1,2,2-tetrafluoroethylthio group, heptafluoropropylthio group, 1,2,2,2-tetrafluoro-1-trifluoromethylethylthio group, nonafluorobutylthio group Etc. are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

In the present specification, the notation of C _a -C _b alkylsulfinyl represents an alkyl-S (O) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylsulfinyl group, ethylsulfinyl group, Specific examples include n-propylsulfinyl group, i-propylsulfinyl group, n-butylsulfinyl group, s-butylsulfinyl group, i-butylsulfinyl group, t-butylsulfinyl group and the like. The range is selected.

In the present specification, the expression C _a -C _b haloalkylsulfinyl represents a haloalkyl-S (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, difluoromethylsulfinyl group, trifluoromethyl Sulfinyl group, bromodifluoromethylsulfinyl group, 2,2,2-trifluoroethylsulfinyl group, 2-bromo-1,1,2,2-tetrafluoroethylsulfinyl group, 1,2,2,2-tetrafluoro- Specific examples include 1-trifluoromethylethylsulfinyl group, nonafluorobutylsulfinyl group and the like, and each is selected within the range of the designated number of carbon atoms.

The notation of C _a -C _b alkylsulfonyl in the present specification represents an alkyl-SO ₂ — group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as methanesulfonyl group, ethanesulfonyl group, n- Specific examples include propylsulfonyl group, i-propylsulfonyl group, n-butylsulfonyl group, s-butylsulfonyl group, i-butylsulfonyl group, t-butylsulfonyl group, n-pentylsulfonyl group, n-hexylsulfonyl group and the like. Each of which is selected for each specified number of carbon atoms.

The notation of C _a -C _b haloalkylsulfonyl in the present specification represents a haloalkyl-SO ₂ -group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as a difluoromethanesulfonyl group, a trifluoromethanesulfonyl group, Chlorodifluoromethanesulfonyl group, bromodifluoromethanesulfonyl group, 2,2,2-trifluoroethanesulfonyl group, 1,1,2,2-tetrafluoroethanesulfonyl group, 1,1,2-trifluoro-2-chloroethane A sulfonyl group etc. are mentioned as a specific example, It selects in the range of each designated carbon atom number.

The notation of C _a -C _b alkylamino in the present specification represents an amino group in which one of the hydrogen atoms is substituted with an alkyl group having the above meaning consisting of _a to _b carbon atoms, for example, a methylamino group , Ethylamino group, n-propylamino group, i-propylamino group, n-butylamino group, i-butylamino group, t-butylamino group and the like. Selected by range.

In the present specification, the notation of di (C _a -C _b alkyl) amino has the above-mentioned meaning that the number of carbon atoms, which may be the same or different from each other, is ab. Represents an amino group substituted by an alkyl group, for example, dimethylamino group, ethyl (methyl) amino group, diethylamino group, n-propyl (methyl) amino group, i-propyl (methyl) amino group, di (n-propyl) Specific examples include amino groups, n-butyl (methyl) amino groups, i-butyl (methyl) amino groups, t-butyl (methyl) amino groups, and the like, each selected within the range of the specified number of carbon atoms. .

In the present specification, the expression C _a -C _b alkylcarbonyl represents an alkyl-C (O) -group having the above-mentioned meaning consisting of _{a- b} carbon atoms, for example, CH ₃ C (O) -group. , CH ₃ CH ₂ C (O)-group, CH ₃ CH ₂ CH ₂ C (O)-group, (CH ₃ ) ₂ CHC (O)-group, CH ₃ (CH ₂ ) ₃ C (O)-group , (CH ₃ ) ₂ CHCH ₂ C (O)-group, CH ₃ CH ₂ CH (CH ₃ ) C (O)-group, (CH ₃ ) ₃ CC (O)-group, CH ₃ (CH ₂ ) ₄ Specific examples include C (O) — group, CH ₃ (CH ₂ ) ₅ C (O) — group, etc., and each is selected within the range of the designated number of carbon atoms.

The notation of C _a -C _b haloalkylcarbonyl in the present specification represents a haloalkyl-C (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, FCH ₂ C (O) -group , ClCH ₂ C (O)-group, F ₂ CHC (O)-group, Cl ₂ CHC (O)-group, CF ₃ C (O)-group, ClCF ₂ C (O)-group, BrCF ₂ C ( O)-group, CCl ₃ C (O)-group, CF ₃ CF ₂ C (O)-group, ClCH ₂ CH ₂ CH ₂ C (O)-group, CF ₃ CF ₂ CF ₂ C (O)-group , ClCH ₂ C (CH ₃ ) ₂ C (O) — groups and the like are listed as specific examples, and each is selected within the range of the designated number of carbon atoms.

In the present specification, the expression C _a -C _b cycloalkylcarbonyl represents a cycloalkyl-C (O) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, cyclopropyl-C (O )-Group, 1-methylcyclopropyl-C (O)-group, 2-methylcyclopropyl-C (O)-group, 2,2-dimethylcyclopropyl-C (O)-group, cyclobutyl-C (O ) -Groups, cyclopentyl-C (O) -groups, cyclohexyl-C (O) -groups, etc., are given as specific examples, each selected within the range of the number of carbon atoms specified.

The notation of C _a -C _b alkoxycarbonyl in the present specification represents an alkyl-OC (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, CH ₃ OC (O) -group , CH ₃ CH ₂ OC (O)-group, CH ₃ CH ₂ CH ₂ OC (O)-group, (CH ₃ ) ₂ CHOC (O)-group, CH ₃ (CH ₂ ) ₃ OC (O)-group , (CH ₃ ) ₂ CHCH ₂ OC (O) — group, (CH ₃ ) ₃ COC (O) — group, and the like are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

In the present specification, the expression C _a -C _b haloalkoxycarbonyl represents a haloalkyl-OC (O) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as ClCH ₂ CH ₂ OC (O ) -Groups, CF ₃ CH ₂ OC (O) -groups and the like are listed as specific examples, each selected within the range of the number of carbon atoms specified.

In the present specification, the expression C _a -C _b alkylthiocarbonyl represents an alkyl-SC (O) -group having the above-mentioned meaning consisting of _{a- b} carbon atoms, for example, CH ₃ SC (O) -group CH ₃ CH ₂ SC (O)-group, CH ₃ CH ₂ CH ₂ SC (O)-group, (CH ₃ ) ₂ CHSC (O)-group, CH ₃ (CH ₂ ) ₃ SC (O)-group , (CH ₃ ) ₂ CHCH ₂ SC (O) — group, (CH ₃ ) ₃ CSC (O) — group, and the like are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

The notation of C _a -C _b alkoxythiocarbonyl in the present specification represents an alkyl-OC (S) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, CH ₃ OC (S) — Group, CH ₃ CH ₂ OC (S)-group, CH ₃ CH ₂ CH ₂ OC (S)-group, (CH ₃ ) ₂ CHOC (S)-group, CH ₃ (CH ₂ ) ₃ OC (S)- Specific examples include a group, (CH ₃ ) ₂ CHCH ₂ OC (S) — group, (CH ₃ ) ₃ COC (S) — group, etc., and each is selected within the range of the designated number of carbon atoms.

The notation of C _a -C _b alkylaminocarbonyl in the present specification represents a carbamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, CH ₃ NHC (O) - _{group, CH 3 CH 2 NHC (O} ) - _{group, CH 3 CH 2 CH 2 NHC} (O) - _{group, (CH 3) 2 CHNHC (} O) - group, CH ₃ (CH _{2) 3} NHC (O)-group, (CH ₃ ) ₂ CHCH ₂ NHC (O)-group, CH ₃ CH ₂ CH (CH ₃ ) NHC (O)-group, (CH ₃ ) ₃ CNHC (O)-group, etc. Specific examples are given, each selected in the range of the specified number of carbon atoms.

In the present specification, the notation of di (C _a -C _b alkyl) aminocarbonyl means in the above-mentioned meaning that the number of carbon atoms which may be the same or different from each other is _a to _b. Represents a carbamoyl group substituted by an alkyl group, for example, a (CH ₃ ) ₂ NC (O) — group, a CH ₃ CH ₂ N (CH ₃ ) C (O) — group, a (CH ₃ CH ₂ ) ₂ NC ( Specific examples include (O)-group, (CH ₃ CH ₂ CH ₂ ) ₂ NC (O)-group, (CH ₃ CH ₂ CH ₂ CH ₂ ) ₂ NC (O)-group, etc. Selected in the range of the number of carbon atoms.

In the present specification, the notation of C _a -C _b alkylaminothiocarbonyl represents a thiocarbamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, CH ₃ NHC (S) - _{group, CH 3 CH 2 NHC (S} ) - _{group, CH 3 CH 2 CH 2 NHC} (S) - _{group, (CH 3) 2 CHNHC (} S) - group, CH ₃ (CH ₂ ) ₃ NHC (S) -group, (CH ₃ ) ₂ CHCH ₂ NHC (S) -group, CH ₃ CH ₂ CH (CH ₃ ) NHC (S) -group, (CH ₃ ) ₃ CNHC (S) -group Etc. are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

The notation of di (C _a -C _b alkyl) aminothiocarbonyl in the present specification means the above-mentioned meaning that the number of carbon atoms that may be the same or different from each other is a to b. Represents a thiocarbamoyl group substituted by an alkyl group such as (CH ₃ ) ₂ NC (S) — group, CH ₃ CH ₂ N (CH ₃ ) C (S) — group, (CH ₃ CH ₂ ) ₂ Specific examples include NC (S) -group, (CH ₃ CH ₂ CH ₂ ) ₂ NC (S) -group, (CH ₃ CH ₂ CH ₂ CH ₂ ) ₂ NC (S) -group, and the like. Selected within the specified number of carbon atoms.

The notation of C _a -C _b alkylaminosulfonyl in the present specification represents a sulfamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, CH ₃ NHSO ₂ - group, CH ₃ CH ₂ NHSO ₂ - _{group, CH 3 CH 2 CH 2 NHSO} 2 - _{group, (CH 3) 2 CHNHSO 2} - _{group, CH 3 (CH 2) 3} NHSO 2 - group, (CH ₃ ) ₂ CHCH ₂ NHSO ₂ -group, CH ₃ CH ₂ CH (CH ₃ ) NHSO ₂ -group, (CH ₃ ) ₃ CNHSO ₂ -group, etc., are given as specific examples, and within each specified number of carbon atoms Selected.

In the present specification, the notation of di (C _a -C _b alkyl) aminosulfonyl means in the above meaning that the number of carbon atoms that may be the same or different from each other is _a to _b. Represents a sulfamoyl group substituted by an alkyl group, such as (CH ₃ ) ₂ NSO ₂ — group, CH ₃ CH ₂ N (CH ₃ ) SO ₂ — group, (CH ₃ CH ₂ ) ₂ NSO ₂ — group, ( Specific examples include CH ₃ CH ₂ CH ₂ ) ₂ NSO ₂ — group, (CH ₃ CH ₂ CH ₂ CH ₂ ) ₂ NSO ₂ — group, etc., and each is selected within the range of the designated number of carbon atoms.

The notation of di (C _a -C _b alkyl) phosphoryl in the present specification has the above-mentioned meaning that the number of carbon atoms, which may be both the same or different from each other, consists of _a to _b. Represents a phosphoryl group substituted by an alkyl group, for example, (CH ₃ O) ₂ P (O) -group, (CH ₃ CH ₂ O) ₂ P (O) -group, etc. In the range of the number of carbon atoms.

In the present specification, the notation of di (C _a -C _b alkyl) thiophosphoryl means in the above-mentioned meaning that the number of carbon atoms which may be the same or different from each other may be ab. Represents a thiophosphoryl group substituted by a certain alkyl group, for example, (CH ₃ O) ₂ P (S) -group, (CH ₃ CH ₂ O) ₂ P (S) -group, etc. Is selected within the range of the specified number of carbon atoms.

In the present specification, the notation of tri (C _a -C _b alkyl) silyl is substituted with an alkyl group having the above-mentioned meanings each having the same or different number of carbon atoms from _a to _b . Represents a silyl group, for example, trimethylsilyl group, triethylsilyl group, tri (n-propyl) silyl group, ethyldimethylsilyl group, n-propyldimethylsilyl group, n-butyldimethylsilyl group, i-butyldimethylsilyl group, t- Specific examples include a butyldimethylsilyl group and the like, and each butyldimethylsilyl group is selected within a range of each designated number of carbon atoms.

The notation of C _a -C _b alkylsulfonyloxy in the present specification represents an alkylsulfonyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as a CH ₃ SO ₂ —O— group, CH ₃ CH ₂ SO ₂ -O- group, CH ₃ CH ₂ CH ₂ SO ₂ -O- group, (CH ₃ ) ₂ CHSO ₂ -O- group, CH ₃ (CH ₂ ) ₃ SO ₂ -O- group, Specific examples include (CH ₃ ) ₂ CHCH ₂ SO ₂ —O— group, CH ₃ CH ₂ CH (CH ₃ ) SO ₂ —O— group, (CH ₃ ) ₃ CSO ₂ —O— group, etc. Is selected within the range of the specified number of carbon atoms.

The notation of C _a -C _b haloalkylsulfonyloxy in the present specification represents a haloalkylsulfonyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as CF ₃ SO ₂ —O— group, A CF ₃ CF ₂ SO ₂ —O— group or the like is given as a specific example, and is selected within the range of each designated number of carbon atoms.

The notation of C _a -C _b alkylsulfonylamino in the present specification represents an alkylsulfonyl-NH— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, CH ₃ SO ₂ —NH— group, CH ₃ CH ₂ SO ₂ -NH- group, CH ₃ CH ₂ CH ₂ SO ₂ -NH- group, (CH ₃ ) ₂ CHSO ₂ -NH- group, CH ₃ (CH ₂ ) ₃ SO ₂ -NH- group, Specific examples include (CH ₃ ) ₂ CHCH ₂ SO ₂ -NH- group, CH ₃ CH ₂ CH (CH ₃ ) SO ₂ -NH- group, (CH ₃ ) ₃ CSO ₂ -NH- group, Is selected within the range of the specified number of carbon atoms.

The notation of C _a -C _b haloalkylsulfonylamino in the present specification represents a haloalkylsulfonyl-NH— group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as CF ₃ SO ₂ —NH— group, Specific examples include CF ₃ CF ₂ SO ₂ —NH— groups, etc., each selected within the range of the specified number of carbon atoms.

C _a -C _b cycloalkyl (C _d -C _e ) alkyl, C _a -C _b alkoxy (C _d -C _e ) alkyl, C _a -C _b haloalkoxy (C _d -C _e ) alkyl as used herein , C _a -C _b alkylthio (C _d -C _e ) alkyl, C _a -C _b haloalkylthio (C _d -C _e ) alkyl, C _a -C _b alkylsulfinyl (C _d -C _e ) alkyl, C _a -C _b haloalkylsulfinyl (C _d ~C _e) alkyl, C _a -C _b alkylsulfonyl (C _d ~C _e) alkyl, C _a -C _b haloalkylsulfonyl (C _d ~C _e) alkyl, C _a -C _b alkylcarbonyl (C _d -C _e ) alkyl, C _a -C _b haloalkylcarbonyl (C _d -C _e ) alkyl, C _a -C _b alkoxycarbonyl (C _d -C _e ) alkyl, C _a -C _b halo alkoxycarbonyl (C _d -C _e) alkyl, C _a -C _b alkylaminocarbonyl (C _d -C _e) alkyl, di (C _a -C _b alkyl) aminocarbonyl (C _d C _e) alkyl, tri (C _a -C _b alkyl) silyl (C _d -C _e) alkyl, phenyl (C _d -C _e) alkyl, phenyl substituted by _{(Z) p1 (C d ~C} e) The notation such as alkyl, L- (C _d -C _e ) alkyl or M- (C _d -C _e ) alkyl is any C _a -C _b cycloalkyl group, C _a -C _b , each having the above meaning. Alkoxy group, C _a -C _b haloalkoxy group, C _a -C _b alkylthio group, C _a -C _b haloalkylthio group, C _a -C _b alkylsulfinyl group, C _a -C _b haloalkylsulfinyl group, C _a- C _b alkylsulfonyl group, C _a -C _b haloalkylsulfonyl group, C _a -C _b alkylcarbonyl group, C _a -C _b haloalkylcarbonyl group, C _a -C _b alkoxycarbonyl group, C _a -C _b haloalkoxycarbonyl Group, C _a -C _b alkylaminocarbonyl group, di (C _a -C _b alkyl) aminocarbonyl group, tri ( C _a -C _b alkyl) silyl group, phenyl group, phenyl group substituted by (Z) _p1 , L group or M group, the hydrogen atom bonded to the carbon atom is arbitrarily substituted by d ~ e represents a linear or branched hydrocarbon group consisting of e, and is selected within the range of the respective designated number of carbon atoms.

Optionally substituted by R ⁷ herein (C _a ~C _b) alkyl, optionally substituted by R ¹⁶ (C _a ~C _b) alkyl, optionally substituted by R ²¹ (C _a ~ C _b) alkyl, optionally substituted by R ²⁵ (C _a ~C _b) optionally substituted by alkyl or R ³³ (C _a ~C _b) representation of alkyl, any R ^7, R ^16, R ²¹ , R ²⁵ or R ³³ represents a linear or branched hydrocarbon group consisting of a to b carbon atoms in which hydrogen atoms bonded to carbon atoms are arbitrarily substituted, and each designation In the range of the number of carbon atoms. At this time, when two or more substituents R ⁷ , R ¹⁶ , R ²¹ , R ²⁵ or R ³³ on each (C _a -C _b ) alkyl group are present, each R ⁷ , R ¹⁶ , R ^{21 is present.} , R ²⁵ or R ³³ may be the same as or different from each other.

In the present specification, the notation of hydroxy (C _d -C _e ) haloalkyl, C _a -C _b alkoxy (C _d -C _e ) haloalkyl or C _a -C _b haloalkoxy (C _d -C _e ) haloalkyl is a hydroxyl group, A C _a -C _b alkoxy group as defined above or a haloalkyl group as defined above consisting of d to e carbon atoms optionally substituted by a C _a -C _b haloalkoxy group as defined above. For example, 2,2,2-trifluoro-1-hydroxy-1- (trifluoromethyl) ethyl group, 2,2,2-trifluoro-1-methoxy-1- (trifluoromethyl) ethyl group, 2 , 2,2-Trifluoro-1- (2,2,2-trifluoroethoxy) -1- (trifluoromethyl) ethyl group, 3- (1,2-dichloro-1,2,2-trifluoroethoxy ) -1,1,2,2,3,3-hexafluoropropyl group and the like are listed as specific examples, and each group is selected within the range of the designated number of carbon atoms.

Optionally substituted by R ²¹ herein (C _a ~C _b) notation haloalkyl, a haloalkyl group having a carbon atom number which is optionally substituted by R ²¹ is the meaning of consisting a~b pieces Selected and selected for each specified number of carbon atoms. At this time, when two or more substituents R ²¹ on each (C _a -C _b ) haloalkyl group are present, each R ²¹ may be the same as or different from each other.

The R ⁷ herein optionally substituted (C _a ~C _b) cycloalkyl, optionally substituted by R ¹⁶ (C _a ~C _b) cycloalkyl, optionally substituted by R ²¹ (C _a -C _b) cycloalkyl, notation (C _{a ~C b)} cycloalkyl such as optionally substituted by optionally substituted (C _{a ~C b)} cycloalkyl or R ³³ by R ²⁵ is, R ⁷ , R ¹⁶ , R ²¹ , R ²⁵ or R ³³ represents a cycloalkyl group having the above-mentioned meaning consisting of a to b carbon atoms. At this time, the substitution by R ⁷ , R ¹⁶ , R ²¹ , R ²⁵ or R ³³ may be a ring structure part, a side chain part or both, and When two or more substituents R ⁷ , R ¹⁶ , R ²¹ , R ²⁵ or R ³³ on the (C _a -C _b ) cycloalkyl group are present, each R ⁷ , R ¹⁶ , R ²¹ , R ²⁵ Alternatively, R ³³ may be the same as or different from each other.

Herein is optionally substituted by R ²¹ (C _a ~C _b) representation of halocycloalkyl are defined above in which the carbon atoms which is optionally substituted by R ²¹ is composed of a~b number halo Represents a cycloalkyl group. At this time, the substitution by R ²¹ may be a ring structure part, a side chain part, or both of them, and each (C _a -C _b ) halocycloalkyl group. When two or more of the above substituents R ²¹ are present, each R ²¹ may be the same as or different from each other.

Notation such as phenyl (C _d ~C _e) alkenyl substituted by phenyl (C _d ~C _e) alkenyl or (Z) _p1 in the present specification, by a phenyl group or (Z) _p1 is a meaning of each of the It represents an alkenyl group having the above-mentioned meaning consisting of d to e carbon atoms optionally substituted with a substituted phenyl group, and is selected in the range of each designated number of carbon atoms.

Optionally substituted by R ⁷ herein (C _a ~C _b) alkenyl, optionally substituted by R ¹⁶ (C _a ~C _b) alkenyl, optionally substituted by R ²¹ (C _a ~ C _b) alkenyl, optionally substituted by R ²⁵ (C _a ~C _b) optionally substituted by alkenyl or R ³³ (C _a ~C _b) notation ^{alkenyl, R 7, R 16, R} 21 , R ²⁵ or R ³³ represents an alkenyl group having the above-mentioned meaning, wherein the number of carbon atoms is optionally substituted by a to b, and is selected in the range of each designated number of carbon atoms. At this time, when two or more substituents R ⁷ , R ¹⁶ , R ²¹ , R ²⁵ or R ³³ on each (C _a -C _b ) alkenyl group are present, each R ⁷ , R ¹⁶ , R ^{21 is present.} , R ²⁵ or R ³³ may be the same as or different from each other.

Phenyl (C _d ~C _e) notation alkynyl or (Z) phenyl substituted by _p1 (C _d ~C _e) alkynyl herein, optionally by phenyl substituted by phenyl or (Z) _p1 Represents an alkynyl group having the above-mentioned meaning, wherein the number of carbon atoms substituted is from d to e, and is selected within the range of each designated number of carbon atoms.

Optionally substituted by R ⁷ herein (C _a ~C _b) alkynyl, optionally substituted by R ¹⁶ (C _a ~C _b) alkynyl, optionally substituted by R ²¹ (C _a ~ C _b) alkynyl, optionally substituted by R ²⁵ (C _a ~C _b) optionally substituted by alkynyl, or R ³³ (C _a ~C _b) notation ^{alkynyl, R 7, R 16, R} 21 , R ²⁵ or R ³³ represents an alkynyl group having the above-mentioned meaning, wherein the number of carbon atoms is optionally substituted by a to b, and is selected in the range of each designated number of carbon atoms. At this time, when two or more substituents R ⁷ , R ¹⁶ , R ²¹ , R ²⁵ or R ³³ on each (C _a -C _b ) alkynyl group are present, each R ⁷ , R ¹⁶ , R ^{21 is present.} , R ²⁵ or R ³³ may be the same as or different from each other.

Phenyl (C _a ~C _b) notation alkoxy or (Z) phenyl substituted by _p1 (C _a ~C _b) alkoxy in the present specification is arbitrarily by a phenyl group substituted by a phenyl group or (Z) _p1 Represents a (C _a -C _b ) alkoxy group as defined above, and the (C _a -C _b ) alkoxy group includes, for example, a —CH ₂ O— group, a —CH (CH ₃ ) O— group, — Specific examples include C (CH ₃ ) ₂ O— group, —CH ₂ CH ₂ O— group, —CH (CH ₃ ) CH ₂ O— group, —C (CH ₃ ) ₂ CH ₂ O— group and the like. , Each selected range of carbon atoms.

In the present specification, C _a -C _b haloalkoxy (C _d -C _e ) haloalkoxy is represented by the number of carbon atoms optionally substituted by the C _a -C _b haloalkoxy group as defined above being _{d- e} Represents a haloalkoxy group having the above-mentioned meaning, such as 1,1,2-trifluoro-2-trifluoromethoxyethoxy group, 1,1,2-trifluoro-2-heptafluoropropyloxyethoxy group, etc. Are given as specific examples and are selected in the range of each designated number of carbon atoms.

Phenyl notation (C _a ~C _b) phenyl substituted by alkylcarbonyl or _{(Z) p1 (C a ~C} b) alkylcarbonyl herein, a phenyl group substituted by a phenyl group or (Z) _p1 Represents a (C _a -C _b ) alkylcarbonyl group having the above meaning optionally substituted by, for example, as _a (C _a -C _b ) alkylcarbonyl group, for example, a —CH ₂ C (O) — group, —CH (CH ₃ ) C (O)-group, -C (CH ₃ ) ₂ C (O)-group, -CH ₂ CH ₂ C (O)-group, -CH (CH ₃ ) CH ₂ C (O)-group, -C (CH ₃ ) ₂ CH ₂ C (O)-group, -CH ₂ CH (CH ₃ ) C (O)-group, -CH ₂ C (CH ₃ ) ₂ C (O)-group, -CH ₂ Specific examples include CH ₂ CH ₂ C (O) — groups and the like, each selected within the range of the specified number of carbon atoms.

Representation of substituted phenyl (C _a ~C _b) alkoxycarbonyl by phenyl (C _a ~C _b) alkoxycarbonyl or (Z) _p1 in the present specification, a phenyl group substituted by a phenyl group or (Z) _p1 Represents a (C _a -C _b ) alkoxycarbonyl group having the above meaning optionally substituted by, for example, a (C _a -C _b ) alkoxycarbonyl group such as a —CH ₂ OC (O) — group, —CH (CH ₃ ) OC (O)-group, -C (CH ₃ ) ₂ OC (O)-group, -CH ₂ CH ₂ OC (O)-group, -CH (CH ₃ ) CH ₂ OC (O)-group, Specific examples include —C (CH ₃ ) ₂ CH ₂ OC (O) — group and the like, and each is selected within the range of the number of carbon atoms specified.

In this specification
[R ² represents that, together with R ¹ , a C ₂ -C ₆ alkylene chain may be formed to form a 3- to 7-membered ring with the nitrogen atom to which the alkylene chain is bonded. May contain one oxygen atom, sulfur atom or nitrogen atom,
[R ¹⁷ and R ¹⁸ together form a C _{4 to} C ₇ alkylene chain to form a 5- to 8-membered ring together with the nitrogen atom to which the alkylene chain is bonded. May contain one oxygen or sulfur atom,
[Represents that R ²⁶ and R ²⁷ may form a C ₂ -C ₅ alkylene chain together to form a 3- to 6-membered ring together with the nitrogen atom to which the R ²⁶ and R ²⁷ are bonded. May contain one oxygen or sulfur atom,
[Represents that R ²⁹ and R ³⁰ together form a C ₂ -C ₅ alkylene chain to form a 3- to 6-membered ring together with the nitrogen atom to which the alkylene chain is bonded. May contain one oxygen, sulfur or nitrogen atom,
as well as
[Represents that R ³⁴ and R ³⁵ together form a C ₂ -C ₅ alkylene chain to form a 3- to 6-membered ring with the nitrogen atom to which it is bonded. May contain one oxygen or sulfur atom,
Specific examples of the notation include, for example, aziridine, azetidine, pyrrolidine, oxazolidine, thiazolidine, imidazolidine, piperidine, morpholine, thiomorpholine, piperazine, homopiperidine, heptamethyleneimine, etc. Selected.

In this specification
[R ⁹ and R ¹⁰ together form a C _{2 to} C ₆ alkylene chain, which indicates that a 3 to 7 membered ring may be formed with the atoms to be bonded. May contain one oxygen, sulfur or nitrogen atom,
Specific examples of the notation include, for example, aziridine, azetidine, azetidin-2-one, pyrrolidine, pyrrolidin-2-one, oxazolidine, oxazolidine-2-one, thiazolidine, thiazolidine-2-one, imidazolidine, imidazolidine-2- ON, piperidine, piperidin-2-one, morpholine, tetrahydro-1,3-oxazin-2-one, thiomorpholine, tetrahydro-1,3-thiazin-2-one, piperazine, tetrahydropyrimidin-2-one, homopiperidine , Homopiperidin-2-one and the like, and each is selected within the range of the designated number of atoms.

In this specification
[R ¹¹ represents that, together with R ⁹ , a C ₂ -C ₄ alkylene chain may be formed to form a 5- to 7-membered ring with the atoms to be bonded. May contain one atom, sulfur atom or nitrogen atom,
Specific examples of the notation include, for example, isoxazoline, 1,4,2-dioxazoline, 1,4,2-oxathiazoline, 1,2,4-oxadiazoline, dihydro-1,2-oxazine, dihydro-1, 4,2-dioxazine, dihydro-1,4,2-oxathiazine, dihydro-4H-1,2,4-oxadiazine, tetrahydro-1,2-oxazepine, etc. are selected, each selected within the specified number of atoms Is done.

In the compounds included in the present invention, examples of the substituent represented by W ¹ or W ² include an oxygen atom or a sulfur atom, and among these, an oxygen atom is preferable.

  In the compounds included in the present invention, examples of the range of the substituent represented by X include the following groups. At this time, when m represents an integer of 2 or more in each of the following cases, each X may be the same as or different from each other.

  That is, X-I: a halogen atom.

  X-II: cyano and nitro.

X-III: C ₁ ~C ₆ alkyl and C ₁ -C ₆ haloalkyl.

X-IV: C ₁ ~C ₆ alkoxy, C ₁ -C ₆ haloalkoxy and C ₁ -C ₆ alkylsulfonyloxy.

XV: C ₁ ~C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl and C ₁ -C ₆ haloalkylsulfonyl.

X-VI: m represents an integer of 2 or more, two Xs are adjacent, and two adjacent Xs form —OCH ₂ O— or —OCH ₂ CH ₂ O— Forms a 5- or 6-membered ring with the carbon atom to which it is attached. In this case, a hydrogen atom is a halogen atom attached to each carbon atom forming the ring may be optionally substituted by C ₁ -C ₄ alkyl or C ₁ -C ₄ haloalkyl group.

  In the compound included in the present invention, m representing the number of substituents represented by X includes an integer of 0 to 4. Among these, m is preferably 0, 1 or 2.

  In the compounds included in the present invention, examples of the range of the substituent represented by Y include the following groups. At this time, when n represents an integer of 2 or more in each of the following cases, each Y may be the same as or different from each other.

  That is, Y-I: a halogen atom.

Y-II: C ₁ ~C ₆ alkyl.

Y-III: C ₁ ~C ₆ haloalkyl, hydroxy (C ₁ ~C ₆₎ alkyl and C ₁ -C ₄ alkoxy (C ₁ ~C ₄₎ alkyl.

Y-IV: C ₁ ~C ₆ alkoxy and C ₁ -C ₆ haloalkoxy.

YV: C ₁ ~C ₆ alkylthio and C ₁ -C ₆ haloalkylthio.

Y-VI: C ₁ ~C ₆ alkyl amino and di (C ₁ -C ₆ alkyl) amino.

  In the compounds included in the present invention, n representing the number of substituents represented by Y includes an integer of 0 to 4, and among these, n is preferably 0, 1 or 2.

In the compounds included in the present invention, examples of the range of the substituent represented by R ¹ include the following groups.

That is, R ¹ -I: C ₁ -C ₈ alkyl and C ₃ -C ₈ cycloalkyl.

R ¹ -II: C ₁ -C ₈ alkyl optionally substituted by —OR ²⁶ [where R ²⁶ is C ₁ -C ₆ alkyl, C ₁ -C ₆ alkylaminocarbonyl or di (C ₁ -C ₆ Alkyl) aminocarbonyl. ].

R ¹ -III: C ₁ -C ₈ alkyl optionally substituted by —CH═NOH or —CH═NOR ³¹ [where R ³¹ represents C ₁ -C ₆ alkyl. ].

R ¹ -IV: in C ₁ -C ₈ alkyl [wherein optionally substituted by R ^16, R ¹⁶ represents -OR ^26, R ²⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₄ alkoxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkylthio (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, substituted by (Z) _p1 phenyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₃ -C ₆ cycloalkylcarbonyl, -C (O) N (R 30) R 29, di ( C ₁ -C ₆ alkyl) represents phosphoryl, di (C ₁ -C ₆ alkyl) thiophosphoryl, tri (C ₁ -C ₄ alkyl) silyl, phenyl substituted by phenyl or (Z) _p1, R ²⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C _{1 ~C 4)} alkyl, C ₁ -C ₄ alkylthio (C _{1 ~C 4)} alkyl, phenyl (C _{1 ~C 4)} alkyl, (Z) _p1 Replaced by Alkylsulfonyl (C ₁ ~C ₄₎ represents alkyl, C ₃ -C ₆ cycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, phenyl substituted by phenyl or (Z) _p1, R ³⁰ is hydrogen or represents an atom or C ₁ -C ₆ alkyl, or, by the R ²⁹ and R ³⁰ form a C ₂ -C ₅ alkylene chain together, form a 3-6 membered ring together with the nitrogen atom attached In this case, this alkylene chain may contain one oxygen atom or sulfur atom. ], M-4, M-5, M-14, M-15 and M-16.

R ¹ -V: by R ¹⁶ C ₁ ~C ₈ alkyl [wherein optionally substituted, R ¹⁶ is cyano, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ alkylaminocarbonyl, di (C ₁ ~ C ₆ alkyl) aminocarbonyl, represents -C (R ³²⁾ = NOH or ^{-C (R 32) = NOR 31} , R 31 is C ₁ -C ₆ alkyl, phenyl (C ₁ -C ₄₎ alkyl or (Z ) represents phenyl (C ₁ -C ₄ ) alkyl substituted by _{p 1} , and R ³² represents a hydrogen atom or C ₁ -C ₆ alkyl. ].

R ¹ -VI: optionally substituted C ₁ -C ₈ alkyl [wherein the R ^16, R ¹⁶ is a halogen atom, C ₃ -C ₆ cycloalkyl, tri (C ₁ -C ₆ alkyl) silyl, phenyl, (Z) represents phenyl, L-1, L-2, L-3, L-4, L-45, L-46, L-47 or M substituted by _p1 . ].

R _¹ -VII: C ^{1 ~C} ₆ alkyl, C ₁ -C ₄ alkylthio (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkylsulfinyl (C ₁ ~C ₄₎ alkyl and C ₁ -C ₄ alkylsulfonyl (C ₁ ~C ₄₎ alkyl.

R ¹ -VIII: C ₃ ~C ₈ alkenyl and C ₃ -C ₈ alkynyl.

R ¹ -IX: C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylsulfinyl (C ₁ -C ₄ ) alkyl and C ₁ -C ₄ alkylsulfonyl (C ₁ -C ₄ ) Alkyl.

R ¹ -X: (C ₁ -C ₈ ) alkyl optionally substituted by —N (R ²⁷ ) R ²⁶ , wherein R ²⁶ is C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ alkylsulfonyl or It represents di (C ₁ -C ₆ alkyl) thiophosphoryl, and R ²⁷ represents a hydrogen atom or C ₁ -C ₆ alkyl. ].

R _¹ -XI: C ¹ ~C ₈ alkyl [wherein optionally substituted by R ^16, R ¹⁶ represents -S (O) _{r R} ²⁸ or ^{_{-SO 2 N (R 30) R}} 29, R 28 the C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, hydroxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkoxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkylthio (C ₁ ~ C ₄₎ alkyl, C ₁ -C ₄ alkylcarbonyl (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkoxycarbonyl (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkylaminocarbonyl (C ₁ -C ₄₎ alkyl, di (C ₁ -C ₄ alkyl) aminocarbonyl (C ₁ -C ₄₎ alkyl, tri (C ₁ -C ₄ alkyl) silyl (C ₁ -C ₄₎ alkyl, phenyl (C ₁ -C ₄ ) substituted alkyl, by (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, C ₁ -C ₆ alkylthio, phenyl, (Z) _p1 Phenyl, L-21, L-35, L-45 or L-4 8, r represents an integer of 0 to 2, R ²⁹ represents C _{1 to} C ₆ alkyl, and R ³⁰ represents a hydrogen atom or C _{1 to} C ₆ alkyl. ], M-8, M-9, M-17, M-18 and M-19.

R ¹ XII: by R ¹⁶ is C ₁ -C ₈ alkyl [here was an optionally substituted, R ¹⁶ represents ^{-N (R 27) R 26,} R 26 is C ₁ -C ₆ alkylcarbonyl, C ₃ -C ₆ cycloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl, C ₁ -C ₆ alkylsulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl, phenylsulfonyl, (Z) represents phenylsulfonyl or di (C ₁ -C ₆ alkyl) thiophosphoryl substituted by _{p 1} , and R ²⁷ represents a hydrogen atom or C ₁ -C ₆ alkyl. ], M-13, M-21 and M-22.

R ¹ -XIII: A 3- to 7-membered ring formed by combining R ¹ and R ² is aziridine, azetidine, pyrrolidine, oxazolidine, thiazolidine, piperidine, morpholine, thiomorpholine and homopiperidine.

R ¹ -XIV: C ₁ -C ₆ alkyl, C ₁ -C ₄ alkyl optionally substituted by —OR ²⁶ [where R ²⁶ is C ₁ -C ₄ alkyl, C ₁ -C ₄ alkylaminocarbonyl or Represents di (C ₁ -C ₄ alkyl) aminocarbonyl. ], C ₁ -C ₄ alkylthio (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkylsulfinyl (C ₁ ~C ₄₎ alkyl and C ₁ -C ₄ alkylsulfonyl (C ₁ ~C ₄₎ alkyl, - (C ₁ -C ₄ ) alkyl optionally substituted by N (R ²⁷ ) R ²⁶ , wherein R ²⁶ is C ₁ -C ₄ alkoxycarbonyl, C ₁ -C ₄ alkylsulfonyl or di (C ₁ -C ₄ alkyl) thiophosphoryl, R ²⁷ represents a hydrogen atom or C ₁ -C ₄ alkyl. And C ₁ -C ₄ alkyl optionally substituted by —CH═NOH or —CH═NOR ³¹ , wherein R ³¹ represents C ₁ -C ₄ alkyl. ].

In the compounds included in the present invention, examples of the range of substituents represented by R ² and R ³ include the following groups.

That is, R ² -I or R ³ -I: a hydrogen atom.

R ² -II or R ³ -II: hydrogen atom and C ₁ -C ₆ alkyl.

R ² -III or R ³ -III: hydrogen atom, C ₁ -C ₄ alkoxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₄ alkylthio (C ₁ ~C ₄₎ alkyl and C ₁ -C ₄ alkylsulfonyl (C ₁ ~C ₄₎ alkyl.

R ² -IV or R ³ -IV: a hydrogen atom, C ₃ -C ₆ alkenyl and C ₃ -C ₆ alkynyl.

R ² -V or R ³ -V: hydrogen atom, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z) phenylthio and -SN substituted by _p1 (R ¹⁸⁾ R ¹⁷ [wherein R ¹⁷ represents C ₁ -C ₆ alkyl, C ₁ -C ₆ alkoxycarbonyl (C ₁ -C ₄ ) alkyl or C ₁ -C ₆ alkoxycarbonyl, and R ¹⁸ represents C ₁ -C ₆ alkyl Or R ¹⁷ and R ¹⁸ together form a C _{4 to} C ₅ alkylene chain to form a 5- or 6-membered ring with the nitrogen atom to which it is bound, Sometimes this alkylene chain may contain one oxygen or sulfur atom and may be optionally substituted with a methyl or methoxy group. ].

In the compound included in the present invention, examples of the range of the substituent represented by R ⁴ include the following groups.

That is, R ⁴ -I: C ₁ -C ₆ alkyl and C ₁ -C ₆ haloalkyl.

R ⁴ -II: C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl and C ₃ -C ₈ halocycloalkyl.

R ⁴ -III: optionally substituted by R ²¹ (C ₁ ~C ₆₎ optionally substituted by alkyl and R ²¹ (C ₁ ~C ₆₎ haloalkyl [wherein, R ²¹ is cyano, C ₃ ~ C ₆ cycloalkyl, C ₃ -C ₆ halocycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z) _p1 phenoxy substituted by, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z) phenylthio substituted by _p1, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, phenylsulfonyl, (Z) phenylsulfonyl substituted by _p1, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino, phenylamino, (Z) phenylamino substituted by _p1, C ₁ ~ C ₆ alkoxycarbonyl , Phenyl, (Z) phenyl substituted by _p1 , L-1 to L-5, L-8 to L-24, L-36, L-39, L-45 to L-52 or L-53 . ].

R ⁴ -IV: C ₃ -C ₆ haloalkenyl, C ₃ -C ₆ haloalkynyl, phenyl and phenyl substituted by (Z) _p1 .

In the compounds included in the present invention, examples of the range of the substituent represented by R ⁵ include the following groups.

_{^{That, R 5 -I: (C 1}} ~C 6) alkyl, optionally substituted by R ²¹ optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, optionally substituted by R ²¹ ( optionally substituted by C ₂ -C ₆₎ alkenyl and R ²¹ (C ₂ ~C ₆₎ alkynyl [where, R ²¹ is C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z ) _p1 phenoxy substituted by, phenylthio, phenylthio substituted by (Z) _p1, phenylsulfonyl, (Z) phenylsulfonyl substituted by _p1, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl ) amino, phenylamino, (Z) phenylamino substituted by _p1, C ₁ -C ₆ alkoxycarbonyl, phenyl, phenyl substituted by _{(Z) p1, L-1~L} -5, L-8~L -24, L-36, L-39, L-45 to L-52 or L-53. ].

R ⁵ -II: optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, R ²¹ (C ₂ -C ₆₎ optionally substituted by alkenyl and R ²¹ (C ₂ ~C ₆₎ alkynyl [where, R ²¹ is cyano, C ₃ -C ₆ cycloalkyl, C ₃ -C ₆ halocycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, substituted by (Z) _p1 phenoxy substituted by, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z) _p1 phenylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, phenylsulfonyl, phenylsulfonyl substituted by (Z) _p1, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ A Kill) amino, phenylamino, (Z) phenylamino substituted by _p1, C ₁ -C ₆ alkoxycarbonyl, phenyl, (Z) phenyl substituted by _{p1, L-1~L-5,} L-8~ L-24, L-36, L-39, L-45 to L-52 or L-53 is represented. ].

R ⁵ -III: phenyl, (Z) phenyl substituted by _p1, (Z) phenoxyphenyl phenyl substituted by _p1, (Z) pyridyloxy phenyl substituted by _{p1, L-1~L-4,} L- 8 to L-13, L-15 to L-23, L-45 to L-52 and L-53.

R ⁵ -IV: C ₃ ~C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, phenyl, (Z) phenyl substituted by _p1, phenoxyphenyl substituted by (Z) _p1, by (Z) _p1 Substituted pyridyloxyphenyl, L-1 to L-4, L-8 to L-13, L-15 to L-23, L-25 to L-35, L-37, L-38, L-40 , L-43 to L-58, M-4, M-5, M-8, M-9, M-14 to M-18 and M-19.

R ⁵ -V: cyano, -C (O) OR ⁹ , -C (O) SR ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) NHR ¹⁰ and -C (S) N (R ¹⁰ ) R ⁹ [where R ⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl , C ₃ -C ₆ cycloalkyl (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ substituted by (Z) _p1 alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, phenyl which is substituted by phenyl or (Z) _p1, or R ¹⁰ represents a hydrogen atom or a C ₁ -C ₆ alkyl, or the R ⁹ and R ¹⁰ Together form a C _{4 to} C ₅ alkylene chain to form a 5-membered or 6-membered ring with the nitrogen atom to which the alkylene chain is bonded. Indicates that one atom may be included. ].

R ⁵ -VI: Forms a C ₂ -C ₃ alkylene chain together with Y present at the adjacent position, thereby forming a 5- to 6-membered ring condensed with the benzene ring. At this time, the alkylene chain is oxygen atoms, it may contain one sulfur atom or nitrogen atom may be optionally substituted and the halogen atom or a C ₁ -C ₆ haloalkyl group.

In the compounds included in the present invention, examples of the range of the substituent represented by R ⁶ include the following groups.

That is, R ⁶ -I: a hydrogen atom.

R ⁶ -II: a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylcarbonyl and tri (C ₁ -C ₄ alkyl) silyl.

R ⁶ -III: hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl, cyano (C ₁ ~C ₆₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ ~ C ₆ haloalkenyl, phenyl (C ₃ -C ₆₎ alkenyl, (Z) phenyl substituted by _p1 (C ₃ ~C ₆₎ alkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, phenyl ( C ₃ -C ₆₎ alkynyl, (Z) phenyl substituted by _p1 (C ₃ ~C _{6) ^{alkynyl, -S (O) 2 R 9}} , -C (O) R 9, -C (O) NHR 10 , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ [where R ⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ cycloalkyl (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, it is substituted by (Z) _p1 Represents phenyl (C ₁ -C ₄ ) alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, phenyl or phenyl substituted by (Z) _p1 , and R ¹⁰ represents a hydrogen atom or C Represents _{1 to} C ₆ alkyl, or R ⁹ and R ¹⁰ together form a C _{4 to} C ₅ alkylene chain to form a 5- or 6-membered ring with the nitrogen atom to which it is attached. In this case, this alkylene chain may contain one oxygen atom or one sulfur atom. ], -Si (R ¹³ ) (R ¹⁴ ) R ¹² [wherein R ¹² represents C ₁ -C ₆ alkyl, phenyl or phenyl substituted by (Z) _{p 1} , and R ¹³ and R ¹⁴ are each independently and it represents a C ₁ -C ₆ alkyl. ], -P (O) (OR ²² ) ₂ and -P (S) (OR ²² ) ₂ [wherein R ²² represents C ₁ -C ₆ alkyl. ].

Each group which shows the range of each substituent in these compounds included in the present invention can be arbitrarily combined, and each represents the range of the present compound. Examples of combinations of ranges for R ¹ , R ⁴ , R ⁵ and R ⁶ include the combinations shown in Table 1 below. However, the combinations in Table 1 are for illustrative purposes, and the present invention is not limited to these.
Table 1 Table 1 (continued)
―――――――――――――――――― ――――――――――――――――――
R ¹ R ⁴ R ⁵ R ⁶ R ¹ R ⁴ R ⁵ R ⁶
―――――――――――――――――― ――――――――――――――――――
R ¹ -IR ⁴ -IR ⁵ -IR ⁶ -IR ¹ -VIII R ⁴ -IR ⁵ -IR ⁶ -I
R ¹ -IR ⁴ -IR ⁵ -IR ⁶ -II R ¹ -VIII R ⁴ -IR ⁵ -IR ⁶ -II
R ¹ -IR ⁴ -IR ⁵ -III R ⁶ -IR ¹ -VIII R ⁴ -IR ⁵ -III R ⁶ -I
R ¹ -IR ⁴ -IR ⁵ -III R ⁶ -II R ¹ -VIII R ⁴ -IR ⁵ -III R ⁶ -II
R ¹ -IR ⁴ -IR ⁵ -VI R ⁶ -IR ¹ -VIII R ⁴ -IR ⁵ -VI R ⁶ -I
R ¹ -IR ⁴ -IR ⁵ -VI R ⁶ -II R ¹ -VIII R ⁴ -IR ⁵ -VI R ⁶ -II
^{R 1 -II R 4 -IR 5 -IR} 6 -IR 1 -IX R 4 -IR 5 -IR 6 -I
^{R 1 -II R 4 -IR 5 -IR} 6 -II R 1 -IX R 4 -IR 5 -IR 6 -II
^{R 1 -II R 4 -IR 5 -III} R 6 -IR 1 -IX R 4 -IR 5 -III R 6 -I
^{R 1 -II R 4 -IR 5 -III} R 6 -II R 1 -IX R 4 -IR 5 -III R 6 -II
^{R 1 -II R 4 -IR 5 -III} R 6 -III R 1 -IX R 4 -IR 5 -III R 6 -III
R ¹ -II R ⁴ -IR ⁵ -IV R ⁶ -IR ¹ -IX R ⁴ -IR ⁵ -IV R ⁶ -I
R ¹ -II R ⁴ -IR ⁵ -IV R ⁶ -II R ¹ -IX R ⁴ -IR ⁵ -IV R ⁶ -II
R ¹ -II R ⁴ -IR ⁵ -VR ⁶ -IR ¹ -IX R ⁴ -IR ⁵ -VR ⁶ -I
R ¹ -II R ⁴ -IR ⁵ -VR ⁶ -II R ¹ -IX R ⁴ -IR ⁵ -VR ⁶ -II
R ¹ -II R ⁴ -IR ⁵ -VI R ⁶ -IR ¹ -IX R ⁴ -IR ⁵ -VI R ⁶ -I
R ¹ -II R ⁴ -IR ⁵ -VI R ⁶ -II R ¹ -IX R ⁴ -IR ⁵ -VI R ⁶ -II
R ¹ -II R ⁴ -II R ⁵ -IR ⁶ -IR ¹ -IX R ⁴ -II R ⁵ -IR ⁶ -I
R ¹ -II R ⁴ -II R ⁵ -IR ⁶ -II R ¹ -IX R ⁴ -II R ⁵ -IR ⁶ -II
R ¹ -II R ⁴ -II R ⁵ -III R ⁶ -IR ¹ -IX R ⁴ -II R ⁵ -III R ⁶ -I
R ¹ -II R ⁴ -II R ⁵ -III R ⁶ -II R ¹ -IX R ⁴ -II R ⁵ -III R ⁶ -II
^{R 1 -II R 4 -II R 5} -III R 6 -III R 1 -IX R 4 -II R 5 -III R 6 -III
R ¹ -II R ⁴ -II R ⁵ -IV R ⁶ -IR ¹ -IX R ⁴ -II R ⁵ -IV R ⁶ -I
R ¹ -II R ⁴ -II R ⁵ -IV R ⁶ -II R ¹ -IX R ⁴ -II R ⁵ -IV R ⁶ -II
R ¹ -II R ⁴ -II R ⁵ -VR ⁶ -IR ¹ -IX R ⁴ -II R ⁵ -VR ⁶ -I
R ¹ -II R ⁴ -II R ⁵ -VR ⁶ -II R ¹ -IX R ⁴ -II R ⁵ -VR ⁶ -II
R ¹ -II R ⁴ -II R ⁵ -VI R ⁶ -IR ¹ -IX R ⁴ -II R ⁵ -VI R ⁶ -I
R ¹ -II R ⁴ -II R ⁵ -VI R ⁶ -II R ¹ -IX R ⁴ -II R ⁵ -VI R ⁶ -II
^{R 1 -II R 4 -III R 5} -III R 6 -IR 1 -IX R 4 -III R 5 -III R 6 -I
^{R 1 -II R 4 -III R 5} -III R 6 -II R 1 -IX R 4 -III R 5 -III R 6 -II
R ¹ -II R ⁴ -IV R ⁵ -III R ⁶ -IR ¹ -IX R ⁴ -IV R ⁵ -III R ⁶ -I
^{R 1 -III R 4 -IR 5 -IR} 6 -IR 1 -XR 4 -IR 5 -IR 6 -I
^{R 1 -III R 4 -IR 5 -IR} 6 -II R 1 -XR 4 -IR 5 -IR 6 -II
^{R 1 -III R 4 -IR 5 -III} R 6 -IR 1 -XR 4 -IR 5 -III R 6 -I
^{R 1 -III R 4 -IR 5 -III} R 6 -II R 1 -XR 4 -IR 5 -III R 6 -II
^{R 1 -III R 4 -IR 5 -III} R 6 -III R 1 -XR 4 -IR 5 -III R 6 -III
^{R 1 -III R 4 -IR 5 -IV} R 6 -IR 1 -XR 4 -IR 5 -IV R 6 -I
^{R 1 -III R 4 -IR 5 -IV} R 6 -II R 1 -XR 4 -IR 5 -IV R 6 -II
^{R 1 -III R 4 -IR 5 -VR} 6 -IR 1 -XR 4 -IR 5 -VR 6 -I
^{R 1 -III R 4 -IR 5 -VR} 6 -II R 1 -XR 4 -IR 5 -VR 6 -II
^{R 1 -III R 4 -IR 5 -VI} R 6 -IR 1 -XR 4 -IR 5 -VI R 6 -I
^{R 1 -III R 4 -IR 5 -VI} R 6 -II R 1 -XR 4 -IR 5 -VI R 6 -II
^{R 1 -III R 4 -II R 5} -IR 6 -IR 1 -XR 4 -II R 5 -IR 6 -I
^{R 1 -III R 4 -II R 5} -IR 6 -II R 1 -XR 4 -II R 5 -IR 6 -II
^{R 1 -III R 4 -II R 5} -III R 6 -IR 1 -XR 4 -II R 5 -III R 6 -I
^{R 1 -III R 4 -II R 5} -III R 6 -II R 1 -XR 4 -II R 5 -III R 6 -II
^{R 1 -III R 4 -II R 5} -III R 6 -III R 1 -XR 4 -II R 5 -III R 6 -III
R ¹ -III R ⁴ -II R ⁵ -IV R ⁶ -IR ¹ -XR ⁴ -II R ⁵ -IV R ⁶ -I
R ¹ -III R ⁴ -II R ⁵ -IV R ⁶ -II R ¹ -XR ⁴ -II R ⁵ -IV R ⁶ -II
R ¹ -III R ⁴ -II R ⁵ -VR ⁶ -IR ¹ -XR ⁴ -II R ⁵ -VR ⁶ -I
R ¹ -III R ⁴ -II R ⁵ -VR ⁶ -II R ¹ -XR ⁴ -II R ⁵ -VR ⁶ -II
R ¹ -III R ⁴ -II R ⁵ -VI R ⁶ -IR ¹ -XR ⁴ -II R ⁵ -VI R ⁶ -I
R ¹ -III R ⁴ -II R ⁵ -VI R ⁶ -II R ¹ -XR ⁴ -II R ⁵ -VI R ⁶ -II
^{R 1 -III R 4 -III R 5} -III R 6 -IR 1 -XR 4 -III R 5 -III R 6 -I
^{R 1 -III R 4 -III R 5} -III R 6 -II R 1 -XR 4 -III R 5 -III R 6 -II
^{R 1 -III R 4 -IV R 5} -III R 6 -IR 1 -XR 4 -IV R 5 -III R 6 -I
R ¹ -IV R ⁴ -IR ⁵ -IR ⁶ -IR ¹ -XI R ⁴ -IR ⁵ -IR ⁶ -I
R ¹ -IV R ⁴ -IR ⁵ -III R ⁶ -IR ¹ -XI R ⁴ -IR ⁵ -III R ⁶ -I
R ¹ -IV R ⁴ -IR ⁵ -III R ⁶ -II R ¹ -XI R ⁴ -IR ⁵ -III R ⁶ -II
R ¹ -IV R ⁴ -IR ⁵ -VI R ⁶ -IR ¹ -XI R ⁴ -IR ⁵ -VI R ⁶ -I
R ¹ -VR ⁴ -IR ⁵ -IR ⁶ -IR ¹ -XII R ⁴ -IR ⁵ -IR ⁶ -I
R ¹ -VR ⁴ -IR ⁵ -III R ⁶ -IR ¹ -XII R ⁴ -IR ⁵ -III R ⁶ -I
R ¹ -VR ⁴ -IR ⁵ -III R ⁶ -II R ¹ -XII R ⁴ -IR ⁵ -III R ⁶ -II
R ¹ -VR ⁴ -IR ⁵ -VI R ⁶ -IR ¹ -XII R ⁴ -IR ⁵ -VI R ⁶ -I
^{R 1 -VI R 4 -IR 5 -IR} 6 -IR 1 -XIII R 4 -IR 5 -IR 6 -I
^{R 1 -VI R 4 -IR 5 -III} R 6 -IR 1 -XIII R 4 -IR 5 -III R 6 -I
^{R 1 -VI R 4 -IR 5 -III} R 6 -II R 1 -XIII R 4 -IR 5 -III R 6 -II
R ¹ -VI R ⁴ -IR ⁵ -VI R ⁶ -IR ¹ -XIII R ⁴ -IR ⁵ -VI R ⁶ -I
^{R 1 -VII R 4 -IR 5 -IR} 6 -IR 1 -XIV R 4 -IR 5 -IR 6 -I
^{R 1 -VII R 4 -IR 5 -IR} 6 -II R 1 -XIV R 4 -IR 5 -IR 6 -II
^{R 1 -VII R 4 -IR 5 -IR} 6 -III R 1 -XIV R 4 -IR 5 -IR 6 -III
^{R 1 -VII R 4 -IR 5 -II} R 6 -IR 1 -XIV R 4 -IR 5 -II R 6 -I
^{R 1 -VII R 4 -IR 5 -II} R 6 -II R 1 -XIV R 4 -IR 5 -II R 6 -II
^{R 1 -VII R 4 -IR 5 -III} R 6 -IR 1 -XIV R 4 -IR 5 -III R 6 -I
^{R 1 -VII R 4 -IR 5 -III} R 6 -II R 1 -XIV R 4 -IR 5 -III R 6 -II
^{R 1 -VII R 4 -IR 5 -III} R 6 -III R 1 -XIV R 4 -IR 5 -III R 6 -III
^{R 1 -VII R 4 -IR 5 -IV} R 6 -IR 1 -XIV R 4 -IR 5 -IV R 6 -I
^{R 1 -VII R 4 -IR 5 -IV} R 6 -II R 1 -XIV R 4 -IR 5 -IV R 6 -II
^{R 1 -VII R 4 -IR 5 -IV} R 6 -III R 1 -XIV R 4 -IR 5 -IV R 6 -III
^{R 1 -VII R 4 -IR 5 -VR} 6 -IR 1 -XIV R 4 -IR 5 -VR 6 -I
^{R 1 -VII R 4 -IR 5 -VR} 6 -II R 1 -XIV R 4 -IR 5 -VR 6 -II
^{R 1 -VII R 4 -IR 5 -VI} R 6 -IR 1 -XIV R 4 -IR 5 -VI R 6 -I
^{R 1 -VII R 4 -IR 5 -VI} R 6 -II R 1 -XIV R 4 -IR 5 -VI R 6 -II
^{R 1 -VII R 4 -IR 5 -VI} R 6 -III R 1 -XIV R 4 -IR 5 -VI R 6 -III
^{R 1 -VII R 4 -II R 5} -IR 6 -IR 1 -XIV R 4 -II R 5 -IR 6 -I
^{R 1 -VII R 4 -II R 5} -IR 6 -II R 1 -XIV R 4 -II R 5 -IR 6 -II
^{R 1 -VII R 4 -II R 5} -II R 6 -IR 1 -XIV R 4 -II R 5 -II R 6 -I
^{R 1 -VII R 4 -II R 5} -III R 6 -IR 1 -XIV R 4 -II R 5 -III R 6 -I
^{R 1 -VII R 4 -II R 5} -III R 6 -II R 1 -XIV R 4 -II R 5 -III R 6 -II
^{R 1 -VII R 4 -II R 5} -IV R 6 -IR 1 -XIV R 4 -II R 5 -IV R 6 -I
R ¹ -VII R ⁴ -II R ⁵ -IV R ⁶ -II R ¹ -XIV R ⁴ -II R ⁵ -IV R ⁶ -II
^{R 1 -VII R 4 -II R 5} -VR 6 -IR 1 -XIV R 4 -II R 5 -VR 6 -I
^{R 1 -VII R 4 -II R 5} -VI R 6 -IR 1 -XIV R 4 -II R 5 -VI R 6 -I
R ¹ -VII R ⁴ -II R ⁵ -VI R ⁶ -II R ¹ -XIV R ⁴ -II R ⁵ -VI R ⁶ -II
^{R 1 -VII R 4 -III R 5} -IR 6 -IR 1 -XIV R 4 -III R 5 -IR 6 -I
^{R 1 -VII R 4 -III R 5} -IR 6 -II R 1 -XIV R 4 -III R 5 -IR 6 -II
^{R 1 -VII R 4 -III R 5} -III R 6 -IR 1 -XIV R 4 -III R 5 -III R 6 -I
^{R 1 -VII R 4 -III R 5} -III R 6 -II R 1 -XIV R 4 -III R 5 -III R 6 -II
^{R 1 -VII R 4 -III R 5} -IV R 6 -IR 1 -XIV R 4 -III R 5 -IV R 6 -I
^{R 1 -VII R 4 -III R 5} -VR 6 -IR 1 -XIV R 4 -III R 5 -VR 6 -I
^{R 1 -VII R 4 -III R 5} -VI R 6 -IR 1 -XIV R 4 -III R 5 -VI R 6 -I
^{R 1 -VII R 4 -IV R 5} -IR 6 -IR 1 -XIV R 4 -IV R 5 -IR 6 -I
^{R 1 -VII R 4 -IV R 5} -IR 6 -II R 1 -XIV R 4 -IV R 5 -IR 6 -II
^{R 1 -VII R 4 -IV R 5} -III R 6 -IR 1 -XIV R 4 -IV R 5 -III R 6 -I
^{R 1 -VII R 4 -IV R 5} -III R 6 -II R 1 -XIV R 4 -IV R 5 -III R 6 -II
^{R 1 -VII R 4 -IV R 5} -IV R 6 -IR 1 -XIV R 4 -IV R 5 -IV R 6 -I
^{R 1 -VII R 4 -IV R 5} -VR 6 -IR 1 -XIV R 4 -IV R 5 -VR 6 -I
^{R 1 -VII R 4 -IV R 5} -VI R 6 -IR 1 -XIV R 4 -IV R 5 -VI R 6 -I
―――――――――――――――――― ――――――――――――――――――
The compound of the present invention can be produced, for example, by the following method.

  Manufacturing method A

General formula (4) [wherein W ¹ , W ² , X, Y, R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. And a compound represented by the general formula (5): wherein R ¹ and R ² represent the same meaning as described above. In a solvent inert to the reaction or in the absence of a solvent, if necessary, in the presence of a catalyst, R ³ is a hydrogen atom in the general formula (1). A certain general formula (1-1) [wherein W ¹ , W ² , X, Y, R ¹ , R ² , R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. This invention compound represented by this can be obtained.

  As the amount of the reaction substrate, 1 to 50 equivalents of the compound represented by the general formula (5) can be used per 1 equivalent of the compound represented by the general formula (4).

  In the case of using a solvent, any solvent may be used as long as it does not inhibit the progress of the reaction. For example, aromatic hydrocarbons such as benzene, toluene and xylene, aliphatic hydrocarbons such as hexane and heptane, cyclohexane, etc. Alicyclic hydrocarbons, aromatic halogenated hydrocarbons such as chlorobenzene and dichlorobenzene, fats such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, 1,1,1-trichloroethane, trichloroethylene and tetrachloroethylene Group halogenated hydrocarbons, ethers such as diethyl ether, 1,2-dimethoxyethane, tetrahydrofuran and 1,4-dioxane, esters such as ethyl acetate and ethyl propionate, dimethylformamide, dimethylacetamide, N-methyl- Amides such as 2-pyrrolidone, formic acid, acetic acid, propylene Carboxylic acids such as on acid, amines such as triethylamine, tributylamine, N, N-dimethylaniline, pyridines such as pyridine and picoline, alcohols such as methanol, ethanol and ethylene glycol, acetonitrile, dimethyl sulfoxide, sulfolane, 1 , 3-dimethyl-2-imidazolidinone and water. These solvents may be used alone or as a mixture of two or more thereof.

  When using a catalyst, examples of the reaction catalyst include mineral acids such as hydrochloric acid, sulfuric acid, and nitric acid, and organic acids such as formic acid, acetic acid, propionic acid, trifluoroacetic acid, methanesulfonic acid, benzenesulfonic acid, and p-toluenesulfonic acid. Acid addition salts of amines such as triethylamine hydrochloride, pyridine hydrochloride, Lewis acids such as zinc chloride, zinc iodide, titanium tetrachloride, cerium chloride, ytterbium triflate, boron trifluoride-ether complex, 0.001 to 1 equivalent can be used with respect to the compound represented by (4).

  The reaction temperature can be set to an arbitrary temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrarily within the range of 5 minutes to 100 hours. Can be set.

  In general, for example, 1 to 10 equivalents of the compound represented by the general formula (5) is used per 1 equivalent of the compound represented by the general formula (4), and no solvent is used. The reaction is preferably carried out in a temperature range of 50 ° C. to the reflux temperature of the reaction mixture using a solvent such as dioxane for 30 minutes to 24 hours.

  Manufacturing method B

Formula (6) [wherein W ² , X, Y, R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. And a compound represented by the general formula (5): wherein R ¹ and R ² represent the same meaning as described above. And a compound represented by the general formula (1-2) in which W ¹ is an oxygen atom and R ³ is a hydrogen atom in the general formula (1). In the formula, W ² , X, Y, R ¹ , R ² , R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. This invention compound represented by this can be obtained.

  Manufacturing method C

General formula (7) [wherein W ¹ , X, R ¹ and m represent the same meaning as described above. And a compound represented by the general formula (8): wherein Y, R ³ , R ⁴ , R ⁵ , R ⁶ and n have the same meaning as described above. And a compound represented by the general formula (1-3) in which W ² is an oxygen atom and R ² is a hydrogen atom in the general formula (1). In the formula, W ¹ , X, Y, R ¹ , R ³ , R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. This invention compound represented by this can be obtained.

  Manufacturing method D

General formula (9) [wherein W ² , X, Y, R ³ , R ⁴ , R ⁵ , R ⁶ , m, and n represent the same meaning as described above. And a compound represented by the general formula (5): wherein R ¹ and R ² represent the same meaning as described above. In the general formula (1), the compound represented by the general formula (1) is reacted with a compound in a solvent inert to the reaction or without a solvent, if necessary, in the presence of a base. General formula (1-4) wherein ¹ is an oxygen atom [wherein W ² , X, Y, R ¹ , R ² , R ³ , R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above] Represents. This invention compound represented by this can be obtained.

  The amount of the reaction substrate may be 1 to 100 equivalents of the compound represented by the general formula (5) with respect to 1 equivalent of the compound represented by the general formula (9).

  The condensing agent is not particularly limited as long as it is used for ordinary amide synthesis. For example, Mukaiyama reagent (2-chloro-N-methylpyridinium iodide), DCC (1,3-dicyclohexylcarbodiimide), WSC (1 -Ethyl-3- (3-dimethylaminopropyl) -carbodiimide hydrochloride), CDI (carbonyldiimidazole), dimethylpropynylsulfonium bromide, propargyltriphenylphosphonium bromide, DEPC (diethyl cyanophosphate), etc. 1-4 equivalent can be used with respect to the compound represented by these.

  In the case of using a solvent, any solvent may be used as long as it does not inhibit the progress of the reaction. For example, aromatic hydrocarbons such as benzene, toluene and xylene, aliphatic hydrocarbons such as hexane and heptane, cyclohexane, etc. Alicyclic hydrocarbons, aromatic halogenated hydrocarbons such as chlorobenzene and dichlorobenzene, fats such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, 1,1,1-trichloroethane, trichloroethylene and tetrachloroethylene Group halogenated hydrocarbons, ethers such as diethyl ether, 1,2-dimethoxyethane, tetrahydrofuran and 1,4-dioxane, esters such as ethyl acetate and ethyl propionate, dimethylformamide, dimethylacetamide, N-methyl- Amides such as 2-pyrrolidone, triethylamine, Examples include amines such as tributylamine and N, N-dimethylaniline, pyridines such as pyridine and picoline, acetonitrile, and dimethyl sulfoxide. These solvents may be used alone or as a mixture of two or more thereof.

  Although the addition of a base is not always necessary, when a base is used, examples of the base used include alkali metal hydroxides such as sodium hydroxide and potassium hydroxide, alkali metals such as sodium carbonate, potassium carbonate and sodium hydrogen carbonate. Organic bases such as carbonate, triethylamine, tributylamine, N, N-dimethylaniline, pyridine, 4- (dimethylamino) pyridine, imidazole, 1,8-diazabicyclo [5,4,0] -7-undecene, etc. 1 to 4 equivalents can be used with respect to the compound represented by the general formula (9).

  The reaction temperature can be set to an arbitrary temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrarily within the range of 5 minutes to 100 hours. Can be set.

  In general, for example, 1 to 20 equivalents of the compound represented by the general formula (5) and 1 to 4 equivalents of WSC (1-ethyl-3-ethyl) with respect to 1 equivalent of the compound represented by the general formula (9). (3-dimethylaminopropyl) -carbodiimide hydrochloride), CDI (carbonyldiimidazole) and other condensing agents. If necessary, 1-4 equivalents of potassium carbonate, triethylamine, pyridine, 4- (dimethylamino) pyridine, etc. In the presence of a base, the reaction is carried out for 10 minutes to 24 hours using no solvent or a solvent such as dichloromethane, chloroform, diethyl ether, tetrahydrofuran, 1,4-dioxane, etc., in the range of 0 ° C. to the reflux temperature of these solvents. Is preferred.

  Manufacturing method E

General formula (10) [wherein W ¹ , X, R ¹ , R ² and m represent the same meaning as described above. And a compound represented by the general formula (8): wherein Y, R ³ , R ⁴ , R ⁵ , R ⁶ and n have the same meaning as described above. And a compound represented by general formula (1-5) in which W ² is an oxygen atom in general formula (1) [wherein W ¹ , X, Y, R ¹ , R ² , R ³ , R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above. This invention compound represented by this can be obtained.

  Manufacturing method F

Formula (11) [wherein X, R ¹ and m represent the same meaning as described above. ] After regioselective lithiation according to a known method described in the literature, for example, the method described in Chemical Reviews [Chem. Rev.] 1990, 90, 879, etc. (12) [wherein W ² , Y, R ⁴ , R ⁵ , R ⁶ and n represent the same meaning as described above. In general formula (1), W ¹ is an oxygen atom, and R ² and R ³ are hydrogen atoms. In the general formula (1-6), W ² , X, Y, R ¹ , R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. This invention compound represented by this can be obtained. R-Li represents an alkyl lithium reagent such as butyl lithium.

  Manufacturing method G

General formula (13) [wherein X, Y, R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. And a compound represented by the general formula (14): wherein W ¹ and R ¹ have the same meaning as described above. In the general formula (1), W ² is an oxygen atom, and R ² and R ³ are hydrogen atoms. -7) [wherein W ¹ , X, Y, R ¹ , R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. This invention compound represented by this can be obtained. R-Li represents an alkyl lithium reagent such as butyl lithium.

  Manufacturing method H

In general formula (1), W ² is an oxygen atom and R ³ is a hydrogen atom. General formula (1-8) [wherein W ¹ , X, Y, R ¹ , R ² , R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above. The compound of the present invention represented by the general formula (15) [wherein R ³ represents the same meaning as described above, J ¹ represents a chlorine atom, a bromine atom, an iodine atom, a C ₁ -C ₄ alkylcarbonyloxy group ( For example, pivaloyloxy group), C ₁ -C ₄ alkyl sulfonate group (e.g., methanesulfonyloxy group), C ₁ -C ₄ haloalkylsulfonate group (e.g., trifluoromethanesulfonyloxy group), an aryl sulfonate group (e.g., benzenesulfonyloxy Group, p-toluenesulfonyloxy group) or an azolyl group (for example, imidazol-1-yl group). In the general formula (1), W ¹ is an oxygen atom by reacting the compound represented by the formula (1) with a solvent inert to the reaction if necessary in the presence of a base. Formula (1-5) [wherein W ¹ , X, Y, R ¹ , R ² , R ³ , R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. This invention compound represented by this can be obtained.

  As the amount of the reaction substrate, 1 to 50 equivalents of the compound represented by the general formula (15) can be used per 1 equivalent of the compound represented by the general formula (1-8).

  In the case of using a solvent, any solvent may be used as long as it does not inhibit the progress of the reaction. For example, aromatic hydrocarbons such as benzene, toluene and xylene, aliphatic hydrocarbons such as hexane and heptane, cyclohexane, etc. Alicyclic hydrocarbons, aromatic halogenated hydrocarbons such as chlorobenzene and dichlorobenzene, fats such as dichloromethane, chloroform, carbon tetrachloride, 1,2-dichloroethane, 1,1,1-trichloroethane, trichloroethylene and tetrachloroethylene Group halogenated hydrocarbons, ethers such as diethyl ether, 1,2-dimethoxyethane, tetrahydrofuran and 1,4-dioxane, esters such as ethyl acetate and ethyl propionate, dimethylformamide, dimethylacetamide, N-methyl- Amides such as 2-pyrrolidone, triethylamine, Amines such as tributylamine and N, N-dimethylaniline, pyridines such as pyridine and picoline, alcohols such as methanol, ethanol and ethylene glycol, acetonitrile, dimethyl sulfoxide, sulfolane, 1,3-dimethyl-2-imidazolide Non- and water are listed. These solvents may be used alone or as a mixture of two or more thereof.

  When a base is used, examples of the base used include alkali metal hydrides such as sodium hydride and potassium hydride, alkali metal hydroxides such as sodium hydroxide and potassium hydroxide, sodium ethoxide, potassium tertiary butoxide and the like. Alkali metal alkoxides, alkali metal amides such as lithium diisopropylamide, lithium hexamethyldisilazane, sodium amide, organometallic compounds such as tertiary butyl lithium, alkali metal carbonates such as sodium carbonate, potassium carbonate, sodium bicarbonate Organic bases such as triethylamine, tributylamine, N, N-dimethylaniline, pyridine, 4- (dimethylamino) pyridine, imidazole, 1,8-diazabicyclo [5,4,0] -7-undecene, etc. 1 to the compound represented by (1-8) It can be used equivalents.

  The reaction temperature can be set to an arbitrary temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrarily within the range of 5 minutes to 100 hours. Can be set.

  In general, for example, 1 to 10 equivalents of the compound represented by the general formula (15) is used per 1 equivalent of the compound represented by the general formula (1-8), tetrahydrofuran, 1,4-dioxane, acetonitrile In a polar solvent such as N, N-dimethylformamide, sodium hydride, potassium tertiary butoxide, potassium hydroxide, potassium carbonate, triethylamine, pyridine and the like are represented by the general formula (1-8) as a base if necessary. It is preferable to perform the reaction for 10 minutes to 24 hours in a temperature range of 0 to 90 ° C. using 1 to 3 equivalents per 1 equivalent of the compound.

  Manufacturing method I

In general formula (1), W ¹ is an oxygen atom and R ² is a hydrogen atom. General formula (1-9) [wherein W ² , X, Y, R ¹ , R ³ , R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above. The compound of the present invention represented by general formula (16): wherein R ² and J ¹ represent the same meaning as described above. And a compound represented by the general formula (1-4) in which W ¹ is an oxygen atom in the general formula (1) [wherein W ² , X, Y, R ¹ , R ² , R ³ , R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above. This invention compound represented by this can be obtained.

  In production method A to production method I, the reaction mixture after completion of the reaction is directly concentrated, or dissolved in an organic solvent, concentrated after washing with water, or poured into ice water, followed by normal post-treatment such as extraction after organic solvent extraction. Of the present invention can be obtained. Moreover, when the necessity for purification arises, it can be separated and purified by any purification method such as recrystallization, column chromatograph, thin layer chromatograph, liquid chromatographic fractionation and the like.

The compound represented by general formula (4-1) in which W ¹ and W ² are oxygen atoms in general formula (4), which is a raw material compound for manufacturing the compound of the present invention in production method A, is as follows: Can be synthesized.

  Reaction formula 1

That is, in the general formula (17) [wherein X and m represent the same meaning as described above. And a compound represented by the general formula (8-1) in which R ³ is a hydrogen atom in the general formula (8) [wherein Y, R ⁴ , R ⁵ , R ⁶ and n represent the same meaning as described above] . And the compound represented by the literature, for example, Berichte der Deutschen Hemischen Gesellshaft [Ber. Dtsch. Chem. Ges.] 1907, 40, 3177, Journal of the. Chemical Society [J. Chem. Soc.] 1954, 2023, Journal of the Chemical Society Perkin Transactions, 1 [J. Chem. Soc. Perkin Trans. 1] 1994, 2975 In the general formula (4), W ¹ and W ² are oxygen atoms in the general formula (4-1) [wherein X, Y, R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above. ] Can be easily synthesized.

  Some of the compounds represented by the general formula (5) used in Production Method A, Production Method B, and Production Method D are known compounds, and some of them are commercially available. Others, for example, Chemical and Pharmaceutical Bulletin [Chem. Pharm. Bull.] 1982, 30, 1921, Journal of the American Chemical Society [J. Am Chem. Soc.] 1986, 108, 3811, the method described in International Patent Application Publication (WO 01/23350) and the like, and other primary or secondary alkylamines described in the literature. It can be synthesized according to the synthesis method.

  In the production method B, the compound represented by the general formula (6), which is a raw material compound for producing the compound of the present invention, can be synthesized as follows.

  Reaction formula 2

That is, in the general formula (9), R ³ is a hydrogen atom, the general formula (9-1) [wherein W ² , X, Y, R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above. Represents. ], For example, Journal of the American Chemical Society [J. Am. Chem. Soc.] 1975, Vol. 97, 5582, Journal of Medicinal Chemistry [J. Med. Chem.] 1967, 10, 982, The Journal of Organic Chemistry [J. Org. Chem.] 1963, 28, By cyclization according to the method described on page 2018, etc., general formula (6) [wherein W ² , X, Y, R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above] Represents. ] Can be easily synthesized.

  In Production Method C, the compound represented by the general formula (7), which is a raw material compound for producing the compound of the present invention, can be synthesized as follows.

  Reaction formula 3

That is, in general formula (10), general formula (10-1) wherein R ² is a hydrogen atom [wherein W ¹ , X, R ¹ and m represent the same meaning as described above. The compound represented by the general formula (7) [wherein W ¹ , X, R ¹ and m represent the same meaning as described above]. ] Can be easily synthesized.

  The compound represented by the general formula (8) used in the production method C and the production method E can be synthesized using, for example, the methods represented by the following reaction formulas 4 to 7.

  Reaction formula 4

General formula (18) [wherein Y, R ³ , R ⁴ and n represent the same meaning as described above, and P is generally an acetyl group, a pivaloyl group, a benzoyl group, a tertiary butoxycarbonyl group, a benzyloxycarbonyl group, etc. The protecting group of the amino group used is represented. And a compound represented by the general formula (19) [wherein R ⁵ represents the same meaning as described above. Or a general formula (20) [wherein R ⁵ represents the same meaning as described above, and J ² represents a halogen atom such as a bromine atom or an iodine atom. And the Grignard reactant represented by the literature, for example, Heterocycles 1994, 39, 801, Journal of the American Chemical Society [J. Am. Chem. Soc.] 1988, 110, 1862, Tetrahedron 1960, 11, 252; Tetrahedron Lett. 1995, 36, 9117, etc. And then reacting according to the general formula (8-2) wherein R ⁶ is a hydrogen atom in the general formula (8). Y, R ³ , R ⁴ , R ⁵ and n have the same meaning as described above. The compound represented by this can be obtained.

Further, in the general formula (21) [wherein Y, R ³ , R ⁵ , n and P represent the same meaning as described above. And a compound represented by the general formula (22), wherein R ⁴ represents the same meaning as described above. Or a general formula (23) wherein R ⁴ and J ² represent the same meaning as described above. The compound represented by the general formula (8-2) can also be obtained by reacting with a Grignard reactant represented by the same conditions as described above.

  Some of the lithium reactants represented by general formula (19) and general formula (22) used here are known compounds, and some of them are available as commercial products. In addition, other halogen-metal exchange reactions described in the literature, such as Bulletin of the Chemical Society of Japan [Bull. Chem. Soc. Jpn.] 1990, 63, 3719 Page, The Journal of Organic Chemistry [J. Org. Chem.] 1983, Vol. 48, p. 1449, etc., can be easily synthesized from the corresponding known halides.

  Some of the Grignard reagents represented by the general formula (20) and the general formula (23) are known compounds, and some of them are available as commercial products. In addition, other methods for preparing general Grignard reagents described in the literature, such as Angewante Chemie Int. Ed. Engl., 1969, Vol. 8, 279 Page, The Journal of Organic Chemistry [J. Org. Chem.] 1989, 54, 4413, etc., and can be easily synthesized from the corresponding known halides.

  Reaction formula 5

General formula (21) [wherein Y, R ³ , R ⁵ , n and P represent the same meaning as described above. The compound represented by formula (24) is reacted with a compound represented by the formula (24) according to a known method described in the literature, for example, a method described in Synlett, p. 233, 2003, or a known method. General formula (25) [wherein J ³ represents a hydrogen atom, a bromine atom, a trimethylsilyl group or the like. ] And known methods described in the literature, for example, The Journal of Organic Chemistry [J. Org. Chem.] 2000, 65, 8848 and 2001, 66, 1436 Tetrahedron, 1989, Vol. 45, p. 1423, and the like, followed by deprotection of each protecting group by a commonly used method to give a compound represented by the general formula (8) Wherein R ⁴ is a trifluoromethyl group and R ⁶ is a hydrogen atom (wherein Y, R ³ , R ⁵ and n are as defined above). The compound represented by this can be obtained.

  Reaction formula 6

General formula (26) [wherein Y, R ³ , n, J ² and P represent the same meaning as described above. ] After lithiation of the compound represented by the literature, for example, by lithiation, general formula (27) [wherein R ⁴ and R ⁵ represent the same meaning as described above. The method described in Tetrahedron Lett. 1995, Vol. 36, page 9117, etc., or after forming a Grignard reactant, is represented by the general formula (27). According to the method described in Tetrahedron, 1960, 11, 252; The Journal of Organic Chemistry [J. Org. Chem.] 1988, 53, 754, etc. Then, each protecting group is deprotected by a commonly used method to give a general formula (8-2) wherein R ⁶ is a hydrogen atom in the general formula (8) [wherein Y, R ³ , R ⁴ , R ⁵ and n have the same meaning as described above. The compound represented by this can be obtained. R-Li represents an alkyl lithium reagent such as butyl lithium.

  Reaction formula 7

General formula (28) obtained as an intermediate in reaction formula 4, reaction formula 5 and reaction formula 6, wherein Y, R ³ , R ⁴ , R ⁵ , n and P have the same meaning as described above. And a compound represented by the general formula (29): wherein R ⁶ and J ¹ represent the same meaning as described above. And a compound represented by the general formula (8) [wherein Y, R ³ , R ⁴ , R ⁵ and n represent the same meaning as described above, and R ⁶ represents the above meaning other than a hydrogen atom. The compound represented by this can be obtained.

  In production method D, the compound represented by general formula (9), which is a raw material compound for producing the compound of the present invention, is synthesized using, for example, the method represented by the following reaction formula 8 or 9 can do.

  Reaction formula 8

General formula (17) [wherein X and m represent the same meaning as described above. And a compound represented by the general formula (8): wherein Y, R ³ , R ⁴ , R ⁵ , R ⁶ and n have the same meaning as described above. And a compound represented by the general formula (9-2) wherein W ² is an oxygen atom in the general formula (9) [wherein X, Y, R ³ , R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. The compound represented by this can be obtained.

  Reaction formula 9

General formula (13) [wherein X, Y, R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. In accordance with a known method described in the literature, for example, a method described in Chemical Reviews [Chem. Rev.] 1990, 90, 879, etc., after regioselective lithiation, By reacting with carbon dioxide, general formula (9-3) in which W ² is an oxygen atom and R ³ is a hydrogen atom in general formula (9) [wherein X, Y, R ⁴ , R ⁵ , R ⁶ , m and n have the same meaning as described above. The compound represented by this can be obtained. R-Li represents an alkyl lithium reagent such as butyl lithium.

  In the production method E, the compound represented by the general formula (10), which is a raw material compound for producing the compound of the present invention, is synthesized using, for example, the method represented by the following reaction formula 10 or 11 it can.

  Reaction formula 10

General formula (17) [wherein X and m represent the same meaning as described above. And a compound represented by the general formula (5): wherein R ¹ and R ² represent the same meaning as described above. And a compound represented by the general formula (10-2) in which W ¹ is an oxygen atom in the general formula (10) [wherein X, R ¹ , R ² and m represent the same meaning as described above. The compound represented by this can be obtained.

  Reaction formula 11

Formula (11) [wherein X, R ¹ and m represent the same meaning as described above. In the general formula (10), W ¹ is an oxygen atom and R ² is a hydrogen atom in the general formula (10-3) [wherein X, R ¹ and m represent the same meaning as described above. The compound represented by this can be obtained. R-Li represents an alkyl lithium reagent such as butyl lithium.

  In the production method F, some of the compounds represented by the general formula (11) which are raw material compounds for producing the compound of the present invention are known compounds, and some of them are commercially available. In addition, other methods known in the literature, for example, Bulletin of the Chemical Society of Japan [Bull. Chem. Soc. Jpn.] 1985, 58, 3291, The Journal Of organic chemistry [J. Org. Chem.] 1991, 56, 2395, Tetrahedron Lett. 1994, 35, 2113, International Patent Application Publication (WO 98/23581) It can be easily synthesized according to the method described in Japanese Patent Publication No.

  The compound represented by the general formula (12) used in production method F can be synthesized as follows.

  Reaction formula 12

That is, in general formula (8), R ³ is a hydrogen atom. General formula (8-1) [wherein Y, R ⁴ , R ⁵ , R ⁶ and n represent the same meaning as described above. And a compound represented by the general formula (30): wherein W ² represents an oxygen atom or a sulfur atom. And a commercially available phosgene, thioosgen or an equivalent thereof, for example, known methods described in the literature, for example, Angewante Chemie International Edition in English [Angew. Chem. Int. Ed. Engl.] 1987 26, 894 and 1995, 34, 2497, The Journal of Organic Chemistry [J. Org. Chem.] 1976, 41, 2070, Synthesis 1988, 990 Tetrahedron Lett. 1997, 38, 919, and the like, by reacting according to the method described in general formula (12) [wherein W ² , Y, R ⁴ , R ⁵ , R ⁶ and n have the same meaning as described above. ] Can be easily synthesized.

  In Production Method G, the compound represented by General Formula (13), which is a raw material compound for producing the compound of the present invention, can be synthesized as follows.

  Reaction formula 13

That is, in the general formula (31) [wherein X and m represent the same meaning as described above. And a compound represented by the general formula (8-1) in which R ³ is a hydrogen atom in the general formula (8) [wherein Y, R ⁴ , R ⁵ , R ⁶ and n represent the same meaning as described above] . Or a compound represented by the general formula (31) by a known method (for example, thionyl chloride, phosphorus pentachloride or oxalyl chloride). The corresponding carboxylic acid chloride using a chlorinating agent) is reacted with a compound represented by the general formula (8-1) to give a general formula (13) [wherein X, Y, R ⁴ , R ⁵ , R ⁶ , m and n represent the same meaning as described above. ] Can be easily synthesized.

  The compounds represented by the general formula (31) used here are known compounds, and some of them are available as commercial products.

  Some of the compounds represented by the general formula (14) used in production method G are known compounds, and some of them are commercially available. Other than that, general synthesis methods described in the literature, for example, The Journal of Organic Chemistry [J. Org. Chem.] 1996, 61, 3883, 3929 and 6575, Tetra It can be easily synthesized according to the method described in Tetrahedron Lett. 1999, 40, 363, 6121, etc.

  Compound represented by general formula (15) used in production method H, compound represented by general formula (16) used in production method I, and compound represented by general formula (29) used in reaction formula 7 Some of these are known compounds, some of which are commercially available. Other than the above, general synthesis methods described in the literature, for example, Chemistry Letters [Chem. Lett.] 1976, 373 pages, Journal of the American Chemical Society [J. Am. Chem. Soc.] 1964, 86, 4383, The Journal of Organic Chemistry [J. Org. Chem.] 1976, 41, 4028 and 1978, 43, 3244, Organic Synthesis [Org. Synth.] 1988, Collective Volume 6, p. 101, Tetrahedron Lett. 1972, p. 4339, British Patent (GB 2,161,802), European Patent (EP 0,051,273), etc. It can be easily synthesized according to the method described in 1.

  Some of the compounds represented by the general formula (17) are known compounds, and some of them are commercially available. Others can be synthesized as follows, for example.

  Reaction formula 14

  That is, in the general formula (32) [wherein X and m represent the same meaning as described above, and R represents a lower alkyl group such as a methyl group or an ethyl group. The compound represented by the general hydrolysis reaction described in the literature, for example, Angewante Chem. 1951, 63, 329, Journal of the American Chemical Society [J. Am. Chem. Soc.] 1929, 51, 1865, etc. In accordance with the general formula (33) [wherein X and m represent the same meaning as described above. ], Followed by a general dehydration cyclization reaction described in the literature, such as The Journal of Organic Chemistry [J. Org. Chem.] 1987, 52, 129, etc. In the general formula (17), wherein X and m are as defined above. The compound represented by this can be obtained.

  The compounds represented by the general formula (32) used here are known compounds, and some of them are available as commercial products.

  The compound represented by the general formula (18) can be synthesized, for example, as follows.

  Reaction formula 15

That is, the known general formula (34) [wherein Y, R ³ , n and P represent the same meaning as described above. And a known general formula (35) [wherein R ⁴ represents the same meaning as described above, and J ⁴ represents a leaving group such as a halogen atom, a trifluoromethanesulfonyloxy group, a 2-pyridyloxy group, or the like. Represents. ] Or a known general formula (36) [wherein R ⁴ represents the same meaning as described above. The general aromatic ring acylation reaction described in the literature, for example, Chemistry Letters [Chem. Lett.] 1990, p. 783, The Journal of Organic Chemistry [J. Org] Chem.] 1991, 56, 1963, etc., by reacting in accordance with the general formula (18) [wherein Y, R ³ , R ⁴ , n and P have the same meaning as described above. Represents. The compound represented by this can be obtained.

Alternatively, the general formula (26) [wherein Y, R ³ , n, J ² and P represent the same meaning as described above. ], After lithiation of the compound represented by the literature, for example, known general formula (37) [wherein R ⁴ represents the same meaning as described above, J ⁵ represents a halogen atom, a hydroxyl group, metal salts _{(e.g., -OLi, -ONa), C 1} ~C 4 alkoxy group (e.g., methoxy group, ethoxy group), di (C ₁ -C ₄ alkyl) amino group (e.g., diethylamino group), C ₁ ~ C ₄ alkoxy (C ₁ -C ₄ alkyl) amino group (for example, O, N-dimethylhydroxyamino group) or cyclic amino group (for example, piperidin-1-yl group, morpholin-4-yl group, 4-methylpiperazine) -1-yl group). Or the known compound represented by the general formula (36) [J. Am. Chem. Soc.] 1955, 77, 3657 Tetrahedron Lett. 1980, 21, 2129 and 1991, 32, 2003, US Patent Application Publication (US 5,514,816), etc., or Grignard reactant Heterocycles 1987, 25, 221, Synthetic Communications [Synth. Communication, which is formed and then reacted with a compound represented by general formula (37) or a compound represented by general formula (36) In accordance with the method described in 1985, 15, 1291 and 1990, 20, 1469, German Patent Application Publication (DE 19727042), etc. To obtain a compound represented by the general formula (18).

  The compound represented by the general formula (21) can be synthesized in the same manner as the compound represented by the general formula (18).

  The compound represented by the general formula (26) can be synthesized, for example, as follows.

  Reaction formula 16

That is, the known general formula (38) [wherein Y, R ³ , n and J ² represent the same meaning as described above. The substituted aniline represented by the general method described in the literature, for example, Journal of Medicinal Chemistry [J. Med. Chem.] 1996, 39, 673 and 1997, 40, 3542, etc. In the general formula (26), Y, R ³ , n, J ² and P have the same meaning as described above. The compound represented by this can be obtained.

  Some of the compounds represented by the general formula (27) are known compounds, and some of them are commercially available. Other compounds can be synthesized in the same manner as the compound represented by the general formula (18).

  In each of these reactions, after the completion of the reaction, each of the production intermediates that are the raw material compounds of Production Method A to Production Method I can be obtained by performing a general post-treatment.

  In addition, each production intermediate produced by these methods can be used as it is in the subsequent step without isolation and purification.

  Specific examples of the compound included in the present invention include compounds shown in Tables 2 to 5. However, the compounds in Tables 2 to 5 are for illustrative purposes, and the present invention is not limited thereto.

In the table, “Et” represents an ethyl group. Similarly, n-Pr and Pr-n are normal propyl groups, i-Pr and Pr-i are isopropyl groups, and c-Pr and Pr-c are Cyclopropyl group, n-Bu and Bu-n are normal butyl groups, s-Bu and Bu-s are secondary butyl groups, i-Bu and Bu-i are isobutyl groups, t-Bu and Bu-t Is a tertiary butyl group, c-Bu and Bu-c are cyclobutyl groups, n-Pen and Pen-n are normal pentyl groups, c-Pen and Pen-c are cyclopentyl groups, n-Hex and Hex- n is a normal hexyl group, c-Hex and Hex-c are cyclohexyl groups, Oct is an octyl group, Ph is a phenyl group, 1-Naph is a 1-naphthyl group, 2-Naph is a 2-naphthyl group. Respectively,
The aromatic heterocycles represented by L-1a to L-55a in the table each represent the following structure,

For example, the notation of (L-16a) CHF ₂ represents a 1-difluoromethylpyrazol-4-yl group, and the notation of (L-45c) CF ₃ represents a 5-trifluoromethylpyridin-2-yl group .

  The aliphatic heterocycles represented by M-4a to M-22a in the table each represent the following structure,

For example, the notation (M-22a) C (O) OCH ₃ represents a 1-methoxycarbonylpiperidin-4-yl group.

  Further, T-1 to T-24 in the table each represent the following structure.

Table 2

―――――――――――――――――――――――――――――――――――――――
R²        R¹                           R^Four               R^Five
―――――――――――――――――――――――――――――――――――――――
H CH_Three                          CF_Three              CF₂O (Ph-4-Cl)
H CH_Three                          CF_Three              CH = CH (Ph-4-Cl)
H CH_Three                          CF_Three              CH = CH (Ph-4-OCF_Three)
H CH_Three                          CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH_Three                          CF_Three              Ph-4-F
H CH_Three                          CF_Three              Ph-4-Cl
H CH_Three                          CF_Three              Ph-4-Br
H CH_Three                          CF_Three              Ph-4-I
H CH_Three                          CF_Three              Ph-4-CF_Three
H CH_Three                          CF_Three              Ph-4-OCHF₂
H CH_Three                          CF_Three              Ph-4-OCF_Three
H CH_Three                          CF_Three              Ph-4-OCF₂Br
H CH_Three                          CF_Three              Ph-4-OCF₂CHF₂
H CH_Three                          CF_Three              Ph-4-OCF₂CHFCl
H CH_Three                          CF_Three              Ph-4-OCF₂CHFCF_Three
H CH_Three                          CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH_Three                          CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH_Three                          CF_Three              Ph-4-O (L-45e)
H CH_Three                          CF_Three              Ph-3,4-Cl₂
H CH_Three                          CF_Three              Ph (-3-OCF₂O-4-)
H CH_Three                          CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH_Three                          CF_Three             (L-45c) Cl
H CH_Three                          CF_Three             (L-45c) Br
H CH_Three                          CF_Three             (L-45c) CF_Three
H CH_Three                          CF_Three              L-45e
H CH_Three                          CF_Three              L-45f
H CH_Three                          CF_Three             (L-46c) Cl
H CH_Three                          CF_Three             (L-46c) Br
H CH_Three                          CF_Three             (L-46c) CF_Three
H CH_Three                          CF_Three              L-46d
CH_Three       CH_Three                          CF_Three              Ph-4-Br
CH_Three       CH_Three                          CF_Three              Ph-4-CF_Three
CH_Three       CH_Three                          CF_Three              Ph-4-OCF_Three
CH_Three       CH_Three                          CF_Three             (L-45c) CF_Three
H Et CH_Three              Ph-4-Cl
H Et CH_Three              Ph-4-CF_Three
H Et CH_Three              Ph-4-OCF_Three
H Et CH_Three             (L-45c) Cl
H Et CH_Three             (L-45c) Br
H Et CH_Three             (L-45c) CF_Three
H Et Et Ph-4-Br
H Et n-Pr Ph-4-CF_Three
H Et i-Pr Ph-4-OCF_Three
H Et c-Pr (L-45c) CF_Three
H Et CHF₂             Ph-4-Br
H Et CF_Three              CF₂O (Ph-4-Cl)
H Et CF_Three              CH = CH (Ph-4-Cl)
H Et CF_Three              CH = CH (Ph-4-OCF_Three)
H Et CF_Three              CH = CH (Ph-3,4-Cl₂)
H Et CF_Three              Ph-4-F
H Et CF_Three              Ph-4-Cl
H Et CF_Three              Ph-4-Br
H Et CF_Three              Ph-4-I
H Et CF_Three              Ph-4-CF_Three
H Et CF_Three              Ph-4-OCHF₂
H Et CF_Three              Ph-4-OCF_Three
H Et CF_Three              Ph-4-OCF₂Br
H Et CF_Three              Ph-4-OCF₂CHF₂
H Et CF_Three              Ph-4-OCF₂CHFCl
H Et CF_Three              Ph-4-OCF₂CHFCF_Three
H Et CF_Three              Ph-4-OCF₂CHFOCF_Three
H Et CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H Et CF_Three              Ph-4-O (L-45g)
H Et CF_Three              Ph-3,4-Cl₂
H Et CF_Three              Ph (-3-OCF₂O-4-)
H Et CF_Three              Ph (-3-OCF₂CF₂O-4-)
H Et CF_Three             (L-45c) Cl
H Et CF_Three             (L-45c) Br
H Et CF_Three             (L-45c) CF_Three
H Et CF_Three              L-45e
H Et CF_Three              L-45f
H Et CF_Three             (L-46c) Cl
H Et CF_Three             (L-46c) Br
H Et CF_Three             (L-46c) CF_Three
H Et CF_Three              L-46d
H Et CF₂Cl Ph-4-CF_Three
H Et CF₂Br Ph-4-OCF_Three
H Et CF₂CF_Three          (L-45c) CF_Three
H Et CF₂CF₂CF_Three        Ph-4-Br
H Et CF₂OCH_Three          Ph-4-CF_Three
H Et CF₂SCH_Three          Ph-4-OCF_Three
Et Et CH_Three              Ph-4-Br
Et Et CH_Three              Ph-4-CF_Three
Et Et CH_Three              Ph-4-OCF_Three
Et Et CH_Three             (L-45c) Cl
Et Et CH_Three             (L-45c) Br
Et Et CH_Three             (L-45c) CF_Three
Et Et CF_Three              CF₂O (Ph-4-Cl)
Et Et CF_Three              CH = CH (Ph-4-Cl)
Et Et CF_Three              CH = CH (Ph-4-OCF_Three)
Et Et CF_Three              CH = CH (Ph-3,4-Cl₂)
Et Et CF_Three              Ph-4-F
Et Et CF_Three              Ph-4-Cl
Et Et CF_Three              Ph-4-Br
Et Et CF_Three              Ph-4-I
Et Et CF_Three              Ph-4-CF_Three
Et Et CF_Three              Ph-4-OCHF₂
Et Et CF_Three              Ph-4-OCF_Three
Et Et CF_Three              Ph-4-OCF₂Br
Et Et CF_Three              Ph-4-OCF₂CHF₂
Et Et CF_Three              Ph-4-OCF₂CHFCl
Et Et CF_Three              Ph-4-OCF₂CHFCF_Three
Et Et CF_Three              Ph-4-OCF₂CHFOCF_Three
Et Et CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
Et Et CF_Three              Ph-4-O (L-45g)
Et Et CF_Three              Ph-3,4-Cl₂
Et Et CF_Three              Ph (-3-OCF₂O-4-)
Et Et CF_Three              Ph (-3-OCF₂CF₂O-4-)
Et Et CF_Three             (L-45c) Cl
Et Et CF_Three             (L-45c) Br
Et Et CF_Three             (L-45c) CF_Three
Et Et CF_Three              L-45e
Et Et CF_Three              L-45f
Et Et CF_Three             (L-46c) Cl
Et Et CF_Three             (L-46c) Br
Et Et CF_Three             (L-46c) CF_Three
Et Et CF_Three              L-46d
H n-Pr CH_Three              Ph-4-Br
H n-Pr CH_Three              Ph-4-CF_Three
H n-Pr CH_Three              Ph-4-OCF_Three
H n-Pr CH_Three             (L-45c) Cl
H n-Pr CH_Three             (L-45c) Br
H n-Pr CH_Three             (L-45c) CF_Three
H n-Pr Et (L-45c) CF_Three
H n-Pr n-Pr Ph-4-Br
H n-Pr i-Pr Ph-4-CF_Three
H n-Pr c-Pr Ph-4-OCF_Three
H n-Pr CHF₂            (L-45c) CF_Three
H n-Pr CF_Three              CF₂O (Ph-4-Cl)
H n-Pr CF_Three              CH = CH (Ph-4-Cl)
H n-Pr CF_Three              CH = CH (Ph-4-OCF_Three)
H n-Pr CF_Three              CH = CH (Ph-3,4-Cl₂)
H n-Pr CF_Three              Ph-4-F
H n-Pr CF_Three              Ph-4-Cl
H n-Pr CF_Three              Ph-4-Br
H n-Pr CF_Three              Ph-4-I
H n-Pr CF_Three              Ph-4-CF_Three
H n-Pr CF_Three              Ph-4-OCHF₂
H n-Pr CF_Three              Ph-4-OCF_Three
H n-Pr CF_Three              Ph-4-OCF₂Br
H n-Pr CF_Three              Ph-4-OCF₂CHF₂
H n-Pr CF_Three              Ph-4-OCF₂CHFCl
H n-Pr CF_Three              Ph-4-OCF₂CHFCF_Three
H n-Pr CF_Three              Ph-4-OCF₂CHFOCF_Three
H n-Pr CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H n-Pr CF_Three              Ph-4-O (L-45g)
H n-Pr CF_Three              Ph-3,4-Cl₂
H n-Pr CF_Three              Ph (-3-OCF₂O-4-)
H n-Pr CF_Three              Ph (-3-OCF₂CF₂O-4-)
H n-Pr CF_Three             (L-45c) Cl
H n-Pr CF_Three             (L-45c) Br
H n-Pr CF_Three             (L-45c) CF_Three
H n-Pr CF_Three              L-45e
H n-Pr CF_Three              L-45f
H n-Pr CF_Three             (L-46c) Cl
H n-Pr CF_Three             (L-46c) Br
H n-Pr CF_Three             (L-46c) CF_Three
H n-Pr CF_Three              L-46d
H n-Pr CF₂Cl Ph-4-Br
H n-Pr CF₂Br Ph-4-CF_Three
H n-Pr CF₂CF_Three           Ph-4-OCF_Three
H n-Pr CF₂CF₂CF_Three       (L-45c) CF_Three
H n-Pr CF₂OCH_Three          Ph-4-Br
H n-Pr CF₂SCH_Three          Ph-4-CF_Three
CH_Three       n-Pr CF_Three              Ph-4-Br
CH_Three       n-Pr CF_Three              Ph-4-CF_Three
CH_Three       n-Pr CF_Three              Ph-4-OCF_Three
CH_Three       n-Pr CF_Three             (L-45c) CF_Three
Et n-Pr CF_Three              Ph-4-OCF_Three
n-Pr n-Pr CF_Three             (L-45c) CF_Three
H i-Pr CH_Three              CF₂O (Ph-4-Cl)
H i-Pr CH_Three              CH = CH (Ph-4-Cl)
H i-Pr CH_Three              CH = CH (Ph-4-OCF_Three)
H i-Pr CH_Three              CH = CH (Ph-3,4-Cl₂)
H i-Pr CH_Three              Ph-4-F
H i-Pr CH_Three              Ph-4-Cl
H i-Pr CH_Three              Ph-4-Br
H i-Pr CH_Three              Ph-4-I
H i-Pr CH_Three              Ph-4-CF_Three
H i-Pr CH_Three              Ph-4-OCHF₂
H i-Pr CH_Three              Ph-4-OCF_Three
H i-Pr CH_Three              Ph-4-OCF₂Br
H i-Pr CH_Three              Ph-4-OCF₂CHF₂
H i-Pr CH_Three              Ph-4-OCF₂CHFCl
H i-Pr CH_Three              Ph-4-OCF₂CHFCF_Three
H i-Pr CH_Three              Ph-4-OCF₂CHFOCF_Three
H i-Pr CH_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CH_Three              Ph-4-O (L-45g)
H i-Pr CH_Three              Ph-3,4-Cl₂
H i-Pr CH_Three              Ph (-3-OCF₂O-4-)
H i-Pr CH_Three              Ph (-3-OCF₂CF₂O-4-)
H i-Pr CH_Three             (L-45c) Cl
H i-Pr CH_Three             (L-45c) Br
H i-Pr CH_Three             (L-45c) CF_Three
H i-Pr CH_Three              L-45e
H i-Pr CH_Three              L-45f
H i-Pr CH_Three             (L-46c) Cl
H i-Pr CH_Three             (L-46c) Br
H i-Pr CH_Three             (L-46c) CF_Three
H i-Pr CH_Three              L-46d
H i-Pr Et CF₂O (Ph-4-Cl)
H i-Pr Et CH = CH (Ph-4-Cl)
H i-Pr Et CH = CH (Ph-4-OCF_Three)
H i-Pr Et CH = CH (Ph-3,4-Cl₂)
H i-Pr Et Ph-4-Cl
H i-Pr Et Ph-4-Br
H i-Pr Et Ph-4-CF_Three
H i-Pr Et Ph-4-OCF_Three
H i-Pr Et Ph-4-OCF₂Br
H i-Pr Et Ph-4-OCF₂CHFCF_Three
H i-Pr Et Ph-4-OCF₂CHFOCF_Three
H i-Pr Et Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr Et Ph-4-O (L-45g)
H i-Pr Et Ph-3,4-Cl₂
H i-Pr Et Ph (-3-OCF₂O-4-)
H i-Pr Et Ph (-3-OCF₂CF₂O-4-)
H i-Pr Et (L-45c) Br
H i-Pr Et (L-45c) CF_Three
H i-Pr Et L-45e
H i-Pr Et L-45f
H i-Pr Et (L-46c) Br
H i-Pr Et (L-46c) CF_Three
H i-Pr Et L-46d
H i-Pr n-Pr CF₂O (Ph-4-Cl)
H i-Pr n-Pr CH = CH (Ph-4-Cl)
H i-Pr n-Pr CH = CH (Ph-4-OCF_Three)
H i-Pr n-Pr CH = CH (Ph-3,4-Cl₂)
H i-Pr n-Pr Ph-4-Cl
H i-Pr n-Pr Ph-4-Br
H i-Pr n-Pr Ph-4-CF_Three
H i-Pr n-Pr Ph-4-OCF_Three
H i-Pr n-Pr Ph-4-OCF₂Br
H i-Pr n-Pr Ph-4-OCF₂CHFCF_Three
H i-Pr n-Pr Ph-4-OCF₂CHFOCF_Three
H i-Pr n-Pr Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr n-Pr Ph-4-O (L-45g)
H i-Pr n-Pr Ph-3,4-Cl₂
H i-Pr n-Pr Ph (-3-OCF₂O-4-)
H i-Pr n-Pr Ph (-3-OCF₂CF₂O-4-)
H i-Pr n-Pr (L-45c) Br
H i-Pr n-Pr (L-45c) CF_Three
H i-Pr n-Pr L-45e
H i-Pr n-Pr L-45f
H i-Pr n-Pr (L-46c) Br
H i-Pr n-Pr (L-46c) CF_Three
H i-Pr n-Pr L-46d
H i-Pr i-Pr CF₂O (Ph-4-Cl)
H i-Pr i-Pr CH = CH (Ph-4-Cl)
H i-Pr i-Pr CH = CH (Ph-4-OCF_Three)
H i-Pr i-Pr CH = CH (Ph-3,4-Cl₂)
H i-Pr i-Pr Ph-4-Cl
H i-Pr i-Pr Ph-4-Br
H i-Pr i-Pr Ph-4-CF_Three
H i-Pr i-Pr Ph-4-OCF_Three
H i-Pr i-Pr Ph-4-OCF₂Br
H i-Pr i-Pr Ph-4-OCF₂CHFCF_Three
H i-Pr i-Pr Ph-4-OCF₂CHFOCF_Three
H i-Pr i-Pr Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr i-Pr Ph-4-O (L-45g)
H i-Pr i-Pr Ph-3,4-Cl₂
H i-Pr i-Pr Ph (-3-OCF₂O-4-)
H i-Pr i-Pr Ph (-3-OCF₂CF₂O-4-)
H i-Pr i-Pr (L-45c) Br
H i-Pr i-Pr (L-45c) CF_Three
H i-Pr i-Pr L-45e
H i-Pr i-Pr L-45f
H i-Pr i-Pr (L-46c) Br
H i-Pr i-Pr (L-46c) CF_Three
H i-Pr i-Pr L-46d
H i-Pr c-Pr CF₂O (Ph-4-Cl)
H i-Pr c-Pr CH = CH (Ph-4-Cl)
H i-Pr c-Pr CH = CH (Ph-4-OCF_Three)
H i-Pr c-Pr CH = CH (Ph-3,4-Cl₂)
H i-Pr c-Pr Ph-4-Cl
H i-Pr c-Pr Ph-4-Br
H i-Pr c-Pr Ph-4-CF_Three
H i-Pr c-Pr Ph-4-OCF_Three
H i-Pr c-Pr Ph-4-OCF₂Br
H i-Pr c-Pr Ph-4-OCF₂CHFCF_Three
H i-Pr c-Pr Ph-4-OCF₂CHFOCF_Three
H i-Pr c-Pr Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr c-Pr Ph-4-O (L-45g)
H i-Pr c-Pr Ph-3,4-Cl₂
H i-Pr c-Pr Ph (-3-OCF₂O-4-)
H i-Pr c-Pr Ph (-3-OCF₂CF₂O-4-)
H i-Pr c-Pr (L-45c) Br
H i-Pr c-Pr (L-45c) CF_Three
H i-Pr c-Pr L-45e
H i-Pr c-Pr L-45f
H i-Pr c-Pr (L-46c) Br
H i-Pr c-Pr (L-46c) CF_Three
H i-Pr c-Pr L-46d
H i-Pr n-Bu Ph-4-Br
H i-Pr s-Bu Ph-4-CF_Three
H i-Pr i-Bu Ph-4-OCF_Three
H i-Pr c-Bu (L-45c) CF_Three
H i-Pr n-Pen Ph-4-Br
H i-Pr c-Pen Ph-4-CF_Three
H i-Pr n-Hex Ph-4-OCF_Three
H i-Pr c-Hex (L-45c) CF_Three
H i-Pr CH₂F Ph-4-Br
H i-Pr CH₂Cl Ph-4-CF_Three
H i-Pr CH₂Br Ph-4-OCF_Three
H i-Pr CHF₂             CF₂O (Ph-4-Cl)
H i-Pr CHF₂             CH = CH (Ph-4-Cl)
H i-Pr CHF₂             CH = CH (Ph-4-OCF_Three)
H i-Pr CHF₂             CH = CH (Ph-3,4-Cl₂)
H i-Pr CHF₂             Ph-4-F
H i-Pr CHF₂             Ph-4-Cl
H i-Pr CHF₂             Ph-4-Br
H i-Pr CHF₂             Ph-4-I
H i-Pr CHF₂             Ph-4-CF_Three
H i-Pr CHF₂             Ph-4-OCHF₂
H i-Pr CHF₂             Ph-4-OCF_Three
H i-Pr CHF₂             Ph-4-OCF₂Br
H i-Pr CHF₂             Ph-4-OCF₂CHF₂
H i-Pr CHF₂             Ph-4-OCF₂CHFCl
H i-Pr CHF₂             Ph-4-OCF₂CHFCF_Three
H i-Pr CHF₂             Ph-4-OCF₂CHFOCF_Three
H i-Pr CHF₂             Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CHF₂             Ph-4-O (L-45g)
H i-Pr CHF₂             Ph-3,4-Cl₂
H i-Pr CHF₂             Ph (-3-OCF₂O-4-)
H i-Pr CHF₂             Ph (-3-OCF₂CF₂O-4-)
H i-Pr CHF₂            (L-45c) Cl
H i-Pr CHF₂            (L-45c) Br
H i-Pr CHF₂            (L-45c) CF_Three
H i-Pr CHF₂             L-45e
H i-Pr CHF₂             L-45f
H i-Pr CHF₂            (L-46c) Cl
H i-Pr CHF₂            (L-46c) Br
H i-Pr CHF₂            (L-46c) CF_Three
H i-Pr CHF₂             L-46d
H i-Pr CHFCl (L-45c) CF_Three
H i-Pr CHFBr Ph-4-Br
H i-Pr CF_Three              T-1
H i-Pr CF_Three              T-2
H i-Pr CF_Three              T-3
H i-Pr CF_Three              T-4
H i-Pr CF_Three              T-5
H i-Pr CF_Three              CH₂OCH_Three
H i-Pr CF_Three              CH₂OEt
H i-Pr CF_Three              CH₂OPr-n
H i-Pr CF_Three              CH₂OPr-i
H i-Pr CF_Three              CH₂OBu-n
H i-Pr CF_Three              CH₂OCH₂CF_Three
H i-Pr CF_Three              CH₂OCH₂CF₂CF_Three
H i-Pr CF_Three              CH₂OCH (CF_Three)₂
H i-Pr CF_Three              CH₂OC (O) (Ph-2-Cl)
H i-Pr CF_Three              CH₂OC (O) (Ph-3-Cl)
H i-Pr CF_Three              CH₂OC (O) (Ph-4-Cl)
H i-Pr CF_Three              CH₂OPh
H i-Pr CF_Three              CH₂O (Ph-4-F)
H i-Pr CF_Three              CH₂O (Ph-2-Cl)
H i-Pr CF_Three              CH₂O (Ph-3-Cl)
H i-Pr CF_Three              CH₂O (Ph-4-Cl)
H i-Pr CF_Three              CH₂O (Ph-4-Br)
H i-Pr CF_Three              CH₂O (Ph-4-CF_Three)
H i-Pr CF_Three              CH₂O (Ph-4-OCF_Three)
H i-Pr CF_Three              CH₂CH₂OCH_Three
H i-Pr CF_Three              CF₂OPh
H i-Pr CF_Three              CF₂O (Ph-3-F)
H i-Pr CF_Three              CF₂O (Ph-4-F)
H i-Pr CF_Three              CF₂O (Ph-2-Cl)
H i-Pr CF_Three              CF₂O (Ph-3-Cl)
H i-Pr CF_Three              CF₂O (Ph-4-Cl)
H i-Pr CF_Three              CF₂O (Ph-3-Br)
H i-Pr CF_Three              CF₂O (Ph-4-Br)
H i-Pr CF_Three              CF₂O (Ph-3-CF_Three)
H i-Pr CF_Three              CF₂O (Ph-4-CF_Three)
H i-Pr CF_Three              CF₂O (Ph-3-OCF_Three)
H i-Pr CF_Three              CF₂O (Ph-4-OCF_Three)
H i-Pr CF_Three              M-4a
H i-Pr CF_Three              M-5a
H i-Pr CF_Three              CH₂SCH_Three
H i-Pr CF_Three              CH₂SO₂CH_Three
H i-Pr CF_Three              CH₂SCF_Three
H i-Pr CF_Three              CH₂SO₂CF_Three
H i-Pr CF_Three              CH₂SPh
H i-Pr CF_Three              CH₂S (Ph-3-Cl)
H i-Pr CF_Three              CH₂S (Ph-4-Cl)
H i-Pr CF_Three              CH₂SO₂(Ph-3-Cl)
H i-Pr CF_Three              CH₂SO₂(Ph-4-Cl)
H i-Pr CF_Three              CH₂CH₂SCH_Three
H i-Pr CF_Three              CH₂CH₂SO₂CH_Three
H i-Pr CF_Three              CH₂CH (CH_Three) SCH_Three
H i-Pr CF_Three              CH₂CH (CH_Three) SEt
H i-Pr CF_Three              CH₂CH₂SCF_Three
H i-Pr CF_Three              CH₂N (CH_Three)₂
H i-Pr CF_Three              CH₂NHPh
H i-Pr CF_Three              CH₂NH (Ph-3-Cl)
H i-Pr CF_Three              CH₂NH (Ph-4-Cl)
H i-Pr CF_Three              CF₂C (O) OEt
H i-Pr CF_Three              CH₂CH₂Ph
H i-Pr CF_Three              CH₂CH₂(Ph-3-Cl)
H i-Pr CF_Three              CH₂CH₂(Ph-4-Cl)
H i-Pr CF_Three              CH (CH_Three) CH₂Ph
H i-Pr CF_Three              CH₂(L-5a)
H i-Pr CF_Three              CH₂(L-14a)
H i-Pr CF_Three              CH₂(L-24a)
H i-Pr CF_Three              CH₂(L-36a)
H i-Pr CF_Three              T-22
H i-Pr CF_Three              T-23
H i-Pr CF_Three              T-24
H i-Pr CF_Three              C (O) OCH_Three
H i-Pr CF_Three              C (O) OEt
H i-Pr CF_Three              C (O) OPr-n
H i-Pr CF_Three              C (O) OPr-i
H i-Pr CF_Three              C (O) OBu-n
H i-Pr CF_Three              C (O) OBu-t
H i-Pr CF_Three              C (O) OCH₂CF_Three
H i-Pr CF_Three              C (O) SEt
H i-Pr CF_Three              C (O) N (CH_Three)₂
H i-Pr CF_Three              CH = CHPh
H i-Pr CF_Three              CH = CH (Ph-3-F)
H i-Pr CF_Three              CH = CH (Ph-4-F)
H i-Pr CF_Three              CH = CH (Ph-2-Cl)
H i-Pr CF_Three              CH = CH (Ph-3-Cl)
H i-Pr CF_Three              CH = CH (Ph-4-Cl)
H i-Pr CF_Three              CH = CH (Ph-3-Br)
H i-Pr CF_Three              CH = CH (Ph-4-Br)
H i-Pr CF_Three              CH = CH (Ph-3-CF_Three)
H i-Pr CF_Three              CH = CH (Ph-4-CF_Three)
H i-Pr CF_Three              CH = CH (Ph-3-OCF_Three)
H i-Pr CF_Three              CH = CH (Ph-4-OCF_Three)
H i-Pr CF_Three              CH = CH (Ph-3-SCH_Three)
H i-Pr CF_Three              CH = CH (Ph-4-SCH_Three)
H i-Pr CF_Three              CH = CH (Ph-3-SO₂CH_Three)
H i-Pr CF_Three              CH = CH (Ph-4-SO₂CH_Three)
H i-Pr CF_Three              CH = CH (Ph-3,4-F₂)
H i-Pr CF_Three              CH = CH (Ph-3-F-4-Cl)
H i-Pr CF_Three              CH = CH (Ph-3,4-Cl₂)
H i-Pr CF_Three              CH = CH (Ph-3,4-Br₂)
H i-Pr CF_Three              CH = CH (Ph-3-F-4-CF_Three)
H i-Pr CF_Three              CH = CH (Ph-3-Cl-4-OCF_Three)
H i-Pr CF_Three              CH = CH [Ph (-3-OCF₂O-4-)]
H i-Pr CF_Three              Ph
H i-Pr CF_Three              Ph-3-F
H i-Pr CF_Three              Ph-4-F
H i-Pr CF_Three              Ph-2-Cl
H i-Pr CF_Three              Ph-3-Cl
H i-Pr CF_Three              Ph-4-Cl
H i-Pr CF_Three              Ph-3-Br
H i-Pr CF_Three              Ph-4-Br
H i-Pr CF_Three              Ph-3-I
H i-Pr CF_Three              Ph-4-I
H i-Pr CF_Three              Ph-4-CH_Three
H i-Pr CF_Three              Ph-4-Et
H i-Pr CF_Three              Ph-4-Pr-n
H i-Pr CF_Three              Ph-4-Pr-i
H i-Pr CF_Three              Ph-4-Bu-n
H i-Pr CF_Three              Ph-4-Bu-i
H i-Pr CF_Three              Ph-4-Bu-t
H i-Pr CF_Three              Ph-3-CF_Three
H i-Pr CF_Three              Ph-4-CF_Three
H i-Pr CF_Three              Ph-4-C (CF_Three)₂OH
H i-Pr CF_Three              Ph-4-C (CF_Three)₂OCH_Three
H i-Pr CF_Three              Ph-4-CH₂OCH_Three
H i-Pr CF_Three              Ph-4-CH₂OCH₂CF_Three
H i-Pr CF_Three              Ph-4-CH₂SCH_Three
H i-Pr CF_Three              Ph-4-CH₂S (O) CH_Three
H i-Pr CF_Three              Ph-4-CH₂SO₂CH_Three
H i-Pr CF_Three              Ph-4-CH₂SEt
H i-Pr CF_Three              Ph-4-CH₂S (O) Et
H i-Pr CF_Three              Ph-4-CH₂SO₂Et
H i-Pr CF_Three              Ph-4-CH₂SPr-n
H i-Pr CF_Three              Ph-4-CH₂SO₂Pr-n
H i-Pr CF_Three              Ph-4-CH₂SPr-i
H i-Pr CF_Three              Ph-4-CH₂SO₂Pr-i
H i-Pr CF_Three              Ph-4-CH₂SPr-c
H i-Pr CF_Three              Ph-4-CH₂SO₂Pr-c
H i-Pr CF_Three              Ph-4-CH₂SBu-n
H i-Pr CF_Three              Ph-4-CH₂SO₂Bu-n
H i-Pr CF_Three              Ph-4-CH₂SCF_Three
H i-Pr CF_Three              Ph-4-CH₂S (O) CF_Three
H i-Pr CF_Three              Ph-4-CH₂SO₂CF_Three
H i-Pr CF_Three              Ph-4-CH₂SCH₂CF_Three
H i-Pr CF_Three              Ph-4-OH
H i-Pr CF_Three              Ph-4-OCH_Three
H i-Pr CF_Three              Ph-4-OEt
H i-Pr CF_Three              Ph-4-OPr-n
H i-Pr CF_Three              Ph-4-OPr-i
H i-Pr CF_Three              Ph-4-OBu-n
H i-Pr CF_Three              Ph-4-OBu-t
H i-Pr CF_Three              Ph-4-OCHF₂
H i-Pr CF_Three              Ph-3-OCF_Three
H i-Pr CF_Three              Ph-4-OCF_Three
H i-Pr CF_Three              Ph-4-OCF₂Br
H i-Pr CF_Three              Ph-4-OCH₂CF_Three
H i-Pr CF_Three              Ph-4-OCF₂CHF₂
H i-Pr CF_Three              Ph-4-OCF₂CHFCl
H i-Pr CF_Three              Ph-4-OCF₂CHFBr
H i-Pr CF_Three              Ph-4-OCF₂CF₂Br
H i-Pr CF_Three              Ph-4-OCF₂CFCl₂
H i-Pr CF_Three              Ph-4-OCF₂CCl_Three
H i-Pr CF_Three              Ph-4-OCH₂CF₂CHF₂
H i-Pr CF_Three              Ph-3-OCF₂CHFCF_Three
H i-Pr CF_Three              Ph-4-OCF₂CHFCF_Three
H i-Pr CF_Three              Ph-4-OCH (CF_Three)₂
H i-Pr CF_Three              Ph-4-OCF₂CFBrCF_Three
H i-Pr CF_Three              Ph-3-OCF₂CHFOCF_Three
H i-Pr CF_Three              Ph-4-OCF₂CHFOCF_Three
H i-Pr CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF_Three              Ph-4-OCH₂CH = CH₂
H i-Pr CF_Three              Ph-4-OCH₂CH = CF₂
H i-Pr CF_Three              Ph-4-OCH₂CF = CF₂
H i-Pr CF_Three              Ph-4-OCH₂CH = CCl₂
H i-Pr CF_Three              Ph-4-OCH₂CCl = CCl₂
H i-Pr CF_Three              Ph-4-OCH₂Ph
H i-Pr CF_Three              Ph-4-OSO₂CH_Three
H i-Pr CF_Three              Ph-4-OSO₂Et
H i-Pr CF_Three              Ph-4-OSO₂Pr-n
H i-Pr CF_Three              Ph-4-OSO₂Pr-i
H i-Pr CF_Three              Ph-4-OSO₂Bu-n
H i-Pr CF_Three              Ph-4-OSO₂CHCl₂
H i-Pr CF_Three              Ph-4-OSO₂CF_Three
H i-Pr CF_Three              Ph-4-OSO₂CH₂CF_Three
H i-Pr CF_Three              Ph-3-O (Ph-4-Cl)
H i-Pr CF_Three              Ph-4-O (Ph-4-Cl)
H i-Pr CF_Three              Ph-4-O (Ph-4-Br)
H i-Pr CF_Three              Ph-4-O (Ph-4-CF_Three)
H i-Pr CF_Three              Ph-4-O (L-21b) Br
H i-Pr CF_Three              Ph-4-O (L-21b) CF_Three
H i-Pr CF_Three              Ph-3-O (L-45c) Br
H i-Pr CF_Three              Ph-4-O (L-45c) Br
H i-Pr CF_Three              Ph-3-O (L-45c) CF_Three
H i-Pr CF_Three              Ph-4-O (L-45c) CF_Three
H i-Pr CF_Three              Ph-3-O (L-45e)
H i-Pr CF_Three              Ph-4-O (L-45e)
H i-Pr CF_Three              Ph-3-O (L-48b) Br
H i-Pr CF_Three              Ph-4-O (L-48b) Br
H i-Pr CF_Three              Ph-4-SCH_Three
H i-Pr CF_Three              Ph-4-S (O) CH_Three
H i-Pr CF_Three              Ph-4-SO₂CH_Three
H i-Pr CF_Three              Ph-4-SEt
H i-Pr CF_Three              Ph-4-S (O) Et
H i-Pr CF_Three              Ph-4-SO₂Et
H i-Pr CF_Three              Ph-4-SPr-n
H i-Pr CF_Three              Ph-4-S (O) Pr-n
H i-Pr CF_Three              Ph-4-SO₂Pr-n
H i-Pr CF_Three              Ph-4-SPr-i
H i-Pr CF_Three              Ph-4-S (O) Pr-i
H i-Pr CF_Three              Ph-4-SO₂Pr-i
H i-Pr CF_Three              Ph-4-SBu-n
H i-Pr CF_Three              Ph-4-S (O) Bu-n
H i-Pr CF_Three              Ph-4-SO₂Bu-n
H i-Pr CF_Three              Ph-4-SBu-t
H i-Pr CF_Three              Ph-4-S (O) Bu-t
H i-Pr CF_Three              Ph-4-SO₂Bu-t
H i-Pr CF_Three              Ph-4-SCH₂F
H i-Pr CF_Three              Ph-4-S (O) CH₂F
H i-Pr CF_Three              Ph-4-SO₂CH₂F
H i-Pr CF_Three              Ph-4-SCHF₂
H i-Pr CF_Three              Ph-4-S (O) CHF₂
H i-Pr CF_Three              Ph-4-SO₂CHF₂
H i-Pr CF_Three              Ph-3-SCF_Three
H i-Pr CF_Three              Ph-4-SCF_Three
H i-Pr CF_Three              Ph-4-S (O) CF_Three
H i-Pr CF_Three              Ph-4-SO₂CF_Three
H i-Pr CF_Three              Ph-4-SCF₂Cl
H i-Pr CF_Three              Ph-4-S (O) CF₂Cl
H i-Pr CF_Three              Ph-4-SO₂CF₂Cl
H i-Pr CF_Three              Ph-4-SCF₂Br
H i-Pr CF_Three              Ph-4-S (O) CF₂Br
H i-Pr CF_Three              Ph-4-SO₂CF₂Br
H i-Pr CF_Three              Ph-3-S (Ph-4-Cl)
H i-Pr CF_Three              Ph-4-S (Ph-4-Cl)
H i-Pr CF_Three              Ph-4-S (Ph-4-Br)
H i-Pr CF_Three              Ph-4-S (Ph-4-CF_Three)
H i-Pr CF_Three              Ph-4-S (L-45c) Br
H i-Pr CF_Three              Ph-4-S (L-45c) CF_Three
H i-Pr CF_Three              Ph-4-S (L-45e)
H i-Pr CF_Three              Ph-4-S (L-48b) Br
H i-Pr CF_Three              Ph-4-NO₂
H i-Pr CF_Three              Ph-4-N (CH_Three)₂
H i-Pr CF_Three              Ph-4-N (Et)₂
H i-Pr CF_Three              Ph-4- (T-16)
H i-Pr CF_Three              Ph-4-CN
H i-Pr CF_Three              Ph-4-C (O) OCH_Three
H i-Pr CF_Three              Ph-4-C (O) NH₂
H i-Pr CF_Three              Ph-4-C (O) NHCH_Three
H i-Pr CF_Three              Ph-4-C (O) NHEt
H i-Pr CF_Three              Ph-4-C (O) N (CH_Three)₂
H i-Pr CF_Three              Ph-4-C (S) NH₂
H i-Pr CF_Three              Ph-3-Ph
H i-Pr CF_Three              Ph-4-Ph
H i-Pr CF_Three              Ph-4- (L-5a)
H i-Pr CF_Three              Ph-4- (L-14a)
H i-Pr CF_Three              Ph-4- (L-24a)
H i-Pr CF_Three              Ph-4- (L-36a)
H i-Pr CF_Three              Ph-2,4-F₂
H i-Pr CF_Three              Ph-3,4-F₂
H i-Pr CF_Three              Ph-2-Cl-4-F
H i-Pr CF_Three              Ph-3-Cl-4-F
H i-Pr CF_Three              Ph-2-F-4-Cl
H i-Pr CF_Three              Ph-3-F-4-Cl
H i-Pr CF_Three              Ph-2,4-Cl₂
H i-Pr CF_Three              Ph-3,4-Cl₂
H i-Pr CF_Three              Ph-3,5-Cl₂
H i-Pr CF_Three              Ph-3-Br-4-F
H i-Pr CF_Three              Ph-2-F-4-Br
H i-Pr CF_Three              Ph-3,4-Br₂
H i-Pr CF_Three              Ph-3-CH_Three-4-F
H i-Pr CF_Three              Ph-3-F-4-CH_Three
H i-Pr CF_Three              Ph-3,4- (CH_Three)₂
H i-Pr CF_Three              Ph-3-CF_Three-4-F
H i-Pr CF_Three              Ph-3-CF_Three-4-Cl
H i-Pr CF_Three              Ph-2-F-4-CF_Three
H i-Pr CF_Three              Ph-3-F-4-CF_Three
H i-Pr CF_Three              Ph-2-Cl-4-CF_Three
H i-Pr CF_Three              Ph-3-Br-4-OCH_Three
H i-Pr CF_Three              Ph-3-F-4-OCHF₂
H i-Pr CF_Three              Ph-3-Cl-4-OCHF₂
H i-Pr CF_Three              Ph-3-Br-4-OCHF₂
H i-Pr CF_Three              Ph-3-F-4-OCF_Three
H i-Pr CF_Three              Ph-3-Cl-4-OCF_Three
H i-Pr CF_Three              Ph-3-Br-4-OCF_Three
H i-Pr CF_Three              Ph-3-F-4-OCF₂Br
H i-Pr CF_Three              Ph-3-Cl-4-OCF₂Br
H i-Pr CF_Three              Ph-3-Br-4-OCF₂Br
H i-Pr CF_Three              Ph-3-F-4-OCF₂CHF₂
H i-Pr CF_Three              Ph-3-Cl-4-OCF₂CHF₂
H i-Pr CF_Three              Ph-3-Br-4-OCF₂CHF₂
H i-Pr CF_Three              Ph-3-F-4-OCF₂CHFCl
H i-Pr CF_Three              Ph-3-Cl-4-OCF₂CHFCl
H i-Pr CF_Three              Ph-3-Br-4-OCF₂CHFCl
H i-Pr CF_Three              Ph-3-F-4-OCF₂CHFCF_Three
H i-Pr CF_Three              Ph-3-Cl-4-OCF₂CHFCF_Three
H i-Pr CF_Three              Ph-3-Br-4-OCF₂CHFCF_Three
H i-Pr CF_Three              Ph-3-F-4-OCF₂CHFOCF_Three
H i-Pr CF_Three              Ph-3-Cl-4-OCF₂CHFOCF_Three
H i-Pr CF_Three              Ph-3-Br-4-OCF₂CHFOCF_Three
H i-Pr CF_Three              Ph-3-CH_Three-4-OCF₂CHFOCF_Three
H i-Pr CF_Three         Ph-3-F-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF_Three         Ph-3-Cl-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF_Three         Ph-3-Br-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF_Three              Ph (-3-OCF₂O-4-)
H i-Pr CF_Three              Ph (-3-OCF₂CF₂O-4-)
H i-Pr CF_Three              Ph-3-OPh-4-F
H i-Pr CF_Three              Ph-3-NO₂-4-F
H i-Pr CF_Three              Ph-3-NO₂-4-Cl
H i-Pr CF_Three              Ph-3-CN-4-F
H i-Pr CF_Three              Ph-2,3,4-F_Three
H i-Pr CF_Three              Ph-2,4,5-F_Three
H i-Pr CF_Three              Ph-3,4,5-F_Three
H i-Pr CF_Three              Ph-2,3-F₂-4-CH_Three
H i-Pr CF_Three              Ph-2,3-F₂-4-CF_Three
H i-Pr CF_Three              Ph-3,4-F₂-5-CF_Three
H i-Pr CF_Three              Ph-2-F-3-Cl-5-CF_Three
H i-Pr CF_Three              Ph-3,5-Cl₂-4-OCH_Three
H i-Pr CF_Three              1-Naph
H i-Pr CF_Three              2-Naph
H i-Pr CF_Three              L-1a
H i-Pr CF_Three             (L-1b) Br
H i-Pr CF_Three             (L-1c) Cl
H i-Pr CF_Three             (L-1c) Br
H i-Pr CF_Three             (L-1c) I
H i-Pr CF_Three             (L-1c) CF_Three
H i-Pr CF_Three             (L-1c) SCH_Three
H i-Pr CF_Three             (L-1c) SO₂CH_Three
H i-Pr CF_Three             (L-1c) NO₂
H i-Pr CF_Three              L-2a
H i-Pr CF_Three             (L-2b) Br
H i-Pr CF_Three              L-3a
H i-Pr CF_Three             (L-3b) Cl
H i-Pr CF_Three             (L-3b) Br
H i-Pr CF_Three             (L-3b) SCH_Three
H i-Pr CF_Three             (L-3b) SO₂CH_Three
H i-Pr CF_Three             (L-3c) F
H i-Pr CF_Three             (L-3c) Cl
H i-Pr CF_Three             (L-3c) Br
H i-Pr CF_Three             (L-3c) I
H i-Pr CF_Three             (L-3c) CF_Three
H i-Pr CF_Three             (L-3c) SCH_Three
H i-Pr CF_Three             (L-3c) SO₂CH_Three
H i-Pr CF_Three             (L-3c) NO₂
H i-Pr CF_Three             (L-3c) CN
H i-Pr CF_Three              L-3d
H i-Pr CF_Three              L-4a
H i-Pr CF_Three             (L-4b) Cl
H i-Pr CF_Three             (L-4b) Br
H i-Pr CF_Three             (L-4b) NO₂
H i-Pr CF_Three             (L-4b) CN
H i-Pr CF_Three             (L-6a) Cl
H i-Pr CF_Three             (L-6a) Br
H i-Pr CF_Three             (L-6b) Cl
H i-Pr CF_Three             (L-6b) Br
H i-Pr CF_Three             (L-6b) NO₂
H i-Pr CF_Three              L-8a
H i-Pr CF_Three              L-10a
H i-Pr CF_Three             (L-10b) Cl
H i-Pr CF_Three             (L-10b) Br
H i-Pr CF_Three             (L-10b) SCH_Three
H i-Pr CF_Three              L-11a
H i-Pr CF_Three             (L-15a) CHF₂
H i-Pr CF_Three             (L-15b) CF_Three
H i-Pr CF_Three             (L-16a) CHF₂
H i-Pr CF_Three             (L-16a) CF₂Br
H i-Pr CF_Three             (L-17a) Cl
H i-Pr CF_Three              L-19a
H i-Pr CF_Three              L-20a
H i-Pr CF_Three              L-21a
H i-Pr CF_Three             (L-21b) Cl
H i-Pr CF_Three             (L-21b) Br
H i-Pr CF_Three             (L-21b) I
H i-Pr CF_Three             (L-21b) CF_Three
H i-Pr CF_Three             (L-21b) NO₂
H i-Pr CF_Three              L-22a
H i-Pr CF_Three             (L-22b) Cl
H i-Pr CF_Three             (L-22b) CF_Three
H i-Pr CF_Three             (L-22b) SCH_Three
H i-Pr CF_Three              L-23a
H i-Pr CF_Three             (L-23b) Cl
H i-Pr CF_Three             (L-23b) Br
H i-Pr CF_Three             (L-23b) SCH_Three
H i-Pr CF_Three             (L-23b) NO₂
H i-Pr CF_Three             (L-23c) Cl
H i-Pr CF_Three             (L-23c) Br
H i-Pr CF_Three             (L-23c) SCH_Three
H i-Pr CF_Three             (L-25a) Cl
H i-Pr CF_Three             (L-25a) Br
H i-Pr CF_Three             (L-25a) I
H i-Pr CF_Three             (L-25a) CF_Three
H i-Pr CF_Three              L-25b
H i-Pr CF_Three             (L-30a) SCH_Three
H i-Pr CF_Three             (L-31a) Cl
H i-Pr CF_Three             (L-31a) Br
H i-Pr CF_Three             (L-31a) SCH_Three
H i-Pr CF_Three             (L-34a) Ph
H i-Pr CF_Three             (L-35a) Ph
H i-Pr CF_Three             (L-38a) Cl
H i-Pr CF_Three             (L-38a) Br
H i-Pr CF_Three             (L-38a) NO₂
H i-Pr CF_Three              L-45a
H i-Pr CF_Three             (L-45b) Cl
H i-Pr CF_Three             (L-45c) F
H i-Pr CF_Three             (L-45c) Cl
H i-Pr CF_Three             (L-45c) Br
H i-Pr CF_Three             (L-45c) I
H i-Pr CF_Three             (L-45c) CF_Three
H i-Pr CF_Three             (L-45c) NO₂
H i-Pr CF_Three             (L-45d) F
H i-Pr CF_Three             (L-45d) Cl
H i-Pr CF_Three             (L-45d) Br
H i-Pr CF_Three              L-45e
H i-Pr CF_Three              L-45f
H i-Pr CF_Three              L-46a
H i-Pr CF_Three             (L-46b) Br
H i-Pr CF_Three             (L-46c) F
H i-Pr CF_Three             (L-46c) Cl
H i-Pr CF_Three             (L-46c) Br
H i-Pr CF_Three             (L-46c) I
H i-Pr CF_Three             (L-46c) CF_Three
H i-Pr CF_Three             (L-46c) CH₂SCH_Three
H i-Pr CF_Three             (L-46c) CH₂SO₂CH_Three
H i-Pr CF_Three             (L-46c) OCH₂CF_Three
H i-Pr CF_Three             (L-46c) OCH (CF_Three)₂
H i-Pr CF_Three             (L-46c) OSO₂CH_Three
H i-Pr CF_Three             (L-46c) SCH_Three
H i-Pr CF_Three             (L-46c) SO₂CH_Three
H i-Pr CF_Three             (L-46c) SEt
H i-Pr CF_Three             (L-46c) SPr-i
H i-Pr CF_Three             (L-46c) CN
H i-Pr CF_Three              L-46d
H i-Pr CF_Three              L-47a
H i-Pr CF_Three             (L-47b) F
H i-Pr CF_Three             (L-47b) Cl
H i-Pr CF_Three              L-47c
H i-Pr CF_Three              L-47d
H i-Pr CF_Three              L-48a
H i-Pr CF_Three             (L-48b) Br
H i-Pr CF_Three              L-50a
H i-Pr CF_Three             (L-50b) Cl
H i-Pr CF_Three             (L-50b) Br
H i-Pr CF_Three             (L-50b) I
H i-Pr CF_Three             (L-50b) SCH_Three
H i-Pr CF_Three             (L-50b) SO₂CH_Three
H i-Pr CF_Three              L-51a
H i-Pr CF_Three             (L-51b) Cl
H i-Pr CF_Three             (L-51b) SCH_Three
H i-Pr CF_Three              L-53a
H i-Pr CF_Three              L-55a
H i-Pr CF₂Cl CF₂O (Ph-4-Cl)
H i-Pr CF₂Cl CH = CH (Ph-4-Cl)
H i-Pr CF₂Cl CH = CH (Ph-4-OCF_Three)
H i-Pr CF₂Cl CH = CH (Ph-3,4-Cl₂)
H i-Pr CF₂Cl Ph-4-F
H i-Pr CF₂Cl Ph-4-Cl
H i-Pr CF₂Cl Ph-4-Br
H i-Pr CF₂Cl Ph-4-I
H i-Pr CF₂Cl Ph-4-CF_Three
H i-Pr CF₂Cl Ph-4-OCHF₂
H i-Pr CF₂Cl Ph-4-OCF_Three
H i-Pr CF₂Cl Ph-4-OCF₂Br
H i-Pr CF₂Cl Ph-4-OCF₂CHF₂
H i-Pr CF₂Cl Ph-4-OCF₂CHFCl
H i-Pr CF₂Cl Ph-4-OCF₂CHFCF_Three
H i-Pr CF₂Cl Ph-4-OCF₂CHFOCF_Three
H i-Pr CF₂Cl Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF₂Cl Ph-4-O (L-45g)
H i-Pr CF₂Cl Ph-3,4-Cl₂
H i-Pr CF₂Cl Ph (-3-OCF₂O-4-)
H i-Pr CF₂Cl Ph (-3-OCF₂CF₂O-4-)
H i-Pr CF₂Cl (L-45c) Cl
H i-Pr CF₂Cl (L-45c) Br
H i-Pr CF₂Cl (L-45c) CF_Three
H i-Pr CF₂Cl L-45e
H i-Pr CF₂Cl L-45f
H i-Pr CF₂Cl (L-46c) Cl
H i-Pr CF₂Cl (L-46c) Br
H i-Pr CF₂Cl (L-46c) CF_Three
H i-Pr CF₂Cl L-46d
H i-Pr CFCl₂            Ph-4-CF_Three
H i-Pr CF₂Br CF₂O (Ph-4-Cl)
H i-Pr CF₂Br CH = CH (Ph-4-Cl)
H i-Pr CF₂Br CH = CH (Ph-4-OCF_Three)
H i-Pr CF₂Br CH = CH (Ph-3,4-Cl₂)
H i-Pr CF₂Br Ph-4-F
H i-Pr CF₂Br Ph-4-Cl
H i-Pr CF₂Br Ph-4-Br
H i-Pr CF₂Br Ph-4-I
H i-Pr CF₂Br Ph-4-CF_Three
H i-Pr CF₂Br Ph-4-OCHF₂
H i-Pr CF₂Br Ph-4-OCF_Three
H i-Pr CF₂Br Ph-4-OCF₂Br
H i-Pr CF₂Br Ph-4-OCF₂CHF₂
H i-Pr CF₂Br Ph-4-OCF₂CHFCl
H i-Pr CF₂Br Ph-4-OCF₂CHFCF_Three
H i-Pr CF₂Br Ph-4-OCF₂CHFOCF_Three
H i-Pr CF₂Br Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF₂Br Ph-4-O (L-45g)
H i-Pr CF₂Br Ph-3,4-Cl₂
H i-Pr CF₂Br Ph (-3-OCF₂O-4-)
H i-Pr CF₂Br Ph (-3-OCF₂CF₂O-4-)
H i-Pr CF₂Br (L-45c) Cl
H i-Pr CF₂Br (L-45c) Br
H i-Pr CF₂Br (L-45c) CF_Three
H i-Pr CF₂Br L-45e
H i-Pr CF₂Br L-45f
H i-Pr CF₂Br (L-46c) Cl
H i-Pr CF₂Br (L-46c) Br
H i-Pr CF₂Br (L-46c) CF_Three
H i-Pr CF₂Br L-46d
H i-Pr CFClBr Ph-4-OCF_Three
H i-Pr CFBr₂           (L-45c) CF_Three
H i-Pr CF₂CHF₂          Ph-4-Br
H i-Pr CF₂CF_Three           CF₂O (Ph-4-Cl)
H i-Pr CF₂CF_Three           CH = CH (Ph-4-Cl)
H i-Pr CF₂CF_Three           CH = CH (Ph-4-OCF_Three)
H i-Pr CF₂CF_Three           CH = CH (Ph-3,4-Cl₂)
H i-Pr CF₂CF_Three           Ph-4-F
H i-Pr CF₂CF_Three           Ph-4-Cl
H i-Pr CF₂CF_Three           Ph-4-Br
H i-Pr CF₂CF_Three           Ph-4-I
H i-Pr CF₂CF_Three           Ph-4-CF_Three
H i-Pr CF₂CF_Three           Ph-4-OCHF₂
H i-Pr CF₂CF_Three           Ph-4-OCF_Three
H i-Pr CF₂CF_Three           Ph-4-OCF₂Br
H i-Pr CF₂CF_Three           Ph-4-OCF₂CHF₂
H i-Pr CF₂CF_Three           Ph-4-OCF₂CHFCl
H i-Pr CF₂CF_Three           Ph-4-OCF₂CHFCF_Three
H i-Pr CF₂CF_Three           Ph-4-OCF₂CHFOCF_Three
H i-Pr CF₂CF_Three           Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF₂CF_Three           Ph-4-O (L-45g)
H i-Pr CF₂CF_Three           Ph-3,4-Cl₂
H i-Pr CF₂CF_Three           Ph (-3-OCF₂O-4-)
H i-Pr CF₂CF_Three           Ph (-3-OCF₂CF₂O-4-)
H i-Pr CF₂CF_Three          (L-45c) Cl
H i-Pr CF₂CF_Three          (L-45c) Br
H i-Pr CF₂CF_Three          (L-45c) CF_Three
H i-Pr CF₂CF_Three           L-45e
H i-Pr CF₂CF_Three           L-45f
H i-Pr CF₂CF_Three          (L-46c) Cl
H i-Pr CF₂CF_Three          (L-46c) Br
H i-Pr CF₂CF_Three          (L-46c) CF_Three
H i-Pr CF₂CF_Three           L-46d
H i-Pr CF₂CF₂Cl Ph-4-CF_Three
H i-Pr CFClCF_Three          Ph-4-OCF_Three
H i-Pr CFClCF₂Cl (L-45c) CF_Three
H i-Pr CF₂CF₂Br Ph-4-Br
H i-Pr CFBrCF_Three          Ph-4-CF_Three
H i-Pr CF₂CHFCF_Three        Ph-4-OCF_Three
H i-Pr CF₂CF₂CF_Three        CF₂O (Ph-4-Cl)
H i-Pr CF₂CF₂CF_Three        CH = CH (Ph-4-Cl)
H i-Pr CF₂CF₂CF_Three        CH = CH (Ph-4-OCF_Three)
H i-Pr CF₂CF₂CF_Three        CH = CH (Ph-3,4-Cl₂)
H i-Pr CF₂CF₂CF_Three        Ph-4-F
H i-Pr CF₂CF₂CF_Three        Ph-4-Cl
H i-Pr CF₂CF₂CF_Three        Ph-4-Br
H i-Pr CF₂CF₂CF_Three        Ph-4-I
H i-Pr CF₂CF₂CF_Three        Ph-4-CF_Three
H i-Pr CF₂CF₂CF_Three        Ph-4-OCHF₂
H i-Pr CF₂CF₂CF_Three        Ph-4-OCF_Three
H i-Pr CF₂CF₂CF_Three        Ph-4-OCF₂Br
H i-Pr CF₂CF₂CF_Three        Ph-4-OCF₂CHF₂
H i-Pr CF₂CF₂CF_Three        Ph-4-OCF₂CHFCl
H i-Pr CF₂CF₂CF_Three        Ph-4-OCF₂CHFCF_Three
H i-Pr CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF_Three
H i-Pr CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF₂CF₂CF_Three        Ph-4-O (L-45g)
H i-Pr CF₂CF₂CF_Three        Ph-3,4-Cl₂
H i-Pr CF₂CF₂CF_Three        Ph (-3-OCF₂O-4-)
H i-Pr CF₂CF₂CF_Three        Ph (-3-OCF₂CF₂O-4-)
H i-Pr CF₂CF₂CF_Three       (L-45c) Cl
H i-Pr CF₂CF₂CF_Three       (L-45c) Br
H i-Pr CF₂CF₂CF_Three       (L-45c) CF_Three
H i-Pr CF₂CF₂CF_Three        L-45e
H i-Pr CF₂CF₂CF_Three        L-45f
H i-Pr CF₂CF₂CF_Three       (L-46c) Cl
H i-Pr CF₂CF₂CF_Three       (L-46c) Br
H i-Pr CF₂CF₂CF_Three       (L-46c) CF_Three
H i-Pr CF₂CF₂CF_Three        L-46d
H i-Pr CF (CF_Three)₂        (L-45c) CF_Three
H i-Pr CF₂CFClCF₂Cl Ph-4-Br
H i-Pr CF₂CFBrCF₂Cl Ph-4-CF_Three
H i-Pr CF₂CF₂CF₂CHF₂    Ph-4-OCF_Three
H i-Pr CF₂CF₂CF₂CF_Three    (L-45c) CF_Three
H i-Pr CF (CF_ThreeCF₂CF_Three    Ph-4-Br
H i-Pr CF₂CF₂CF₂CF₂Cl Ph-4-CF_Three
H i-Pr CF₂CF₂CF₂CF₂CF₂CF_Three      Ph-4-OCF_Three
H i-Pr T-1 (L-45c) CF_Three
H i-Pr T-2 Ph-4-Br
H i-Pr CH₂OCH_Three          Ph-4-CF_Three
H i-Pr CH₂OEt Ph-4-OCF_Three
H i-Pr CH₂OCH₂CF_Three      (L-45c) CF_Three
H i-Pr CH₂OCH (CF_Three)₂     Ph-4-Br
H i-Pr CF₂OCH_Three          CF₂O (Ph-4-Cl)
H i-Pr CF₂OCH_Three          CH = CH (Ph-4-Cl)
H i-Pr CF₂OCH_Three          CH = CH (Ph-4-OCF_Three)
H i-Pr CF₂OCH_Three          CH = CH (Ph-3,4-Cl₂)
H i-Pr CF₂OCH_Three          Ph-4-F
H i-Pr CF₂OCH_Three          Ph-4-Cl
H i-Pr CF₂OCH_Three          Ph-4-Br
H i-Pr CF₂OCH_Three          Ph-4-I
H i-Pr CF₂OCH_Three          Ph-4-CF_Three
H i-Pr CF₂OCH_Three          Ph-4-OCHF₂
H i-Pr CF₂OCH_Three          Ph-4-OCF_Three
H i-Pr CF₂OCH_Three          Ph-4-OCF₂Br
H i-Pr CF₂OCH_Three          Ph-4-OCF₂CHF₂
H i-Pr CF₂OCH_Three          Ph-4-OCF₂CHFCl
H i-Pr CF₂OCH_Three          Ph-4-OCF₂CHFCF_Three
H i-Pr CF₂OCH_Three          Ph-4-OCF₂CHFOCF_Three
H i-Pr CF₂OCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF₂OCH_Three          Ph-4-O (L-45g)
H i-Pr CF₂OCH_Three          Ph-3,4-Cl₂
H i-Pr CF₂OCH_Three          Ph (-3-OCF₂O-4-)
H i-Pr CF₂OCH_Three          Ph (-3-OCF₂CF₂O-4-)
H i-Pr CF₂OCH_Three         (L-45c) Cl
H i-Pr CF₂OCH_Three         (L-45c) Br
H i-Pr CF₂OCH_Three         (L-45c) CF_Three
H i-Pr CF₂OCH_Three          L-45e
H i-Pr CF₂OCH_Three          L-45f
H i-Pr CF₂OCH_Three         (L-46c) Cl
H i-Pr CF₂OCH_Three         (L-46c) Br
H i-Pr CF₂OCH_Three         (L-46c) CF_Three
H i-Pr CF₂OCH_Three          L-46d
H i-Pr CF₂OCF₂CF₂CF_Three         Ph-4-CF_Three
H i-Pr CF₂OCF₂CF₂OCF_Three        Ph-4-OCF_Three
H i-Pr CF (CF_Three) OCH_Three          (L-45c) CF_Three
H i-Pr CF (CF_ThreeOCF₂CF₂CF_Three     Ph-4-Br
H i-Pr CH₂SCH_Three          Ph-4-CF_Three
H i-Pr CH₂SO₂CH_Three        Ph-4-OCF_Three
H i-Pr CH₂SEt (L-45c) CF_Three
H i-Pr CH₂SCF_Three          Ph-4-Br
H i-Pr CH₂SPh Ph-4-CF_Three
H i-Pr CH₂CH₂SCH_Three       Ph-4-OCF_Three
H i-Pr CH₂CH₂SCF_Three      (L-45c) CF_Three
H i-Pr CF₂SCH_Three          CF₂O (Ph-4-Cl)
H i-Pr CF₂SCH_Three          CH = CH (Ph-4-Cl)
H i-Pr CF₂SCH_Three          CH = CH (Ph-4-OCF_Three)
H i-Pr CF₂SCH_Three          CH = CH (Ph-3,4-Cl₂)
H i-Pr CF₂SCH_Three          Ph-4-F
H i-Pr CF₂SCH_Three          Ph-4-Cl
H i-Pr CF₂SCH_Three          Ph-4-Br
H i-Pr CF₂SCH_Three          Ph-4-I
H i-Pr CF₂SCH_Three          Ph-4-CF_Three
H i-Pr CF₂SCH_Three          Ph-4-OCHF₂
H i-Pr CF₂SCH_Three          Ph-4-OCF_Three
H i-Pr CF₂SCH_Three          Ph-4-OCF₂Br
H i-Pr CF₂SCH_Three          Ph-4-OCF₂CHF₂
H i-Pr CF₂SCH_Three          Ph-4-OCF₂CHFCl
H i-Pr CF₂SCH_Three          Ph-4-OCF₂CHFCF_Three
H i-Pr CF₂SCH_Three          Ph-4-OCF₂CHFOCF_Three
H i-Pr CF₂SCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H i-Pr CF₂SCH_Three          Ph-4-O (L-45g)
H i-Pr CF₂SCH_Three          Ph-3,4-Cl₂
H i-Pr CF₂SCH_Three          Ph (-3-OCF₂O-4-)
H i-Pr CF₂SCH_Three          Ph (-3-OCF₂CF₂O-4-)
H i-Pr CF₂SCH_Three         (L-45c) Cl
H i-Pr CF₂SCH_Three         (L-45c) Br
H i-Pr CF₂SCH_Three         (L-45c) CF_Three
H i-Pr CF₂SCH_Three          L-45e
H i-Pr CF₂SCH_Three          L-45f
H i-Pr CF₂SCH_Three         (L-46c) Cl
H i-Pr CF₂SCH_Three         (L-46c) Br
H i-Pr CF₂SCH_Three         (L-46c) CF_Three
H i-Pr CF₂SCH_Three          L-46d
H i-Pr CF₂SEt Ph-4-Br
H i-Pr CF₂SPr-n Ph-4-CF_Three
H i-Pr CF₂SPr-i Ph-4-OCF_Three
H i-Pr CF₂SCH₂Ph (L-45c) CF_Three
H i-Pr CF₂SPh Ph-4-Br
H i-Pr CF₂C (O) OEt Ph-4-CF_Three
H i-Pr CF₂SO₂N (CH_Three)₂    Ph-4-OCF_Three
H i-Pr CN (L-45c) CF_Three
H i-Pr C (O) OCH_Three         Ph-4-Br
H i-Pr C (O) OEt Ph-4-CF_Three
H i-Pr C (O) OPr-n Ph-4-OCF_Three
H i-Pr C (O) OPr-i (L-45c) CF_Three
H i-Pr C (O) OBu-n Ph-4-Br
H i-Pr C (O) OBu-t Ph-4-CF_Three
H i-Pr C (O) SEt Ph-4-OCF_Three
H i-Pr C (O) NH₂         (L-45c) CF_Three
H i-Pr C (S) NH₂          Ph-4-Br
H i-Pr C (CH_Three) = NOCH_Three     Ph-4-CF_Three
H i-Pr Ph Ph-4-OCF_Three
H i-Pr Ph-4-F (L-45c) CF_Three
H i-Pr Ph-4-Cl Ph-4-Br
H i-Pr Ph-4-CF_Three         Ph-4-CF_Three
H i-Pr Ph-4-OCF_Three        Ph-4-OCF_Three
CH_Three       i-Pr CF_Three              Ph-4-Br
CH_Three       i-Pr CF_Three              Ph-4-CF_Three
CH_Three       i-Pr CF_Three              Ph-4-OCF_Three
CH_Three       i-Pr CF_Three             (L-45c) CF_Three
Et i-Pr CF_Three             (L-45c) CF_Three
i-Pr i-Pr CF_Three              Ph-4-Br
CH₂OCH_Three   i-Pr CF_Three              Ph-4-CF_Three
CH₂OEt i-Pr CF_Three              Ph-4-OCF_Three
H c-Pr CF_Three              CF₂O (Ph-4-Cl)
H c-Pr CF_Three              CH = CH (Ph-4-Cl)
H c-Pr CF_Three              CH = CH (Ph-4-OCF_Three)
H c-Pr CF_Three              CH = CH (Ph-3,4-Cl₂)
H c-Pr CF_Three              Ph-4-F
H c-Pr CF_Three              Ph-4-Cl
H c-Pr CF_Three              Ph-4-Br
H c-Pr CF_Three              Ph-4-I
H c-Pr CF_Three              Ph-4-CF_Three
H c-Pr CF_Three              Ph-4-OCHF₂
H c-Pr CF_Three              Ph-4-OCF_Three
H c-Pr CF_Three              Ph-4-OCF₂Br
H c-Pr CF_Three              Ph-4-OCF₂CHF₂
H c-Pr CF_Three              Ph-4-OCF₂CHFCl
H c-Pr CF_Three              Ph-4-OCF₂CHFCF_Three
H c-Pr CF_Three              Ph-4-OCF₂CHFOCF_Three
H c-Pr CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H c-Pr CF_Three              Ph-4-O (L-45g)
H c-Pr CF_Three              Ph-3,4-Cl₂
H c-Pr CF_Three              Ph (-3-OCF₂O-4-)
H c-Pr CF_Three              Ph (-3-OCF₂CF₂O-4-)
H c-Pr CF_Three             (L-45c) Cl
H c-Pr CF_Three             (L-45c) Br
H c-Pr CF_Three             (L-45c) CF_Three
H c-Pr CF_Three              L-45e
H c-Pr CF_Three              L-45f
H c-Pr CF_Three             (L-46c) Cl
H c-Pr CF_Three             (L-46c) Br
H c-Pr CF_Three             (L-46c) CF_Three
H c-Pr CF_Three              L-46d
H n-Bu CF_Three              CH = CH (Ph-4-Cl)
H n-Bu CF_Three              Ph-4-Cl
H n-Bu CF_Three              Ph-4-Br
H n-Bu CF_Three              Ph-4-CF_Three
H n-Bu CF_Three              Ph-4-OCF_Three
H n-Bu CF_Three              Ph-4-OCF₂Br
H n-Bu CF_Three              Ph-4-OCF₂CHFCF_Three
H n-Bu CF_Three              Ph-4-OCF₂CHFOCF_Three
H n-Bu CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H n-Bu CF_Three              Ph-4-O (L-45g)
H n-Bu CF_Three              Ph-3,4-Cl₂
H n-Bu CF_Three              Ph (-3-OCF₂O-4-)
H n-Bu CF_Three              Ph (-3-OCF₂CF₂O-4-)
H n-Bu CF_Three             (L-45c) CF_Three
H n-Bu CF_Three              L-45f
H n-Bu CF_Three             (L-46c) CF_Three
H n-Bu CF_Three              L-46d
H i-Bu CF_Three             (L-45c) CF_Three
CH_Three       i-Bu CF_Three              Ph-4-Br
H CH₂Pr-c CF_Three              Ph-4-CF_Three
H s-Bu CH_Three              Ph-4-Br
H s-Bu CH_Three              Ph-4-CF_Three
H s-Bu CH_Three              Ph-4-OCF_Three
H s-Bu CH_Three             (L-45c) Cl
H s-Bu CH_Three             (L-45c) Br
H s-Bu CH_Three             (L-45c) CF_Three
H s-Bu Et Ph-4-OCF_Three
H s-Bu n-Pr (L-45c) CF_Three
H s-Bu i-Pr Ph-4-Br
H s-Bu c-Pr Ph-4-CF_Three
H s-Bu CHF₂             Ph-4-OCF_Three
H s-Bu CF_Three              CF₂O (Ph-4-Cl)
H s-Bu CF_Three              CH = CH (Ph-4-Cl)
H s-Bu CF_Three              CH = CH (Ph-4-OCF_Three)
H s-Bu CF_Three              CH = CH (Ph-3,4-Cl₂)
H s-Bu CF_Three              Ph-4-F
H s-Bu CF_Three              Ph-4-Cl
H s-Bu CF_Three              Ph-4-Br
H s-Bu CF_Three              Ph-4-I
H s-Bu CF_Three              Ph-4-CF_Three
H s-Bu CF_Three              Ph-4-OCHF₂
H s-Bu CF_Three              Ph-4-OCF_Three
H s-Bu CF_Three              Ph-4-OCF₂Br
H s-Bu CF_Three              Ph-4-OCF₂CHF₂
H s-Bu CF_Three              Ph-4-OCF₂CHFCl
H s-Bu CF_Three              Ph-4-OCF₂CHFCF_Three
H s-Bu CF_Three              Ph-4-OCF₂CHFOCF_Three
H s-Bu CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H s-Bu CF_Three              Ph-4-O (L-45g)
H s-Bu CF_Three              Ph-3,4-Cl₂
H s-Bu CF_Three              Ph (-3-OCF₂O-4-)
H s-Bu CF_Three              Ph (-3-OCF₂CF₂O-4-)
H s-Bu CF_Three             (L-45c) Cl
H s-Bu CF_Three             (L-45c) Br
H s-Bu CF_Three             (L-45c) CF_Three
H s-Bu CF_Three              L-45e
H s-Bu CF_Three              L-45f
H s-Bu CF_Three             (L-46c) Cl
H s-Bu CF_Three             (L-46c) Br
H s-Bu CF_Three             (L-46c) CF_Three
H s-Bu CF_Three              L-46d
H s-Bu CF₂Cl (L-45c) CF_Three
H s-Bu CF₂Br Ph-4-Br
H s-Bu CF₂CF_Three           Ph-4-CF_Three
H s-Bu CF₂CF₂CF_Three        Ph-4-OCF_Three
H s-Bu CF₂OCH_Three         (L-45c) CF_Three
H s-Bu CF₂SCH_Three          Ph-4-Br
H t-Bu CH_Three              Ph-4-Br
H t-Bu CH_Three              Ph-4-CF_Three
H t-Bu CH_Three              Ph-4-OCF_Three
H t-Bu CH_Three             (L-45c) Cl
H t-Bu CH_Three             (L-45c) Br
H t-Bu CH_Three             (L-45c) CF_Three
H t-Bu Et Ph-4-CF_Three
H t-Bu n-Pr Ph-4-OCF_Three
H t-Bu i-Pr (L-45c) CF_Three
H t-Bu c-Pr Ph-4-Br
H t-Bu CHF₂             Ph-4-CF_Three
H t-Bu CF_Three              CF₂O (Ph-4-Cl)
H t-Bu CF_Three              CH = CH (Ph-4-Cl)
H t-Bu CF_Three              CH = CH (Ph-4-OCF_Three)
H t-Bu CF_Three              CH = CH (Ph-3,4-Cl₂)
H t-Bu CF_Three              Ph-4-F
H t-Bu CF_Three              Ph-4-Cl
H t-Bu CF_Three              Ph-4-Br
H t-Bu CF_Three              Ph-4-I
H t-Bu CF_Three              Ph-4-CF_Three
H t-Bu CF_Three              Ph-4-OCHF₂
H t-Bu CF_Three              Ph-4-OCF_Three
H t-Bu CF_Three              Ph-4-OCF₂Br
H t-Bu CF_Three              Ph-4-OCF₂CHF₂
H t-Bu CF_Three              Ph-4-OCF₂CHFCl
H t-Bu CF_Three              Ph-4-OCF₂CHFCF_Three
H t-Bu CF_Three              Ph-4-OCF₂CHFOCF_Three
H t-Bu CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H t-Bu CF_Three              Ph-4-O (L-45g)
H t-Bu CF_Three              Ph-3,4-Cl₂
H t-Bu CF_Three              Ph (-3-OCF₂O-4-)
H t-Bu CF_Three              Ph (-3-OCF₂CF₂O-4-)
H t-Bu CF_Three             (L-45c) Cl
H t-Bu CF_Three             (L-45c) Br
H t-Bu CF_Three             (L-45c) CF_Three
H t-Bu CF_Three              L-45e
H t-Bu CF_Three              L-45f
H t-Bu CF_Three             (L-46c) Cl
H t-Bu CF_Three             (L-46c) Br
H t-Bu CF_Three             (L-46c) CF_Three
H t-Bu CF_Three              L-46d
H t-Bu CF₂Cl Ph-4-OCF_Three
H t-Bu CF₂Br (L-45c) CF_Three
H t-Bu CF₂CF_Three           Ph-4-Br
H t-Bu CF₂CF₂CF_Three        Ph-4-CF_Three
H t-Bu CF₂OCH_Three          Ph-4-OCF_Three
H t-Bu CF₂SCH_Three         (L-45c) CF_Three
H c-Bu CF_Three              Ph-4-Br
H n-Pen CF_Three              Ph-4-CF_Three
H CH₂CH₂Pr-i CF_Three              Ph-4-OCF_Three
H CH₂CH (CH_Three) Et CF_Three             (L-45c) CF_Three
H CH₂Bu-t CF_Three              Ph-4-Br
H CH (CH_Three) Pr-n CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) Pr-n CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) Pr-n CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) Pr-n CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) Pr-n CF_Three              Ph-4-F
H CH (CH_Three) Pr-n CF_Three              Ph-4-Cl
H CH (CH_Three) Pr-n CF_Three              Ph-4-Br
H CH (CH_Three) Pr-n CF_Three              Ph-4-I
H CH (CH_Three) Pr-n CF_Three              Ph-4-CF_Three
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCHF₂
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCF_Three
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) Pr-n CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) Pr-n CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) Pr-n CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) Pr-n CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) Pr-n CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) Pr-n CF_Three             (L-45c) Cl
H CH (CH_Three) Pr-n CF_Three             (L-45c) Br
H CH (CH_Three) Pr-n CF_Three             (L-45c) CF_Three
H CH (CH_Three) Pr-n CF_Three              L-45e
H CH (CH_Three) Pr-n CF_Three              L-45f
H CH (CH_Three) Pr-n CF_Three             (L-46c) Cl
H CH (CH_Three) Pr-n CF_Three             (L-46c) Br
H CH (CH_Three) Pr-n CF_Three             (L-46c) CF_Three
H CH (CH_Three) Pr-n CF_Three              L-46d
H CH (CH_Three) Pr-i CF_Three              Ph-4-CF_Three
H CH (Et)₂                      CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂Et CF_Three              Ph-4-Br
H C (CH_Three)₂Et CF_Three              Ph-4-CF_Three
H C (CH_Three)₂Et CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂Et CF_Three             (L-45c) CF_Three
H c-Pen CF_Three             (L-45c) CF_Three
H n-Hex CF_Three              Ph-4-Br
H CH (CH_Three) Bu-i CF_Three              Ph-4-CF_Three
H C (CH_Three)₂Pr-n CF_Three              Ph-4-Br
H C (CH_Three)₂Pr-n CF_Three              Ph-4-CF_Three
H C (CH_Three)₂Pr-n CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂Pr-n CF_Three             (L-45c) CF_Three
H c-Hex CF_Three              Ph-4-OCF_Three
H CH₂Hex-c CF_Three             (L-45c) CF_Three
H Oct CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂Bu-t CF_Three              Ph-4-CF_Three
 -CH₂CH₂CH₂CH₂-CF_Three              Ph-4-OCF_Three
 -CH₂CH₂CH₂CH₂CH₂-CF_Three             (L-45c) CF_Three
 -CH₂CH₂CH (CH_Three) CH₂CH₂-CF_Three              Ph-4-Br
 -CH₂CH (CH_Three) CH₂CH (CH_Three) CH₂-CF_Three              Ph-4-CF_Three
 -CH₂CH₂CH₂CH₂CH₂CH₂-CF_Three              Ph-4-OCF_Three
H CH₂CH₂F CF_Three             (L-45c) CF_Three
H CH₂CH₂Cl CF_Three              Ph-4-Br
H CH₂CF_Three                       CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂F CF_Three              Ph-4-Br
H CH (CH_Three) CH₂F CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂F (S) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂F CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂F CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂Cl CF_Three              Ph-4-Br
H CH (CH_Three) CH₂Cl CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂Cl CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂Cl CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂Br CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂Br (R) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂Br (S) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂Cl CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂Cl CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂Cl CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂Cl CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂Br CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CHBrCH₂Br CF_Three              Ph-4-Br
H CH₂OCH_Three                      CF_Three              Ph-4-CF_Three
H CH₂CH₂OCH_Three                   CF_Three              Ph-4-OCF_Three
H CH₂CH₂OEt CF_Three             (L-45c) CF_Three
CH₂CH₂OEt CH₂CH₂OEt CF_Three              Ph-4-Br
H CH₂CH₂OC (O) NHEt CF_Three              Ph-4-CF_Three
H CH₂CH₂OPh CF_Three              Ph-4-OCF_Three
H CH₂CH₂O (Ph-2-Cl) CF_Three             (L-45c) CF_Three
H CH₂CH₂O (Ph-3-Cl) CF_Three              Ph-4-Br
H CH₂CH₂O (Ph-4-Cl) CF_Three              Ph-4-CF_Three
H CH₂CH (OH) CH_Three                 CF_Three              Ph-4-OCF_Three
H CH₂CH (OH) Et CF_Three             (L-45c) CF_Three
H CH₂CH (OH) Ph CF_Three              Ph-4-Br
H CH₂CH (OH) CH₂Ph CF_Three              Ph-4-CF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              CH = CH (Ph-4-Cl)
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-Cl
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-Br
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-CF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-OCF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-OCF₂Br
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-OCF₂CHFCF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-4-O (L-45g)
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph-3,4-Cl₂
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph (-3-OCF₂O-4-)
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three             (L-45c) CF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              L-45f
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three             (L-46c) CF_Three
H CH₂C (CH_Three)₂OSi (CH_Three)_Three          CF_Three              L-46d
H CH₂CH (OEt)₂                  CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OH CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OH (R) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OH (S) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OCH_Three               CH_Three              Ph-4-Br
H CH (CH_Three) CH₂OCH_Three               CH_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OCH_Three               CH_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OCH_Three               CH_Three             (L-45c) Cl
H CH (CH_Three) CH₂OCH_Three               CH_Three             (L-45c) Br
H CH (CH_Three) CH₂OCH_Three               CH_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OCH_Three               Et Ph-4-Br
H CH (CH_Three) CH₂OCH_Three               n-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂OCH_Three               i-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂OCH_Three               c-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂OCH_Three               CHF₂             Ph-4-Br
H CH (CH_Three) CH₂OCH_Three               CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂OCH_Three               CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OCH_Three               CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂OCH_Three               CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-F
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-I
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OCH_Three               CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OCH_Three               CF_Three             (L-45c) Cl
H CH (CH_Three) CH₂OCH_Three               CF_Three             (L-45c) Br
H CH (CH_Three) CH₂OCH_Three               CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OCH_Three               CF_Three              L-45e
H CH (CH_Three) CH₂OCH_Three               CF_Three              L-45f
H CH (CH_Three) CH₂OCH_Three               CF_Three             (L-46c) Cl
H CH (CH_Three) CH₂OCH_Three               CF_Three             (L-46c) Br
H CH (CH_Three) CH₂OCH_Three               CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OCH_Three               CF_Three              L-46d
H CH (CH_Three) CH₂OCH_Three               CF₂Cl Ph-4-CF_Three
H CH (CH_Three) CH₂OCH_Three               CF₂Br Ph-4-OCF_Three
H CH (CH_Three) CH₂OCH_Three               CF₂CF_Three          (L-45c) CF_Three
H CH (CH_Three) CH₂OCH_Three               CF₂CF₂CF_Three        Ph-4-Br
H CH (CH_Three) CH₂OCH_Three               CF₂OCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂OCH_Three               CF₂SCH_Three          Ph-4-OCF_Three
H CH (CH_Three) CH₂OEt CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OPr-n CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OBu-i CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OCH₂CH₂OCH_Three        CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OCH₂CH₂SCH_Three        CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OCH₂CH₂SEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OCH₂Ph CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) CH_Three           CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) CF_Three           CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-F
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) NHCH_Three         CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) NHEt CH_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHEt CH_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CH_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHEt CH_Three             (L-45c) Cl
H CH (CH_Three) CH₂OC (O) NHEt CH_Three             (L-45c) Br
H CH (CH_Three) CH₂OC (O) NHEt CH_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHEt Et (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHEt n-Pr Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHEt i-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHEt c-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHEt CHF₂            (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-F
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-I
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHEt CF_Three             (L-45c) Cl
H CH (CH_Three) CH₂OC (O) NHEt CF_Three             (L-45c) Br
H CH (CH_Three) CH₂OC (O) NHEt CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              L-45e
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) NHEt CF_Three             (L-46c) Cl
H CH (CH_Three) CH₂OC (O) NHEt CF_Three             (L-46c) Br
H CH (CH_Three) CH₂OC (O) NHEt CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) NHEt CF₂Cl Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHEt CF₂Br Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF₂CF_Three           Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF₂CF₂CF_Three       (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHEt CF₂OCH_Three          Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHEt CF₂SCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-n CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-i CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPr-c CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) NHBu-t CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂CF_Three      CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂CH₂OCH_Three  CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHCH₂CH₂SCH_Three  CF_Three              Ph-4-CF_Three 
H CH (CH_Three) CH₂OC (O) NHCH₂CH₂CH₂SCH_Three      CF_Three       Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂CH = CH₂   CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂Ph CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) NHCH₂(Ph-4-Cl) CF_Three       Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHCH₂(Ph-4-OCH_Three) CF_Three       Ph-4-CF_Three 
H CH (CH_Three) CH₂OC (O) NHCH₂(L-46a) CF_Three       Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHCH₂(L-47a) CF_Three      (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) NHPh CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) NHPh CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) NHPh CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              L-45f
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OC (O) N (Et)₂        CF_Three              L-46d
H CH (CH_Three) CH₂OC (O) N (Pr-i)₂      CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) N (CH_Three) Ph CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OC (O) (T-16) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OC (O) (T-19) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OC (O) (T-20) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OC (O) (T-21) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OP (O) (OEt)₂        CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              L-45f
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OP (S) (OCH_Three)₂       CF_Three              L-46d
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              L-45f
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂OP (S) (OEt)₂        CF_Three              L-46d
H CH (CH_Three) CH₂OPh CF_Three              Ph-4-Br
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              L-45f
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂O (Ph-4-Cl) CF_Three              L-46d
H CH (CH_Three) CH₂O (Ph-3-CF_Three) CF_Three              Ph-4-CF_Three
H CH (Et) CH₂OH CF_Three              Ph-4-OCF_Three
H CH (Et) CH₂OCH_Three                CF_Three             (L-45c) CF_Three
H CH (Ph) CH₂OH CF_Three              Ph-4-Br
H CH (Ph) CH₂OH (R) CF_Three              Ph-4-Br
H CH (Ph-2-Cl) CH₂OH CF_Three              Ph-4-CF_Three
H CH (Ph-4-Cl) CH₂OH CF_Three              Ph-4-OCF_Three
H CH (Ph-4-Ph) CH₂OH CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OH CF_Three              Ph-4-Br
H CH (CH_Three) CH₂OCH_Three               CH_Three              Ph-4-Br
H C (CH_Three)₂CH₂OCH_Three               CH_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OCH_Three               CH_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OCH_Three               CH_Three             (L-45c) Cl
H C (CH_Three)₂CH₂OCH_Three               CH_Three             (L-45c) Br
H C (CH_Three)₂CH₂OCH_Three               CH_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OCH_Three               Et Ph-4-CF_Three
H C (CH_Three)₂CH₂OCH_Three               n-Pr Ph-4-OCF_Three
H C (CH_Three)₂CH₂OCH_Three               i-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂OCH_Three               c-Pr Ph-4-Br
H C (CH_Three)₂CH₂OCH_Three               CHF₂             Ph-4-CF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂OCH_Three               CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂OCH_Three               CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂OCH_Three               CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-F
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-I
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCHF₂
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFCl
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂OCH_Three               CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂OCH_Three               CF_Three             (L-45c) Cl
H C (CH_Three)₂CH₂OCH_Three               CF_Three             (L-45c) Br
H C (CH_Three)₂CH₂OCH_Three               CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              L-45e
H C (CH_Three)₂CH₂OCH_Three               CF_Three              L-45f
H C (CH_Three)₂CH₂OCH_Three               CF_Three             (L-46c) Cl
H C (CH_Three)₂CH₂OCH_Three               CF_Three             (L-46c) Br
H C (CH_Three)₂CH₂OCH_Three               CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂OCH_Three               CF_Three              L-46d
H C (CH_Three)₂CH₂OCH_Three               CF₂Cl Ph-4-OCF_Three
H C (CH_Three)₂CH₂OCH_Three               CF₂Br (L-45c) CF_Three
H C (CH_Three)₂CH₂OCH_Three               CF₂CF_Three           Ph-4-Br
H C (CH_Three)₂CH₂OCH_Three               CF₂CF₂CF_Three        Ph-4-CF_Three
H C (CH_Three)₂CH₂OCH_Three               CF₂OCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂OCH_Three               CF₂SCH_Three         (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) CH_Three           CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) CF_Three           CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CH_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CH_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CH_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CH_Three             (L-45c) Cl
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CH_Three             (L-45c) Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CH_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         Et Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         n-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         i-Pr Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         c-Pr Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CHF₂             Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-F
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-I
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCHF₂
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHFCl
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three             (L-45c) Cl
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three             (L-45c) Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              L-45e
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              L-45f
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three             (L-46c) Cl
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three             (L-46c) Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF_Three              L-46d
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF₂Cl (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF₂Br Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF₂CF_Three           Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF₂CF₂CF_Three        Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF₂OCH_Three         (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH_Three         CF₂SCH_Three          Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-F
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              L-45f
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHEt CF_Three              L-46d
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              L-45f
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-n CF_Three              L-46d
H C (CH_Three)₂CH₂OC (O) NHPr-i CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHPr-c CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂CF_Three      CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂CH₂OCH_Three  CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHCH₂CH₂SCH_Three  CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂CH₂CH₂SCH_Three      CF_Three       Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂CH = CH₂   CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              L-45f
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂OC (O) NHCH₂Ph CF_Three              L-46d
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              L-45f
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂OC (O) N (CH_Three)₂       CF_Three              L-46d
H C (CH_Three)₂CH₂OP (S) (OCH_Three)₂       CF_Three              Ph-4-OCF_Three
H CH₂CH₂CH₂OH CF_Three             (L-45c) CF_Three
H CH₂CH₂CH₂OCH_Three                CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂OCH_Three            CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂CH₂OEt CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂CH₂OEt CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              L-45f
H CH (CH_Three) CH₂CH₂OEt CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂CH₂OEt CF_Three              L-46d
H CH (CH_Three) CH₂CH₂OPr-n CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂OBu-i CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂CH₂OCH₂CF_Three         CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂OCH₂CH₂OCH_Three     CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂OC (O) NHEt CF_Three              Ph-4-OCF_Three
H CH₂CH₂CH₂CH₂OC (O) NHEt CF_Three             (L-45c) CF_Three
H CH₂CH₂CH₂CH₂OC (O) NHPr-i CF_Three              Ph-4-Br
H CH₂CH₂CH₂CH₂CH₂OC (O) NHEt CF_Three              Ph-4-CF_Three
H T-10 CF_Three              Ph-4-OCF_Three
H M-4a CF_Three             (L-45c) CF_Three
H M-5a CF_Three              Ph-4-Br
H CH₂(M-7a) CF_Three              Ph-4-CF_Three
H CH₂(M-16a) CF_Three              Ph-4-OCF_Three
 -CH₂CH₂OCH₂CH₂-CF_Three             (L-45c) CF_Three
H CH₂SCH_Three                      CF_Three              Ph-4-Br
H CH₂CH₂SCH_Three                   CF_Three              Ph-4-CF_Three
H CH₂CH₂SEt CF_Three              Ph-4-OCF_Three
H CH₂CH₂SPr-i CF_Three             (L-45c) CF_Three
H CH₂CH (CH_Three) SCH_Three               CF_Three              Ph-4-Br
H CH₂CH (CH_Three) SO₂CH_Three             CF_Three              Ph-4-CF_Three
H CH₂CH (CH_Three) SEt CF_Three              Ph-4-OCF_Three
H CH₂CH (CH_Three) SO₂Et CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SH CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CH_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CH_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CH_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CH_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-F
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-I
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CH_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CH_Three             (L-45c) Cl
H CH (CH_Three) CH₂SCH_Three               CH_Three             (L-45c) Br
H CH (CH_Three) CH₂SCH_Three               CH_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CH_Three              L-45e
H CH (CH_Three) CH₂SCH_Three               CH_Three              L-45f
H CH (CH_Three) CH₂SCH_Three               CH_Three             (L-46c) Cl
H CH (CH_Three) CH₂SCH_Three               CH_Three             (L-46c) Br
H CH (CH_Three) CH₂SCH_Three               CH_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CH_Three              L-46d
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               Et Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               Et Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               Et Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               Et Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               Et (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               n-Pr Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               n-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               n-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               n-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               i-Pr Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               i-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               i-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               i-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               c-Pr Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               c-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               c-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               c-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               n-Bu Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂F Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂Cl (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂Br Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CHF₂             Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CHF₂            (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CHF₂             L-45f
H CH (CH_Three) CH₂SCH_Three               CHF₂            (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CHF₂             L-46d
H CH (CH_Three) CH₂SCH_Three               CHFCl Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CHFBr Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              c-Pr
H CH (CH_Three) CH₂SCH_Three               CF_Three              c-Bu
H CH (CH_Three) CH₂SCH_Three               CF_Three              c-Pen
H CH (CH_Three) CH₂SCH_Three               CF_Three              c-Hex
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-1
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-2
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-3
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-4
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-5
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OCH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OEt
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OPr-n
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OPr-i
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OBu-n
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OC (O) (Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OC (O) (Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OC (O) (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂OPh
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-2-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-3-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-4-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-2-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-3-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-4-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-2-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-3-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-4-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-2-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-3-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂O (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂OPh
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-2-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-3-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-4-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-2-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-3-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-4-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-2-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-3-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-4-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-2-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-3-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂O (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂S (Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂S (Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂S (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂SO₂(Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂SO₂(Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂SO₂(Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂N (CH_Three)₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂NH (Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂NH (Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂NH (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CF₂C (O) OEt
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂(L-5a)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂(L-14a)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂(L-24a)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂(L-36a)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂CH₂Ph
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂CH₂(Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂CH₂(Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH₂CH₂(Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-22
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-23
H CH (CH_Three) CH₂SCH_Three               CF_Three              T-24
H CH (CH_Three) CH₂SCH_Three               CF_Three              C (O) OEt
H CH (CH_Three) CH₂SCH_Three               CF_Three              C (O) OBu-t
H CH (CH_Three) CH₂SCH_Three               CF_Three              C (O) OCH₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-2-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-4-F)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-2-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-2-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-2-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-2-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-2-SCH_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-SCH_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-4-SCH_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-2-SO₂CH_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-SO₂CH_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-4-SO₂CH_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3,4-F₂)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-F-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3,4-Br₂)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-F-4-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH (Ph-3-Cl-4-OCF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              CH = CH [Ph (-3-OCF₂O-4-)]
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-I
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-Bu-t
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three(R) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three(S) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCH₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFBr
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CF₂Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CFCl₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CCl_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCH₂CF₂CHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCH (CF_Three)₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CFBrCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OSO₂CH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OSO₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-O (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-O (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-O (Ph-4-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-O (Ph-4-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-O (L-45c) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-O (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-O (L-45e)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-O (L-45e)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-O (L-48b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-SCH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-SO₂CH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-S (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-S (Ph-4-Cl)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-S (Ph-4-Br)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-S (Ph-4-CF_Three)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-S (L-45c) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-S (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-S (L-45e)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-S (L-48b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-NO₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-CN
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,3-F₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,4-F₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,5-F₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,5-F₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-Cl-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-3-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,3-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,5-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,5-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-4-Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-5-Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,4-Br₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,5-Br₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-CH_Three-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-CH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-5-CH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,4- (CH_Three)₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,4- (CH_Three)₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-3-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-CF_Three-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-CF_Three-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-5-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-5-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-Cl-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,5- (CF_Three)₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-OCHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHFCl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHFCl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHFCl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-CH_Three-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three         Ph-3-F-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three         Ph-3-Cl-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three         Ph-3-Br-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-OPh-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-NO₂-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-NO₂-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-5-NO₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3-CN-4-F
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,3,4-F_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,3,5-F_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,4,5-F_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,4,5-F_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,3-F₂-4-CH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2,3-F₂-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,4-F₂-5-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-2-F-3-Cl-5-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-3,5-Cl₂-4-OCH_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              1-Naph
H CH (CH_Three) CH₂SCH_Three               CF_Three              2-Naph
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-1b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-1c) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-1c) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-1c) I
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-1c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-2b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3b) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3c) F
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3c) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3c) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3c) I
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-3c) CN
H CH (CH_Three) CH₂SCH_Three               CF_Three              L-3d
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-4b) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-4b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-4b) CN
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-10b) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-10b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-15b) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-16a) CHF₂
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-16a) CF₂Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-17a) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-21b) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-21b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-21b) I
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-21b) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-22b) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-22b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-23b) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-23b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-23c) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-23c) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-31a) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-31a) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-45c) F
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-45c) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-45c) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-45c) I
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three              L-45e
H CH (CH_Three) CH₂SCH_Three               CF_Three              L-45f
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-46c) F
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-46c) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-46c) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-46c) I
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-46c) OCH₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-46c) OCH (CF_Three)₂
H CH (CH_Three) CH₂SCH_Three               CF_Three              L-46d
H CH (CH_Three) CH₂SCH_Three               CF_Three              L-47a
H CH (CH_Three) CH₂SCH_Three               CF_Three              L-47d
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-48b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-50b) Cl
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-50b) Br
H CH (CH_Three) CH₂SCH_Three               CF_Three             (L-51b) Cl
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂Cl Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂Cl (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Cl L-45f
H CH (CH_Three) CH₂SCH_Three               CF₂Cl (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Cl L-46d
H CH (CH_Three) CH₂SCH_Three               CFCl₂           (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂Br Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂Br (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br L-45f
H CH (CH_Three) CH₂SCH_Three               CF₂Br (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂Br L-46d
H CH (CH_Three) CH₂SCH_Three               CFClBr Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CFBr₂            Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CHF₂          Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three          (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           L-45f
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three          (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF_Three           L-46d
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂Cl (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CFClCF_Three          Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CFClCF₂Cl Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂Br Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CFBrCF_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CHFCF_Three        Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three       (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        L-45f
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three       (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF_Three        L-46d
H CH (CH_Three) CH₂SCH_Three               CF (CF_Three)₂         Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂CF₂CF₂CF_Three     Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               T-1 (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               T-2 Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CH₂OCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂OEt Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂OCH₂CF_Three      (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂OCH (CF_Three)₂     Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          L-45f
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three         (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂OCH_Three          L-46d
H CH (CH_Three) CH₂SCH_Three               CH₂SCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂SO₂CH_Three        Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CH₂SCF_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-Cl
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂Br
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-4-O (L-45g)
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph-3,4-Cl₂
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          L-45f
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three         (L-46c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH_Three          L-46d
H CH (CH_Three) CH₂SCH_Three               CF₂SEt Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂SPr-n Ph-4-CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SPr-i Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SCH₂Ph (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               CF₂SPh Ph-4-Br
H CH (CH_Three) CH₂SCH_Three               CF₂C (O) OEt Ph-4-CF_Three 
H CH (CH_Three) CH₂SCH_Three               CF₂SO₂N (CH_Three)₂    Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH_Three               C (O) OEt (L-45c) CF_Three
H CH (CH_Three) CH₂SCH_Three               C (O) SEt Ph-4-Br
CH_Three       CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-CF_Three
Et CH (CH_Three) CH₂SCH_Three               CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CH_Three              Ph-4-Br
H CH (CH_Three) CH₂S (O) CH_Three            CH_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CH_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CH_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-Cl)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-Br)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-CF_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-OCF_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-Br)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-CF_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-OCF_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-F)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-SCH_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-SO₂CH_Three)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-F
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-2-Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-I
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCH₂CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OSO₂CH_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-OSO₂CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-4-O (L-45e)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-2,4-F₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-F
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-2-F-4-Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-2,4-Cl₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3,5-Cl₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-F
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-2-F-4-Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3,4-Br₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-CH_Three-4-F
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-CF_Three-4-F
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-CF_Three-4-Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-2-F-4-CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-2-Cl-4-CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHFCl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHFCl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHFCl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3-CH_Three-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three         Ph-3-F-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three         Ph-3-Cl-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three         Ph-3-Br-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              Ph-3,4-F₂-5-CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              2-Naph
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-1b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-1c) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-1c) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-1c) CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-2b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-3b) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-3b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-3c) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-3c) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-3c) CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              L-3d
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-4b) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-4b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-10b) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-10b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-15b) CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-16a) CHF₂
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-16a) CF₂Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-17a) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-21b) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-21b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-21b) CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-22b) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-22b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-23b) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-23b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-23c) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-23c) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-31a) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-31a) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-45c) F
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-45c) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-45c) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              L-45e
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              L-45f
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-46c) F
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-46c) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-46c) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              L-46d
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              L-47a
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three              L-47d
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-48b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-50b) Cl
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-50b) Br
H CH (CH_Three) CH₂S (O) CH_Three            CF_Three             (L-51b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-I
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three             (L-45c) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three             (L-45c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              L-45e
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three             (L-46c) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three             (L-46c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH_Three              L-46d
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             Et Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             Et (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             n-Pr Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             n-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             n-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             n-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             i-Pr Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             i-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             i-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             i-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             c-Pr Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             c-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             c-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             c-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             n-Bu (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH₂F Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CH₂Cl Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH₂Br Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂            (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂            (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHF₂             L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CHFCl (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CHFBr Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              c-Pr
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              c-Bu
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              c-Pen
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              c-Hex
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-1
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-2
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-3
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-4
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-5
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OCH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OEt
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OPr-n
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OPr-i
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OBu-n
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OC (O) (Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OC (O) (Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OC (O) (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂OPh
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂OPh
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂S (Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂S (Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂S (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂SO₂(Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂SO₂(Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂SO₂(Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂N (CH_Three)₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂NH (Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂NH (Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂NH (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CF₂C (O) OEt
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂(L-5a)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂(L-14a)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂(L-24a)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂(L-36a)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂CH₂Ph
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂CH₂(Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂CH₂(Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH₂CH₂(Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-22
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-23
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              T-24
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              C (O) OEt
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              C (O) OBu-t
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              C (O) OCH₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-F)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-SCH_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-SCH_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-SCH_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-SO₂CH_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-SO₂CH_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-SO₂CH_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3,4-F₂)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-F-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3,4-Br₂)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-F-4-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-Cl-4-OCF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              CH = CH [Ph (-3-OCF₂O-4-)]
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-I
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-Bu-t
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCH₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFBr
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CFCl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CCl_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCH₂CF₂CHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCH (CF_Three)₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CFBrCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OSO₂CH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-OSO₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-O (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-O (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-O (Ph-4-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-O (Ph-4-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-45c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-O (L-45e)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-45e)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-48b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-SCH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-SO₂CH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-S (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-S (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-S (Ph-4-Br)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-S (Ph-4-CF_Three)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-45c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-45e)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-48b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-NO₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-4-CN
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,3-F₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,4-F₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,5-F₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,5-F₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-Cl-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-3-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,3-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,5-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,5-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,4-Br₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,5-Br₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-CH_Three-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-CH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-CH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,4- (CH_Three)₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,4- (CH_Three)₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-3-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-CF_Three-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-CF_Three-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-5-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-Cl-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,5- (CF_Three)₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHFCl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHFCl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHFCl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-CH_Three-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three         Ph-3-F-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three         Ph-3-Cl-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three         Ph-3-Br-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-OPh-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-NO₂-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-NO₂-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-NO₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3-CN-4-F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,3,4-F_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,3,5-F_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,4,5-F_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,4,5-F_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,3-F₂-4-CH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2,3-F₂-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,4-F₂-5-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-2-F-3-Cl-5-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              Ph-3,5-Cl₂-4-OCH_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              1-Naph
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              2-Naph
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-1b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-1c) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-1c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-1c) I
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-1c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-2b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3c) F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3c) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3c) I
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-3c) CN
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              L-3d
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-4b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-4b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-4b) CN
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-10b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-10b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-15b) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-16a) CHF₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-16a) CF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-17a) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-21b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-21b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-21b) I
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-21b) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-22b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-22b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-23b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-23b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-23c) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-23c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-31a) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-31a) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-45c) F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-45c) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-45c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-45c) I
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              L-45e
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-46c) F
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-46c) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-46c) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-46c) I
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-46c) OCH₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-46c) OCH (CF_Three)₂
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              L-47a
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three              L-47d
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-48b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-50b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-50b) Br
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-51b) Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Cl L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CFCl₂            Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂Br L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CFClBr Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CFBr₂           (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CHF₂          Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three          (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three          (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF_Three           L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂Cl Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CFClCF_Three          Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CFClCF₂Cl (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂Br Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CFBrCF_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CHFCF_Three        Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three       (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three       (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF_Three        L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CF (CF_Three)₂        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂CF₂CF₂CF_Three     Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             T-1 Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             T-2 Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH₂OCH_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH₂OEt Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CH₂OCH₂CF_Three       Ph-4-CF_Three 
H CH (CH_Three) CH₂SO₂CH_Three             CH₂OCH (CF_Three)₂     Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three         (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂OCH_Three          L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CH₂SCH_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CH₂SO₂CH_Three        Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CH₂SCF_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-Cl
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three         (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          L-45f
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three         (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH_Three          L-46d
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SEt Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SPr-n (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SPr-i Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SCH₂Ph Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SPh Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂C (O) OEt (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF₂SO₂N (CH_Three)₂    Ph-4-Br
H CH (CH_Three) CH₂SO₂CH_Three             C (O) OEt Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH_Three             C (O) SEt Ph-4-OCF_Three
H CH (CH_Three) CH₂SEt CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SEt (R) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SEt (S) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SEt CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂SEt CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SEt CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SEt CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SEt CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SEt CF_Three              L-45f
H CH (CH_Three) CH₂SEt CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SEt CF_Three              L-46d
H CH (CH_Three) CH₂S (O) Et CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-Br
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂S (O) Et CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂S (O) Et CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (O) Et CF_Three              L-45f
H CH (CH_Three) CH₂S (O) Et CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂S (O) Et CF_Three              L-46d
H CH (CH_Three) CH₂SO₂Et CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂Et CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂Et CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂Et CF_Three              L-45f
H CH (CH_Three) CH₂SO₂Et CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂Et CF_Three              L-46d
H CH (CH_Three) CH₂SPr-n CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SPr-n CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SPr-n CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SPr-n CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SPr-i CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂Pr-i CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SBu-n CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SBu-i CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SBu-i CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SBu-i CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SBu-i CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SBu-t CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SBu-t CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SBu-t CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SBu-t CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂Bu-t CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SHex-n CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SHex-c CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH₂CF_Three            CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (O) CH₂CF_Three         CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH₂CF_Three          CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SCH₂CH₂OH CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH₂CH₂OCH_Three        CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (O) CH₂CH₂OCH_Three     CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH₂CH₂OCH_Three      CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SCH₂CH₂OEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂S (O) CH₂CH₂OEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂CH₂CH₂OEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH₂CH₂OC (O) CF_Three    CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SCH₂CH₂SCH_Three        CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH₂Si (CH_Three)_Three       CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH₂Si (CH_Three)_Three       CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SCH₂Si (CH_Three)_Three       CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SCH₂Si (CH_Three)_Three       CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SCH₂C (O) CH_Three        CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SCH₂CH₂C (O) OCH_Three    CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (O) CH₂CH₂C (O) OCH_Three CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂CH₂CH₂C (O) OCH_Three  CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH₂C (O) N (Et)₂     CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (O) CH₂C (O) N (Et)₂  CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH₂C (O) N (Et)₂   CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SCH₂(Ph-2,4-Cl₂) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SCH₂CH = CH₂         CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SCH₂C≡CH CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SC (O) CH_Three           CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SSCH_Three              CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SSCH_Three              CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              L-45f
H CH (CH_Three) CH₂SSCH_Three              CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SSCH_Three              CF_Three              L-46d
H CH (CH_Three) CH₂SS (Ph-2-NO₂) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂NH₂             CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH_Three           CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH_Three           CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH_Three           CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH_Three           CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-F
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHEt (S) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂NHEt CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂NHEt CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              L-45f
H CH (CH_Three) CH₂SO₂NHEt CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂NHEt CF_Three              L-46d
H CH (CH_Three) CH₂SO₂NHPr-n CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHPr-i CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHBu-n CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂NHBu-t CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂CH₂Cl CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH₂CH₂OH CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂CH₂OCH_Three    CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH₂CH₂SCH_Three    CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂CH₂S (O) CH_Three      CF_Three         Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH₂CH₂SO₂CH_Three       CF_Three        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) CH₂SCH_Three     CF_Three         Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) CH₂SCH_Three(S, S) CF_Three     Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) CH₂S (O) CH_Three      CF_Three     Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) CH₂S (O) CH_Three(S, S) CF_Three    (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) CH₂SO₂CH_Three       CF_Three     Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) CH₂SO₂CH_Three(S, S) CF_Three     Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHC (CH_Three)₂CH₂SCH_Three     CF_Three         Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) C (O) NH₂     CF_Three        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) C (O) NHCH_Three   CF_Three         Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) C (O) NHEt CF_Three         Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂CH = CH₂     CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH₂C≡CH CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂Ph CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH₂Ph (S) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-2-F) CF_Three         Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-2-Cl) CF_Three        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-2-Br) CF_Three         Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-2-OCH_Three) CF_Three         Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-3-OCH_Three) CF_Three         Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-4-OCH_Three) CF_Three        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-4-SCF_Three) CF_Three         Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-2-NO₂) CF_Three         Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-3-NO₂) CF_Three         Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-4-NO₂) CF_Three        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-3-CN) CF_Three         Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH₂(Ph-4-CN) CF_Three         Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(L-45a) CF_Three         Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(L-46a) CF_Three        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂(L-47a) CF_Three         Ph-4-Br
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) Ph CF_Three         Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) Ph (R) CF_Three         Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂NHCH (CH_Three) Ph (S) CF_Three        (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂NHCH₂CH₂Ph CF_Three         Ph-4-Br
H CH (CH_Three) CH₂SO₂NH (Ph-2-OCH_Three) CF_Three         Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂N (CH_Three)₂         CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂N (CH_Three)₂         CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂N (CH_Three)₂         CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂N (CH_Three)₂         CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂N (CH_Three) Et CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-F
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂(S) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              L-45f
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂SO₂N (Et)₂          CF_Three              L-46d
H CH (CH_Three) CH₂SO₂(T-19) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂(T-20) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂(T-21) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂N (CH_Three) CH₂Ph CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂N (Et) CH₂Ph CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SC (O) NHEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SC (O) N (CH_Three)₂       CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SC (O) N (Et)₂        CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SC (S) NHCH_Three         CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SC (S) NHEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SC (S) N (CH_Three)₂       CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SPh CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SPh CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SPh CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SPh CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (L-21a) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂(L-21a) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (L-45a) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂S (L-45a) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (L-45a) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (L-45a) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (O) (L-45a) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂S (O) (L-45a) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂S (O) (L-45a) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (O) (L-45a) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂SO₂(L-45a) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂(L-45a) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂(L-45a) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂(L-45a) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (L-48a) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂S (O) (L-48a) CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂SO₂(L-48a) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂S (L-48b) CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂S (O) (L-48b) CF_Three              Ph-4-Br
H CH (CH_Three) CH₂SO₂(L-48b) CF_Three              Ph-4-CF_Three
H CH (Et) CH₂SCH_Three                CF_Three             (L-45c) CF_Three
H CH (CH₂SCH_Three)₂                 CF_Three              Ph-4-Br
H CH (Ph) CH₂SCH_Three                CF_Three              Ph-4-CF_Three
H CH (Ph) CH₂S (O) CH_Three             CF_Three              Ph-4-OCF_Three
H CH (Ph) CH₂SO₂CH_Three              CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH (CH_Three) SCH_Three           CF_Three              Ph-4-Br
H CH (CH_Three) CH (CH_Three) SO₂CH_Three         CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH (CH_Three) SEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH (CH_Three) SO₂Et CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CH_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CH_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CH_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-F
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-I
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCHF₂
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CH_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CH_Three             (L-45c) Cl
H C (CH_Three)₂CH₂SCH_Three               CH_Three             (L-45c) Br
H C (CH_Three)₂CH₂SCH_Three               CH_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              L-45e
H C (CH_Three)₂CH₂SCH_Three               CH_Three              L-45f
H C (CH_Three)₂CH₂SCH_Three               CH_Three             (L-46c) Cl
H C (CH_Three)₂CH₂SCH_Three               CH_Three             (L-46c) Br
H C (CH_Three)₂CH₂SCH_Three               CH_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH_Three              L-46d
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               Et Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               Et Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               Et Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               Et Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               Et (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               n-Pr Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               n-Pr Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               n-Pr Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               n-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               i-Pr Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               i-Pr Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               i-Pr Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               i-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               c-Pr Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               c-Pr Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               c-Pr Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               c-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               n-Bu Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CH₂F Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH₂Cl Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CH₂Br (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CHF₂             Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CHF₂            (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             L-45f
H C (CH_Three)₂CH₂SCH_Three               CHF₂            (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CHF₂             L-46d
H C (CH_Three)₂CH₂SCH_Three               CHFCl Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CHFBr Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              c-Pr
H C (CH_Three)₂CH₂SCH_Three               CF_Three              c-Bu
H C (CH_Three)₂CH₂SCH_Three               CF_Three              c-Pen
H C (CH_Three)₂CH₂SCH_Three               CF_Three              c-Hex
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-1
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-2
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-3
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-4
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-5
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OCH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OEt
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OPr-n
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OPr-i
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OBu-n
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OC (O) (Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OC (O) (Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OC (O) (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂OPh
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-2-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-3-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-4-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-2-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-3-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-4-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-2-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-3-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-2-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-3-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂O (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂OPh
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-2-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-3-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-4-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-2-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-3-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-4-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-2-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-3-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-2-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-3-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂O (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂S (Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂S (Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂S (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂SO₂(Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂SO₂(Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂SO₂(Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂N (CH_Three)₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂NH (Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂NH (Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂NH (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CF₂C (O) OEt
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂(L-5a)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂(L-14a)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂(L-24a)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂(L-36a)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂CH₂Ph
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂CH₂(Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂CH₂(Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH₂CH₂(Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-22
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-23
H C (CH_Three)₂CH₂SCH_Three               CF_Three              T-24
H C (CH_Three)₂CH₂SCH_Three               CF_Three              C (O) OEt
H C (CH_Three)₂CH₂SCH_Three               CF_Three              C (O) OBu-t
H C (CH_Three)₂CH₂SCH_Three               CF_Three              C (O) OCH₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-2-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-4-F)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-2-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-2-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-2-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-2-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-2-SCH_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-SCH_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-4-SCH_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-2-SO₂CH_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-SO₂CH_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-4-SO₂CH_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3,4-F₂)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-F-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3,4-Br₂)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-F-4-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH (Ph-3-Cl-4-OCF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              CH = CH [Ph (-3-OCF₂O-4-)]
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-I
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-Bu-t
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCH₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFBr
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CFCl₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CCl_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCH₂CF₂CHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCH (CF_Three)₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CFBrCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OSO₂CH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-OSO₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-O (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-O (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-O (Ph-4-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-O (L-45c) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-O (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-O (L-45e)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-O (L-45e)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-O (L-48b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-SCH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-SO₂CH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-S (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-S (Ph-4-Cl)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-S (Ph-4-Br)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-S (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-S (L-45c) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-S (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-S (L-45e)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-S (L-48b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-NO₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-4-CN
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,3-F₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,4-F₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,5-F₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,5-F₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-Cl-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-3-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,3-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,5-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,5-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-5-Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,4-Br₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,5-Br₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-CH_Three-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-CH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-5-CH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,4- (CH_Three)₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,4- (CH_Three)₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-3-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-CF_Three-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-CF_Three-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-5-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-5-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-Cl-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,5- (CF_Three)₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-OCHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-F-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Cl-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-Br-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-CH_Three-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three         Ph-3-F-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three         Ph-3-Cl-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three         Ph-3-Br-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-OPh-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-NO₂-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-NO₂-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-5-NO₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3-CN-4-F
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,3,4-F_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,3,5-F_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,4,5-F_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,4,5-F_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,3-F₂-4-CH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2,3-F₂-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,4-F₂-5-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-2-F-3-Cl-5-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              Ph-3,5-Cl₂-4-OCH_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              1-Naph
H C (CH_Three)₂CH₂SCH_Three               CF_Three              2-Naph
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-1b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-1c) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-1c) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-1c) I
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-1c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-2b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3c) F
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3c) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3c) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3c) I
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-3c) CN
H C (CH_Three)₂CH₂SCH_Three               CF_Three              L-3d
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-4b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-4b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-4b) CN
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-10b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-10b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-15b) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-16a) CHF₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-16a) CF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-17a) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-21b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-21b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-21b) I
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-21b) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-22b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-22b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-23b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-23b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-23c) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-23c) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-31a) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-31a) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-45c) F
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-45c) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-45c) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-45c) I
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three              L-45e
H C (CH_Three)₂CH₂SCH_Three               CF_Three              L-45f
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-46c) F
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-46c) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-46c) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-46c) I
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-46c) OCH₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-46c) OCH (CF_Three)₂
H C (CH_Three)₂CH₂SCH_Three               CF_Three              L-46d
H C (CH_Three)₂CH₂SCH_Three               CF_Three              L-47a
H C (CH_Three)₂CH₂SCH_Three               CF_Three              L-47d
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-48b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-50b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-50b) Br
H C (CH_Three)₂CH₂SCH_Three               CF_Three             (L-51b) Cl
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl L-45f
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Cl L-46d
H C (CH_Three)₂CH₂SCH_Three               CFCl₂            Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂Br Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂Br (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br L-45f
H C (CH_Three)₂CH₂SCH_Three               CF₂Br (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂Br L-46d
H C (CH_Three)₂CH₂SCH_Three               CFClBr (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CFBr₂            Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂CHF₂          Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three          (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           L-45f
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three          (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF_Three           L-46d
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂Cl Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CFClCF_Three         (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CFClCF₂Cl Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂Br Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CFBrCF_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CHFCF_Three       (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three       (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        L-45f
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three       (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF_Three        L-46d
H C (CH_Three)₂CH₂SCH_Three               CF (CF_Three)₂         Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂CF₂CF₂CF_Three     Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               T-1 Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               T-2 (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH₂OCH_Three          Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CH₂OEt Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH₂OCH₂CF_Three       Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CH₂OCH (CF_Three)₂    (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three         (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          L-45f
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three         (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂OCH_Three          L-46d
H C (CH_Three)₂CH₂SCH_Three               CH₂SCH_Three          Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CH₂SO₂CH_Three        Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CH₂SCF_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-Cl
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three         (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          L-45f
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three         (L-46c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH_Three          L-46d
H C (CH_Three)₂CH₂SCH_Three               CF₂SEt (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SPr-n Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂SPr-i Ph-4-CF_Three 
H C (CH_Three)₂CH₂SCH_Three               CF₂SCH₂Ph Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂SPh (L-45c) CF_Three
H C (CH_Three)₂CH₂SCH_Three               CF₂C (O) OEt Ph-4-Br
H C (CH_Three)₂CH₂SCH_Three               CF₂SO₂N (CH_Three)₂    Ph-4-CF_Three 
H C (CH_Three)₂CH₂SCH_Three               C (O) OEt Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH_Three               C (O) SEt (L-45c) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CH_Three              Ph-4-Br
H C (CH_Three)₂CH₂S (O) CH_Three            CH_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CH_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CH_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-Br)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH₂O (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-Br)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CF₂O (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-F)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-SCH_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-4-SO₂CH_Three)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-F
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-2-Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-I
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three(-) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three(+) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCH₂CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFCl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OSO₂CH_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-OSO₂CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-4-O (L-45e)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-2,4-F₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-F
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-2-F-4-Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-2,4-Cl₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3,5-Cl₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-F
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-2-F-4-Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3,4-Br₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-CH_Three-4-F
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-CF_Three-4-F
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-CF_Three-4-Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-2-F-4-CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-2-Cl-4-CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHFCl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHFCl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHFCl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-F-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Cl-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-Br-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3-CH_Three-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three         Ph-3-F-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three         Ph-3-Cl-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three         Ph-3-Br-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              Ph-3,4-F₂-5-CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              2-Naph
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-1b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-1c) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-1c) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-1c) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-2b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-3b) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-3b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-3c) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-3c) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-3c) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              L-3d
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-4b) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-4b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-10b) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-10b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-15b) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-16a) CHF₂
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-16a) CF₂Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-17a) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-21b) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-21b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-21b) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-22b) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-22b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-23b) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-23b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-23c) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-23c) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-31a) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-31a) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-45c) F
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-45c) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-45c) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              L-45e
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              L-45f
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-46c) F
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-46c) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-46c) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              L-46d
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              L-47a
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three              L-47d
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-48b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-50b) Cl
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-50b) Br
H C (CH_Three)₂CH₂S (O) CH_Three            CF_Three             (L-51b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-I
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three             (L-45c) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three             (L-45c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              L-45e
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three             (L-46c) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three             (L-46c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH_Three              L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             Et Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             Et (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             n-Pr Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             n-Pr Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             n-Pr Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             n-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             i-Pr Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             i-Pr Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             i-Pr Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             i-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             c-Pr Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             c-Pr Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             c-Pr Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             c-Pr (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             n-Bu Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂F (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂Cl Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂Br Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂            (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂            (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHF₂             L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CHFCl Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CHFBr (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              c-Pr
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              c-Bu
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              c-Pen
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              c-Hex
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-1
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-2
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-3
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-4
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-5
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OCH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OEt
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OPr-n
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OPr-i
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OBu-n
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OC (O) (Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OC (O) (Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OC (O) (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂OPh
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-2-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-3-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂O (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂OPh
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-2-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-3-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂O (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂S (Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂S (Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂S (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂SO₂(Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂SO₂(Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂SO₂(Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂N (CH_Three)₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂NH (Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂NH (Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂NH (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CF₂C (O) OEt
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂(L-5a)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂(L-14a)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂(L-24a)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂(L-36a)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂CH₂Ph
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂CH₂(Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂CH₂(Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH₂CH₂(Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-22
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-23
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              T-24
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              C (O) OEt
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              C (O) OBu-t
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              C (O) OCH₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-F)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-SCH_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-SCH_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-SCH_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-2-SO₂CH_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-SO₂CH_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-4-SO₂CH_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3,4-F₂)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-F-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3,4-Br₂)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-F-4-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH (Ph-3-Cl-4-OCF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              CH = CH [Ph (-3-OCF₂O-4-)]
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-I
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-Bu-t
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCH₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFBr
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CFCl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CCl_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCH₂CF₂CHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCH (CF_Three)₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CFBrCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OSO₂CH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-OSO₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-O (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-O (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-O (Ph-4-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-O (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-45c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-O (L-45e)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-45e)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-O (L-48b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-SCH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-SO₂CH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-S (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-S (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-S (Ph-4-Br)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-S (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-45c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-45e)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-S (L-48b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-NO₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-4-CN
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,3-F₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,4-F₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,5-F₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,5-F₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-Cl-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-3-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,3-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,5-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,5-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,4-Br₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,5-Br₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-CH_Three-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-CH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-CH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,4- (CH_Three)₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,4- (CH_Three)₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-3-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-CF_Three-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-CF_Three-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-5-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-Cl-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,5- (CF_Three)₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHFCl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-F-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Cl-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-Br-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-CH_Three-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three         Ph-3-F-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three         Ph-3-Cl-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three         Ph-3-Br-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-OPh-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-NO₂-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-NO₂-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-5-NO₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3-CN-4-F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,3,4-F_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,3,5-F_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,4,5-F_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,4,5-F_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,3-F₂-4-CH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2,3-F₂-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,4-F₂-5-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-2-F-3-Cl-5-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              Ph-3,5-Cl₂-4-OCH_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              1-Naph
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              2-Naph
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-1b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-1c) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-1c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-1c) I
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-1c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-2b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3c) F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3c) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3c) I
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-3c) CN
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              L-3d
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-4b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-4b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-4b) CN
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-10b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-10b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-15b) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-16a) CHF₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-16a) CF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-17a) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-21b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-21b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-21b) I
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-21b) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-22b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-22b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-23b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-23b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-23c) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-23c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-31a) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-31a) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-45c) F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-45c) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-45c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-45c) I
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              L-45e
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-46c) F
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-46c) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-46c) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-46c) I
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-46c) OCH₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-46c) OCH (CF_Three)₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              L-47a
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three              L-47d
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-48b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-50b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-50b) Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF_Three             (L-51b) Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Cl L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CFCl₂            Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂Br L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CFClBr Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CFBr₂            Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CHF₂         (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three          (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three          (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF_Three           L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂Cl Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CFClCF_Three          Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CFClCF₂Cl Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂Br (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CFBrCF_Three          Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CHFCF_Three        Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three       (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three       (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF_Three        L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CF (CF_Three)₂         Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂CF₂CF₂CF_Three    (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             T-1 Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             T-2 Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂OCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂OEt (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂OCH₂CF_Three       Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂OCH (CF_Three)₂     Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three         (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three         (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂OCH_Three          L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂SCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂SO₂CH_Three       (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CH₂SCF_Three          Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-Cl
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three         (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          L-45f
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three         (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH_Three          L-46d
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SEt Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SPr-n Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SPr-i (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SCH₂Ph Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SPh Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂C (O) OEt Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             CF₂SO₂N (CH_Three)₂   (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂CH_Three             C (O) OEt Ph-4-Br
H C (CH_Three)₂CH₂SO₂CH_Three             C (O) SEt Ph-4-CF_Three
H C (CH_Three)₂CH₂SEt CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SEt CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SEt CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SEt CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SEt CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SEt CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SEt CF_Three              L-45f
H C (CH_Three)₂CH₂SEt CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SEt CF_Three              L-46d
H C (CH_Three)₂CH₂S (O) Et CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂S (O) Et CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂S (O) Et CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂S (O) Et CF_Three              L-45f
H C (CH_Three)₂CH₂S (O) Et CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂S (O) Et CF_Three              L-46d
H C (CH_Three)₂CH₂SO₂Et CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂Et CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂Et CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂Et CF_Three              L-45f
H C (CH_Three)₂CH₂SO₂Et CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂Et CF_Three              L-46d
H C (CH_Three)₂CH₂SPr-n CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SPr-n CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SPr-n CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SPr-n CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂S (O) Pr-n CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂Pr-n CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂Pr-n CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂Pr-n CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂Pr-n CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SPr-i CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SPr-i CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SPr-i CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SPr-i CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂S (O) Pr-i CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂Pr-i CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SBu-t CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂S (O) Bu-t CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SCH₂(Ph-4-Cl) CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂NH₂             CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂NHCH_Three           CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂NHEt CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂NHEt CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂NHEt CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂NHEt CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂OCH_Three    CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂OC (O) CH_Three      CF_Three       (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂SCH_Three    CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂S (O) CH_Three       CF_Three        Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂SO₂CH_Three  CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂SEt CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂S (O) Et CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂SO₂Et CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂SPh CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂S (O) Ph CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂NHCH₂CH₂SO₂Ph CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂NHCH₂Ph CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂N (CH_Three)₂         CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂N (CH_Three)₂         CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂N (CH_Three)₂         CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂N (CH_Three)₂         CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-F
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              L-45f
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SO₂N (Et)₂          CF_Three              L-46d
H C (CH_Three)₂CH₂SO₂(T-19) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂SO₂(T-21) CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂SPh CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂S (O) Ph CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂SO₂Ph CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂S (L-45a) CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂S (O) (L-45a) CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂SO₂(L-45a) CF_Three              Ph-4-CF_Three
H CH₂CH₂CH₂SCH_Three                CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂SCH_Three            CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂SCH_Three            CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂SCH_Three            CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂SCH_Three            CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂CH₂S (O) CH_Three         CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂S (O) CH_Three         CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂S (O) CH_Three         CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂S (O) CH_Three         CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂CH₂SO₂CH_Three          CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂SO₂CH_Three          CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂SO₂CH_Three          CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂SO₂CH_Three          CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂CH₂SEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂SEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂SEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂SEt CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂CH₂S (O) Et CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂S (O) Et CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂S (O) Et CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂S (O) Et CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂CH₂SO₂Et CF_Three              Ph-4-Br
H CH (CH_Three) CH₂CH₂SO₂Et CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂CH₂SO₂Et CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH₂SO₂Et CF_Three             (L-45c) CF_Three
H CH (Et) CH₂CH₂SCH_Three             CF_Three             (L-45c) CF_Three
H CH (CH₂OH) CH₂CH₂SCH_Three          CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂CH₂SCH_Three            CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂CH₂SEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (CH₂)_ThreeSCH_Three            CF_Three              Ph-4-Br
H CH (CH_Three) (CH₂)_ThreeSCH_Three            CF_Three              Ph-4-CF_Three
H CH (CH_Three) (CH₂)_ThreeSCH_Three            CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (CH₂)_ThreeSCH_Three            CF_Three             (L-45c) CF_Three
H CH (CH_Three) (CH₂)_ThreeS (O) CH_Three         CF_Three             (L-45c) CF_Three
H CH (CH_Three) (CH₂)_ThreeSO₂CH_Three          CF_Three              Ph-4-Br
H CH (CH_Three) (CH₂)_ThreeSO₂CH_Three          CF_Three              Ph-4-CF_Three
H CH (CH_Three) (CH₂)_ThreeSO₂CH_Three          CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (CH₂)_ThreeSO₂CH_Three          CF_Three             (L-45c) CF_Three
H CH (CH_Three) (CH₂)_ThreeSEt CF_Three              Ph-4-Br
H CH (CH_Three) (CH₂)_ThreeSEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) (CH₂)_ThreeSEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (CH₂)_ThreeSEt CF_Three             (L-45c) CF_Three
H CH (CH_Three) (CH₂)_ThreeS (O) Et CF_Three              Ph-4-Br
H CH (CH_Three) (CH₂)_ThreeSO₂Et CF_Three              Ph-4-Br
H CH (CH_Three) (CH₂)_ThreeSO₂Et CF_Three              Ph-4-CF_Three
H CH (CH_Three) (CH₂)_ThreeSO₂Et CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (CH₂)_ThreeSO₂Et CF_Three             (L-45c) CF_Three
H C (CH_Three)₂(CH₂)_ThreeSCH_Three            CF_Three              Ph-4-CF_Three
H C (CH_Three)₂(CH₂)_ThreeS (O) CH_Three         CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂SO₂CH_Three             CF_Three             (L-45c) CF_Three
H C (CH_Three)₂(CH₂)_ThreeSEt CF_Three              Ph-4-Br
H C (CH_Three)₂(CH₂)_ThreeS (O) Et CF_Three              Ph-4-CF_Three
H C (CH_Three)₂(CH₂)_ThreeSO₂Et CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂(CH₂)_ThreeSO₂NHCH_Three        CF_Three             (L-45c) CF_Three
H C (CH_Three)₂(CH₂)_ThreeSO₂NHEt CF_Three              Ph-4-Br
H C (CH_Three)₂(CH₂)_ThreeSO₂N (CH_Three)₂      CF_Three              Ph-4-CF_Three
H C (CH_Three)₂(CH₂)_ThreeSO₂N (Et)₂       CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂CH₂CH (CH_Three) SCH_Three     CF_Three             (L-45c) CF_Three
H CH (CH_Three) (CH₂)_FourSCH_Three            CF_Three              Ph-4-Br
H CH (CH_Three) (CH₂)_FourSO₂CH_Three          CF_Three              Ph-4-CF_Three
H CH (CH_Three) (CH₂)_FourSEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (CH₂)_FourS (O) Et CF_Three             (L-45c) CF_Three
H CH (CH_Three) (CH₂)_FourSO₂Et CF_Three              Ph-4-Br
H T-6 CF_Three              Ph-4-CF_Three
H T-7 CF_Three              Ph-4-OCF_Three
H T-8 CF_Three             (L-45c) CF_Three
H T-9 CF_Three              Ph-4-Br
H T-11 CF_Three              Ph-4-CF_Three
H T-12 CF_Three              Ph-4-OCF_Three
H T-13 CF_Three             (L-45c) CF_Three
H T-14 CF_Three              Ph-4-Br
H T-15 CF_Three              Ph-4-CF_Three
H M-8a CF_Three              Ph-4-OCF_Three
H M-9a CF_Three             (L-45c) CF_Three
H M-9b CF_Three              Ph-4-Br
H M-9c CF_Three              Ph-4-CF_Three
H M-19a CF_Three              Ph-4-OCF_Three
H CH₂NHC (O) OCH_Three                CF_Three             (L-45c) CF_Three
H CH₂NHC (O) OEt CF_Three              Ph-4-Br
H CH₂NHC (O) OPr-i CF_Three              Ph-4-Br
H CH₂NHC (O) OPr-i CF_Three              Ph-4-CF_Three
H CH₂NHC (O) OPr-i CF_Three              Ph-4-OCF_Three
H CH₂NHC (O) OPr-i CF_Three             (L-45c) CF_Three
H CH₂CH₂NHC (O) CH_Three              CF_Three              Ph-4-CF_Three
H CH₂CH₂NHC (O) N (CH_Three)₂          CF_Three              Ph-4-OCF_Three
H CH₂CH₂NHC (O) Ph CF_Three             (L-45c) CF_Three
H CH₂CH₂N (CH_Three) OCH_Three             CF_Three              Ph-4-Br
H CH (CH_Three) CH₂NHC (O) CH_Three          CF_Three              Ph-4-Br
H CH (CH_Three) CH₂NHC (O) CH_Three          CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂NHC (O) CH_Three          CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂NHC (O) CH_Three          CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂NHC (O) Et CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂NHC (O) OCH_Three         CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂NHC (O) N (CH_Three)₂      CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂NHC (S) NHEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂NHSO₂CH_Three           CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂NHSO₂Et CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂NHSO₂Ph CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂NHSO₂N (CH_Three)₂       CF_Three              Ph-4-Br
H CH (CH_Three) CH₂NHP (S) (OCH_Three)₂      CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂NHP (S) (OEt)₂       CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂N (CH_Three)₂            CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CH_Three              Ph-4-Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CH_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CH_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CH_Three             (L-45c) Cl
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CH_Three             (L-45c) Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CH_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       Et Ph-4-Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       n-Pr Ph-4-CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       i-Pr Ph-4-OCF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       c-Pr (L-45c) CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CHF₂             Ph-4-Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-F
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-Cl
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-I
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCHF₂
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three             (L-45c) Cl
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three             (L-45c) Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              L-45e
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              L-45f
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three             (L-46c) Cl
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three             (L-46c) Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF_Three              L-46d
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF₂Cl Ph-4-CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF₂Br Ph-4-OCF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF₂CF_Three          (L-45c) CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF₂CF₂CF_Three        Ph-4-Br
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF₂OCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH₂N (CH_Three) SO₂CH_Three       CF₂SCH_Three          Ph-4-OCF_Three
H C (CH_Three)₂CH₂NHC (O) CH_Three          CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂NHC (O) Et CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂NHC (O) Pr-c CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂NHC (O) Bu-t CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂NHC (O) CF_Three          CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂NHC (O) Ph CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-F
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-Cl
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              L-45f
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH₂NHC (O) OCH_Three         CF_Three              L-46d
H C (CH_Three)₂CH₂NHC (O) OEt CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH₂NHC (O) OPr-n CF_Three              Ph-4-OCF_Three
H CH₂CH₂CH₂NHC (O) OCH_Three          CF_Three             (L-45c) CF_Three
H CH₂CH₂CH₂NHC (O) OBu-t CF_Three              Ph-4-Br
H CH₂CH₂CH₂N (CH_Three)₂             CF_Three              Ph-4-CF_Three
H CH₂CH₂CH₂N (CH_Three) OCH_Three          CF_Three              Ph-4-OCF_Three
H (M-22a) CHO CF_Three             (L-45c) CF_Three
H (M-22a) C (O) CH_Three                CF_Three              Ph-4-Br
H (M-22a) C (O) OCH_Three               CF_Three              Ph-4-CF_Three
H (M-22a) C (O) OEt CF_Three              Ph-4-OCF_Three
H (M-22a) C (O) SCH_Three               CF_Three             (L-45c) CF_Three
H CH₂Si (CH_Three)_Three                  CF_Three              Ph-4-Br
H C (CH_Three)₂CHO CF_Three              Ph-4-CF_Three
H CH (CH_Three) C (O) CH_Three               CF_Three              Ph-4-OCF_Three
H CH (CHO) CH₂SO₂CH_Three             CF_Three             (L-45c) CF_Three
H C (CH_Three) (CHO) CH₂SO₂CH_Three         CF_Three              Ph-4-Br
H C (CH_Three) (CHO) CH₂SO₂Et CF_Three              Ph-4-CF_Three
H CH₂CH = NOCH_Three                  CF_Three              Ph-4-OCF_Three
H CH₂C (Ph) = NOCH_Three               CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH = NOCH_Three              CH_Three              Ph-4-Br
H CH (CH_Three) CH = NOCH_Three              CH_Three              Ph-4-CF_Three
H CH (CH_Three) CH = NOCH_Three              CH_Three              Ph-4-OCF_Three
H CH (CH_Three) CH = NOCH_Three              CH_Three             (L-45c) Cl
H CH (CH_Three) CH = NOCH_Three              CH_Three             (L-45c) Br
H CH (CH_Three) CH = NOCH_Three              CH_Three             (L-45c) CF_Three
H CH (CH_Three) CH = NOCH_Three              Et Ph-4-Br
H CH (CH_Three) CH = NOCH_Three              n-Pr Ph-4-CF_Three
H CH (CH_Three) CH = NOCH_Three              i-Pr Ph-4-OCF_Three
H CH (CH_Three) CH = NOCH_Three              c-Pr (L-45c) CF_Three
H CH (CH_Three) CH = NOCH_Three              CHF₂             Ph-4-Br
H CH (CH_Three) CH = NOCH_Three              CF_Three              CF₂O (Ph-4-Cl)
H CH (CH_Three) CH = NOCH_Three              CF_Three              CH = CH (Ph-4-Cl)
H CH (CH_Three) CH = NOCH_Three              CF_Three              CH = CH (Ph-4-Br)
H CH (CH_Three) CH = NOCH_Three              CF_Three              CH = CH (Ph-4-CF_Three)
H CH (CH_Three) CH = NOCH_Three              CF_Three              CH = CH (Ph-4-OCF_Three)
H CH (CH_Three) CH = NOCH_Three              CF_Three              CH = CH (Ph-3,4-Cl₂)
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-F
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-Cl
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-Br
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-I
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCHF₂
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCF₂Br
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHF₂
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHFCl
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHFCF_Three
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHFOCF_Three
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-4-O (L-45g)
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-3,4-F₂
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-3-F-4-Cl
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph-3,4-Cl₂
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph (-3-OCF₂O-4-)
H CH (CH_Three) CH = NOCH_Three              CF_Three              Ph (-3-OCF₂CF₂O-4-)
H CH (CH_Three) CH = NOCH_Three              CF_Three             (L-45c) Cl
H CH (CH_Three) CH = NOCH_Three              CF_Three             (L-45c) Br
H CH (CH_Three) CH = NOCH_Three              CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH = NOCH_Three              CF_Three              L-45e
H CH (CH_Three) CH = NOCH_Three              CF_Three              L-45f
H CH (CH_Three) CH = NOCH_Three              CF_Three             (L-46c) Cl
H CH (CH_Three) CH = NOCH_Three              CF_Three             (L-46c) Br
H CH (CH_Three) CH = NOCH_Three              CF_Three             (L-46c) CF_Three
H CH (CH_Three) CH = NOCH_Three              CF_Three              L-46d
H CH (CH_Three) CH = NOCH_Three              CF₂Cl Ph-4-CF_Three
H CH (CH_Three) CH = NOCH_Three              CF₂Br Ph-4-OCF_Three
H CH (CH_Three) CH = NOCH_Three              CF₂CF_Three          (L-45c) CF_Three
H CH (CH_Three) CH = NOCH_Three              CF₂CF₂CF_Three        Ph-4-Br
H CH (CH_Three) CH = NOCH_Three              CF₂OCH_Three          Ph-4-CF_Three
H CH (CH_Three) CH = NOCH_Three              CF₂SCH_Three          Ph-4-OCF_Three
H CH (CH_Three) CH = NOPr-n CF_Three              Ph-4-Br
H CH (CH_Three) CH = NOPr-n CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH = NOPr-n CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH = NOPr-n CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH = NOCH₂Pr-c CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH = NOCH₂CH₂OEt CF_Three              Ph-4-Br
H CH (CH_Three) CH = NOCH₂CH₂SEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH = NOCH₂CH = CH₂        CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH = NOCH₂Ph CF_Three             (L-45c) CF_Three
H CH (CH_Three) C (CH_Three) = NOCH_Three          CF_Three              Ph-4-Br
H C (CH_Three)₂CH = NOH CF_Three              Ph-4-Br
H C (CH_Three)₂CH = NOH CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH = NOH CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH = NOH CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              CF₂O (Ph-4-Cl)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              CH = CH (Ph-4-Br)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              CH = CH (Ph-4-CF_Three)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              CH = CH (Ph-4-OCF_Three)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              CH = CH (Ph-3,4-Cl₂)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-F
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-Cl
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-Br
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHF₂
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-3,4-F₂
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-3-F-4-Cl
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH = NOCH_Three              CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH = NOCH_Three              CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              L-45f
H C (CH_Three)₂CH = NOCH_Three              CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH = NOCH_Three              CF_Three              L-46d
H C (CH_Three)₂CH = NOEt CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH = NOCH₂C (O) OBu-t CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH = NOCH₂C (O) N (Et)₂    CF_Three             (L-45c) CF_Three
H C (CH_Three) (CH₂SO₂CH_Three) CH = NOH CF_Three              Ph-4-Br
H C (CH_Three) (CH₂SO₂Et) CH = NOH CF_Three              Ph-4-CF_Three
H CH₂CH₂CH = NOCH_Three               CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂CH = NOCH_Three           CF_Three             (L-45c) CF_Three
H CH₂CH₂CH₂CH = NOEt CF_Three              Ph-4-Br
H CH₂C (O) OEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) C (O) OCH_Three              CF_Three              Ph-4-OCF_Three
H CH (CH_Three) C (O) OEt CF_Three             (L-45c) CF_Three
H CH₂CH₂C (O) OEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂C (O) OEt CF_Three              Ph-4-CF_Three
H CH (CH_Three) C (O) NHEt CF_Three              Ph-4-OCF_Three
H CH (CH_Three) C (O) NHPr-n CF_Three             (L-45c) CF_Three
H CH (CH_Three) C (O) NHBu-n CF_Three              Ph-4-Br
H CH (CH_Three) C (O) NHCH₂Ph CF_Three              Ph-4-CF_Three
H CH (CH_Three) C (O) N (CH_Three)₂           CF_Three              Ph-4-OCF_Three
H CH (CH_Three) C (O) N (Et)₂            CF_Three             (L-45c) CF_Three
H CH (CH_Three) C (O) N (Pr-n)₂          CF_Three              Ph-4-Br
H CH (CH_Three) C (O) (T-16) CF_Three              Ph-4-CF_Three
H CH (CH_Three) C (O) (T-17) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) C (O) (T-18) CF_Three             (L-45c) CF_Three
H CH (CH_Three) C (O) (T-19) CF_Three              Ph-4-Br
H CH (CH_Three) C (O) (T-20) CF_Three              Ph-4-CF_Three
H CH (CH_Three) C (O) (T-21) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂C (O) NHCH_Three          CF_Three             (L-45c) CF_Three
H CH (CH_Three) CH₂C (O) NHEt CF_Three              Ph-4-Br
H CH (CH_Three) CH₂C (O) N (CH_Three)₂        CF_Three              Ph-4-CF_Three
H CH (CH_Three) CH₂C (O) N (Et)₂         CF_Three              Ph-4-OCF_Three
H CH (CH_Three) CH₂C (O) N (CH_Three) Ph CF_Three             (L-45c) CF_Three
H CH (CH_Three) CN CF_Three              Ph-4-Br
H C (CH_Three)₂CN CF_Three              Ph-4-CF_Three
H CH₂CH = CH₂                    CF_Three              Ph-4-OCF_Three
CH₂CH = CH₂ CH₂CH = CH₂                    CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-Cl
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-Br
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-CF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂CH = CH₂                CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂CH = CH₂                CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂CH = CH₂                CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂CH = CH₂                CF_Three             (L-45c) CF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              L-45f
H C (CH_Three)₂CH = CH₂                CF_Three             (L-46c) CF_Three
H C (CH_Three)₂CH = CH₂                CF_Three              L-46d
H C (CH_Three)₂CH = CHC (O) NHEt CF_Three              Ph-4-Br
H C (CH_Three)₂CH = CHPh (E) CF_Three              Ph-4-CF_Three
H CH₂C≡CH CF_Three              Ph-4-OCF_Three
CH_Three       CH₂C≡CH CF_Three              Ph-4-Br
CH_Three       CH₂C≡CH CF_Three              Ph-4-CF_Three
CH_Three       CH₂C≡CH CF_Three              Ph-4-OCF_Three
CH_Three       CH₂C≡CH CF_Three             (L-45c) CF_Three
H C (CH_Three)₂C≡CH CF_Three              CH = CH (Ph-4-Cl)
H C (CH_Three)₂C≡CH CF_Three              Ph-4-Cl
H C (CH_Three)₂C≡CH CF_Three              Ph-4-Br
H C (CH_Three)₂C≡CH CF_Three              Ph-4-CF_Three
H C (CH_Three)₂C≡CH CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂C≡CH CF_Three              Ph-4-OCF₂Br
H C (CH_Three)₂C≡CH CF_Three              Ph-4-OCF₂CHFCF_Three
H C (CH_Three)₂C≡CH CF_Three              Ph-4-OCF₂CHFOCF_Three
H C (CH_Three)₂C≡CH CF_Three              Ph-4-OCF₂CHFOCF₂CF₂CF_Three
H C (CH_Three)₂C≡CH CF_Three              Ph-4-O (L-45g)
H C (CH_Three)₂C≡CH CF_Three              Ph-3,4-Cl₂
H C (CH_Three)₂C≡CH CF_Three              Ph (-3-OCF₂O-4-)
H C (CH_Three)₂C≡CH CF_Three              Ph (-3-OCF₂CF₂O-4-)
H C (CH_Three)₂C≡CH CF_Three             (L-45c) CF_Three
H C (CH_Three)₂C≡CH CF_Three              L-45f
H C (CH_Three)₂C≡CH CF_Three             (L-46c) CF_Three
H C (CH_Three)₂C≡CH CF_Three              L-46d
H C (CH_Three)₂C≡CPh CF_Three             (L-45c) CF_Three
H C (CH_Three)₂C≡C (Ph-4-CH_Three) CF_Three              Ph-4-Br
H C (CH_Three)₂C≡C (Ph-4-CF_Three) CF_Three              Ph-4-CF_Three
H C (CH_Three)₂C≡C (Ph-4-OCH_Three) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂C≡C (Ph-4-OCF_Three) CF_Three             (L-45c) CF_Three
H C (CH_Three)₂C≡C (Ph-2,4-F₂) CF_Three              Ph-4-Br
H C (CH_Three)₂C≡C (Ph-2,4-Cl₂) CF_Three              Ph-4-CF_Three
H C (CH_Three)₂C≡C (Ph-2,6-Cl₂) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂C≡C (1-Naph) CF_Three             (L-45c) CF_Three
H C (CH_Three)₂C≡C (L-3a) CF_Three              Ph-4-Br
H C (CH_Three)₂C≡C (L-4a) CF_Three              Ph-4-CF_Three
H C (CH_Three)₂C≡C (L-45a) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂C≡C (L-45g) CF_Three             (L-45c) CF_Three
H C (CH_Three)₂C≡C (L-46a) CF_Three              Ph-4-Br
H CH₂Ph CF_Three              Ph-4-CF_Three
CH_Three       CH₂Ph CF_Three              Ph-4-OCF_Three
Et CH₂Ph CF_Three             (L-45c) CF_Three
H CH₂(Ph-2-F) CF_Three              Ph-4-Br
CH_Three       CH₂(Ph-2-F) CF_Three              Ph-4-CF_Three
H CH₂(Ph-2-Cl) CF_Three              Ph-4-OCF_Three
H CH₂(Ph-3-Cl) CF_Three             (L-45c) CF_Three
CH_Three       CH₂(Ph-3-Cl) CF_Three              Ph-4-Br
H CH₂(Ph-4-Cl) CF_Three              Ph-4-CF_Three
H CH₂(Ph-2-CH_Three) CF_Three              Ph-4-OCF_Three
H CH₂(Ph-3-CH_Three) CF_Three             (L-45c) CF_Three
H CH₂(Ph-4-CH_Three) CF_Three              Ph-4-Br
H CH₂(Ph-2-CF_Three) CF_Three              Ph-4-CF_Three
H CH₂(Ph-2-OCH_Three) CF_Three              Ph-4-OCF_Three
H CH₂(Ph-3-OCH_Three) CF_Three             (L-45c) CF_Three
H CH₂(Ph-4-OCH_Three) CF_Three              Ph-4-Br
H CH₂(Ph-4-OCF_Three) CF_Three              Ph-4-CF_Three
H CH₂(Ph-2,3-Cl₂) CF_Three              Ph-4-OCF_Three
H CH₂(Ph-2,4-Cl₂) CF_Three             (L-45c) CF_Three
H CH₂(Ph-3,4-Cl₂) CF_Three              Ph-4-Br
H CH₂(L-45a) CF_Three              Ph-4-CF_Three
H CH₂(L-46a) CF_Three              Ph-4-OCF_Three
H CH₂(L-47a) CF_Three             (L-45c) CF_Three
H CH (CH_Three) Ph CF_Three              Ph-4-Br
H CH (CH_Three) Ph (R) CF_Three              Ph-4-CF_Three
H CH (CH_Three) Ph (S) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (Ph-2-Cl) CF_Three             (L-45c) CF_Three
H CH (CH_Three) (Ph-3-Cl) CF_Three              Ph-4-Br
H CH (CH_Three) (Ph-4-Cl) CF_Three              Ph-4-CF_Three
H CH (CH_Three) (L-1a) CF_Three              Ph-4-OCF_Three
H CH (CH_Three) (L-3a) CF_Three             (L-45c) CF_Three
H CH (CH_Three) (L-45a) CF_Three              Ph-4-Br
H C (CH_Three)₂Ph CF_Three              Ph-4-CF_Three
H C (CH_Three)₂(Ph-3-Cl) CF_Three              Ph-4-OCF_Three
H C (CH_Three)₂(Ph-4-Cl) CF_Three             (L-45c) CF_Three
H CH₂CH₂Ph CF_Three              Ph-4-Br
H CH₂CH₂(Ph-2-Cl) CF_Three              Ph-4-CF_Three
H CH₂CH₂(Ph-3-Cl) CF_Three              Ph-4-OCF_Three
H CH₂CH₂(Ph-4-Cl) CF_Three             (L-45c) CF_Three
H CH₂CH₂(L-46a) CF_Three              Ph-4-Br
H C (CH_Three)₂CH₂Ph CF_Three              Ph-4-CF_Three
H CH₂CH₂CH₂Ph CF_Three              Ph-4-OCF_Three
H OCH_Three                         CF_Three             (L-45c) CF_Three
H OPr-n CF_Three              Ph-4-Br
H OCH₂CH = CHCl CF_Three              Ph-4-CF_Three
H OCH₂Ph CF_Three              Ph-4-OCF_Three
H NHCHO CF_Three             (L-45c) CF_Three
H NHC (O) CH_Three                    CF_Three              Ph-4-Br
H NHC (O) Ph CF_Three              Ph-4-CF_Three
H NHC (O) OCH_Three                   CF_Three              Ph-4-OCF_Three
H NHC (O) OPh CF_Three             (L-45c) CF_Three
H NHC (O) OCH₂Ph CF_Three              Ph-4-Br
H N (CH_Three)₂                      CF_Three              Ph-4-CF_Three
H N (CH_Three) CHO CF_Three              Ph-4-OCF_Three
H N (CH_Three) C (O) CH_Three                CF_Three             (L-45c) CF_Three
H N (CH_Three) C (O) OCH_Three               CF_Three              Ph-4-Br
―――――――――――――――――――――――――――――――――――――――
Table 3
  In the table, substituent (X)_mAnd (Y)_nThe numbers representing the substitution positions correspond to the positions of the numbers described in the following structural formulas, and the symbol “-” represents no substitution.

―――――――――――――――――――――――――――――――――――――――
(X) _m (Y) _n R ⁴ R ⁵ R ⁶
―――――――――――――――――――――――――――――――――――――――
− 2-CH ₃ CF ₃ Ph-4-Br H
5-F 2-CH ₃ CF ₃ Ph-4-CF ₃ H
6-F 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3,4-F ₂ 2-CH ₃ CF ₃ Ph-4-Br H
3,4-F ₂ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3,4-F ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3,4-F ₂ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3,6-F ₂ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
4,5-F ₂ 2-CH ₃ CF ₃ Ph-4-Br H
4-Cl 2-CH ₃ CF ₃ Ph-4-CF ₃ H
5-Cl 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
6-Cl 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-Cl-4-F 2-CH ₃ CF ₃ Ph-4-Br H
3-Cl-4-F 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-Cl-4-F 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-Cl-4-F 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3,4-Cl ₂ 2-CH ₃ CH ₃ Ph-4-Br H
3,4-Cl ₂ 2-CH ₃ CH ₃ Ph-4-CF ₃ H
3,4-Cl ₂ 2-CH ₃ CH ₃ Ph-4-OCF ₃ H
3,4-Cl ₂ 2-CH ₃ CH ₃ (L-45c) Cl H
3,4-Cl ₂ 2-CH ₃ CH ₃ (L-45c) Br H
3,4-Cl ₂ 2-CH ₃ CH ₃ (L-45c) CF ₃ H
3,4-Cl ₂ 2-CH ₃ CH ₃ (L-45c) CF ₃ H
3,4-Cl ₂ 2-CH ₃ n-Pr Ph-4-Br H
3,4-Cl ₂ 2-CH ₃ i-Pr Ph-4-CF ₃ H
3,4-Cl ₂ 2-CH ₃ c-Pr Ph-4-OCF ₃ H
3,4-Cl ₂ 2-CH ₃ CHF ₂ (L-45c) CF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) H
3,4-Cl ₂ 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) H
3,4-Cl ₂ 2-CH ₃ CF ₃ CH = CH (Ph-4-Br) H
3,4-Cl ₂ 2-CH ₃ CF ₃ CH = CH (Ph-4-CF ₃ ) H
3,4-Cl ₂ 2-CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) H
3,4-Cl ₂ 2-CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-FH
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-Cl H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-Br H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-IH
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCHF ₂ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCl H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-4-O (L-45g) H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-3,4-F ₂ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-3-F-4-Cl H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) H
3,4-Cl ₂ 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) H
3,4-Cl ₂ 2-CH ₃ CF ₃ (L-45c) Cl H
3,4-Cl ₂ 2-CH ₃ CF ₃ (L-45c) Br H
3,4-Cl ₂ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ L-45e H
3,4-Cl ₂ 2-CH ₃ CF ₃ L-45f H
3,4-Cl ₂ 2-CH ₃ CF ₃ (L-46c) Cl H
3,4-Cl ₂ 2-CH ₃ CF ₃ (L-46c) Br H
3,4-Cl ₂ 2-CH ₃ CF ₃ (L-46c) CF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₃ L-46d H
3,4-Cl ₂ 2-CH ₃ CF ₂ Cl Ph-4-Br H
3,4-Cl ₂ 2-CH ₃ CF ₂ Br Ph-4-CF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₂ CF ₃ Ph-4-OCF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₂ CF ₂ CF ₃ (L-45c) CF ₃ H
3,4-Cl ₂ 2-CH ₃ CF ₂ OCH ₃ Ph-4-Br H
3,4-Cl ₂ 2-CH ₃ CF ₂ SCH ₃ Ph-4-CF ₃ H
3,5-Cl ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3,6-Cl ₂ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
5,6-Cl ₂ 2-CH ₃ CF ₃ Ph-4-Br H
6-Br 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3,4-Br ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3,6-Br ₂ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
5,6-Br ₂ 2-CH ₃ CF ₃ Ph-4-Br H
3-I 2-I CF ₃ Ph-4-CF ₃ H
3-I 2-CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) CH ₃
3-I 2-CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) C (O) CH ₃
3-I 2-CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) C (O) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Br) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Br) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Br) C (O) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-Br) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-CF ₃ ) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-CF ₃ ) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-CF ₃ ) C (O) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-CF ₃ ) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) C (O) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) C (O) CH ₃
3-I 2-CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-F CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-F CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-FC (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-F Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-Cl CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Cl CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Cl C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Cl Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br Et
3-I 2-CH ₃ CF ₃ Ph-4-Br n-Pr
3-I 2-CH ₃ CF ₃ Ph-4-Br i-Pr
3-I 2-CH ₃ CF ₃ Ph-4-Br n-Bu
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ CF ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ OEt
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ SCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ CH = CH ₂
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ CH = CF ₂
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ CH = CCl ₂
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ CF = CF ₂
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ CCl = CCl ₂
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ C≡CH
3-I 2-CH ₃ CF ₃ Ph-4-Br CH ₂ Ph
3-I 2-CH ₃ CF ₃ Ph-4-Br C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br C (O) Bu-t
3-I 2-CH ₃ CF ₃ Ph-4-Br C (O) SCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br C (S) SEt
3-I 2-CH ₃ CF ₃ Ph-4-Br Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-Br Si (CH ₃ ) ₂ Bu-t
3-I 2-CH ₃ CF ₃ Ph-4-Br Si (CH ₃ ) ₂ Ph
3-I 2-CH ₃ CF ₃ Ph-4-I CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-I CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-IC (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-I Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ Et
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ n-Pr
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ i-Pr
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ n-Bu
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ CF ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ OEt
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ SCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ CH = CH ₂
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ CH = CF ₂
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ CH = CCl ₂
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ CF = CF ₂
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ CCl = CCl ₂
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ C≡CH
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ CH ₂ Ph
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ C (O) Bu-t
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ C (O) SCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ C (S) SEt
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ Si (CH ₃ ) ₂ Bu-t
3-I 2-CH ₃ CF ₃ Ph-4-CF ₃ Si (CH ₃ ) ₂ Ph
3-I 2-CH ₃ CF ₃ Ph-4-CHF ₂ CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CHF ₂ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CHF ₂ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-CHF ₂ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ Et
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ n-Pr
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ i-Pr
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ n-Bu
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ CF ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ OEt
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ SCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ CH = CH ₂
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ CH = CF ₂
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ CH = CCl ₂
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ CF = CF ₂
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ CCl = CCl ₂
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ C≡CH
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ CH ₂ Ph
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ C (O) Bu-t
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ C (O) SCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ C (S) SEt
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ Si (CH ₃ ) ₂ Bu-t
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ Si (CH ₃ ) ₂ Ph
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCl CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCl CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCl C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCl Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-4-O (L-45g) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-O (L-45g) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-4-O (L-45g) C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-4-O (L-45g) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-F ₂ CH ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-F ₂ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-F ₂ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-F ₂ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-3-F-4-Cl CH ₃
3-I 2-CH ₃ CF ₃ Ph-3-F-4-Cl CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-3-F-4-Cl C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-3-F-4-Cl Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ CH ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) CH ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) CH ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) C (O) CH ₃
3-I 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ (L-45c) Cl CH ₃
3-I 2-CH ₃ CF ₃ (L-45c) Cl CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ (L-45c) Cl C (O) CH ₃
3-I 2-CH ₃ CF ₃ (L-45c) Cl Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ (L-45c) Br CH ₃
3-I 2-CH ₃ CF ₃ (L-45c) Br CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ (L-45c) Br C (O) CH ₃
3-I 2-CH ₃ CF ₃ (L-45c) Br Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ Et
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ n-Pr
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ i-Pr
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ n-Bu
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ CF ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ OEt
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ SCH ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ CH = CH ₂
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ CH = CF ₂
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ CH = CCl ₂
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ CF = CF ₂
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ CCl = CCl ₂
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ C≡CH
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ CH ₂ Ph
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ C (O) CH ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ C (O) Bu-t
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ C (O) SCH ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ C (S) SEt
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ Si (CH ₃ ) ₂ Bu-t
3-I 2-CH ₃ CF ₃ (L-45c) CF ₃ Si (CH ₃ ) ₂ Ph
3-I 2-CH ₃ CF ₃ L-45e CH ₃
3-I 2-CH ₃ CF ₃ L-45e CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ L-45e C (O) CH ₃
3-I 2-CH ₃ CF ₃ L-45e Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ L-45f CH ₃
3-I 2-CH ₃ CF ₃ L-45f CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ L-45f C (O) CH ₃
3-I 2-CH ₃ CF ₃ L-45f Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ (L-46c) Cl CH ₃
3-I 2-CH ₃ CF ₃ (L-46c) Cl CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ (L-46c) Cl C (O) CH ₃
3-I 2-CH ₃ CF ₃ (L-46c) Cl Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ (L-46c) Br CH ₃
3-I 2-CH ₃ CF ₃ (L-46c) Br CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ (L-46c) Br C (O) CH ₃
3-I 2-CH ₃ CF ₃ (L-46c) Br Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ (L-46c) CF ₃ CH ₃
3-I 2-CH ₃ CF ₃ (L-46c) CF ₃ CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ (L-46c) CF ₃ C (O) CH ₃
3-I 2-CH ₃ CF ₃ (L-46c) CF ₃ Si (CH ₃ ) ₃
3-I 2-CH ₃ CF ₃ L-46d CH ₃
3-I 2-CH ₃ CF ₃ L-46d CH ₂ OCH ₃
3-I 2-CH ₃ CF ₃ L-46d C (O) CH ₃
3-I 2-CH ₃ CF ₃ L-46d Si (CH ₃ ) ₃
3-I 2-Pr-n CF ₃ Ph-4-OCF ₃ H
3-I 2-Pr-i CF ₃ (L-45c) CF ₃ H
3-I 2-Bu-n CF ₃ Ph-4-Br H
3-I 2-CF ₃ CF ₃ Ph-4-CF ₃ H
3-I 2-CF ₂ CF ₃ CF ₃ Ph-4-OCF ₃ H
3-I 2-CH ₂ OH CF ₃ Ph-4-Br H
3-I 2-CH ₂ OH CF ₃ Ph-4-CF ₃ H
3-I 2-CH ₂ OH CF ₃ Ph-4-OCF ₃ H
3-I 2-CH ₂ OH CF ₃ (L-45c) CF ₃ H
3-I 2-CH ₂ OCH ₃ CF ₃ (L-45c) CF ₃ H
3-I 2-CH ₂ SCH ₃ CF ₃ Ph-4-Br H
3-I 2-OCH ₃ CF ₃ Ph-4-Br H
3-I 2-OCH ₃ CF ₃ Ph-4-CF ₃ H
3-I 2-OCH ₃ CF ₃ Ph-4-OCF ₃ H
3-I 2-OCH ₃ CF ₃ (L-45c) CF ₃ H
3-I 2-OEt CF ₃ Ph-4-CF ₃ H
3-I 2-OPr-i CF ₃ Ph-4-OCF ₃ H
3-I 2-OCF ₃ CF ₃ (L-45c) CF ₃ H
3-I 2-OPh CF ₃ Ph-4-Br H
3-I 2-SCH ₃ CF ₃ Ph-4-Br H
3-I 2-SCH ₃ CF ₃ Ph-4-CF ₃ H
3-I 2-SCH ₃ CF ₃ Ph-4-OCF ₃ H
3-I 2-SCH ₃ CF ₃ (L-45c) CF ₃ H
3-I 2-SO ₂ CH ₃ CF ₃ Ph-4-CF ₃ H
3-I 2-SEt CF ₃ Ph-4-OCF ₃ H
3-I 2-SPr-i CF ₃ (L-45c) CF ₃ H
3-I 2-SCHF ₂ CF ₃ Ph-4-Br H
3-I 2-N (CH ₃ ) ₂ CF ₃ Ph-4-CF ₃ H
3-I 2-CN CF ₃ Ph-4-OCF ₃ H
3-I 2-Ph CF ₃ (L-45c) CF ₃ H
3-I 2- (L-14a) CF ₃ Ph-4-Br H
3-I 2- (L-14b) CF ₃ Ph-4-CF ₃ H
3-I 2- (L-14c) CF ₃ Ph-4-OCF ₃ H
3-I 2- (L-14d) CF ₃ (L-45c) CF ₃ H
3-I 2- (L-14e) CF ₃ Ph-4-Br H
3-I 2- (L-14f) CF ₃ Ph-4-CF ₃ H
3-I 2-CH ₃ -3-F CF ₃ Ph-4-OCF ₃ H
3-I 2-CH ₃ -5-F CF ₃ (L-45c) CF ₃ H
3-I 2-CH ₃ -3-Cl CF ₃ Ph-4-Br H
3-I 2-CH ₃ -5-Cl CF ₃ Ph-4-CF ₃ H
3-I 2,3- (CH ₃ ) ₂ CF ₃ Ph-4-OCF ₃ H
3-I 2,5- (CH ₃ ) ₂ CF ₃ (L-45c) CF ₃ H
3-I 2,6- (CH ₃ ) ₂ CF ₃ Ph-4-Br H
3-I 2-CH ₃ -3-OCH ₃ CF ₃ Ph-4-CF ₃ H
3-I 2-CH ₃ -3-OCHF ₂ CF ₃ Ph-4-OCF ₃ H
3-I 2-CH ₃ -3,5-Cl ₂ CF ₃ (L-45c) CF ₃ H
4-I 2-CH ₃ CF ₃ Ph-4-Br H
5-I 2-CH ₃ CF ₃ Ph-4-CF ₃ H
6-I 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-I-4-Cl 2-CH ₃ CF ₃ (L-45c) CF ₃ H
4-Cl-6-I 2-CH ₃ CF ₃ Ph-4-Br H
5-CH ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
6-CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-Cl-4-CH ₃ 2-CH ₃ CF ₃ Ph-4-Br H
3-Cl-4-CH ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-Cl-4-CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-Cl-4-CH ₃ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
6-Et 2-CH ₃ CF ₃ (L-45c) CF ₃ H
4-CF ₃ 2-CH ₃ CF ₃ Ph-4-Br H
6-CF ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-CF ₂ CF ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-OCH ₃ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
6-OCH ₃ 2-CH ₃ CF ₃ Ph-4-Br H
3-Cl-4-OCH ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-OCH ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
5-OCHF ₂ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
6-OCHF ₂ 2-CH ₃ CF ₃ Ph-4-Br H
5-OCF ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ CH = CH (Ph-4-Br) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ CH = CH (Ph-4-CF ₃ ) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-FH
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-Cl H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-Br H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-O (L-45g) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-3,4-F ₂ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-3-F-4-Cl H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ L-45f H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ (L-46c) CF ₃ H
3-OSO ₂ CH ₃ 2-CH ₃ CF ₃ L-46d H
3-OSO ₂ Et 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-OSO ₂ CF ₃ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ CH = CH (Ph-4-Br) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ CH = CH (Ph-4-CF ₃ ) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-FH
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-Cl H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-Br H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-4-O (L-45g) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-3,4-F ₂ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-3-F-4-Cl H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) H
3-OCF ₂ O-4 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ L-45f H
3-OCF ₂ O-4 2-CH ₃ CF ₃ (L-46c) CF ₃ H
3-OCF ₂ O-4 2-CH ₃ CF ₃ L-46d H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ CH = CH (Ph-4-Cl) H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-Cl H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-Br H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ Br H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFCF ₃ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-4-O (L-45g) H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph-3,4-Cl ₂ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph (-3-OCF ₂ O-4-) H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ Ph (-3-OCF ₂ CF ₂ O-4-) H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ L-45f H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ (L-46c) CF ₃ H
3-OCF ₂ CF ₂ O-4 2-CH ₃ CF ₃ L-46d H
6-SCH ₃ 2-CH ₃ CF ₃ Ph-4-Br H
6-SO ₂ CH ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-SEt 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-SO ₂ Et 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-SPr-i 2-CH ₃ CF ₃ Ph-4-Br H
3-S (O) Pr-i 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-SO ₂ Pr-i 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
6-S (O) CF ₃ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-SCH ₂ CF ₃ 2-CH ₃ CF ₃ Ph-4-Br H
6-SCH ₂ CF ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-S (O) CH ₂ CF ₃ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
6-S (O) CH ₂ CF ₃ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-SO ₂ CH ₂ CF ₃ 2-CH ₃ CF ₃ Ph-4-Br H
3-Cl-6-SCF ₃ 2-CH ₃ CF ₃ Ph-4-CF ₃ H
6-NO ₂ 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-CN 2-CH ₃ CF ₃ (L-45c) CF ₃ H
6-C (O) OCH ₃ 2-CH ₃ CF ₃ Ph-4-Br H
3-C (O) NHPr-i 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-C≡CH 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
3-C≡CSi (CH ₃ ) ₃ 2-CH ₃ CF ₃ (L-45c) CF ₃ H
6-C≡CH 2-CH ₃ CF ₃ Ph-4-Br H
6-Ph 2-CH ₃ CF ₃ Ph-4-CF ₃ H
3-CH = CH-CH = CH-4 2-CH ₃ CF ₃ Ph-4-OCF ₃ H
4-CH = CH-CH = CH-5 2-CH ₃ CF ₃ (L-45c) CF ₃ H
3-Si (CH ₃ ) ₃ 2-CH ₃ CF ₃ Ph-4-Br H
―――――――――――――――――――――――――――――――――――――――
Table 4 In the table, the number representing the substitution position of the substituent (X) _m corresponds to the position of the number described in the following structural formula, and the-sign represents no substitution. .

―――――――――――――――――――――――――――――――――――――――
(X) _m YR ¹ R ⁶
―――――――――――――――――――――――――――――――――――――――
3-F CH ₃ i-Pr H
3-F CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-F CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-F CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-F CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-F CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-F CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-Cl CH ₃ i-Pr H
3-Cl CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-Cl CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-Cl CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-Cl CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-Cl CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-Cl CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3,4-Cl ₂ CH ₃ i-Pr H
3,4-Cl ₂ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3,4-Cl ₂ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3,4-Cl ₂ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3,4-Cl ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3,4-Cl ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3,4-Cl ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-Br CH ₃ i-Pr H
3-Br CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-Br CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-Br CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-Br CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-Br CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-Br CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-I − i-Pr H
3-I − CH (CH ₃ ) CH ₂ SCH ₃ H
3-I − CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-I − CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-I − C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-I − C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-I − C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-IF i-Pr H
3-IF CH (CH ₃ ) CH ₂ SCH ₃ H
3-IF CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-IF CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-IFC (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-IFC (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-IFC (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-I Cl i-Pr H
3-I Cl CH (CH ₃ ) CH ₂ SCH ₃ H
3-I Cl CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-I Cl CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-I Cl C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-I Cl C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-I Cl C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-I Br i-Pr H
3-I Br CH (CH ₃ ) CH ₂ SCH ₃ H
3-I Br CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-I Br CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-I Br C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-I Br C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-I Br C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-I CH ₃ CH ₃ H
3-I CH ₃ Et H
3-I CH ₃ i-Pr H
3-I CH ₃ i-Pr CH ₃
3-I CH ₃ i-Pr CH ₂ OCH ₃
3-I CH ₃ i-Pr C (O) CH ₃
3-I CH ₃ i-Pr Si (CH ₃ ) ₃
3-I CH ₃ s-Bu H
3-I CH ₃ t-Bu H
3-I CH ₃ CH (CH ₃ ) Pr-n H
3-I CH ₃ CH (CH ₃ ) CH ₂ OCH ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) CH ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) NHCH ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) NHEt H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) NHPr-n H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) NHPr-i H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) NHPr-c H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) NHCH ₂ Ph H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) NHPh H
3-I CH ₃ CH (CH ₃ ) CH ₂ OC (O) N (Et) ₂ H
3-I CH ₃ CH (CH ₃ ) CH ₂ OP (S) (OCH ₃ ) ₂ H
3-I CH ₃ CH (CH ₃ ) CH ₂ OP (S) (OEt) ₂ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ OCH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ OC (O) NHCH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ OC (O) NHEt H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ OC (O) NHPr-n H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ OC (O) NHCH ₂ Ph H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ OC (O) N (CH ₃ ) ₂ H
3-I CH ₃ CH (CH ₃ ) CH ₂ CH ₂ OEt H
3-I CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ CH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ CH ₂ OCH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ C (O) CH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ Si (CH ₃ ) ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ CH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ CH ₂ OCH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ C (O) CH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ Si (CH ₃ ) ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CH ₂ OCH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ C (O) CH ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ Si (CH ₃ ) ₃
3-I CH ₃ CH (CH ₃ ) CH ₂ SEt H
3-I CH ₃ CH (CH ₃ ) CH ₂ S (O) Et H
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ Et H
3-I CH ₃ CH (CH ₃ ) CH ₂ SCH ₂ Si (CH ₃ ) ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ SSCH ₃ H
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ NHEt H
3-I CH ₃ CH (CH ₃ ) CH ₂ SO ₂ N (Et) ₂ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ CH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ CH ₂ OCH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ C (O) CH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ Si (CH ₃ ) ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ CH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ CH ₂ OCH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ C (O) CH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ Si (CH ₃ ) ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ CH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ CH ₂ OCH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ C (O) CH ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ Si (CH ₃ ) ₃
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SEt H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) Et H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ Et H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ N (Et) ₂ H
3-I CH ₃ CH (CH ₃ ) CH ₂ N (CH ₃ ) SO ₂ CH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH ₂ NHC (O) OCH ₃ H
3-I CH ₃ CH (CH ₃ ) CH = NOCH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH = NOCH ₃ H
3-I CH ₃ C (CH ₃ ) ₂ CH = CH ₂ H
3-I CH ₃ C (CH ₃ ) ₂ C≡CH H
3-I Et i-Pr H
3-I Et CH (CH ₃ ) CH ₂ SCH ₃ H
3-I Et CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-I Et CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-I Et C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-I Et C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-I Et C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-I OCH ₃ i-Pr H
3-I OCH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-I OCH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-I OCH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-I OCH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-I OCH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-I OCH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-I SCH ₃ i-Pr H
3-I SCH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-I SCH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-I SCH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-I SCH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-I SCH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-I SCH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-CH ₃ CH ₃ i-Pr H
3-CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-CH ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-CF ₃ CH ₃ i-Pr H
3-CF ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-CF ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-CF ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-OCHF ₂ CH ₃ i-Pr H
3-OCHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-OCHF ₂ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-OCHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-OCHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-OCHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-OCHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-OCF ₃ CH ₃ i-Pr H
3-OCF ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-OCF ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-OCF ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-OCF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-OCF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-OCF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-OSO ₂ CH ₃ CH ₃ i-Pr H
3-OSO ₂ CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-OSO ₂ CH ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-OSO ₂ CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-OSO ₂ CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-OSO ₂ CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-OSO ₂ CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-OCF ₂ O-4 CH ₃ i-Pr H
3-OCF ₂ O-4 CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-OCF ₂ O-4 CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-OCF ₂ O-4 CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-OCF ₂ O-4 CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-OCF ₂ O-4 CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-OCF ₂ O-4 CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-SCH ₃ CH ₃ i-Pr H
3-SCH ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-SCH ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-SCH ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-SCH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-SCH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-SCH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-S (O) CH ₃ CH ₃ i-Pr H
3-S (O) CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-S (O) CH ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-S (O) CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-S (O) CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-S (O) CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-S (O) CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-SO ₂ CH ₃ CH ₃ i-Pr H
3-SO ₂ CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-SO ₂ CH ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-SO ₂ CH ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-SO ₂ CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-SO ₂ CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-SO ₂ CH ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-SCHF ₂ CH ₃ i-Pr H
3-SCHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-SCHF ₂ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-SCHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-SCHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-SCHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-SCHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-S (O) CHF ₂ CH ₃ i-Pr H
3-S (O) CHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-S (O) CHF ₂ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-S (O) CHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-S (O) CHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-S (O) CHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-S (O) CHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-SO ₂ CHF ₂ CH ₃ i-Pr H
3-SO ₂ CHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-SO ₂ CHF ₂ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-SO ₂ CHF ₂ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-SO ₂ CHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-SO ₂ CHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-SO ₂ CHF ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-SCF ₃ CH ₃ i-Pr H
3-SCF ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-SCF ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-SCF ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-SCF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-SCF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-SCF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-S (O) CF ₃ CH ₃ i-Pr H
3-S (O) CF ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-S (O) CF ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-S (O) CF ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-S (O) CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-S (O) CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-S (O) CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-SO ₂ CF ₃ CH ₃ i-Pr H
3-SO ₂ CF ₃ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-SO ₂ CF ₃ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-SO ₂ CF ₃ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-SO ₂ CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-SO ₂ CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-SO ₂ CF ₃ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
3-NO ₂ CH ₃ i-Pr H
3-NO ₂ CH ₃ CH (CH ₃ ) CH ₂ SCH ₃ H
3-NO ₂ CH ₃ CH (CH ₃ ) CH ₂ S (O) CH ₃ H
3-NO ₂ CH ₃ CH (CH ₃ ) CH ₂ SO ₂ CH ₃ H
3-NO ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SCH ₃ H
3-NO ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ S (O) CH ₃ H
3-NO ₂ CH ₃ C (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ H
―――――――――――――――――――――――――――――――――――――――
Table 5

―――――――――――――――――――――――――――――――――――――――
R ⁴ Y ² R ⁵ Y ³ R ⁶
―――――――――――――――――――――――――――――――――――――――
CH ₃ H CF ₂ O (Ph-4-Cl) HH
CH ₃ H CH = CH (Ph-4-Cl) HH
CH ₃ H CH = CH (Ph-4-OCF ₃ ) HH
CH ₃ H CH = CH (Ph-3,4-Cl ₂ ) HH
CH ₃ H Ph-4-FHH
CH ₃ H Ph-4-Cl HH
CH ₃ H Ph-4-Br HH
CH ₃ H Ph-4-IHH
CH ₃ H Ph-4-CF ₃ HH
CH ₃ H Ph-4-OCHF ₂ HH
CH ₃ H Ph-4-OCF ₃ HH
CH ₃ H Ph-4-OCF ₂ Br HH
CH ₃ H Ph-4-OCF ₂ CHF ₂ HH
CH ₃ H Ph-4-OCF ₂ CHFCl HH
CH ₃ H Ph-4-OCF ₂ CHFCF ₃ HH
CH ₃ H Ph-4-OCF ₂ CHFOCF ₃ HH
CH ₃ H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CH ₃ H Ph-4-O (L-45g) HH
CH ₃ H Ph-3,4-Cl ₂ HH
CH ₃ H Ph (-3-OCF ₂ O-4-) HH
CH ₃ H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CH ₃ H (L-45c) Cl HH
CH ₃ H (L-45c) Br HH
CH ₃ H (L-45c) CF ₃ HH
CH ₃ H L-45e HH
CH ₃ H L-45f HH
CH ₃ H (L-46c) Cl HH
CH ₃ H (L-46c) Br HH
CH ₃ H (L-46c) CF ₃ HH
CH ₃ H L-46d HH
Et H CF ₂ O (Ph-4-Cl) HH
Et H CH = CH (Ph-4-Cl) HH
Et H CH = CH (Ph-4-OCF ₃ ) HH
Et H CH = CH (Ph-3,4-Cl ₂ ) HH
Et H Ph-4-Cl HH
Et H Ph-4-Br HH
Et H Ph-4-CF ₃ HH
Et H Ph-4-OCF ₃ HH
Et H Ph-4-OCF ₂ Br HH
Et H Ph-4-OCF ₂ CHFCF ₃ HH
Et H Ph-4-OCF ₂ CHFOCF ₃ HH
Et H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
Et H Ph-4-O (L-45g) HH
Et H Ph-3,4-Cl ₂ HH
Et H Ph (-3-OCF ₂ O-4-) HH
Et H Ph (-3-OCF ₂ CF ₂ O-4-) HH
Et H (L-45c) Br HH
Et H (L-45c) CF ₃ HH
Et H L-45e HH
Et H L-45f HH
Et H (L-46c) Br HH
Et H (L-46c) CF ₃ HH
Et H L-46d HH
n-Pr H Ph-4-Br HH
n-Pr H Ph-4-CF ₃ HH
n-Pr H Ph-4-OCF ₃ HH
n-Pr H (L-45c) CF ₃ HH
i-Pr H Ph-4-Br HH
i-Pr H Ph-4-CF ₃ HH
i-Pr H Ph-4-OCF ₃ HH
i-Pr H (L-45c) CF ₃ HH
c-Pr H Ph-4-Br HH
c-Pr H Ph-4-CF ₃ HH
c-Pr H Ph-4-OCF ₃ HH
c-Pr H (L-45c) CF ₃ HH
n-Bu H Ph-4-Br HH
CH ₂ FH Ph-4-CF ₃ HH
CH ₂ Cl H Ph-4-OCF ₃ HH
CH ₂ Br H (L-45c) CF ₃ HH
CHF ₂ H CF ₂ O (Ph-4-Cl) HH
CHF ₂ H CH = CH (Ph-4-Cl) HH
CHF ₂ H CH = CH (Ph-4-OCF ₃ ) HH
CHF ₂ H CH = CH (Ph-3,4-Cl ₂ ) HH
CHF ₂ H Ph-4-FHH
CHF ₂ H Ph-4-Cl HH
CHF ₂ H Ph-4-Br HH
CHF ₂ H Ph-4-IHH
CHF ₂ H Ph-4-CF ₃ HH
CHF ₂ H Ph-4-OCHF ₂ HH
CHF ₂ H Ph-4-OCF ₃ HH
CHF ₂ H Ph-4-OCF ₂ Br HH
CHF ₂ H Ph-4-OCF ₂ CHF ₂ HH
CHF ₂ H Ph-4-OCF ₂ CHFCl HH
CHF ₂ H Ph-4-OCF ₂ CHFCF ₃ HH
CHF ₂ H Ph-4-OCF ₂ CHFOCF ₃ HH
CHF ₂ H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CHF ₂ H Ph-4-O (L-45g) HH
CHF ₂ H Ph-3,4-Cl ₂ HH
CHF ₂ H Ph (-3-OCF ₂ O-4-) HH
CHF ₂ H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CHF ₂ H (L-45c) Cl HH
CHF ₂ H (L-45c) Br HH
CHF ₂ H (L-45c) CF ₃ HH
CHF ₂ H L-45e HH
CHF ₂ H L-45f HH
CHF ₂ H (L-46c) Cl HH
CHF ₂ H (L-46c) Br HH
CHF ₂ H (L-46c) CF ₃ HH
CHF ₂ H L-46d HH
CHFCl H Ph-4-Br HH
CHFBr H Ph-4-CF ₃ HH
CF ₃ H CH ₂ OCH ₃ HH
CF ₃ H CH ₂ OEt HH
CF ₃ H CH ₂ OPr-n HH
CF ₃ H CH ₂ OPr-i HH
CF ₃ H CH ₂ OBu-n HH
CF ₃ H CH ₂ OCH ₂ CF ₃ HH
CF ₃ H CH ₂ OCH ₂ CF ₂ CF ₃ HH
CF ₃ H CH ₂ OCH (CF ₃ ) ₂ HH
CF ₃ H CH ₂ OPh HH
CF ₃ H CH ₂ O (Ph-4-F) HH
CF ₃ H CH ₂ O (Ph-2-Cl) HH
CF ₃ H CH ₂ O (Ph-3-Cl) HH
CF ₃ H CH ₂ O (Ph-4-Cl) HH
CF ₃ H CH ₂ O (Ph-4-Br) HH
CF ₃ H CH ₂ O (Ph-4-CF ₃ ) HH
CF ₃ H CH ₂ O (Ph-2-OCF ₃ ) HH
CF ₃ H CH ₂ O (Ph-3-OCF ₃ ) HH
CF ₃ H CH ₂ O (Ph-4-OCF ₃ ) HH
CF ₃ H CF ₂ OPh HH
CF ₃ H CF ₂ O (Ph-3-F) HH
CF ₃ H CF ₂ O (Ph-4-F) HH
CF ₃ H CF ₂ O (Ph-2-Cl) HH
CF ₃ H CF ₂ O (Ph-3-Cl) HH
CF ₃ H CF ₂ O (Ph-4-Cl) HH
CF ₃ H CF ₂ O (Ph-3-Br) HH
CF ₃ H CF ₂ O (Ph-4-Br) HH
CF ₃ H CF ₂ O (Ph-3-CF ₃ ) HH
CF ₃ H CF ₂ O (Ph-4-CF ₃ ) HH
CF ₃ H CF ₂ O (Ph-3-OCF ₃ ) HH
CF ₃ H CF ₂ O (Ph-4-OCF ₃ ) HH
CF ₃ H CH ₂ SPh HH
CF ₃ H CH ₂ S (Ph-3-Cl) HH
CF ₃ H CH ₂ S (Ph-4-Cl) HH
CF ₃ H CH ₂ SO ₂ (Ph-3-Cl) HH
CF ₃ H CH ₂ SO ₂ (Ph-4-Cl) HH
CF ₃ H CH ₂ N (CH ₃ ) ₂ HH
CF ₃ H CH ₂ NHPh HH
CF ₃ H CH ₂ NH (Ph-3-Cl) HH
CF ₃ H CH ₂ NH (Ph-4-Cl) HH
CF ₃ H CF ₂ C (O) OEt HH
CF ₃ H CH ₂ (L-5a) HH
CF ₃ H CH ₂ (L-14a) HH
CF ₃ H CH ₂ (L-24a) HH
CF ₃ H CH ₂ (L-36a) HH
CF ₃ HC (O) OEt HH
CF ₃ HC (O) OBu-t HH
CF ₃ HC (O) OCH ₂ CF ₃ HH
CF ₃ H CH = CHPh HH
CF ₃ H CH = CH (Ph-3-F) HH
CF ₃ H CH = CH (Ph-4-F) HH
CF ₃ H CH = CH (Ph-2-Cl) HH
CF ₃ H CH = CH (Ph-3-Cl) HH
CF ₃ H CH = CH (Ph-4-Cl) HH
CF ₃ H CH = CH (Ph-3-Br) HH
CF ₃ H CH = CH (Ph-4-Br) HH
CF ₃ H CH = CH (Ph-3-CF ₃ ) HH
CF ₃ H CH = CH (Ph-4-CF ₃ ) HH
CF ₃ H CH = CH (Ph-3-OCF ₃ ) HH
CF ₃ H CH = CH (Ph-4-OCF ₃ ) HH
CF ₃ H CH = CH (Ph-3-SCH ₃ ) HH
CF ₃ H CH = CH (Ph-4-SCH ₃ ) HH
CF ₃ H CH = CH (Ph-3-SO ₂ CH ₃ ) HH
CF ₃ H CH = CH (Ph-4-SO ₂ CH ₃ ) HH
CF ₃ H CH = CH (Ph-3,4-F ₂ ) HH
CF ₃ H CH = CH (Ph-3-F-4-Cl) HH
CF ₃ H CH = CH (Ph-3,4-Cl ₂ ) HH
CF ₃ H CH = CH (Ph-3,4-Br ₂ ) HH
CF ₃ H CH = CH (Ph-3-F-4-CF ₃ ) HH
CF ₃ H CH = CH (Ph-3-Cl-4-OCF ₃ ) HH
CF ₃ H CH = CH [Ph (-3-OCF ₂ O-4-)] HH
CF ₃ H Ph HH
CF ₃ H Ph-2-FHH
CF ₃ H Ph-3-FHH
CF ₃ H Ph-4-FHH
CF ₃ H Ph-2-Cl HH
CF ₃ H Ph-3-Cl HH
CF ₃ H Ph-4-Cl HH
CF ₃ H Ph-3-Br HH
CF ₃ H Ph-4-Br HH
CF ₃ H Ph-4-Br H CH ₃
CF ₃ H Ph-4-Br H Et
CF ₃ H Ph-4-Br H n-Pr
CF ₃ H Ph-4-Br H i-Pr
CF ₃ H Ph-4-Br H n-Bu
CF ₃ H Ph-4-Br H CH ₂ CF ₃
CF ₃ H Ph-4-Br H CH ₂ OCH ₃
CF ₃ H Ph-4-Br H CH ₂ OEt
CF ₃ H Ph-4-Br H CH ₂ SCH ₃
CF ₃ H Ph-4-Br H CH ₂ CH = CH ₂
CF ₃ H Ph-4-Br H CH ₂ CH = CF ₂
CF ₃ H Ph-4-Br H CH ₂ CH = CCl ₂
CF ₃ H Ph-4-Br H CH ₂ CF = CF ₂
CF ₃ H Ph-4-Br H CH ₂ CCl = CCl ₂
CF ₃ H Ph-4-Br H CH ₂ C≡CH
CF ₃ H Ph-4-Br H CH ₂ Ph
CF ₃ H Ph-4-Br H Si (CH ₃ ) ₃
CF ₃ H Ph-4-Br H Si (CH ₃ ) ₂ Bu-t
CF ₃ H Ph-4-Br H Si (CH ₃ ) ₂ Ph
CF ₃ H Ph-4-IHH
CF ₃ H Ph-4-Bu-t HH
CF ₃ H Ph-3-CF ₃ HH
CF ₃ H Ph-4-CF ₃ HH
CF ₃ H Ph-4-CF ₃ H CH ₃
CF ₃ H Ph-4-CF ₃ H Et
CF ₃ H Ph-4-CF ₃ H n-Pr
CF ₃ H Ph-4-CF ₃ H i-Pr
CF ₃ H Ph-4-CF ₃ H n-Bu
CF ₃ H Ph-4-CF ₃ H CH ₂ CF ₃
CF ₃ H Ph-4-CF ₃ H CH ₂ OCH ₃
CF ₃ H Ph-4-CF ₃ H CH ₂ OEt
CF ₃ H Ph-4-CF ₃ H CH ₂ SCH ₃
CF ₃ H Ph-4-CF ₃ H CH ₂ CH = CH ₂
CF ₃ H Ph-4-CF ₃ H CH ₂ CH = CF ₂
CF ₃ H Ph-4-CF ₃ H CH ₂ CH = CCl ₂
CF ₃ H Ph-4-CF ₃ H CH ₂ CF = CF ₂
CF ₃ H Ph-4-CF ₃ H CH ₂ CCl = CCl ₂
CF ₃ H Ph-4-CF ₃ H CH ₂ C≡CH
CF ₃ H Ph-4-CF ₃ H CH ₂ Ph
CF ₃ H Ph-4-CF ₃ H Si (CH ₃ ) ₃
CF ₃ H Ph-4-CF ₃ H Si (CH ₃ ) ₂ Bu-t
CF ₃ H Ph-4-CF ₃ H Si (CH ₃ ) ₂ Ph
CF ₃ H Ph-4-OCH ₃ HH
CF ₃ H Ph-4-OCHF ₂ HH
CF ₃ H Ph-3-OCF ₃ HH
CF ₃ H Ph-4-OCF ₃ HH
CF ₃ H Ph-4-OCF ₃ H CH ₃
CF ₃ H Ph-4-OCF ₃ H Et
CF ₃ H Ph-4-OCF ₃ H n-Pr
CF ₃ H Ph-4-OCF ₃ H i-Pr
CF ₃ H Ph-4-OCF ₃ H n-Bu
CF ₃ H Ph-4-OCF ₃ H CH ₂ CF ₃
CF ₃ H Ph-4-OCF ₃ H CH ₂ OCH ₃
CF ₃ H Ph-4-OCF ₃ H CH ₂ OEt
CF ₃ H Ph-4-OCF ₃ H CH ₂ SCH ₃
CF ₃ H Ph-4-OCF ₃ H CH ₂ CH = CH ₂
CF ₃ H Ph-4-OCF ₃ H CH ₂ CH = CF ₂
CF ₃ H Ph-4-OCF ₃ H CH ₂ CH = CCl ₂
CF ₃ H Ph-4-OCF ₃ H CH ₂ CF = CF ₂
CF ₃ H Ph-4-OCF ₃ H CH ₂ CCl = CCl ₂
CF ₃ H Ph-4-OCF ₃ H CH ₂ C≡CH
CF ₃ H Ph-4-OCF ₃ H CH ₂ Ph
CF ₃ H Ph-4-OCF ₃ H Si (CH ₃ ) ₃
CF ₃ H Ph-4-OCF ₃ H Si (CH ₃ ) ₂ Bu-t
CF ₃ H Ph-4-OCF ₃ H Si (CH ₃ ) ₂ Ph
CF ₃ H Ph-4-OCF ₂ Br HH
CF ₃ H Ph-4-OCH ₂ CF ₃ HH
CF ₃ H Ph-4-OCF ₂ CHF ₂ HH
CF ₃ H Ph-4-OCF ₂ CHFCl HH
CF ₃ H Ph-4-OCF ₂ CHFBr HH
CF ₃ H Ph-4-OCF ₂ CF ₂ Br HH
CF ₃ H Ph-4-OCF ₂ CFCl ₂ HH
CF ₃ H Ph-4-OCF ₂ CCl ₃ HH
CF ₃ H Ph-4-OCH ₂ CF ₂ CHF ₂ HH
CF ₃ H Ph-3-OCF ₂ CHFCF ₃ HH
CF ₃ H Ph-4-OCF ₂ CHFCF ₃ HH
CF ₃ H Ph-4-OCH (CF ₃ ) ₂ HH
CF ₃ H Ph-4-OCF ₂ CFBrCF ₃ HH
CF ₃ H Ph-3-OCF ₂ CHFOCF ₃ HH
CF ₃ H Ph-4-OCF ₂ CHFOCF ₃ HH
CF ₃ H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₃ H Ph-4-OSO ₂ CH ₃ HH
CF ₃ H Ph-4-OSO ₂ CF ₃ HH
CF ₃ H Ph-3-O (Ph-4-Cl) HH
CF ₃ H Ph-4-O (Ph-4-Cl) HH
CF ₃ H Ph-4-O (Ph-4-Br) HH
CF ₃ H Ph-4-O (Ph-4-CF ₃ ) HH
CF ₃ H Ph-4-O (L-45c) Br HH
CF ₃ H Ph-4-O (L-45c) CF ₃ HH
CF ₃ H Ph-3-O (L-45e) HH
CF ₃ H Ph-4-O (L-45e) HH
CF ₃ H Ph-4-O (L-48b) Br HH
CF ₃ H Ph-4-SCH ₃ HH
CF ₃ H Ph-4-SO ₂ CH ₃ HH
CF ₃ H Ph-3-S (Ph-4-Cl) HH
CF ₃ H Ph-4-S (Ph-4-Cl) HH
CF ₃ H Ph-4-S (Ph-4-Br) HH
CF ₃ H Ph-4-S (Ph-4-CF ₃ ) HH
CF ₃ H Ph-4-S (L-45c) Br HH
CF ₃ H Ph-4-S (L-45c) CF ₃ HH
CF ₃ H Ph-4-S (L-45e) HH
CF ₃ H Ph-4-S (L-48b) Br HH
CF ₃ H Ph-4-NO ₂ HH
CF ₃ H Ph-4-CN HH
CF ₃ H Ph-2,3-F ₂ HH
CF ₃ H Ph-2,4-F ₂ HH
CF ₃ H Ph-3,4-F ₂ HH
CF ₃ H Ph-2,5-F ₂ HH
CF ₃ H Ph-3,5-F ₂ HH
CF ₃ H Ph-2-Cl-4-FHH
CF ₃ H Ph-2-F-3-Cl HH
CF ₃ H Ph-3-Cl-4-FHH
CF ₃ H Ph-2-F-4-Cl HH
CF ₃ H Ph-3-F-4-Cl HH
CF ₃ H Ph-2,3-Cl ₂ HH
CF ₃ H Ph-2,4-Cl ₂ HH
CF ₃ H Ph-2,5-Cl ₂ HH
CF ₃ H Ph-3,4-Cl ₂ HH
CF ₃ H Ph-3,5-Cl ₂ HH
CF ₃ H Ph-3-Br-4-FHH
CF ₃ H Ph-2-F-4-Br HH
CF ₃ H Ph-2-F-5-Br HH
CF ₃ H Ph-3,4-Br ₂ HH
CF ₃ H Ph-3,5-Br ₂ HH
CF ₃ H Ph-3-CH ₃ -4-FHH
CF ₃ H Ph-3-F-4-CH ₃ HH
CF ₃ H Ph-2-F-5-CH ₃ HH
CF ₃ H Ph-2,4- (CH ₃ ) ₂ HH
CF ₃ H Ph-3,4- (CH ₃ ) ₂ HH
CF ₃ H Ph-2-F-3-CF ₃ HH
CF ₃ H Ph-3-CF ₃ -4-FHH
CF ₃ H Ph-3-CF ₃ -4-Cl HH
CF ₃ H Ph-2-F-4-CF ₃ HH
CF ₃ H Ph-3-F-4-CF ₃ HH
CF ₃ H Ph-2-F-5-CF ₃ HH
CF ₃ H Ph-3-F-5-CF ₃ HH
CF ₃ H Ph-2-Cl-4-CF ₃ HH
CF ₃ H Ph-3,5- (CF ₃ ) ₂ HH
CF ₃ H Ph-3-Br-4-OCH ₃ HH
CF ₃ H Ph-3-F-4-OCHF ₂ HH
CF ₃ H Ph-3-Cl-4-OCHF ₂ HH
CF ₃ H Ph-3-Br-4-OCHF ₂ HH
CF ₃ H Ph-3-F-4-OCF ₃ HH
CF ₃ H Ph-3-Cl-4-OCF ₃ HH
CF ₃ H Ph-3-Br-4-OCF ₃ HH
CF ₃ H Ph-3-F-4-OCF ₂ Br HH
CF ₃ H Ph-3-Cl-4-OCF ₂ Br HH
CF ₃ H Ph-3-Br-4-OCF ₂ Br HH
CF ₃ H Ph-3-F-4-OCF ₂ CHF ₂ HH
CF ₃ H Ph-3-Cl-4-OCF ₂ CHF ₂ HH
CF ₃ H Ph-3-Br-4-OCF ₂ CHF ₂ HH
CF ₃ H Ph-3-F-4-OCF ₂ CHFCl HH
CF ₃ H Ph-3-Cl-4-OCF ₂ CHFCl HH
CF ₃ H Ph-3-Br-4-OCF ₂ CHFCl HH
CF ₃ H Ph-3-F-4-OCF ₂ CHFCF ₃ HH
CF ₃ H Ph-3-Cl-4-OCF ₂ CHFCF ₃ HH
CF ₃ H Ph-3-Br-4-OCF ₂ CHFCF ₃ HH
CF ₃ H Ph-3-F-4-OCF ₂ CHFOCF ₃ HH
CF ₃ H Ph-3-Cl-4-OCF ₂ CHFOCF ₃ HH
CF ₃ H Ph-3-Br-4-OCF ₂ CHFOCF ₃ HH
CF ₃ H Ph-3-CH ₃ -4-OCF ₂ CHFOCF ₃ HH
CF ₃ H Ph-3-F-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₃ H Ph-3-Cl-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₃ H Ph-3-Br-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₃ H Ph (-3-OCF ₂ O-4-) HH
CF ₃ H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CF ₃ H Ph-3-OPh-4-FHH
CF ₃ H Ph-3-NO ₂ -4-FHH
CF ₃ H Ph-3-NO ₂ -4-Cl HH
CF ₃ H Ph-2-F-5-NO ₂ HH
CF ₃ H Ph-3-CN-4-FHH
CF ₃ H Ph-2,3,4-F ₃ HH
CF ₃ H Ph-2,3,5-F ₃ HH
CF ₃ H Ph-2,4,5-F ₃ HH
CF ₃ H Ph-3,4,5-F ₃ HH
CF ₃ H Ph-2,3-F ₂ -4-CH ₃ HH
CF ₃ H Ph-2,3-F ₂ -4-CF ₃ HH
CF ₃ H Ph-3,4-F ₂ -5-CF ₃ HH
CF ₃ H Ph-2-F-3-Cl-5-CF ₃ HH
CF ₃ H Ph-3,5-Cl ₂ -4-OCH ₃ HH
CF ₃ H 1-Naph HH
CF ₃ H 2-Naph HH
CF ₃ H (L-1b) Br HH
CF ₃ H (L-1c) Cl HH
CF ₃ H (L-1c) Br HH
CF ₃ H (L-1c) IHH
CF ₃ H (L-1c) CF ₃ HH
CF ₃ H (L-2b) Br HH
CF ₃ H (L-3b) Cl HH
CF ₃ H (L-3b) Br HH
CF ₃ H (L-3c) FHH
CF ₃ H (L-3c) Cl HH
CF ₃ H (L-3c) Br HH
CF ₃ H (L-3c) IHH
CF ₃ H (L-3c) CF ₃ HH
CF ₃ H (L-3c) CN HH
CF ₃ H L-3d HH
CF ₃ H (L-4b) Cl HH
CF ₃ H (L-4b) Br HH
CF ₃ H (L-4b) CN HH
CF ₃ H (L-10b) Cl HH
CF ₃ H (L-10b) Br HH
CF ₃ H (L-15b) CF ₃ HH
CF ₃ H (L-16a) CHF ₂ HH
CF ₃ H (L-16a) CF ₂ Br HH
CF ₃ H (L-17a) Cl HH
CF ₃ H (L-21b) Cl HH
CF ₃ H (L-21b) Br HH
CF ₃ H (L-21b) IHH
CF ₃ H (L-21b) CF ₃ HH
CF ₃ H (L-22b) Cl HH
CF ₃ H (L-22b) Br HH
CF ₃ H (L-23b) Cl HH
CF ₃ H (L-23b) Br HH
CF ₃ H (L-23c) Cl HH
CF ₃ H (L-23c) Br HH
CF ₃ H (L-31a) Cl HH
CF ₃ H (L-31a) Br HH
CF ₃ H (L-45c) FHH
CF ₃ H (L-45c) Cl HH
CF ₃ H (L-45c) Br HH
CF ₃ H (L-45c) IHH
CF ₃ H (L-45c) CF ₃ HH
CF ₃ H (L-45c) CF ₃ H CH ₃
CF ₃ H (L-45c) CF ₃ H Et
CF ₃ H (L-45c) CF ₃ H n-Pr
CF ₃ H (L-45c) CF ₃ H i-Pr
CF ₃ H (L-45c) CF ₃ H n-Bu
CF ₃ H (L-45c) CF ₃ H CH ₂ CF ₃
CF ₃ H (L-45c) CF ₃ H CH ₂ OCH ₃
CF ₃ H (L-45c) CF ₃ H CH ₂ OEt
CF ₃ H (L-45c) CF ₃ H CH ₂ SCH ₃
CF ₃ H (L-45c) CF ₃ H CH ₂ CH = CH ₂
CF ₃ H (L-45c) CF ₃ H CH ₂ CH = CF ₂
CF ₃ H (L-45c) CF ₃ H CH ₂ CH = CCl ₂
CF ₃ H (L-45c) CF ₃ H CH ₂ CF = CF ₂
CF ₃ H (L-45c) CF ₃ H CH ₂ CCl = CCl ₂
CF ₃ H (L-45c) CF ₃ H CH ₂ C≡CH
CF ₃ H (L-45c) CF ₃ H CH ₂ Ph
CF ₃ H (L-45c) CF ₃ H Si (CH ₃ ) ₃
CF ₃ H (L-45c) CF ₃ H Si (CH ₃ ) ₂ Bu-t
CF ₃ H (L-45c) CF ₃ H Si (CH ₃ ) ₂ Ph
CF ₃ H L-45e HH
CF ₃ H L-45f HH
CF ₃ H (L-46c) FHH
CF ₃ H (L-46c) Cl HH
CF ₃ H (L-46c) Br HH
CF ₃ H (L-46c) IHH
CF ₃ H (L-46c) CF ₃ HH
CF ₃ H (L-46c) OCH ₂ CF ₃ HH
CF ₃ H (L-46c) OCH (CF ₃ ) ₂ HH
CF ₃ H L-46d HH
CF ₃ H L-47a HH
CF ₃ H L-47d HH
CF ₃ H (L-48b) Br HH
CF ₃ H (L-50b) Cl HH
CF ₃ H (L-50b) Br HH
CF ₃ H (L-51b) Cl HH
CF ₃ -OCF ₂ -HH
CF ₃ -OCF ₂ -H CH ₃
CF ₃ -OCF ₂ -H CH ₂ OCH ₃
CF ₃ -OCF ₂ -H Si (CH ₃ ) ₃
CF ₃ H -CF ₂ O- H
CF ₃ H -CF ₂ O- CH ₃
CF ₃ H -CF ₂ O- CH ₂ OCH ₃
CF ₃ H -CF ₂ O- Si (CH ₃ ) ₃
CF ₂ Cl H CF ₂ O (Ph-4-Cl) HH
CF ₂ Cl H CH = CH (Ph-4-Cl) HH
CF ₂ Cl H CH = CH (Ph-4-OCF ₃ ) HH
CF ₂ Cl H CH = CH (Ph-3,4-Cl ₂ ) HH
CF ₂ Cl H Ph-4-FHH
CF ₂ Cl H Ph-4-Cl HH
CF ₂ Cl H Ph-4-Br HH
CF ₂ Cl H Ph-4-IHH
CF ₂ Cl H Ph-4-CF ₃ HH
CF ₂ Cl H Ph-4-OCHF ₂ HH
CF ₂ Cl H Ph-4-OCF ₃ HH
CF ₂ Cl H Ph-4-OCF ₂ Br HH
CF ₂ Cl H Ph-4-OCF ₂ CHF ₂ HH
CF ₂ Cl H Ph-4-OCF ₂ CHFCl HH
CF ₂ Cl H Ph-4-OCF ₂ CHFCF ₃ HH
CF ₂ Cl H Ph-4-OCF ₂ CHFOCF ₃ HH
CF ₂ Cl H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₂ Cl H Ph-4-O (L-45g) HH
CF ₂ Cl H Ph-3,4-Cl ₂ HH
CF ₂ Cl H Ph (-3-OCF ₂ O-4-) HH
CF ₂ Cl H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CF ₂ Cl H (L-45c) Cl HH
CF ₂ Cl H (L-45c) Br HH
CF ₂ Cl H (L-45c) CF ₃ HH
CF ₂ Cl H L-45e HH
CF ₂ Cl H L-45f HH
CF ₂ Cl H (L-46c) Cl HH
CF ₂ Cl H (L-46c) Br HH
CF ₂ Cl H (L-46c) CF ₃ HH
CF ₂ Cl H L-46d HH
CFCl ₂ H Ph-4-OCF ₃ HH
CF ₂ Br H Ph-4-Cl HH
CF ₂ Br H Ph-4-Br HH
CF ₂ Br H Ph-4-CF ₃ HH
CF ₂ Br H Ph-4-OCF ₃ HH
CF ₂ Br H Ph-4-OCF ₂ Br HH
CF ₂ Br H Ph-4-OCF ₂ CHFCF ₃ HH
CF ₂ Br H Ph-4-OCF ₂ CHFOCF ₃ HH
CF ₂ Br H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₂ Br H Ph-4-O (L-45g) HH
CF ₂ Br H Ph-3,4-Cl ₂ HH
CF ₂ Br H Ph (-3-OCF ₂ O-4-) HH
CF ₂ Br H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CF ₂ Br H (L-45c) CF ₃ HH
CF ₂ Br H L-45f HH
CF ₂ Br H (L-46c) CF ₃ HH
CF ₂ Br H L-46d HH
CFClBr H (L-45c) CF ₃ HH
CFBr ₂ H Ph-4-Br HH
CF ₂ CHF ₂ H Ph-4-CF ₃ HH
CF ₂ CF ₃ H CF ₂ O (Ph-4-Cl) HH
CF ₂ CF ₃ H CH = CH (Ph-4-Cl) HH
CF ₂ CF ₃ H CH = CH (Ph-4-OCF ₃ ) HH
CF ₂ CF ₃ H CH = CH (Ph-3,4-Cl ₂ ) HH
CF ₂ CF ₃ H Ph-4-FHH
CF ₂ CF ₃ H Ph-4-Cl HH
CF ₂ CF ₃ H Ph-4-Br HH
CF ₂ CF ₃ H Ph-4-IHH
CF ₂ CF ₃ H Ph-4-CF ₃ HH
CF ₂ CF ₃ H Ph-4-OCHF ₂ HH
CF ₂ CF ₃ H Ph-4-OCF ₃ HH
CF ₂ CF ₃ H Ph-4-OCF ₂ Br HH
CF ₂ CF ₃ H Ph-4-OCF ₂ CHF ₂ HH
CF ₂ CF ₃ H Ph-4-OCF ₂ CHFCl HH
CF ₂ CF ₃ H Ph-4-OCF ₂ CHFCF ₃ HH
CF ₂ CF ₃ H Ph-4-OCF ₂ CHFOCF ₃ HH
CF ₂ CF ₃ H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₂ CF ₃ H Ph-4-O (L-45g) HH
CF ₂ CF ₃ H Ph-3,4-Cl ₂ HH
CF ₂ CF ₃ H Ph (-3-OCF ₂ O-4-) HH
CF ₂ CF ₃ H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CF ₂ CF ₃ H (L-45c) Cl HH
CF ₂ CF ₃ H (L-45c) Br HH
CF ₂ CF ₃ H (L-45c) CF ₃ HH
CF ₂ CF ₃ H L-45e HH
CF ₂ CF ₃ H L-45f HH
CF ₂ CF ₃ H (L-46c) Cl HH
CF ₂ CF ₃ H (L-46c) Br HH
CF ₂ CF ₃ H (L-46c) CF ₃ HH
CF ₂ CF ₃ H L-46d HH
CF ₂ CF ₂ Cl H Ph-4-OCF ₃ HH
CFClCF ₃ H (L-45c) CF ₃ HH
CFClCF ₂ Cl H Ph-4-Br HH
CF ₂ CF ₂ Br H Ph-4-CF ₃ HH
CFBrCF ₃ H Ph-4-OCF ₃ HH
CF ₂ CHFCF ₃ H (L-45c) CF ₃ HH
CF ₂ CF ₂ CF ₃ H Ph-4-Cl HH
CF ₂ CF ₂ CF ₃ H Ph-4-Br HH
CF ₂ CF ₂ CF ₃ H Ph-4-CF ₃ HH
CF ₂ CF ₂ CF ₃ H Ph-4-OCF ₃ HH
CF ₂ CF ₂ CF ₃ H Ph-4-OCF ₂ Br HH
CF ₂ CF ₂ CF ₃ H Ph-4-OCF ₂ CHFCF ₃ HH
CF ₂ CF ₂ CF ₃ H Ph-4-OCF ₂ CHFOCF ₃ HH
CF ₂ CF ₂ CF ₃ H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₂ CF ₂ CF ₃ H Ph-4-O (L-45g) HH
CF ₂ CF ₂ CF ₃ H Ph-3,4-Cl ₂ HH
CF ₂ CF ₂ CF ₃ H Ph (-3-OCF ₂ O-4-) HH
CF ₂ CF ₂ CF ₃ H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CF ₂ CF ₂ CF ₃ H (L-45c) CF ₃ HH
CF ₂ CF ₂ CF ₃ H L-45f HH
CF ₂ CF ₂ CF ₃ H (L-46c) CF ₃ HH
CF ₂ CF ₂ CF ₃ H L-46d HH
CF (CF ₃ ) ₂ H Ph-4-Br HH
CF ₂ CFClCF ₂ Cl H Ph-4-CF ₃ HH
CF ₂ CFBrCF ₂ Cl H Ph-4-OCF ₃ HH
CF ₂ CF ₂ CF ₂ CHF ₂ H (L-45c) CF ₃ HH
CF ₂ CF ₂ CF ₂ CF ₃ H Ph-4-Br HH
CF (CF ₃ ) CF ₂ CF ₃ H Ph-4-CF ₃ HH
CF ₂ CF ₂ CF ₂ CF ₂ Cl H Ph-4-OCF ₃ HH
T-1 H (L-45c) CF ₃ HH
T-2 H Ph-4-Br HH
CF ₂ OCH ₃ H Ph-4-Cl HH
CF ₂ OCH ₃ H Ph-4-Br HH
CF ₂ OCH ₃ H Ph-4-CF ₃ HH
CF ₂ OCH ₃ H Ph-4-OCF ₃ HH
CF ₂ OCH ₃ H Ph-4-OCF ₂ Br HH
CF ₂ OCH ₃ H Ph-4-OCF ₂ CHFCF ₃ HH
CF ₂ OCH ₃ H Ph-4-OCF ₂ CHFOCF ₃ HH
CF ₂ OCH ₃ H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₂ OCH ₃ H Ph-4-O (L-45g) HH
CF ₂ OCH ₃ H Ph-3,4-Cl ₂ HH
CF ₂ OCH ₃ H Ph (-3-OCF ₂ O-4-) HH
CF ₂ OCH ₃ H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CF ₂ OCH ₃ H (L-45c) CF ₃ HH
CF ₂ OCH ₃ H L-45f HH
CF ₂ OCH ₃ H (L-46c) CF ₃ HH
CF ₂ OCH ₃ H L-46d HH
CF ₂ SCH ₃ H Ph-4-Cl HH
CF ₂ SCH ₃ H Ph-4-Br HH
CF ₂ SCH ₃ H Ph-4-CF ₃ HH
CF ₂ SCH ₃ H Ph-4-OCF ₃ HH
CF ₂ SCH ₃ H Ph-4-OCF ₂ Br HH
CF ₂ SCH ₃ H Ph-4-OCF ₂ CHFCF ₃ HH
CF ₂ SCH ₃ H Ph-4-OCF ₂ CHFOCF ₃ HH
CF ₂ SCH ₃ H Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ HH
CF ₂ SCH ₃ H Ph-4-O (L-45g) HH
CF ₂ SCH ₃ H Ph-3,4-Cl ₂ HH
CF ₂ SCH ₃ H Ph (-3-OCF ₂ O-4-) HH
CF ₂ SCH ₃ H Ph (-3-OCF ₂ CF ₂ O-4-) HH
CF ₂ SCH ₃ H (L-45c) CF ₃ HH
CF ₂ SCH ₃ H L-45f HH
CF ₂ SCH ₃ H (L-46c) CF ₃ HH
CF ₂ SCH ₃ H L-46d HH
CF ₂ SPr-n H Ph-4-CF ₃ HH
CF ₂ SPr-i H Ph-4-OCF ₃ HH
―――――――――――――――――――――――――――――――――――――――
The compounds of the present invention are stored in so-called agricultural pests that harm agricultural and horticultural crops and trees, so-called livestock pests parasitic on livestock and poultry, so-called sanitary pests that cause various adverse effects in human living environments such as houses, and warehouses. It is possible to effectively control low-concentration pests such as so-called stored-grain pests that harm cereals and the like, and mite, nematodes, molluscs, and crustaceans that occur and harm in similar situations.

Specific examples of insects, mites, nematodes, molluscs and crustaceans that can be controlled using the compounds of the present invention include, for example,
Plutella xylostella, Agrotis ipsilon, Agrotis segetum, Helicoverpa armigera, Tobacco moth (Helicoverpa zea), Cotton ball worm (Helicoverpa zea), Tobacco budworm (Heliothis virescens) ), Naranga aenescens, Plusia nigrisigna, Pseudaletia separata, Spodoptera exigua, Spodoptera litura, Spodoptera litura, pod worm Worm (Spodoptera eridania), Tomato horn worm (Manduca quinquemaculata), Tobacco horn worm (Manduca sexta), Grapeberry moss (Endopiza viteana), Ginmon peach moth (Lyonetia prunifoliella malinella), Kinmonhosoga (Phyllonorycter ringone moth) llocnistis citrella), cotton beetle (Pectinophora gossypiella), peach scallop (Carposina niponensis), apple wolfberry (Adoxophyes orana faciata), tea wolfberry (Adoxophyes honmai), chadki (Homona magnamina), ydla molesta, Chilo suppressalis, Cnaphalocrocis medinalis, Hellula undalis, European corn borer (Ostrinia nubilalis), Soybean looper (Pseudoplusia includens), Irrigating tribe (Trichoplusia nitriphan) cunea), Lepidoptera (Pieris rapae crucivora), Lepidoptera (Parnara guttata) and other Lepidoptera pests,
Douganebubui (Anomala cuprea), Japanese beetle (Anomala rufocuprea), Japanese beetle (Popillia japonica), Colorado potato beetle (Lepinotarsa decemlineata), Common beetle (Epilachna varivestis), Japanese horned beetle (Melanotus ramsu) Pepper (Epuraea domina), Henosepilachna vigintioctopunctata, Tenebrio molitor, Tribobrium castaneum, Monchorus turkey ), Leaf beetle (Aulacophora femoralis), rice beetle (Oulema oryzae), Phyllotreta striolata, Cylas formicarius, cotton weevil (Anthonomus grandis), rice weevil (Ethinocnemus squa) Alfata weevil (Hypera postica), rice weevil (Lissorhoptrus oryzophilus), hornbill (Sitophilus zeamais), hornet weevil (Sphenophrus venatus vestius), granary weevil (Sitophilus granarius), Southern corn root worm (Diabata ica) Crustacea pests such as root worms (Diabrotica virgifera), Northern corn root worms (Diabrotica barberi), Aobaarigatatae (Paederus fuscipes),
Sea turtle (Eurydema rugosa), White-headed bug (Eysarcoris ventralis), White-headed bug (Halyomorpha mista), Southern stink bug (Nezara viridula), Spider-headed bug (Leptocorisa chinensis), White-headed bug (Riptortus clam) hemipterus), tarnished plant bug (Lygus lineolaris), cotton-free hopper (Psuedatomoscelis seriatus), azalea (Stephanitis pyrioides), butterfly (Epiacanthus stramineus), tea-nosed leafhopper (Empoasca onukii), potato leaf Empoasca fabae), leafhopper leafhopper (Nephotettix cinctinceps), brown leafhopper (Laodelphax striatellus), leafhopper (Nilaparvata lugens), white leafhopper (Sogatella furcifera), leafworm (Trioza erytreae), leafworm (Trioza erytreae) Bemisia tabaci, Dialeurodes citri, Trialeurodes vaporariorum, Cotton aphid (Aphis gossypii), Aphis pomi, Myphis persicae, Icha pula Scale insects (Icerya purchasi), citrus scale insects (Planococcus citri), scallop scale insects (Pseudococcus comstocki), ruby beetle (Ceroplastes rubens), hornworm scale insects (Unaspis yanonensis), insect lice (Cimex lectularius), etc.
Thrips palma, Thrips tabaci, Thrips tabaci, Thrips tabaci, Thrips tabaci, Thrips tabaci
Drosophila (Dacus dorsalis), Drosophila (Dacus cucurbitae), Drosophila fruit fly (Ceratitis capitata), Green leaf fly (Hydrellia griseola), Drosophila flyfly (Liriomyza bryoniae), Larimyza flies (Liriomyza flies) pomonella, fly Hessian (Mayetiola destructor), housefly (Musca domestica), flies (Stomoxys calcitrans), sheep flies (Melophagus ovinus), bullflies (Hypoderma bovis), dwarf flies (Hypoderma lineatum), opalese vis , Glossina morsitans), Prosimulium yezoensis, cattle fly (Tabanus trigonus), giant fly (Telmatoscopus albipunctatus), red-footed hawk (Leptoconops nipponensis), Acacia (Culex pipiens pallens), Laka (Anopheles hyracanus sinesis) Diptera pests such as,
Bumblebee (Apethymus kuri), Bumblebee (Athalia rosae japonensis), Bumblebee (Neodiprion sertifer), Guntai ant (Eciton burchelli, Eciton schmitti), Black-headed ant (Camponotus japonicus), Mysticia sp. (Solenopsis spp.), Pharaoh ant (Monomorium pharaonis), etc.
Reticulate pests such as black cockroach (Periplaneta fuliginosa), cockroach (Periplaneta japonica), German cockroach (Blattella germanica),
Straight insect pests such as telegryllus emma, kerat (Gryllotalpa africana), locust migratoria, loxta yezoensis, mackerel grasshopper (Schistocerca gregaria),
Termite insect pests such as termites (Coptotermes formosanus), Yamato termites (Reticulitermes speratus), Thai termites (Odontotermes formosanus),
Pesticides such as cat fleas (Ctenocephalidae felis), human fleas (Pulex irritans), and keops mouse fleas (Xenopsylla cheopis),
White-eye pests such as chicken lice (Menacanthus stramineus) and bovine lice (Bovicola bovis),
Lice insect pests such as cattle lice (Haematopinus eurysternus), pig lice (Haematopinus suis), cattle white lice (Linognathus vituli), horned lice (Solenopotes capillatus),
Spider mites (Panonychus citri), apple spider mite (Panonychus ulmi), Kanzawa spider mite (Tetranychus kanzawai), spider mites (Tetranychus urticae), etc.
Acarphylla theae, Scarlet mite (Aculops pelekassi), Scarlet mite (Eriophyes chibaensis), Tulip mite (Aceria tulipae), etc.
Dust mites such as tea dust mite (Polyphaotarsonemus latus), cyclamen dust mite (Steneotarsonemus pallidus),
Acarid mites (Tyrophagus putrescentiae), Robin mite (Rhizoglyphus robini),
Bee mites such as honeybee mite (Varroa jacobsoni),
Ticks, such as the tick (Boophilus microplus), the spider tick (Haemaphysalis longicornis),
Cucumber mites such as sheep cucumber mites (Psoroptes ovis),
Spider mites such as Scaroptes scabiei,
Crustaceans, such as Armadillidium vulgare,
Red-bellied nematode (Prathylenchus penetrans), Kurumi-gure-saenchu (Prathylenchus vulnus), Potato-cyst nematode (Globodera rostochiensis), Soybean-cyst nematode (Heterodera glycines), Red-tailed nematode Nematodes such as (Bursaphelenchus lignicolus),
Mollusks such as Ponacea canaliculata, slug (Incilaria bilineata), Austa despecta sieboldiana, Mishaimai (Euhadra peliomphala),
However, the present invention is not limited to these examples.

  Furthermore, the compound of the present invention is also effective against pests that have developed resistance to existing insecticides such as organophosphorus compounds, carbamate compounds, and pyrethroid compounds.

  That is, the compounds of the present invention are: Diptera, Thripidae, Hemiptera, Lepidoptera, Coleoptera, Hymenoptera, Diptera, Reticulates, Isoptera, Termites, Mites, Lice and Nematodes It is possible to effectively control the insect pests at a low concentration. On the other hand, the compounds of the present invention have extremely useful features that have almost no adverse effects on mammals, fish, crustaceans and beneficial insects.

  When using the compound of the present invention, it is usually mixed with a suitable solid carrier or liquid carrier, and if desired, a surfactant, penetrant, spreading agent, thickener, antifreezing agent, binder, anti-caking agent. , Disintegrating agents, antifoaming agents, preservatives and anti-degradation agents, etc., and soluble concentrate, emulsion (emulsifiable concentrate), wettable powder, water-soluble powder, granular water Water dispersible granule, water soluble granule, suspension concentrate, concentrated emulsion, suspoemulsion, microemulsion, dustable powder ), Granule tablets, and emulsifiable gels, and can be put to practical use. Further, from the viewpoint of labor saving and safety improvement, the preparations of any of the above dosage forms can be provided by being enclosed in a water-soluble package such as a water-soluble capsule and a bag of a water-soluble film.

  Examples of the solid carrier include quartz, calcite, gypsum, dolomite, chalk, kaolinite, pyrophyllite, sericite, halosite, metahalosite, kibushi clay, glazed clay, porcelain stone, siegrite, and allophane. Natural minerals such as shirasu, kira, talc, bentonite, activated clay, acid clay, pumice, attapulgite, zeolite and diatomaceous earth, for example, calcined clay, perlite, shirasu balloon, vermiculite, attapulgus clay and calcined diatomaceous earth Baked products such as magnesium carbonate, calcium carbonate, sodium carbonate, sodium bicarbonate, ammonium sulfate, sodium sulfate, magnesium sulfate, diammonium hydrogen phosphate, ammonium dihydrogen phosphate and potassium chloride, such as glucose, fructose , And Saccharides such as sugar and lactose, polysaccharides such as starch, powdered cellulose and dextrin, organic materials such as urea, urea derivatives, benzoic acid and benzoic acid salts, such as wood flour, cork flour, corn cob, walnut shell and Examples include plants such as tobacco stalks, fly ash, white carbon (for example, hydrous synthetic silica, anhydrous synthetic silica, hydrous synthetic silicate, etc.) and fertilizers.

Examples of the liquid carrier include xylene, alkyl (C ₉ or C ₁₀ etc.) benzene, phenyl xylyl ethane and alkyl (C ₁ or C ₃ etc.) naphthalene and other aromatic hydrocarbons, machine oil, normal paraffin, isoparaffin and Aliphatic hydrocarbons such as naphthene, mixtures of aromatic and aliphatic hydrocarbons such as kerosene, alcohols such as ethanol, isopropanol, cyclohexanol, phenoxyethanol and benzyl alcohol, ethylene glycol, propylene glycol, diethylene glycol, hexylene glycol , Polyhydric alcohols such as polyethylene glycol and polypropylene glycol, propyl cellosolve, butyl cellosolve, phenyl cellosolve, propylene glycol monomethyl ether, propylene Ethers such as recall monoethyl ether, propylene glycol monopropyl ether, propylene glycol monobutyl ether and propylene glycol monophenyl ether, ketones such as acetophenone, cyclohexanone and γ-butyrolactone, fatty acid methyl esters, dialkyl esters of succinic acid, dialkyl esters of glutamic acid, adipine esters such as dialkyl ester and dialkyl phthalate esters, N- alkyl (C _1, C ₈ or C _12, etc.) acid amide pyrrolidone, soybean oil, linseed oil, rapeseed oil, coconut oil, such as cottonseed oil and castor oil Examples include fats and oils, dimethyl sulfoxide and water.

  These solid and liquid carriers may be used alone or in combination of two or more.

  Examples of the surfactant include polyoxyethylene alkyl ether, polyoxyethylene alkyl (mono or di) phenyl ether, polyoxyethylene (mono, di or tri) styryl phenyl ether, polyoxyethylene polyoxypropylene block copolymer, polyoxyethylene Ethylene fatty acid (mono or di) ester, sorbitan fatty acid ester, polyoxyethylene sorbitan fatty acid ester, castor oil ethylene oxide adduct, acetylene glycol, acetylene alcohol, ethylene oxide adduct of acetylene glycol, ethylene oxide adduct of acetylene alcohol and alkyl Nonionic surfactants such as glycosides, alkyl sulfate esters, alkylbenzene sulfonates, lignin sulfonates, Killsulfosuccinate, naphthalenesulfonate, alkylnaphthalenesulfonate, salt of formalin condensate of naphthalenesulfonic acid, salt of formalin condensate of alkylnaphthalenesulfonic acid, polyoxyethylene alkyl ether sulfate or phosphate ester salt, polyoxy Ethylene (mono or di) alkyl phenyl ether sulfate or phosphate ester salt, polyoxyethylene (mono, di or tri) styryl phenyl ether sulfate or phosphate ester salt, polycarboxylate (eg polyacrylate, polymaleate and Copolymers of maleic acid and olefins, etc.) and anionic surfactants such as polystyrene sulfonates, cationic surfactants such as alkylamine salts and alkyl quaternary ammonium salts, amino acid types and beties Amphoteric surfactants such as mold, and silicone-based surfactants and fluorinated surfactants.

  The content of these surfactants is not particularly limited, but is usually preferably in the range of 0.05 to 20 parts by weight with respect to 100 parts by weight of the preparation of the present invention. These surfactants may be used alone or in combination of two or more.

  The application amount of the compound of the present invention varies depending on the application scene, application time, application method, cultivated crops, etc., but generally 0.005 to 50 kg per hectare (ha) is appropriate as the amount of active ingredient.

  Next, formulation examples of the preparation when the compound of the present invention is used are shown. However, the formulation examples of the present invention are not limited to these. In the following formulation examples, “parts” means parts by weight.

[Wettable powder]
Compound of the present invention 0.1 to 80 parts Solid carrier 5 to 98.9 parts Surfactant 1 to 10 parts Others 0 to 5 parts Other examples include anti-caking agents and decomposition inhibitors.

[Milk]
Compound of the present invention 0.1 to 30 parts Liquid carrier 45 to 95 parts Surfactant 4.9 to 15 parts Others 0 to 10 parts Others include, for example, spreading agents, decomposition inhibitors and the like.

[Suspension]
Compound of the present invention 0.1 to 70 parts Liquid carrier 15 to 98.89 parts Surfactant 1 to 12 parts Others 0.01 to 30 parts Others include, for example, antifreezing agents and thickeners.

(Granule wettable powder)
Compound of the present invention 0.1 to 90 parts Solid carrier 0 to 98.9 parts Surfactant 1 to 20 parts Others 0 to 10 parts Others include, for example, binders and decomposition inhibitors.

(Liquid)
Compound of the present invention 0.01 to 70 parts Liquid carrier 20 to 99.99 parts Others 0 to 10 parts Other examples include antifreezing agents and spreading agents.

[Granule]
Compound of the present invention 0.01 to 80 parts Solid carrier 10 to 99.99 parts Others 0 to 10 parts Others include, for example, binders, decomposition inhibitors and the like.

[Dust]
Compound of the present invention 0.01 to 30 parts Solid support 65 to 99.99 parts Others 0 to 5 parts Other examples include a drift inhibitor and a decomposition inhibitor.

  Next, although the formulation example which uses this invention compound as an active ingredient is shown more concretely, this invention is not limited to these.

  In the following formulation examples, “parts” means parts by weight.

[Formulation Example 1] wettable powder Compound No. 1-038 of the present invention 20 parts Pyrophyllite 74 parts Solpol 5039 4 parts (mixture of nonionic surfactant and anionic surfactant: Toho Chemical Co., Ltd.) Product name)
Carplex # 80D 2 parts (Synthetic hydrous silicic acid: Shionogi & Co., Ltd. trade name)
The above is uniformly mixed and ground to obtain a wettable powder.

[Formulation Example 2] Milk Compound of the Present Invention No. 1-038 5 parts Xylene 75 parts N-methylpyrrolidone 15 parts Solpol 2680 5 parts (mixture of nonionic surfactant and anionic surfactant: Toho Chemical Industry (Product name)
The above is uniformly mixed to obtain an emulsion.

[Composition Example 3] Suspension Agent Compound No. 1-038 of this invention 25 parts Agrisol S-710 10 parts (Nonionic surfactant: Kao Corporation trade name)
LUNOX 1000C 0.5 part (anionic surfactant: Toho Chemical Industries, Ltd. trade name)
Xanthan gum 0.2 parts water 64.3 parts After uniformly mixing the above, wet pulverize to make a suspension.

[Composition Example 4] Granule wettable powder Compound No. 1-038 of the present invention 75 parts Hytenol NE-15 5 parts (anionic surfactant: trade name of Daiichi Kogyo Seiyaku Co., Ltd.)
Vanillex N 10 parts (anionic surfactant: Nippon Paper Industries Co., Ltd. trade name)
Carplex # 80D 10 parts (Synthetic hydrous silicic acid: Shionogi Pharmaceutical Co., Ltd. trade name)
After uniformly mixing and pulverizing the above, a small amount of water is added, stirred and mixed, granulated with an extrusion granulator, and dried to obtain a granulated wettable powder.

[Formulation Example 5] Granule Compound No. 1-038 of the present invention 5 parts Bentonite 50 parts Talc 45 parts And dried to form granules.

[Composition Example 6] Powder Compound of the present invention No. 1-038 3 parts Carplex # 80D 0.5 part (synthetic hydrous silicic acid: Shionogi & Co., Ltd. trade name)
Kaolinite 95 parts Diisopropyl phosphate 1.5 parts The above is uniformly mixed and ground to obtain a powder.

  In use, the above preparation is diluted 1 to 10000 times with water or sprayed directly without dilution.

  In addition, when using the compound of the present invention as an agrochemical, other types of herbicides, various insecticides, acaricides, nematicides, fungicides, plant growth regulators, as necessary, when formulated or sprayed, You may mix and apply with a synergist, a fertilizer, a soil improvement agent, etc.

  In particular, when mixed with other pesticides or plant hormones, the cost can be reduced by reducing the amount of applied medicine, the insecticidal spectrum can be expanded by the synergistic action of the mixed drugs, and higher pest control effects can be expected. At this time, a combination with a plurality of known agricultural chemicals is also possible. Examples of the type of agricultural chemical used in combination with the compound of the present invention include compounds described in the Farm Chemicals Handbook 1999 edition. Specific examples of common names are as follows, but the general names are not necessarily limited to these.

  Bactericides: acibenzolar-S-methyl, acylaminobenzamide, amobam, ampropyfos, anilazine, azaconazole, azoxystrobin ( azoxystrobin), benalaxyl, benodanil, benomyl, benthiazole, benzamacril, binapacryl, biapacryl, biphenyl, bitertanol, beoxazine, beoxazine (Bordeaux mixture), blasticidin-S (blasticidin-S), bromoconazole, bupirimate, buthiobate, calcium polysulfide, captafol, captan ) 、 Kappa -Copper oxychloride, carpropamid, carbendazim, carboxin, CGA-279202 (test name), chinomethionat, clobenthiazone, chlorfenazol, Chloroneb, chlorothalonil, chlozolinate, cufraneb, cymoxanil, cyproconazol, cyprodinil, cyprofuram, dazomet deazot ), Dichlorophen, diclobutrazol, diclhlofluanid, diclomedine, dicloran, diethofencarb, diclocymet ), Difenoconazole, diflumetorim, dimethirimol, dimethomorph, diniconazole, dinicoazole-M, dinocap, diphenylamine, diphenylamine, dithiomine , Ditalimfos, dithianon, dodemorph, dodine, drazoxolon, edifenphos, epoxiconazole, etaconazole, ethirimol, etirimol etridiazole), famoxadone, fenarimol, febuconazole, fenamidone, fendazosulam, fenfuram, fe Hexhexamid, fenpiclonil, fenpropidin, fenpropimorph, fentin, ferbam, ferimzone, fluazinam, fludioxonil, fluoro Fluoride, fluquinconazole, flusilazole, flusulfamide, flutolanil, flutriafol, folpet, fosetyl-aluminium, fuberidazole (Fuberidazole), flaxaxyl (fururalaxyl), furametpyr, guazatine, hexachlorobenzene, hexaconazole, hymexazol, imaza Imazalil, imibenconazole, iminoctadine, ipconazole, iprobenfos, iprodione, isoprothiolane, iprovalicarb, cingamycin, kasugamycin (Kresoxim-methyl), mancopper, mancozeb, maneb, maneb, mepanipyrim, mepronil, metalaxyl, metconazole, methasulfocarb, methylasulfocarb (Metiram), metominostrobin, microbutanil, MTF-753 (test name), nabam, nickel bis (dimethyldithiocarbamate), nitroter -Isopropyl (nitrothal-isopropyl), nuarimol, NNF-9425 (test name), octhilinone, offurace, oxadixyl, oxycarboxin, oxypoconazole fumarate (Oxpoconazole fumarate), pefurzoate, penconazole, pencicuron, phthalide, piperalin, polyoxins, potassium hydrogen carbonate, probenazole, prochloraz (Prochloraz), procymidone, propamocarb hydrochloride, propiconazole, propineb, pyrazophos, pyrifenox, pyrimethanil, pyromethanil Pyroquilon, quinomethionate, quinoxyfen, quintozene, RH7281 (study name), sodium hydrogen carbonate, sodium hypochlorite, sulfur, Spiroxamine, tebuconazole, tecnazene, tetraconazole, thiabendazole, thiadiazin / milneb, thifluzamide, thiophanate-methyl, thiophanate-methyl thiram), tolclofos-methyl, tolylfluanid, triadimefon, triadimenol, triazoxide, tricyclazole, tridemorph, triflumi Triflumizole, triforine, triticonazole, validamycin, vinclozolin, zinc sulfate, zineb, ziram and shiitake mycelium extract Such.

  Bactericides: streptomycin, tecloftalam, oxyterracycline and oxolinic acid.

  Nematicides: aldoxycarb, cadusafos, fosthiazate, fosthietan, oxamyl and fenamiphos.

  Acaricides: acequinocyl, amitraz, bifenazate, bromopropylate, chinomethionate, chlorobezilate, clofentezine, cyhexatine, Dicofol, dienochlor, etoxazole, fenazaquin, fenbutatin oxide, fenpropathrin, fenproximate, halfenprox, halfenprox, Hexythiazox, milbemectin, propargite, pyridaben, pyrimidifen and tebufenpyrad.

  Insecticides: abamectin, acephate, acetamipirid, aldicarb, allethrin, azinphos-methyl, bendiocarb, benfuracarb, benfuracarb bensultap), bifenthrin, buprofezin, butocarboxim, carbaryl, carbofuran, carbofuran, carbosulfan, cartap, chlorfenapyr, chlorpyrifos ), Chlorfenvinphos, chlorfluazuron, clothianidin, chromafenozide, chlorpyrifos-methyl, cycloprotorin ( cycloprothrin), cyfluthrin, beta-cyfluthrin, cypermethrin, cyromazine, cyhalothrin, lambda-cyhalothrin, deltamethrin, diafenthiu Ron (diafenthiuron), diazinon, diacloden, diflubenzuron, dimethylvinphos, diofenolan, disulfoton, dimethoate, emamectin-benzoate, emamectin-benzoate EPN, esfenvalerate, ethiofencarb, ethiprole, etofenprox, etrimfos, fenitrothion, fenob Carb (fenobucarb), phenoxycarb (fenoxycarb), fenpropathrin (fenpropathrin), fenvalerate, fipronil, fluacrypyrim (fluacrypyrim), flucythrinate, flufenoxuron, flufenoxuron Flufenprox, tau-fluvalinate, fonophos, formetanate, formothion, furathiocarb, halofenozide, hexaflumuron, hydra Methylnon (hydramethylnon), imidacloprid (isoidaphos), indoxacarb (indoxacarb), isoprocarb (isoprocarb), isoxathion (isoxathion), lufenuron (lufenuron), malathion (ma lathion, metalaldehyde, methamidophos, methidathion, methacrifos, metalcarb, methomyl, metoprene, methoxychlor, methoxyfenozide, monochrome Monofotophos, muscalure, nidinotefuran, nitenpyram, omethoate, oxydemeton-methyl, oxamyl, parathion, parathion-parathion -methyl), permethrin, phenthoate, phothom, phorate, phosalone, phosmet, phosphamidon, pirimicarb b), pirimiphos-methyl, profenofos, protrifenbute, pyrometrozine, pyraclofos, pyriproxyfen, rotenone, sulprofos ), Silafluofen, spinosad, sulfotep, tebfenozide, teflubenzuron, tefluthorin, terbufos, tetrachlorvinphos, iacloprid, iacloprid Thiocyclam, thiodicarb, thiamethoxam, thiofanox, thiometon, tolfenpyrad, tralomethrin, trichlorphone (Trichlorfon), triazuron, triflumuron and vamidion.

  Hereinafter, the present invention will be described in more detail by specifically describing synthesis examples and test examples of the compounds of the present invention as examples, but the present invention is not limited thereto.

[Synthesis example]
Synthesis example 1
N ¹ - [4- [1- hydroxy-1- (5-trifluoromethyl-2-yl) ethyl] -2-methylphenyl] -3-iodo -N ² - isopropyl phthalic acid diamide (present invention compound No .2-001).

Step 1: Preparation of 2-cyano-5-trifluoromethylpyridine 19.4 g of zinc cyanide and tetrakistriphenylphosphine palladium in a solution of 15.0 g of 2-chloro-5-trifluoromethylpyridine in 150 ml of N, N-dimethylformamide 9.6 g was added, and the mixture was stirred at 80 ° C. for 3 hours under a nitrogen atmosphere. After completion of the reaction, the reaction mixture was allowed to cool to room temperature, poured into 300 ml of dilute aqueous ammonia, and extracted with 300 ml of diethyl ether. The organic layer was washed with 200 ml of saturated brine, dried over anhydrous magnesium sulfate, the solvent was distilled off under reduced pressure, and the residue was purified by distillation under reduced pressure (96.0-99.0 ° C./40 mmHg). 9 g was obtained as white crystals.
Melting point: 36.0-38.0 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ 9.00 (bs, 1H), 8.13 (dd, J = 8.3, 2.1 Hz, 1H), 7.87 (d, J = 8.3 Hz, 1H).

Step 2: Preparation of 2-acetyl-5-trifluoromethylpyridine Methylmagnesium bromide in a solution of 4.7 g of 2-cyano-5-trifluoromethylpyridine under nitrogen atmosphere in 40 ml of tetrahydrofuran at −78 ° C. with stirring 35.0 ml of a tetrahydrofuran solution (0.93M) was added dropwise, and after completion of the dropwise addition, the temperature was raised to room temperature and stirring was continued for another 1 hour at room temperature. After completion of the reaction, the reaction mixture was poured into 100 ml of 2N hydrochloric acid and extracted with 200 ml of ethyl acetate. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure to obtain 4.5 g of the desired product as a brown oily substance.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.95 (bs, 1H), 8.16 (d, J = 8.4 Hz, 1H), 8.08 (dd, J = 8.4, 2.1 Hz, 1H), 2.76 ( s, 3H).

Step 3; Preparation of 4- [1-Hydroxy-1- (5-trifluoromethylpyridin-2-yl) ethyl] -2-methylcarbanilide acid-t-butyl 4-Iodo-2-under nitrogen atmosphere 12.5 ml of n-butyllithium (1.57M hexane solution) was added dropwise to a solution of 3.0 g of methylcarbanilide acid-tert-butyl in 40 ml of t-butylmethyl ether with stirring at -50 ° C. Thereafter, the temperature was raised to 0 ° C. and the mixture was further stirred for 30 minutes. Subsequently, this reaction mixture was cooled to -78 ° C, 1.7 g of 2-acetyl-5-trifluoromethylpyridine was added, the temperature was gradually raised to 0 ° C, and stirring was continued for 14 hours at the same temperature. After completion of the reaction, 100 ml of saturated aqueous ammonium chloride solution was added to the reaction mixture, the organic layer was separated, and the aqueous layer was extracted with 100 ml of ethyl acetate. The organic layers were combined and dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 9-2: 3) to obtain 1.3 g of the objective product as a brown solid.
Melting point 132.0-134.5 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.79 (bs, 1H), 7.86 (dd, J = 8.3, 2.1 Hz, 1H), 7.77 (d, J = 8.3 Hz, 1H), 7.42 ( d, J = 8.3Hz, 1H), 7.2-7.3 (m, 2H), 6.24 (bs, 1H), 5.23 (s, 1H), 2.22 (s, 3H), 1.92 (s, 3H), 1.51 (s , 9H).

Step 4; Preparation of 1- (4-amino-3-methylphenyl) -1- (5-trifluoromethylpyridin-2-yl) ethanol 4- [1-hydroxy-1- (5-trifluoromethylpyridine- To 0.4 g of 2-yl) ethyl] -2-methylcarbanilide acid-t-butyl, 3.0 ml of trifluoroacetic acid was added dropwise with stirring under ice cooling. After stirring for 20 minutes at room temperature, 50 ml of saturated aqueous potassium carbonate solution was added under ice cooling, extracted with 30 ml of chloroform, the organic layer was dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. 0.27 g of product was obtained as a brown oil.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.78 (bs, 1H), 7.84 (dd, J = 8.3, 2.1 Hz, 1H), 7.43 (d, J = 8.3 Hz, 1H), 7.05- 7.15 (m, 2H), 6.61 (d, J = 8.3Hz, 1H), 5.15 (s, 1H), 3.59 (bs, 2H), 2.13 (s, 3H), 1.90 (s, 3H).

Step 5; N ¹ - preparation of isopropyl phthalic diamides - [4- [1-hydroxy-1- (4-trifluoromethyl-2-yl) ethyl] -2-methylphenyl] -3-iodo--N ² To a solution of 0.36 g of 3-iodo-N-isopropylphthalamic acid in 5 ml of toluene was added dropwise 0.26 g of trifluoroacetic anhydride at room temperature with stirring. After stirring at the same temperature for 2 hours, the solvent was distilled off under reduced pressure, the residue was dissolved in 3.0 ml of acetonitrile, and 1- (4-amino-3-methylphenyl) -1- (5-trifluoromethyl) was dissolved. 0.27 g of pyridin-2-yl) ethanol was added and stirring was continued at room temperature for 2 hours. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (3: 2) to obtain 0.43 g of the desired product as a brown oily substance. .
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.80 (bs, 1H), 8.29 (bs, 1H), 7.7-8.05 (m, 4H), 7.1-7.5 (m, 4H), 5.84 (d , J = 8.3Hz, 1H), 5.28 (s, 1H), 4.1-4.3 (m, 1H), 2.28 (s, 3H), 1.94 (s, 3H), 1.17 (d, J = 6.6Hz, 6H) .

Synthesis example 2
^{N 1 - [4- [1- (} 4- bromo-difluoromethoxyphenyl) -2,2,2-trifluoro-1-hydroxyethyl] -2-methylphenyl] -3-iodo -N ² - isopropyl phthalic acid diamide (Invention compound No. 1-010).

Step 1: Preparation of 4'-bromodifluoromethoxy-2,2,2-trifluoroacetophenone 2,2,2-trifluoro-4'-hydroxyacetophenone 2.0 g of 1,3-dimethyl-2-imidazolidinone To a 10 ml solution, 0.51 g of 55% oily sodium hydride was added under ice-cooling and stirred at room temperature for 30 minutes. The reaction mixture was then added dropwise to a solution of 11.0 g of dibromodifluoromethane in 10 ml of 1,3-dimethyl-2-imidazolidinone at a rate maintaining the internal temperature of 10 ° C. or lower while stirring with ice cooling. After adding 0.12 g of warm potassium-t-butoxide, stirring was continued for another hour at the same temperature. After completion of the reaction, the reaction mixture was poured into 150 ml of ice water and extracted with 100 ml of diethyl ether. The organic layer was washed with water, dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 19-1: 9) to give 1.83 g of the desired product as a yellow oil.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.16 (d, J = 8.8 Hz, 2H), 7.43 (d, J = 8.8 Hz, 2H).

Step 2; Preparation of 4- [1- (4-Bromodifluoromethoxyphenyl) -2,2,2-trifluoro-1-hydroxyethyl] -2-methylcarbanilide acid-t-butyl 4 under nitrogen atmosphere -Iodo-2-methylcarbanilic acid-t-butyl In a solution of 1.91 g of t-butyl methyl ether in 25 ml, with stirring at -60 ° C, 8.0 ml of n-butyl lithium (1.58 M hexane solution) was added. After the dropwise addition, the temperature was raised to 0 ° C. after completion of the dropwise addition, and the mixture was further stirred for 30 minutes. The reaction mixture was then cooled to -78 ° C, 7.0 g of 4'-bromodifluoromethoxy-2,2,2-trifluoroacetophenone was added, the temperature was gradually raised to 0 ° C, and further 30 minutes at the same temperature. Stirring was continued. After completion of the reaction, the reaction mixture was poured into 100 ml of saturated aqueous ammonium chloride solution, the organic layer was separated, and the aqueous layer was extracted with 50 ml of ethyl acetate. The organic layers were combined and dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 19-1: 4) to obtain 1.0 g of the objective product as a brown oily substance.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300MHz) δ7.87 (d, J = 8.3Hz, 1H), 7.51 (d, J = 8.8Hz, 2H), 7.15-7.35 (m, 4H), 6.32 ( bs, 1H), 3.00 (bs, 1H), 2.24 (s, 3H), 1.52 (s, 9H).

Step 3; Preparation of 1- (4-amino-3-methylphenyl) -1- (4-bromodifluoromethoxyphenyl) -2,2,2-trifluoroethanol 4- [1- (4-Bromodifluoromethoxyphenyl) ) -2,2,2-trifluoro-1-hydroxyethyl] -2-methylcarbanilide acid-t-butyl (1.0 g) was dropwise added with trifluoroacetic acid (3.0 ml) with stirring under ice-cooling. After stirring for 20 minutes at room temperature, 50 ml of saturated aqueous potassium carbonate solution was added under ice cooling, extracted with 50 ml of chloroform, the organic layer was dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. 0.6 g of the product was obtained as brown crystals.
Melting point: 77.5-80.5 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300MHz) δ7.53 (d, J = 8.5Hz, 2H), 7.0-7.25 (m, 4H), 6.61 (d, J = 8.0Hz, 1H), 2.65- 3.15 (bs, 3H), 2.13 (s, 3H).

Step ^{4; N 1 - [4- [} 1- (4- bromo-difluoromethoxyphenyl) -2,2,2-trifluoro-1-hydroxyethyl] -2-methylphenyl] -3-iodo -N ² - isopropyl Preparation of phthalic acid diamide 0.18 g of trifluoroacetic anhydride was added dropwise to a solution of 0.25 g of 3-iodo-N-isopropylphthalamic acid in 5 ml of toluene with stirring at room temperature. After stirring at the same temperature for 1 hour, the solvent was distilled off under reduced pressure, and the residue was dissolved in 3 ml of acetonitrile to give 1- (4-amino-3-methylphenyl) -1- (4-bromodifluoromethoxyphenyl). -2,2,2-trifluoroethanol (0.27 g) was added, and stirring was continued at room temperature for 15 hours. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (2: 3) to obtain 0.13 g of the desired product as brown crystals.
Melting point 97.0-102.5 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ 8.39 (bs, 1H), 8.06 (d, J = 8.8Hz, 1H), 7.96 (d, J = 7.8Hz, 1H), 7.78 (d, J = 8.0Hz, 1H), 7.53 (d, J = 8.8Hz, 2H), 7.1-7.35 (m, 5H), 5.86 (d, J = 8.0Hz, 1H), 4.15-4.3 (m, 1H), 3.16 (s, 1H), 2.30 (s, 3H), 1.17 (d, J = 6.6Hz, 6H).

Synthesis example 3
N ¹ - [4- [2,2,2- trifluoro-1-hydroxy-1- (4-trifluoromethoxyphenyl) ethyl] -2-methylphenyl] -3-iodo -N ² - isopropyl phthalic acid diamide (Invention compound No. 1-009).

Step 1: Preparation of [2,2,2-trifluoro-1-methoxy-1- (4-trifluoromethoxyphenyl) ethyl] trimethylsilane 10.0 g of 1,4-dimethoxymethyl 4-trifluoromethoxybenzoate To a 55 ml solution of ethane, 13.6 g of (trifluoromethyl) trimethylsilane and 0.1 g of cesium fluoride were added with stirring under ice cooling, and the temperature was raised to room temperature over 2 hours with stirring. After further stirring for 1 hour at room temperature, the reaction mixture was poured into 200 ml of ice water, extracted with 200 ml of ethyl acetate, the organic layer was dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with hexane to obtain 16.0 g of the desired product as a colorless oil.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.62 (d, J = 8.5Hz, 2H), 7.23 (d, J = 8.5Hz, 2H), 3.21 (s, 3H), 0.27 (s, 9H).

Step 2: Production of 2,2,2-trifluoro-4′-trifluoromethoxyacetophenone
[2,2,2-trifluoro-1-methoxy-1- (4-trifluoromethoxyphenyl) ethyl] trimethylsilane (16.0 g) in tetrahydrofuran (55 ml) was stirred at room temperature with tetrahydrofuran of tetrabutylammonium fluoride. 9.5 ml of 1M solution was added and stirred at room temperature for 20 minutes. After completion of the reaction, 200 ml of saturated aqueous sodium hydrogen carbonate solution was added to the reaction mixture, extracted with 200 ml of ethyl acetate, the organic layer was dried over anhydrous magnesium sulfate, the solvent was distilled off under reduced pressure, and 10.8 g of the desired product was obtained as a brown oil. Obtained as material.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.15 (d, J = 8.8 Hz, 2H), 7.37 (d, J = 8.8 Hz, 2H).

Step 3; Preparation of 4- [2,2,2-trifluoro-1-hydroxy-1- (4-trifluoromethoxyphenyl) ethyl] -2-methylcarbanilide acid-t-butyl 4 under nitrogen atmosphere -Iodo-2-methylcarbanilic acid-t-butyl 10.0 g of t-butyl methyl ether in 130 ml was stirred at -60 ° C and 41.8 ml of n-butyl lithium (1.58 M hexane solution) was added. After the dropwise addition, the temperature was raised to 0 ° C. after completion of the dropwise addition, and the mixture was further stirred for 30 minutes. The reaction mixture was then cooled to −78 ° C., and 2,2,2-trifluoro-4′-trifluoromethoxyacetophenone (7.75 g) was added, the temperature was gradually raised to 0 ° C., and the temperature was further increased for 30 minutes. Stirring was continued. After completion of the reaction, the reaction mixture was poured into 300 ml of saturated aqueous ammonium chloride solution, the organic layer was separated, and the aqueous layer was extracted with 100 ml of ethyl acetate. The organic layers were combined and dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 19-1: 4) to obtain 9.0 g of the objective product as a colorless oil.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.87 (d, J = 8.5Hz, 1H), 7.50 (d, J = 8.8Hz, 2H), 7.1-7.35 (m, 4H), 6.31 ( bs, 1H), 2.95 (bs, 1H), 2.23 (s, 3H), 1.52 (s, 9H).

Step 4: Production of 1- (4-amino-3-methylphenyl) -2,2,2-trifluoro-1- (4-trifluoromethoxyphenyl) ethanol 4- [2,2,2-trifluoro- 19.0 ml of trifluoroacetic acid was added dropwise to 9.0 g of 1-hydroxy-1- (4-trifluoromethoxyphenyl) ethyl] -2-methylcarbanilide acid-t-butyl under ice-cooling and stirring. After stirring for 30 minutes at room temperature, 200 ml of saturated aqueous potassium carbonate solution was added under ice cooling, extracted with 100 ml of chloroform and 100 ml of ethyl acetate, the organic layers were combined and dried over anhydrous sodium sulfate, and then the solvent was removed under reduced pressure. Was distilled off to obtain 6.8 g of the desired product as yellow crystals.
Melting point 127.0-128.5 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300MHz) δ7.51 (d, J = 8.5Hz, 2H), 7.0-7.25 (m, 4H), 6.60 (d, J = 8.3Hz, 1H), 3.06 ( bs, 3H), 2.13 (s, 3H).

Step 5; N ^1- [4- [2,2,2-trifluoro-1-hydroxy-1- (4-trifluoromethoxyphenyl) ethyl] -2-methylphenyl] -3-iodo-N ² -isopropyl Preparation of phthalic acid diamide 1.0 g of trifluoroacetic anhydride was added dropwise to a solution of 0.2 g of 3-iodo-N-isopropylphthalamic acid in 5 ml of toluene with stirring at room temperature. After stirring at the same temperature for 30 minutes, the solvent was distilled off under reduced pressure, the residue was dissolved in 5 ml of acetonitrile, and 1- (4-amino-3-methylphenyl) -2,2,2-trifluoro-1 -0.2 g of (4-trifluoromethoxyphenyl) ethanol and 1 drop of trifluoroacetic acid were added and stirring was continued for 4 hours at room temperature. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 1) to obtain 0.33 g of the objective product as a colorless resinous substance. It was.
¹ H NMR (CDCl ₃ , Me ₄ Si, 400 MHz) δ 8.39 (bs, 1H), 8.10 (d, J = 8.8Hz, 1H), 7.95 (d, J = 7.6Hz, 1H), 7.80 (d, J = 8.0Hz, 1H), 7.52 (d, J = 8.0Hz, 2H), 7.2-7.35 (m, 5H), 5.90 (d, J = 8.0Hz, 1H), 4.15-4.3 (m, 1H), 3.01 (s, 1H), 2.33 (s, 3H), 1.17 (d, J = 6.6Hz, 6H).

Synthesis example 4
N ^1- [4- [2,2,2-trifluoro-1-hydroxy-1- (2,2,3,3-tetrafluoro-1,4-dioxa-2,3-dihydronaphthalen-6-yl ) Ethyl] -2-methylphenyl] -3-iodo-N ² -isopropylphthalic acid diamide (Compound No. 1-028 of the present invention).

Step 1: Preparation of 2-methyl-4-trifluoroacetylcarbanilic acid-t-butyl In a nitrogen atmosphere, a solution of 10.0 g of 4-iodo-2-methylcarbanilide-t-butyl in 300 ml of diethyl ether was added. While stirring at −10 ° C., 45.0 ml of n-butyllithium (1.5M hexane solution) was added dropwise. After completion of the dropwise addition, the mixture was stirred at the same temperature for 30 minutes. Next, this reaction mixture was cooled to -78 ° C, and 9.5 g of ethyl trifluoroacetate was added dropwise. After completion of the dropwise addition, stirring was continued for another 1 hour at the same temperature. After completion of the reaction, the reaction mixture was heated to −10 ° C. and 100 ml of 2N hydrochloric acid was added and stirred vigorously. Was distilled off. The residue was purified by silica gel column chromatography eluting with diethyl ether-hexane (1: 4) to obtain 3.2 g of the objective product as white crystals.
Melting point: 85.0-87.0 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.25 (d, J = 8.8Hz, 1H), 7.8-8.0 (m, 2H), 6.62 (bs, 1H), 2.32 (s, 3H), 1.55 (s, 9H).

Step 2; 4- [2,2,2-trifluoro-1-hydroxy-1- (2,2,3,3-tetrafluoro-1,4-dioxa-2,3-dihydronaphthalen-6-yl) Preparation of ethyl] -2-methylcarbanilide-t-butyl 2.37 g of 6-bromo-2,2,3,3-tetrafluoro-1,4-dioxa-2,3-dihydronaphthalene under nitrogen atmosphere 5.4 ml of n-butyllithium (1.58 M hexane solution) was added dropwise to a 30 ml solution of t-butyl methyl ether with stirring at -40 ° C. After completion of the dropwise addition, the temperature was raised to 0 ° C and further stirred for 1 hour. . The reaction mixture was then cooled to −50 ° C., and a solution of 1.0 g of 2-methyl-4-trifluoroacetylcarbanilic acid-tert-butyl in 20 ml of t-butyl methyl ether was added dropwise and gradually raised to 0 ° C. Stirring was continued for 1 hour at the same temperature. After completion of the reaction, the reaction mixture was poured into 100 ml of saturated aqueous ammonium chloride solution, the organic layer was separated, and the aqueous layer was extracted with 50 ml of ethyl acetate. The organic layers were combined, dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 4) to obtain 2.3 g of the objective product as a yellow oil.

Step 3; 1- (4-amino-3-methylphenyl) -2,2,2-trifluoro-1- (2,2,3,3-tetrafluoro-1,4-dioxa-2,3-dihydro Preparation of naphthalen-6-yl) ethanol 4- [2,2,2-trifluoro-1-hydroxy-1- (2,2,3,3-tetrafluoro-1,4-dioxa-2,3-dihydro To 2.3 g of naphthalen-6-yl) ethyl] -2-methylcarbanilide acid-t-butyl, 15.0 ml of trifluoroacetic acid was added dropwise with stirring under ice cooling. After stirring for 30 minutes at room temperature, excess trifluoroacetic acid was distilled off under reduced pressure, the residue was dissolved in 100 ml of ethyl acetate, washed with 100 ml of saturated aqueous sodium carbonate solution, saturated brine and then sulfuric anhydride. After dehydration and drying in the order of magnesium, the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (2: 3) and high performance liquid chromatograph eluting with acetonitrile-water (80:20), and 0.5 g of the desired product was obtained as white crystals. Got as.
Melting point: 147.5-150.0 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.33 (s, 1H), 7.24 (d, J = 9.9 Hz, 1H), 7.05-7.1 (m, 3H), 6.58 (d, J = 9.1 Hz, 1H), 3.72 (bs, 2H), 3.45 (bs, 1H), 2.12 (s, 3H).

Step 4; N ^1- [4- [2,2,2-trifluoro-1-hydroxy-1- (2,2,3,3-tetrafluoro-1,4-dioxa-2,3-dihydronaphthalene- 6-yl) ethyl] -2-methylphenyl] -3-iodo-N ² -isopropylphthalic acid diamide 0.15 g of 3-iodo-N-isopropylphthalamic acid in 10 ml of toluene at room temperature with stirring 0.15 g of trifluoroacetic anhydride was added dropwise. After stirring at the same temperature for 30 minutes, the solvent was distilled off under reduced pressure, the residue was dissolved in 3 ml of acetonitrile, and 1- (4-amino-3-methylphenyl) -2,2,2-trifluoro-1 -(2,2,3,3-tetrafluoro-1,4-dioxa-2,3-dihydronaphthalen-6-yl) ethanol (0.15 g) in acetonitrile (5 ml) was added dropwise. Stirring was continued. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (2: 3) to obtain 0.25 g of the desired product as a colorless resinous substance. It was.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.42 (s, 1H), 8.10 (d, J = 8.8 Hz, 1H), 7.9-8.05 (m, 2H), 7.73 (d, J = 7.8 Hz, 1H), 7.05-7.35 (m, 6H), 5.98 (d, J = 8.1Hz, 1H), 4.1-4.25 (m, 1H), 3.69 (s, 1H), 2.28 (s, 3H), 1.16 (d, J = 6.6 Hz, 6H).

Synthesis example 5
N ^1- [4- [2,2,2-Trifluoro-1-hydroxy-1- (4-methanesulfonyloxyphenyl) ethyl] -2-methylphenyl] -3-iodo-N ² -isopropylphthalic acid diamide (Invention compound No. 1-015).

Step 1; Preparation of 4'-hydroxy-3-methyl-4-nitrobenzophenone 4'-methoxy-3-methyl-4-nitrobenzophenone Boron tribromide 2 was added to a solution of 2.0 g of 4'-methoxy-3-methyl-4-nitrobenzophenone in 30 ml of dichloromethane under ice-cooling and stirring. 0.1 ml was added and stirred at room temperature for 20 hours. After completion of the reaction, 2 ml of diethyl ether was added to the reaction mixture and stirred for 10 minutes, then poured into 30 ml of water, and the organic layer was separated. The organic layer was washed with water, dehydrated and dried in the order of saturated saline and then anhydrous sodium sulfate, and reduced pressure. The solvent was distilled off under. The remaining solid was washed with a diisopropyl ether-hexane mixed solvent to obtain 1.8 g of the desired product as pale purple crystals.
Melting point: 146.0-148.0 ° C
¹ H NMR (CDCl ₃ -DMSO-d ₆ , Me ₄ Si, 300 MHz) δ9.71 (bs, 1H), 8.02 (d, J = 8.3 Hz, 1H), 7.55-7.85 (m, 4H), 6.94 ( d, J = 8.3Hz, 2H), 2.68 (s, 3H).

Step 2; Preparation of 4- (3-methyl-4-nitrobenzoyl) phenyl methanesulfonate 4 ml of 4'-hydroxy-3-methyl-4-nitrobenzophenone and 0.20 g of triethylamine 5 ml of N, N-dimethylformamide To the solution, 0.22 g of methanesulfonyl chloride was added with stirring under ice cooling, and the mixture was stirred at the same temperature for 20 minutes. After completion of the reaction, the reaction mixture was poured into 30 ml of water and extracted with 50 ml of diethyl ether. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (2: 5) to obtain 0.54 g of the desired product as a brown oily substance.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ8.05 (d, J = 8.3 Hz, 1H), 7.89 (d, J = 8.8 Hz, 2H), 7.75 (s, 1H), 7.72 (d, J = 8.3Hz, 1H), 7.45 (d, J = 8.8Hz, 2H), 3.25 (s, 3H), 2.66 (s, 3H).

Step 3; Preparation of 4- [1- (4-Amino-3-methylphenyl) -2,2,2-trifluoro-1-hydroxyethyl] phenyl = methanesulfonate 4- (3-Methyl-4-nitrobenzoyl ) To a solution of 0.54 g of phenyl methanesulfonate and 1.5 ml of (trifluoromethyl) trimethylsilane in 3 ml of 1,2-dimethoxyethane, 0.06 g of cesium fluoride is added with stirring under ice cooling, and then the temperature is raised to room temperature. Stirring was continued for another 18 hours. After completion of the reaction, the reaction mixture was poured into 30 ml of water and extracted with 50 ml of diethyl ether. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was dissolved in 3 ml of tetrahydrofuran, and 0.3 ml of a 1M solution of tetrabutylammonium fluoride in tetrahydrofuran was added with stirring at room temperature, followed by stirring at room temperature for 10 minutes. After completion of the reaction, the solvent was distilled off under reduced pressure, 30 ml of water was added, extracted with 30 ml of ethyl acetate, dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the desiccant was filtered off. To the filtrate was added 0.2 g of 5% palladium-carbon, and the mixture was stirred at room temperature for 20 hours in a hydrogen atmosphere. After completion of the reaction, palladium-carbon was filtered off through Celite, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 2 to 2: 3). Purification gave 0.24 g of the desired product as white crystals.
Melting point 137.0-139.0C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.54 (d, J = 8.8Hz, 2H), 7.25 (d, J = 7.7Hz, 2H), 7.11 (s, 1H), 7.09 (d, J = 8.3Hz, 1H), 6.62 (d, J = 9.0Hz, 1H), 3.72 (bs, 2H), 3.16 (s, 3H), 2.94 (bs, 1H), 2.14 (s, 3H).

Step 4: N ^1- [4- [2,2,2-trifluoro-1-hydroxy-1- (4-methanesulfonyloxyphenyl) ethyl] -2-methylphenyl] -3-iodo-N ² -isopropyl Preparation of phthalic acid diamide 0.09 g of trifluoroacetic anhydride was added dropwise to a solution of 0.10 g of 3-iodo-N-isopropylphthalamic acid in 5 ml of toluene with stirring at room temperature. After stirring at the same temperature for 30 minutes, the solvent was distilled off under reduced pressure, the residue was dissolved in 4 ml of acetonitrile, and 4- [1- (4-amino-3-methylphenyl) -2,2,2-trimethyl was dissolved. 0.11 g of fluoro-1-hydroxyethyl] phenyl methanesulfonate and 1 drop of trifluoroacetic acid were added and stirred at room temperature for 18 hours. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 1) to obtain 0.20 g of the desired product as a colorless resinous solid. It was.
Melting point: 111.0-114.0 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ 8.39 (bs, 1H), 8.08 (d, J = 9.1Hz, 1H), 7.97 (d, J = 8.0Hz, 1H), 7.79 (d, J = 7.1Hz, 1H), 7.54 (d, J = 8.8Hz, 2H), 7.15-7.4 (m, 5H), 5.17 (d, J = 8.0Hz, 1H), 4.15-4.3 (m, 1H), 3.17 (s, 3H), 3.07 (s, 1H), 2.30 (s, 3H), 1.17 (d, J = 6.6Hz, 6H).

Synthesis Example 6
N ^1- [4- [3- (4-Chlorophenyl) -1-hydroxy-1-trifluoromethyl-2-propenyl] -2-methylphenyl] -3-iodo-N ² -isopropylphthalic acid diamide (invention) Compound No. 2-018).

Step 1; Preparation of 4- [3- (4-Chlorophenyl) -1-hydroxy-1-trifluoromethyl-2-propenyl] -2-methylcarbanilide acid t-butyl 4-iodo- under nitrogen atmosphere To a solution of 10.0 g of 2-methylcarbanilide acid-t-butyl in 140 ml of t-butylmethyl ether, 41.8 ml of n-butyllithium (1.58 M hexane solution) was added dropwise with stirring at -60 ° C. After completion of the dropwise addition, the temperature was raised to 0 ° C. and further stirred for 30 minutes. The reaction mixture was then cooled to −78 ° C., 7.0 g of 4- (4-chlorophenyl) -1,1,1-trifluoro-3-buten-2-one was added, and the temperature was gradually raised to 0 ° C. Further, stirring was continued for 30 minutes at the same temperature. After completion of the reaction, the reaction mixture was poured into 300 ml of saturated aqueous ammonium chloride solution, the organic layer was separated, and the aqueous layer was extracted with 100 ml of ethyl acetate. The organic layers were combined and dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 9-2: 3) and alumina column chromatography eluting with chloroform to obtain 4.2 g of the objective product as a colorless oily substance. It was.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.90 (d, J = 8.1 Hz, 1H), 7.25-7.5 (m, 6H), 6.82 (d, J = 16.0 Hz, 1H), 6.63 ( d, J = 16.0Hz, 1H), 6.31 (bs, 1H), 2.73 (s, 1H), 2.27 (s, 3H), 1.52 (s, 9H).

Step 2: Production of 1- (4-amino-3-methylphenyl) -3- (4-chlorophenyl) -1-trifluoromethyl-2-propen-1-ol 4- [3- (4-chlorophenyl)- 8.0 ml of trifluoroacetic acid was added dropwise to 4.2 g of 1-hydroxy-1-trifluoromethyl-2-propenyl] -2-methylcarbanilide acid-t-butyl with stirring under ice cooling. After stirring at room temperature for 30 minutes, 150 ml of saturated aqueous potassium carbonate solution was added under ice-cooling, extracted with 100 ml of chloroform, the organic layer was dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The remaining solid was washed with 10 ml of diisopropyl ether to obtain 2.4 g of the desired product as white crystals.
Melting point: 126.5-129.0 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.15-7.4 (m, 6H), 6.83 (d, J = 16.0Hz, 1H), 6.55-6.75 (m, 2H), 2.8-3.5 (broad , 3H), 2.17 (s, 3H).

Step ^{3; N 1 - [4- [} 3- (4- chlorophenyl) -1-hydroxy-1-trifluoromethyl-2-propenyl] -2-methylphenyl] -3-iodo -N ² - isopropyl phthalic acid diamide Preparation of 3-iodo-N-isopropylphthalamic acid 1.86 g of trifluoroacetic anhydride 0.86 g was added dropwise to a 20 ml toluene solution at room temperature with stirring. After stirring at the same temperature for 1 hour, the solvent was distilled off under reduced pressure, the residue was dissolved in 10 ml of acetonitrile, and 1- (4-amino-3-methylphenyl) -3- (4-chlorophenyl) -1- 1.0 g of trifluoromethyl-2-propen-1-ol was added and stirring was continued for 3 hours at room temperature. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 9 to 2: 3) to give 1.50 g of the desired product as white crystals. Got as.
Melting point: 108.0-113.0 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 400 MHz) δ8.38 (s, 1H), 8.07 (d, J = 8.8Hz, 1H), 7.96 (d, J = 8.0Hz, 1H), 7.78 (d, J = 8.0Hz, 1H), 7.15-7.5 (m, 7H), 6.83 (d, J = 16.0Hz, 1H), 6.64 (d, J = 16.0Hz, 1H), 5.85 (d, J = 8.4Hz, 1H), 4.15-4.3 (m, 1H), 2.99 (s, 1H), 2.34 (s, 3H), 1.16 (d, J = 6.4Hz, 6H).

Synthesis example 7
^{N 1 - [4- [1- (} 4- chlorophenyl) -2,2,2-trifluoro-1-methoxyethyl] -2-methylphenyl] -3-iodo -N ² - isopropyl phthalic acid diamide (present invention Compound No. 3-002).

Step 1; Preparation of 4- [1- (4-chlorophenyl) -2,2,2-trifluoro-1-hydroxyethyl] -2-methylcarbanilide acid t-butyl 4-iodo- under nitrogen atmosphere To a solution of 3.0 g of 2-methylcarbanilide acid-t-butyl in 40 ml of t-butylmethyl ether, 12.5 ml of n-butyllithium (1.58 M hexane solution) was added dropwise with stirring at -50 ° C. After completion of the dropwise addition, the temperature was raised to 0 ° C. and further stirred for 30 minutes. The reaction mixture was then cooled to -78 ° C, 1.88 g of 4'-chloro-2,2,2-trifluoroacetophenone was added, the temperature was gradually raised to 0 ° C, and the mixture was further stirred at the same temperature for 30 minutes. Continued. After completion of the reaction, 100 ml of saturated aqueous ammonium chloride solution was added to the reaction mixture, the organic layer was separated, and the aqueous layer was extracted with 100 ml of ethyl acetate. The organic layers were combined and dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 9-2: 3) to obtain 2.96 g of the desired product as a colorless transparent oily substance.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.86 (d, J = 8.7 Hz, 1H), 7.40 (d, J = 8.4 Hz, 2H), 7.15-7.35 (m, 4H), 6.30 ( bs, 1H), 2.93 (s, 1H), 2.22 (s, 3H), 1.52 (s, 9H).

Step 2: Preparation of 1- (4-amino-3-methylphenyl) -1- (4-chlorophenyl) -2,2,2-trifluoroethanol 4- [1- (4-chlorophenyl) -2,2, To 2.96 g of 2-trifluoro-1-hydroxyethyl] -2-methylcarbanilide acid-t-butyl, 6.0 ml of trifluoroacetic acid was added dropwise with stirring under ice cooling. After stirring for 20 minutes at room temperature, 70 ml of saturated aqueous potassium carbonate solution was added under ice cooling, extracted with 100 ml of chloroform, the organic layer was dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. 1.80 g of product was obtained as a brown solid.
Melting point 157.0-160.5 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.45 (d, J = 8.8Hz, 2H), 7.28 (d, J = 8.8Hz, 2H), 7.05-7.15 (m, 2H), 6.60 ( d, J = 8.3Hz, 1H), 5.03 (bs, 1H), 3.74 (bs, 2H), 2.12 (s, 3H).

Step 3; Preparation of 4- [1- (4-Chlorophenyl) -2,2,2-trifluoro-1-methoxyethyl] -2-methylaniline 1- (4-Amino-3-methylphenyl) -1- To a solution of 0.5 g of (4-chlorophenyl) -2,2,2-trifluoroethanol in 3 ml of N, N-dimethylformamide was added 0.073 g of 55% oily sodium hydride with stirring on ice, and at room temperature. The mixture was stirred for 20 minutes, then 0.24 g of methyl iodide was added, and stirring was continued for another 2 hours at the same temperature. After completion of the reaction, the reaction mixture was poured into 20 ml of ice water, extracted with 30 ml of ethyl acetate, the organic layer was dried over anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (2: 3) to obtain 0.44 g of the desired product as a brown oily substance.
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ7.2-7.4 (m, 4H), 6.9-7.1 (m, 3H), 6.62 (d, J = 8.3Hz, 1H), 3.71 (bs, 2H ), 3.27 (s, 3H), 2.14 (s, 3H).

Step ^{4; N 1 - [4- [} 1- (4- chlorophenyl) -2,2,2-trifluoro-1-methoxyethyl] -2-methylphenyl] -3-iodo -N ² - isopropyl phthalic acid diamide Preparation of 0.18 g of trifluoroacetic anhydride was added dropwise to a solution of 0.25 g of 3-iodo-N-isopropylphthalamic acid in 5 ml of toluene with stirring at room temperature. After stirring at the same temperature for 1 hour, the solvent was distilled off under reduced pressure, the residue was dissolved in 3.0 ml of acetonitrile, and 4- [1- (4-chlorophenyl) -2,2,2-trifluoro-1 -Methoxyethyl] -2-methylaniline (0.21 g) was added, and stirring was continued at room temperature for 14 hours. After completion of the reaction, the precipitated crystals were separated by filtration and washed with a small amount of acetonitrile to obtain 0.2 g of the desired product as white crystals.
Melting point 211.5-214.0 ° C
¹ H NMR (CDCl ₃ , Me ₄ Si, 300 MHz) δ 8.35 (bs, 1H), 8.09 (d, J = 8.8Hz, 1H), 7.97 (d, J = 7.6Hz, 1H), 7.79 (d, J = 8.0Hz, 1H), 7.15-7.35 (m, 7H), 5.83 (d, J = 8.0Hz, 1H), 4.15-4.3 (m, 1H), 3.30 (s, 3H), 2.31 (s, 3H ), 1.17 (d, J = 6.6 Hz, 6H).

Synthesis example 8
N ^1- [4- [2- (4-Chlorophenoxy) -1-hydroxy-1-trifluoromethylethyl] -2-methylphenyl] -3-iodo-N ² -isopropylphthalic acid diamide (Compound No. of the present invention) .2-004).

Step 1; Preparation of 4- [2- (4-Chlorophenoxy) -1-hydroxy-1-trifluoromethylethyl] -2-methylcarbanilide acid-t-butyl 2-Methyl-4- (1-tri To a solution of 2.0 g of fluoromethyloxiran-1-yl) carbanilide-t-butyl and 1.5 g of 4-chlorophenol in 30 ml of N, N-dimethylformamide was added 0.45 g of 60% oily sodium hydride under ice-cooling and stirring. Was added and stirred at room temperature for 24 hours. After completion of the reaction, the reaction mixture was poured into 150 ml of ice water and extracted with 100 ml of diethyl ether. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 4) to obtain 2.1 g of the objective product as a colorless oil.

Step ^{2; N 1 - [4- [} 2- (4- chlorophenoxy) -1-hydroxy-1-trifluoromethyl-ethyl] -2-methylphenyl] -3-iodo -N ² - preparation of isopropyl phthalic diamides To 1.0 g of 4- [2- (4-chlorophenoxy) -1-hydroxy-1-trifluoromethylethyl] -2-methylcarbanilide acid-t-butyl, trifluoroacetic acid 5. 0 ml was added dropwise. After stirring for 10 minutes at room temperature, excess trifluoroacetic acid was distilled off under reduced pressure to obtain crude 1- (4-amino-3-methylphenyl) -2- (4-chlorophenoxy) -1 -Trifluoromethylethanol was obtained.

To a 10 ml toluene solution of 0.8 g 3-iodo-N-isopropylphthalamic acid, 0.8 g trifluoroacetic anhydride was added dropwise at room temperature with stirring. After stirring at the same temperature for 30 minutes, the solvent was distilled off under reduced pressure, the residue was dissolved in 20 ml of acetonitrile, and the above crude 1- (4-amino-3-methylphenyl) -2- (4-chlorophenoxy) was dissolved. ) -1-Trifluoromethylethanol was added and stirring was continued at room temperature for 3 hours. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-chloroform (2: 3) to obtain 0.7 g of the desired product as white crystals.
Melting point 90.0-95.0 ° C.

Synthesis Example 9
N ^1- [4- [2- (4-chlorophenoxy) -2,2-difluoro-1-hydroxy-1-trifluoromethylethyl] -2-methylphenyl] -3-iodo-N ² -isopropylphthalic acid Diamide (the present compound No. 2-008).

Step 1; Preparation of 1- (2-bromo-1,1,2,3,3,3-hexafluoropropyloxy) -4-chlorobenzene 2,2-dibromo-1,1,2,3,3,3 -To a solution of 20.0 g of hexafluoropropane and 7.0 g of 4-chlorophenol in 100 ml of N, N-dimethylformamide was added 2.2 g of 60% oily sodium hydride under ice-cooling and stirring for 12 hours at room temperature. did. After completion of the reaction, the reaction mixture was poured into 300 ml of ice water and extracted with 150 ml of diethyl ether. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 4) to obtain 18.0 g of the desired product as a colorless oil.

Step 2: Preparation of 4- [2- (4-chlorophenoxy) -1,2,2-trifluoro-1-trifluoromethylethyl] -2-methylaniline 1- (2-Bromo-1,1,2 , 3,3,3-hexafluoropropyloxy) -4-chlorobenzene (5.0 g) and o-toluidine (1.5 g) in 50 ml of dimethyl sulfoxide, with stirring, 1.8 g of sodium bicarbonate and 3.8 g of sodium dithionite. Was added and stirred at 70 ° C. for 3 hours. After completion of the reaction, the reaction mixture was poured into 300 ml of ice water and extracted with 150 ml of diethyl ether. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 4) to obtain 3.8 g of the desired product as a colorless oil.

Step 3; Preparation of 1- (4-amino-3-methylphenyl) -2- (4-chlorophenoxy) -2,2-difluoro-1-trifluoromethylethanol 4- [2- (4-chlorophenoxy) -1,2,2-trifluoro-1-trifluoromethylethyl] -2-methylaniline in an amount of 2.0 g of 1,4-dioxane in 20 ml was added with 3.0 g of potassium hydroxide and heated under reflux for 2 Stir for hours. After completion of the reaction, the solvent was distilled off under reduced pressure, the residue was poured into 100 ml of ice water and extracted with 100 ml of diethyl ether, and the organic layer was dehydrated and dried in the order of saturated brine and anhydrous magnesium sulfate, and the solvent was removed under reduced pressure. Was distilled off. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (2: 3) to obtain 0.6 g of the desired product as a pale yellow oily substance.

Step ^{4; N 1 - [4- [} 3- (4- chlorophenyl) -1-hydroxy-1-trifluoromethyl-2-propenyl] -2-methylphenyl] -3-iodo -N ² - isopropyl phthalic acid diamide Preparation of 0.6 g of trifluoroacetic anhydride was added dropwise to a solution of 0.6 g of 3-iodo-N-isopropylphthalamic acid in 5 ml of toluene with stirring at room temperature. After stirring at the same temperature for 30 minutes, the solvent was distilled off under reduced pressure, and the residue was dissolved in 10 ml of acetonitrile to give 1- (4-amino-3-methylphenyl) -2- (4-chlorophenoxy) -2. , 2-difluoro-1-trifluoromethylethanol 0.5 g was added and stirring was continued at room temperature for 5 hours. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-chloroform (2: 3) to obtain 0.3 g of the objective product as colorless crystals.
Melting point 65.0-75.0 ° C.

Synthesis Example 10
N ^1- (2,2-difluoro-3-hydroxy-5-methyl-3-trifluoromethyl-2,3-dihydrobenzofuran-6-yl) -3-iodo-N ² -isopropylphthalic acid diamide (invention) Compound No. 4-002).

Step 1; Preparation of 1- (2-bromo-1,1,2,3,3,3-hexafluoropropyloxy) -4-methyl-3-nitrobenzene 2,2-dibromo-1,1,2,3 To a solution of 10.0 g of 1,3,3-hexafluoropropane and 5.0 g of 4-methyl-3-nitrophenol in 100 ml of N, N-dimethylformamide was added 1.4 g of 60% oily sodium hydride under ice-cooling. And stirred at room temperature for 12 hours. After completion of the reaction, the reaction mixture was poured into 300 ml of ice water and extracted with 150 ml of diethyl ether. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 4) to obtain 8.0 g of the desired product as a pale yellow oily substance.

Step 2; Preparation of 5- (2-Bromo-1,1,2,3,3,3-hexafluoropropyloxy) -2-methylaniline 1- (2-Bromo-1,1,2,3,3 , 3-Hexafluoropropyloxy) -4-methyl-3-nitrobenzene To a solution of 8.0 g of ethanol in 100 ml of ethanol at room temperature, 9.5 g of tin chloride dihydrate and 15 ml of concentrated hydrochloric acid were added at the same temperature. For 12 hours. After completion of the reaction, the solvent was distilled off under reduced pressure, the residue was poured into 100 ml of 2N aqueous sodium hydroxide solution and extracted with 100 ml of diethyl ether, and the organic layer was dehydrated, dried and dried over anhydrous magnesium sulfate in this order. The solvent was distilled off under. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (1: 4) to obtain 6.0 g of the desired product as a pale yellow oily substance.

Step 3; Preparation of 6-amino-2,2,3-trifluoro-5-methyl-3-trifluoromethyl-2,3-dihydrobenzofuran 5- (2-bromo-1,1,2,3,3 , 3-Hexafluoropropyloxy) -2-methylaniline to a solution of 6.0 g of dimethyl sulfoxide with stirring, 2.2 g of sodium hydrogen carbonate and 4.5 g of sodium dithionite were added and stirred at 70 ° C. for 3 hours. Stir. After completion of the reaction, the reaction mixture was poured into 300 ml of ice water and extracted with 150 ml of diethyl ether. The organic layer was dehydrated and dried in the order of saturated brine and then anhydrous magnesium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by silica gel column chromatography eluting with ethyl acetate-hexane (3: 7) to obtain 3.0 g of the objective product as a colorless oil.

Step 4: Preparation of 6-amino-2,2-difluoro-3-hydroxy-5-methyl-3-trifluoromethyl-2,3-dihydrobenzofuran 6-amino-2,2,3-trifluoro-5- Treatment of 1.0 g of methyl-3-trifluoromethyl-2,3-dihydrobenzofuran with alumina column chromatography eluting with ethyl acetate-methanol (7: 3) gave 0.6 g of the desired product as white crystals. It was.

Step 5; N ¹ - (2,2- difluoro-3-hydroxy-5-methyl-3-trifluoromethyl-2,3-dihydrobenzofuran-6-yl) -3-iodo -N ² - isopropyl phthalic acid diamide Preparation of 0.6 g of trifluoroacetic anhydride was added dropwise to a solution of 0.6 g of 3-iodo-N-isopropylphthalamic acid in 5 ml of toluene with stirring at room temperature. After stirring at the same temperature for 30 minutes, the solvent was distilled off under reduced pressure, the residue was dissolved in 10 ml of acetonitrile, and 6-amino-2,2-difluoro-3-hydroxy-5-methyl-3-trifluoromethyl was dissolved. 0.5 g of -2,3-dihydrobenzofuran was added and stirring was continued for 5 hours at room temperature. After completion of the reaction, the solvent was distilled off under reduced pressure, and the residue was purified by silica gel column chromatography eluting with ethyl acetate-chloroform (1: 1) to obtain 0.4 g of the objective product as colorless crystals.
Melting point: 144.0-146.0 ° C.

  This invention compound can be manufactured according to the said manufacturing method and an Example. Examples of such compounds are shown in Tables 6 to 10, but the present invention is not limited to these.

In the table, the description of i-Pr represents an isopropyl group. Similarly, s-Bu represents a secondary butyl group, t-Bu represents a tertiary butyl group, Ph represents a phenyl group, and 2-Naph represents 2-butyl. Each represents a naphthyl group,
The aromatic heterocycles represented by L-15b to L-45e in the table each represent the following structure.

For example, the notation [(D-15b) CF ₃ ] represents a 1-methyl-5-trifluoromethylpyrazol-3-yl group, and the notation [CH ₂ (L-36a)] is 1,2, Represents a 4-triazol-1-ylmethyl group.

In the table, * 1 means “resinous” and * 2 means “oily”.
Table 6

―――――――――――――――――――――――――――――――――――――――
No. (X) _m R ³ R ⁴ (Z) _p1 mp (℃)
―――――――――――――――――――――――――――――――――――――――
1-001 3-I i-Pr CH ₃ 4-Cl 177.0-179.0
1-002 3-I i-Pr i-Pr 4-Cl 112.0-115.0
1-003 3-I i-Pr CF ₃ 4-F 192.0-194.0
1-004 3-I i-Pr CF ₃ 3-Cl * 1
1-005 3-I i-Pr CF ₃ 4-Cl 107.5-109.5
1-006 3-I i-Pr CF ₃ 4-Br 110.0-113.0
1-007 3-I i-Pr CF ₃ 4-CF ₃ 112.0-114.0
1-008 3-I i-Pr CF ₃ 4-OCH ₃ 102.0-105.0
1-009 3-I i-Pr CF ₃ 4-OCF ₃ * 1
1-010 3-I i-Pr CF ₃ 4-OCF ₂ Br 97.0-102.5
1-011 3-I i-Pr CF ₃ 4-OCF ₂ CHF ₂ 98.0-101.0
1-012 3-I i-Pr CF ₃ 4-OCF ₂ CHFCF ₃ 98.0-101.0
1-013 3-I i-Pr CF ₃ 4-OCF ₂ CHFOCF ₃ 93.0-96.0
1-014 3-I i-Pr CF ₃ 4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ 78.0-80.0
1-015 3-I i-Pr CF ₃ 4-OSO ₂ CH ₃ 111.0-114.0
1-016 3-I i-Pr CF ₃ 3-O (L-45e) 103.5-107.0
1-017 3-I i-Pr CF ₃ 4-O (L-45e) 107.0-109.0
1-018 3-I i-Pr CF ₃ 4-SCH ₃ 100.0-107.5
1-019 3-I i-Pr CF ₃ 4-SO ₂ CH ₃ 150.0-162.0
1-020 3-I i-Pr CF ₃ 2-F-4-Cl * 1
1-021 3-I i-Pr CF ₃ 2,4-Cl ₂ 120.0-124.0
1-022 3-I i-Pr CF ₃ 3,4-Cl ₂ 112.0-113.0
1-023 3-I i-Pr CF ₃ 3,5-Cl ₂ 195.0-197.0
1-024 3-I i-Pr CF ₃ 3,4-Br ₂ 125.0-131.5
1-025 3-I i-Pr CF ₃ 3-Cl-4-OCHF ₂ * 1
1-026 3-I i-Pr CF ₃ 3-CH ₃ -4-OCF ₂ CHFOCF ₃ 92.0-94.0
1-027 3-I i-Pr CF ₃ 3-OCF ₂ O-4 * 1
1-028 3-I i-Pr CF ₃ 3-OCF ₂ CF ₂ O-4 * 1
1-029 3-I i-Pr CF ₃ 3,5-Cl ₂ -4-OCH ₃ 110.0-116.5
1-030 3-I i-Pr C (O) OCH ₃ 4-Cl 133.5-135.0
1-031 3-I s-Bu CF ₃ 4-OCF ₃ * 1
1-032 3-I t-Bu CF ₃ 4-OCF ₃ 151.0-154.0
1-033 3-I CH (CH ₃ ) CH ₂ SCH ₃ i-Pr 4-Cl 105.0-107.0
1-034 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-F 127.0-130.0
1-035 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3-Cl * 1
1-036 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-Cl 95.5-99.0
1-037 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-Bu-t 107.0-111.0
1-038 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-CF ₃ 101.0-103.0
1-039 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OCH ₃ 97.0-99.0
1-040 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OCF ₃ 112.0-115.0
1-041 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OCF ₂ Br * 1
1-042 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OCF ₂ CHF ₂ 93.0-96.0
1-043 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OCF ₂ CHFCF ₃ 91.0-95.0
1-044 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OCF ₂ CHFOCF ₃ 86.0-89.0
1-045 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ 71.0-72.0
1-046 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-OSO ₂ CH ₃ 97.0-100.0
1-047 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3-O (L-45e) * 1
1-048 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-O (L-45e) 105.0-107.0
1-049 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 4-SO ₂ CH ₃ 117.0-120.0
1-050 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 2-F-4-Cl 116.0-120.0
1-051 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 2,4-Cl ₂ 112.0-116.0
1-052 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3,4-Cl ₂ 99.0-103.0
1-053 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3,5-Cl ₂ 121.0-123.5
1-054 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3,4-Br ₂ 108.0-110.0
1-055 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3-Cl-4-OCHF ₂ * 1
1-056 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3-Cl-4-OCF ₃ 83.0-89.0
1-057 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3-CH ₃ -4-OCF ₂ CHFOCF ₃ 86.0-89.0
1-058 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3-OCF ₂ O-4 * 1
1-059 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3-OCF ₂ CF ₂ O-4 * 1
1-060 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 3,5-Cl ₂ -4-OCH ₃ 110.0-113.5
1-061 3-I CH (CH ₃ ) CH ₂ SCH ₃ C (O) OCH ₃ 4-Cl * 1
1-062 3-I CH (CH ₃ ) CH ₂ S (O) CH ₃ CF ₃ 3-Cl 182.0-184.0
1-063 3-I CH (CH ₃ ) CH ₂ S (O) CH ₃ CF ₃ 4-OCF ₃ 229.0-231.0
1-064 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ i-Pr 4-Cl 122.0-124.0
1-065 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-F 142.0-144.0
1-066 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-Cl 180.0-184.0
1-067 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-CF ₃ 111.0-113.0
1-068 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-OCH ₃ 123.0-126.0
1-069 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-OCF ₃ 218.0-220.0
1-070 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-OCF ₂ Br 115.0-117.5
1-071 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-OCF ₂ CHF ₂ 112.0-115.0
1-072 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-OCF ₂ CHFCF ₃ 144.0-146.0
1-073 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-OCF ₂ CHFOCF ₃ 102.0-105.0
1-074 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 4-O (L-45e) 123.0-124.0
1-075 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 2-F-4-Cl 228.0-230.0
1-076 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 2,4-Cl ₂ 125.0-128.0
1-077 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 3,4-Cl ₂ 112.0-114.0
1-078 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 3,5-Cl ₂ 127.0-132.0
1-079 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 3,4-Br ₂ 133.0-145.0
1-080 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 3-Cl-4-OCHF ₂ * 1
1-081 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 3-CH ₃ -4-OCF ₂ CHFOCF ₃ 116.0-118.0
1-082 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 3-OCF ₂ O-4 193.0-203.0
1-083 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 3-OCF ₂ CF ₂ O-4 * 1
1-084 3-IC (CH ₃ ) ₂ CH ₂ SCH ₃ CF ₃ 4-Cl 172.0-175.0
1-085 3-IC (CH ₃ ) ₂ CH ₂ SCH ₃ CF ₃ 4-OCF ₃ * 1
1-086 3-IC (CH ₃ ) ₂ CH ₂ SCH ₃ CF ₃ 3,4-Cl ₂ 96.0-98.0
1-087 3-IC (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ CF ₃ 4-Cl 126.0-128.0
1-088 3-IC (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ CF ₃ 4-OCF ₃ * 1
1-089 3-IC (CH ₃ ) ₂ CH ₂ SO ₂ CH ₃ CF ₃ 3,4-Cl ₂ 109.0-113.0
1-090 3-IC (CH ₃ ) ₂ C≡CH CF ₃ 4-OCF ₃ * 1
―――――――――――――――――――――――――――――――――――――――
Table 7

―――――――――――――――――――――――――――――――――――――――
No. (X) _m R ³ R ⁴ R ⁵ mp (℃)
―――――――――――――――――――――――――――――――――――――――
2-001 3-I i-Pr CH ₃ (L-45c) CF ₃ * 1
2-002 3-I i-Pr CF ₃ CH ₂ CH ₂ (Ph-4-Cl) 103.5-106.0
2-003 3-I i-Pr CF ₃ CH ₂ OCH ₃ 181.0-184.0
2-004 3-I i-Pr CF ₃ CH ₂ O (Ph-4-Cl) 90.0-95.0
2-005 3-I i-Pr CF ₃ CH ₂ OC (O) (Ph-4-Cl) 180.0-183.0
2-006 3-I i-Pr CF ₃ CF ₂ O (Ph-2-Cl) 86.0-88.0
2-007 3-I i-Pr CF ₃ CF ₂ O (Ph-3-Cl) 82.0-85.0
2-008 3-I i-Pr CF ₃ CF ₂ O (Ph-4-Cl) 65.0-75.0
2-009 3-I i-Pr CF ₃ CH ₂ S (Ph-4-Cl) 80.0-83.0
2-010 3-I i-Pr CF ₃ CH ₂ SO ₂ (Ph-4-Cl) 111.0-113.0
2-011 3-I i-Pr CF ₃ CH ₂ N (CH ₃ ) ₂ 204.0-207.0
2-012 3-I i-Pr CF ₃ CH ₂ NH (Ph-4-Cl) 120.0-122.0
2-013 3-I i-Pr CF ₃ CF ₂ C (O) OEt * 1
2-014 3-I i-Pr CF ₃ CH ₂ (L-36a) 149.0-152.0
2-015 3-I i-Pr CF ₃ C (O) OEt 177.0-178.0
2-016 3-I i-Pr CF ₃ CH = CH (Ph-4-F) 109.0-111.0
2-017 3-I i-Pr CF ₃ CH = CH (Ph-3-Cl) * 1
2-018 3-I i-Pr CF ₃ CH = CH (Ph-4-Cl) 108.0-113.0
2-019 3-I i-Pr CF ₃ CH = CH (Ph-4-OCF ₃ ) 104.0-108.5
2-020 3-I i-Pr CF ₃ CH = CH (Ph-4-SCH ₃ ) * 1
2-021 3-I i-Pr CF ₃ CH = CH (Ph-4-SO ₂ CH ₃ ) 133.0-138.0
2-022 3-I i-Pr CF ₃ CH = CH (Ph-3,4-Cl ₂ ) 111.0-113.0
2-023 3-I i-Pr CF ₃ 2-Naph 113.0-117.0
2-024 3-I i-Pr CF ₃ (L-45c) CF ₃ 107.0-110.0
2-025 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ CF ₂ O (Ph-4-Cl) * 1
2-026 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ CH = CH (Ph-4-F) 98.0-111.0
2-027 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ CH = CH (Ph-3-Cl) * 1
2-028 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ CH = CH (Ph-4-Cl) 103.5-108.0
2-029 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) * 1
2-030 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) 98.0-101.0
2-031 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ 2-Naph * 1
2-032 3-I CH (CH ₃ ) CH ₂ SCH ₃ CF ₃ (L-15b) CF ₃ 94.0-97.0
2-033 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ CF ₂ O (Ph-4-Cl) 131.5-135.0
2-034 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ CH = CH (Ph-4-F) 123.0-125.0
2-035 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ CH = CH (Ph-4-Cl) 128.0-130.5
2-036 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ CH = CH (Ph-4-OCF ₃ ) 120.5-125.0
2-037 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ CH = CH (Ph-3,4-Cl ₂ ) 124.0-128.0
2-038 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CF ₃ 2-Naph * 1
―――――――――――――――――――――――――――――――――――――――
Table 8

―――――――――――――――――――――――――――――――――――――――
No. (X) _m R ³ R ⁵ R ⁶ mp (℃)
―――――――――――――――――――――――――――――――――――――――
3-001 3-I i-Pr CF ₂ O (Ph-4-Cl) CH ₃ 55.0-65.0
3-002 3-I i-Pr Ph-4-Cl CH ₃ 211.5-214.0
3-003 3-I i-Pr Ph-4-Cl CH ₂ OCH ₃ 226.5-229.0
3-004 3-I i-Pr Ph-4-Cl C (O) CH ₃ 212.0-214.0
3-005 3-I i-Pr CH = CH (Ph-4-Cl) CH ₃ * 1
3-006 3-I CH (CH ₃ ) CH ₂ SCH ₃ CH = CH (Ph-4-Cl) CH ₃ * 1
3-007 3-I CH (CH ₃ ) CH ₂ SCH ₃ CH = CH (Ph-4-Cl) CH ₂ OCH ₃ * 1
3-008 3-I CH (CH ₃ ) CH ₂ SCH ₃ Ph-4-Cl CH ₃ 103.0-107.0
3-009 3-I CH (CH ₃ ) CH ₂ SCH ₃ Ph-4-Cl CH ₂ OCH ₃ 185.0-188.5
3-010 3-I CH (CH ₃ ) CH ₂ SCH ₃ Ph-4-Cl Si (CH ₃ ) ₃ 113.0-116.0
3-011 3-I CH (CH ₃ ) CH ₂ SCH ₃ Ph-4-OCH ₃ Si (CH ₃ ) ₃ 99.0-103.0
3-012 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CH = CH (Ph-4-Cl) CH ₃ * 1
3-013 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ CH = CH (Ph-4-Cl) CH ₂ OCH ₃ * 1
3-014 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ Ph-4-Cl CH ₃ 111.0-114.0
3-015 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ Ph-4-Cl CH ₂ OCH ₃ * 1
3-016 3-I CH (CH ₃ ) CH ₂ SO ₂ CH ₃ Ph-4-OCH ₃ Si (CH ₃ ) ₃ 115.0-119.0
―――――――――――――――――――――――――――――――――――――――
Table 9

―――――――――――――――――――――――――――――――――――――――
No. (X) _m R ³ (Y) _n R ⁶ mp (℃)
―――――――――――――――――――――――――――――――――――――――
4-001 3-I i-Pr 2-CH ₃ H 123.0-126.0
4-002 3-I i-Pr 6-CH ₃ H 144.0-146.0
4-003 3-I i-Pr 6-CH ₃ Ph-4-Cl 195.0-198.0
―――――――――――――――――――――――――――――――――――――――
Table 10

―――――――――――――――――――――――――――――――――――――――
No. Y ¹ R ⁴ R ⁵ R ⁶ mp (℃)
―――――――――――――――――――――――――――――――――――――――
5-01 CH ₃ CH ₃ (L-45c) CF ₃ H * 2
5-02 CH ₃ CF ₃ C (O) OEt H * 2
5-03 CH ₃ CF ₃ CH = CH (Ph-4-F) H 97.0-99.0
5-04 CH ₃ CF ₃ Ph-4-Cl H 157.0-160.5
5-05 CH ₃ CF ₃ Ph-4-Cl CH ₃ * 2
5-06 CH ₃ CF ₃ Ph-4-OCH ₃ Si (CH ₃ ) ₃ * 2
5-07 CH ₃ CF ₃ Ph-4-OCF ₂ CHF ₂ H 69.0-72.0
5-08 CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₃ H 70.0-75.0
5-09 CH ₃ CF ₃ Ph-4-OCF ₂ CHFOCF ₂ CF ₂ CF ₃ H * 2
5-10 CH ₃ CF ₃ Ph-4-OSO ₂ CH ₃ H 137.0-139.0
5-11 CH ₃ CF ₃ Ph-2,4-Cl ₂ H 149.0-151.0
5-12 CH ₃ CF ₃ Ph-3-CH ₃ -4-OCF ₂ CHFOCF ₃ H 84.0-87.0
5-13 CH ₃ CF ₃ Ph-3-OCF ₂ CF ₂ O-4 H 147.5-150.0
5-14 CH ₃ CF ₃ (L-45c) CF ₃ H 136.0-138.5
―――――――――――――――――――――――――――――――――――――――
[Test example]
Next, the usefulness of the compound of the present invention as a pest control agent will be specifically described in the following test examples, but the present invention is not limited to these.

Test Example 1 Insecticidal test against a diamondback moth A 10% emulsion of the compound of the present invention (for some compounds, 25% wettable powder) was diluted with water containing a spreading agent to prepare a chemical solution having a concentration of 100 ppm. Immerse kanran leaves in this solution for about 10 seconds, air-dry and place in a petri dish. 10 second-instar larvae of Plutella xylostella are released per petri dish and covered with a hole. Housed in a constant temperature room. The number of dead insects after 6 days was investigated, and the death rate was calculated from the same calculation formula as in Test Example 1. The test was conducted in a two-ward system.

As a result, the following compounds showed 100% mortality.
Compound of the present invention: No.1-001,1-002,1-003,1-004,1-005,1-006,1-007,1-008,1-009,1-010,1-011, 1-012,1-013,1-014,1-015,1-016,1-017,1-018,1-019,1-020,1-021,1-022,1-023,1- 024,1-025,1-026,1-027,1-028,1-029,1-030,1-031,1-032,1-033,1-034,1-035,1-036, 1-037,1-038,1-039,1-040,1-041,1-042,1-043,1-044,1-045,1-046,1-047,1-048,1- 050,1-051,1-052,1-053,1-054,1-055,1-056,1-057,1-058,1-059,1-060,1-061,1-062, 1-063,1-064,1-065,1-066,1-067,1-068,1-069,1-070,1-071,1-072,1-073,1-074,1- 075,1-076,1-077,1-078,1-079,1-080,1-081,1-082,1-083,1-084,1-085,1-086,1-087, 1-088,1-089,1-090,2-001,2-002,2-003,2-004,2-005,2-006,2-007,2-008,2-009,2- 010,2-011,2-012,2-013,2-014,2-015,2-016,2-017,2-018,2-019,2-020,2-021,2-022, 2-023, 2-024, 2-025, 2-026, 2-027, 2-028, 2-029, 2-030, 2-031, 2-032, 2-033, 2-034, 2- 035,2-036,2-037,2-038,3-001,3-002,3-004,3-005,3-006,3-007,3-008,3-009,3-010, 3-011, 3-012, 3-013, 3-014, 3-015, 4-001, 4-002.

Test Example 2 Insecticidal test against Spodoptera litura 10% emulsion of the compound of the present invention (depending on the compound, 25% wettable powder was tested) was diluted with water containing a spreading agent to prepare a chemical solution having a concentration of 100 ppm. Immerse kanran leaves in this chemical for about 10 seconds, air dry and place in a petri dish. 10 second-instar larvae of Spodoptera litura are released per petri dish, and a lid with a hole is opened. Housed in a constant temperature room. The number of dead insects after 6 days was investigated, and the death rate was calculated from the following formula. The test was conducted in a two-ward system.

Death rate (%) = (Number of dead insects / Number of dead insects) × 100
As a result, the following compounds showed a death rate of 80% or more.
Compound of the present invention: No.1-001,1-003,1-005,1-006,1-007,1-009,1-010,1-011,1-012,1-013,1-014, 1-015,1-016,1-017,1-020,1-021,1-022,1-023,1-024,1-025,1-026,1-027,1-028,1- 029,1-031,1-032,1-034,1-035,1-036,1-038,1-040,1-041,1-042,1-043,1-044,1-045, 1-047,1-048,1-050,1-051,1-052,1-053,1-054,1-055,1-056,1-057,1-058,1-059,1- 063,1-065,1-066,1-067,1-069,1-070,1-071,1-072,1-073,1-074,1-075,1-076,1-077, 1-078,1-079,1-080,1-081,1-082,1-083,1-084,1-085,1-086,1-087,1-088,1-089,1- 090,2-001,2-004,2-007,2-008,2-012,2-016,2-017,2-018,2-019,2-020,2-022,2-024, 2-025, 2-026, 2-027, 2-028, 2-029, 2-030, 2-033, 2-034, 2-035, 2-036, 2-037, 3-001, 3- 002,3-004,3-005,3-006,3-007,3-008,3-009,3-010,3-012,3-013,3-014,3-015,4-001, 4-002.

Test Example 3 Insecticidal Test for Chahamaki A 10% emulsion of the compound of the present invention (10% wettable powder was tested depending on the compound) was diluted with water containing a spreading agent to prepare a chemical solution having a concentration of 100 ppm. Soak kanran leaves in this chemical solution for about 10 seconds, air dry and place in a petri dish. In this, 5 second-instar larvae of Homona magnanima are released per petri dish, covered and placed in a constant temperature room at 25 ° C. Accommodated. The number of dead insects after 6 days was investigated, and the death rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

As a result, the following compounds showed a death rate of 80% or more.
Compound of the present invention: No.1-001,1-003,1-004,1-005,1-006,1-007,1-009,1-010,1-011,1-012,1-013, 1-017,1-020,1-021,1-022,1-023,1-024,1-025,1-026,1-027,1-028,1-032,1-034,1- 035,1-036,1-038,1-040,1-041,1-042,1-043,1-044,1-045,1-048,1-050,1-051,1-052, 1-053,1-054,1-056,1-057,1-058,1-059,1-062,1-063,1-065,1-066,1-067,1-069,1- 070,1-071,1-072,1-073,1-075,1-076,1-077,1-078,1-079,1-081,1-082,1-083,1-084, 1-085,1-086,1-088,1-089,2-008,2-016,2-018,2-019,2-024,2-029,2-033,2-035,3- 001,3-002,3-008,3-009,3-014,3-015,4-001,4-002.

Test Example 4 Insecticidal test against cucumber potato beetle A 10% emulsion of the compound of the present invention (10% wettable powder depending on the compound) was diluted with water containing a spreading agent to prepare a chemical solution having a concentration of 500 ppm. Soak cucumber leaves in this chemical solution for about 10 seconds, air-dry and place in a petri dish. 5 second-instar larvae of Aulacophora femoralis are released per petri dish, covered and placed in a constant temperature room at 25 ° C. Accommodated. The number of dead insects after 6 days was investigated, and the death rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

As a result, the following compounds showed 100% mortality.
Compound of the present invention: No.1-001,1-004,1-005,1-006,1-007,1-009,1-010,1-011,1-012,1-013,1-014, 1-016,1-017,1-018,1-020,1-022,1-023,1-024,1-025,1-026,1-027,1-028,1-031,1- 032,1-035,1-036,1-038,1-040,1-041,1-042,1-043,1-044,1-045,1-047,1-048,1-050, 1-052,1-053,1-054,1-055,1-056,1-057,1-058,1-059,1-062,1-063,1-064,1-066,1- 067,1-068,1-069,1-070,1-071,1-072,1-073,1-074,1-075,1-077,1-078,1-079,1-080, 1-081,1-082,1-083,1-084,1-085,1-086,1-087,1-088,1-089,2-001,2-004,2-008,2- 009,2-010,2-016,2-017,2-018,2-019,2-021,2-022,2-024,2-025,2-026,2-028,2-029, 2-030,2-033,2-034,2-035,2-036,2-037,3-001,3-005,3-006,3-007,3-008,3-010,3- 012,3-013,3-014,4-001,4-002.

Test Example 5 Insecticidal test against Spodoptera litura (Comparative test)
A 10% emulsion of the compound of the present invention and the comparative compound was diluted with water containing a spreading agent to prepare a chemical solution having a predetermined concentration. Immerse kanran leaves in this chemical for about 10 seconds, air-dry and place in a petri dish. In this, 7 third-instar larvae of Spodoptera litura are released per petri dish, and a lid with a hole is opened. Housed in a constant temperature room. Artificial feed (1 cm ³ ) was added 2 days after the treatment, the number of dead insects after 6 days was investigated, and the death rate was calculated from the following formula. The test was conducted in a two-ward system.

Death rate (%) = (Number of dead insects / Number of dead insects) × 100
Table 11 shows the death rate of each test compound at each predetermined concentration.
Table 11 ――――――――――――――――――――――――――――――――――――
Test compound concentration (ppm)
33 10 3 1 0.3 0.1
――――――――――――――――――――――――――――――――――――
Compound of the present invention No.1-036 100 100 100 85.7 28.6 14.3
Compound of the present invention No.1-084 100 100 71.4 21.3 0
Compound No.1-087 100 100 100 71.4 21.3 0
Comparative compound A 0
――――――――――――――――――――――――――――――――――――
Comparative compound A: European Patent Application No. 1006107, Compound No. 472

The substituted benzanilide compound according to the present invention exhibits excellent pest control activity, particularly insecticidal / miticidal activity, and is extremely useful with little adverse effect on non-target organisms such as mammals, fish and beneficial insects. A compound.

Claims (8)

General formula (1):

[Wherein, W ¹ and W ² each independently represent an oxygen atom or a sulfur atom,
X is a halogen atom, cyano, nitro, _{azido, -SCN, -SF 5, C 1} ~C 6 alkyl, optionally substituted by R ⁷ (C ₁ ~C ₆₎ alkyl, C ₃ -C ₈ cycloalkyl , optionally substituted by R ⁷ (C ₃ ~C ₈₎ cycloalkyl, C ₂ -C ₆ alkenyl, optionally substituted by R ⁷ (C ₂ ~C ₆₎ alkenyl, C ₃ -C ₈ cycloalkenyl , C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₂ -C ₆ alkynyl, optionally substituted by R ⁷ (C ₂ ~C ₆₎ ^{alkynyl, -OH, -OR 8, -OS (} O) 2 R 8, -SH, -S (O) _r R ⁸ , -CHO, -C (O) R ⁹ , -C (O) OR ⁹ , -C (O) SR ⁹ , -C (O) NHR ¹⁰ , -C ( O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , -CH = NOR ¹¹ , -C (R ⁹ ) = NOR ¹¹ , -S (O) ₂ OR ⁹ , -S (O) ₂ NHR ¹⁰ , -S (O) ₂ N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴⁾ R ^12, phenyl, (Z) phenyl substituted by _p1, represents L or M, when m represents 2, 3 or 4, each X May be the or different from each other the same as each other,
Further, when two Xs are adjacent to each other, the two adjacent Xs are -CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ O-, -CH ₂ OCH _2- , -OCH ₂ O-, -CH ₂ CH ₂ S-, -CH ₂ SCH _2- , -CH ₂ CH ₂ N (R ¹⁵ )-, -CH ₂ N (R ¹⁵ ) CH _2- , -CH ₂ CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ CH ₂ O-, -CH ₂ CH ₂ OCH _2- , -CH ₂ OCH ₂ O-, -OCH ₂ CH ₂ O-, -OCH ₂ CH ₂ S-, -CH ₂ CH = CH-,- OCH = CH-, -SCH = CH-, -N (R ¹⁵ ) CH = CH-, -OCH = N-, -SCH = N-, -N (R ¹⁵ ) CH = N-, -N (R ¹⁵ By forming N = CH-, -CH = CHCH = CH-, -OCH ₂ CH = CH-, -N = CHCH = CH-, -N = CHCH = N- or -N = CHN = CH- A 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each of two Xs is bonded. At this time, the hydrogen atom bonded to each carbon atom forming the ring is optionally substituted by Z. In addition, when simultaneously substituted with two or more Z, each Z may be the same as or different from each other,
Y is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, optionally substituted by R ⁷ (C ₁ ~C ₆₎ alkyl, C ₃ -C ₈ cycloalkyl, -OR ^8, -S (O ) _r R ⁸ , —NH ₂ , C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino or —Si (R ¹³ ) (R ¹⁴ ) R ¹² , n is 2, 3 or 4 Each Y may be the same as or different from each other;
Further, when two Ys are adjacent to each other, the two adjacent Ys are —CH ₂ CH ₂ CH ₂ —, —CH ₂ CH ₂ O—, —CH ₂ OCH ₂ —, —OCH ₂ O—, —CH ₂ CH ₂ S-, -CH ₂ SCH _2- , -SCH ₂ S-, -CH ₂ CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ CH ₂ O-, -CH ₂ CH ₂ OCH ₂ -,- By forming CH ₂ OCH ₂ O-, -OCH ₂ CH ₂ O-, -OCH ₂ CH ₂ S-, -SCH ₂ CH ₂ S-, -OCH = N- or -SCH = N- A 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each Y is bonded, and at this time, the hydrogen atom bonded to each carbon atom forming the ring may be optionally substituted by Z Furthermore, when two or more Z are substituted at the same time, each Z may be the same as or different from each other,
R ¹ is hydrogen atom, cyano, optionally substituted by C ₁ -C ₁₂ alkyl, optionally substituted by R ¹⁶ (C ₁ ~C ₁₂₎ alkyl, C ₃ -C ₁₂ cycloalkyl, R ¹⁶ ( C ₃ -C ₁₂₎ cycloalkyl, C ₃ -C ₁₂ alkenyl, optionally substituted by R ¹⁶ (C ₃ ~C ₁₂₎ alkenyl, C ₃ -C ₁₂ cycloalkenyl, C ₃ -C ₁₂ halo cycloalkenyl, C ₃ -C ₁₂ alkynyl, optionally substituted by R ¹⁶ (C ₃ ~C ₁₂₎ alkynyl, -OH, C ₁ -C ₈ alkoxy, C ₃ -C ₈ alkenyloxy, C ₃ -C ₈ haloalkenyloxy , phenoxy, (Z) _p1 phenoxy substituted by phenyl (C ₁ ~C ₄₎ alkoxy, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ ^{alkoxy, -N (R 20) R 19} , Phenyl, (Z) represents phenyl, L or M substituted by _p1 ,
R ² and R ³ are each independently a hydrogen atom, cyano, C ₁ -C ₁₂ alkyl, (C ₁ -C ₁₂ ) alkyl optionally substituted with R ¹⁶ , C ₃ -C ₁₂ alkenyl, C _3- C ₁₂ haloalkenyl, C ₃ -C ₁₂ alkynyl, C ₃ -C ₁₂ haloalkynyl, -OH, C ₁ -C ₈ alkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z) phenylthio substituted by _{p1, -S (O) 2 R} 9, -SN (R 18) R 17, -S (O) 2 N (R 10) R 9, -N (R 20) R 19, -C (O) R ⁹ , -C (O) OR ⁹ , -C (O) SR ⁹ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) N (R 10) R 9, or represents phenyl which is substituted by phenyl or (Z) _p1, or, R ² is formed a C ₂ -C ₆ alkylene chain together with R ¹ This represents that a 3- to 7-membered ring may be formed together with the nitrogen atom to be bonded. At this time, the alkylene chain has an oxygen atom, a sulfur atom or a nitrogen atom. Pieces comprise may, and halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ haloalkyl group, C ₁ -C ₆ alkoxy group, C ₁ -C ₆ alkylcarbonyl group or a C ₁ -C ₆ alkoxycarbonyl group Optionally substituted by
R ⁴ is optionally substituted by C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, R ²¹ (C ₁ ~C ₆₎ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, optionally substituted by R ²¹ (C ₃ ~C ₈₎ cycloalkyl, optionally substituted by R ²¹ (C ₃ ~C ₈₎ halocycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, phenyl, phenyl substituted by (Z) _p1, L or Represents M,
R ⁵ is cyano, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, R ²¹ (C ₃ -C ₈₎ cycloalkyl, optionally substituted optionally substituted by R ²¹ (C _{3 ~C 8)} halocycloalkyl, the R ²¹ (C ₂ ~C ₆₎ alkenyl, C ₃ -C ₈ cycloalkyl alkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ ^{alkynyl, -OR 8, -S (O)} r R 8, -N (R 10) R 9, -CHO, -C (O) R ⁹ , -CH = NOR ¹¹ , -C (R ⁹ ) = NOR ¹¹ , -C (O) OR ⁹ , -C (O) SR ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , phenyl, (Z) phenyl substituted by _p1, biphenyl, biphenyl substituted by (Z) _p1, phenoxyphenyl, phenoxyphenyl substituted by (Z) _p1, Pirijiruo Shifeniru, (Z) pyridyloxy phenyl substituted by _p1, phenylthiophenyl, (Z) phenylthio phenyl substituted by _p1, phenylsulfinyl phenyl, phenylsulfinyl phenyl substituted by (Z) _p1, phenylsulfonyl phenyl, (Z) phenylsulfonyl phenyl substituted by _p1, or represents L or M, or by forming a C ₂ -C ₃ alkylene chain together with Y being present on the adjacent position, it is condensed with a benzene ring Represents that a 5- to 6-membered ring may be formed, in which case the alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and optionally by a halogen atom or a C ₁ -C ₆ haloalkyl group May be replaced,
R ⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~ C ₆ ) haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, phenyl (C ₃ -C ₆ ) alkenyl, (Z) phenyl substituted by _p1 (C ₃ -C ₆₎ alkenyl, C ₃ -C ₈ cycloalkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, phenyl (C ₃ ~C ₆₎ alkynyl, phenyl substituted by (Z) _p1 (C ₃ -C _{6) ^{alkynyl, -S (O) 2 R 9}} , -C (O) R 9, -C (O) OR 9, -C (O) SR 9, -C (S) OR 9, -C (S) SR ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ or M,
L represents an aromatic heterocycle represented by any one of formulas L-1 to L-58,

M represents a saturated heterocyclic ring represented by any one of formulas M-1 to M-28;

Z is a halogen atom, cyano, nitro, _{azido, -SCN, -SF 5, C 1} ~C 6 alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkoxy (C ₁ ~C ₃₎ alkyl, cyano (C ₁ ~C ₆₎ alkyl, hydroxy (C ₁ ~C ₃₎ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ ~C ₃₎ haloalkyl, C ₁ -C ₃ haloalkoxy (C _{1 ~C 3)} haloalkyl, C ₁ -C ₃ alkylthio (C _{1 ~C 3)} alkyl, C ₁ -C ₃ haloalkylthio (C _{1 ~C 3)} alkyl, C ₁ -C ₃ alkylsulfinyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₃ haloalkylsulfinyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₃ alkylsulfonyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₃ haloalkyl sulfonyl (C ₁ ~C ₃₎ alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₂ -C ₆ alkenyl, C ₂ -C ₆ haloalkenyl, C ₃ -C ₈ Cycloalkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₂ -C ₆ alkynyl, C ₂ -C ₆ haloalkynyl, -OH, C ₁ ~C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₃ haloalkoxy (C ₁ ~C ₃₎ haloalkoxy, C ₂ -C ₆ alkenyloxy, C ₂ -C ₆ haloalkenyloxy, C ₃ -C ₆ alkynyloxy, C ₃ -C ₆ haloalkynyloxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, -SH, C ₁ ~C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, -NH _2, C ₁ ~C ₆ alkyl amino, di (C ₁ -C ₆ alkyl) amino, C ₁ -C ₆ alkylsulfonylamino, C ₁ -C ₆ haloalkylsulfonyl amino, C ₁ -C ₆ an alkoxycarbonyl Boniru, C ₁ -C _{6 haloalkoxycarbonyl, -C (O) NH 2,} C 1 ~C 6 alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) _{aminocarbonyl, -C (S) NH 2,} C 1 -C ₆ alkylaminosulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl or a tri (C ₁ -C ₆ alkyl) a silyl, when p1, p2, p3 or p4 represents an integer of 2 or more, each of the Z may be the same as or different from each other,
Further, when two Zs are adjacent to each other, the two adjacent Zs are -CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ O-, -CH ₂ OCH _2- , -OCH ₂ O-, -CH ₂ CH ₂ S-, -CH ₂ SCH _2- , -CH ₂ CH ₂ CH ₂ CH ₂ CH _2- , -CH ₂ CH ₂ CH ₂ O-, -CH ₂ CH ₂ OCH _2- , -CH ₂ OCH ₂ O- , -OCH ₂ CH ₂ O-, -OCH ₂ CH ₂ S- or -CH = CHCH = CH- to form a 5-membered or 6-membered ring with the carbon atom to which each of the two Z bonds may be, at this time, the hydrogen atoms bonded to each carbon atom forming the ring may be optionally substituted by halogen atom or C ₁ -C ₆ alkyl group,
R ⁷ is a halogen atom, cyano, C _{3 to} C ₈ cycloalkyl, C _{3 to} C ₈ halocycloalkyl, —OH, —OR ⁸ , —SH, —S (O) _r R ⁸ , —N (R ¹⁰ ) R ⁹ , -N (R ¹⁰ ) CHO, -N (R ¹⁰ ) C (O) R ⁹ , -N (R ¹⁰ ) C (O) OR ⁹ , -N (R ¹⁰ ) C (O) SR ⁹ , -N (R ¹⁰ ) C (S) OR ⁹ , -N (R ¹⁰ ) C (S) SR ⁹ , -N (R ¹⁰ ) S (O) ₂ R ⁹ , -C (O) OR ⁹ ,- C (O) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , phenyl, (Z) represents phenyl, L or M substituted by _p1 ;
R ⁸ is optionally substituted by C ₁ -C ₆ alkyl, optionally substituted by R ²⁵ (C ₁ ~C ₆₎ alkyl, C ₃ -C ₈ cycloalkyl, R ²⁵ (C ₃ ~C ₈ ) cycloalkyl, C ₂ -C ₆ alkenyl, optionally substituted by R ²⁵ (C ₂ ~C ₆₎ alkenyl, C ₃ -C ₈ cycloalkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₃ -C ₆ It represents alkynyl, optionally substituted by R ²⁵ (C ₃ ~C ₆₎ alkynyl, phenyl, phenyl, L or M, which is substituted by (Z) _p1,
R ⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ cycloalkyl (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylthio (C _{1 ~C 4)} alkyl, cyano (C _{1 ~C 6)} alkyl, phenyl (C _{1 ~C 4)} alkyl, (Z) phenyl substituted by _p1 (C _{1 ~C 4)} Alkyl, L- (C ₁ -C ₄ ) alkyl, M- (C ₁ -C ₄ ) alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ represents haloalkenyl, C ₃ -C ₆ alkynyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁰ represents a hydrogen atom or C ₁ -C ₆ alkyl, or R ⁹ and R ¹⁰ together form a C ₂ -C ₆ alkylene chain to form 3-7 together with the atoms to be bonded. indicates that the members may form a ring, this time the alkylene chain an oxygen atom, may contain one sulfur atom or a nitrogen atom, and a halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ alkoxy group, a formyl group, may be optionally substituted by C ₁ -C ₆ alkylcarbonyl group or a C ₁ -C ₆ alkoxycarbonyl group,
R ¹¹ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, or represents C ₃ -C ₆ alkynyl or C ₃ -C ₆ haloalkynyl, or, R ¹¹ is C ₂ -C ₄ alkylene together with R ⁹ By forming a chain, it represents that a 5- to 7-membered ring may be formed together with the atoms to be bonded. At this time, the alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and a halogen atom. or it may be optionally substituted by C ₁ -C ₆ alkyl group,
R ¹² represents C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ alkenyl, phenyl or phenyl substituted by (Z) _p1 ;
R ¹³ and R ¹⁴ each independently represent C ₁ -C ₆ alkyl or C ₁ -C ₆ haloalkyl,
R ¹⁵ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxycarbonyl (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ haloalkoxycarbonyl (C ₁ -C ₄₎ alkyl, phenyl (C ₁ -C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ -C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ ~ C ₆ represents alkynyl, C ₃ -C ₆ haloalkynyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁶ is a halogen atom, cyano, nitro, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, -OR ²⁶ , -N (R ²⁷ ) R ²⁶ , -SH, -S (O) _r R ²⁸ , -SO ₂ NHR ³⁰ , -SO ₂ N (R ³⁰ ) R ²⁹ , -CHO, -C (O) R ²⁹ , -C (O) OH, -C (O) OR ²⁹ , -C (O ) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) OR ²⁹ , -C (R ³² ) = NOH, -C (R ³² ) = NOR ³¹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , -P (phenyl) ₂ , -P (O) (phenyl) ₂ , phenyl, (Z) represents phenyl, L or M substituted by _p1 ,
R ¹⁷ is C ₁ -C ₁₂ alkyl, C ₁ -C ₁₂ haloalkyl, C ₁ -C ₁₂ alkoxy (C ₁ -C ₁₂ ) alkyl, cyano (C ₁ -C ₁₂ ) alkyl, C ₁ -C ₁₂ alkoxycarbonyl (C ₁ ~C ₁₂₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₁₂ alkenyl, C ₃ -C ₁₂ halo represents alkenyl, C ₃ -C ₁₂ alkynyl, C ₃ -C ₁₂ haloalkynyl, C ₁ -C ₁₂ alkylcarbonyl, C ₁ -C ₁₂ alkoxycarbonyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁸ is C ₁ -C ₁₂ alkyl, C ₁ -C ₁₂ haloalkyl, C ₁ -C ₁₂ alkoxy (C ₁ -C ₁₂ ) alkyl, cyano (C ₁ -C ₁₂ ) alkyl, C ₁ -C ₁₂ alkoxycarbonyl (C ₁ ~C ₁₂₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₁₂ alkenyl, C ₃ -C ₁₂ halo alkenyl, C ₃ -C ₁₂ alkynyl, C ₃ -C ₁₂ haloalkynyl, or represents phenyl which is substituted by phenyl or (Z) _p1, or, C ₄ -C ₇ and R ¹⁷ and R ¹⁸ together By forming an alkylene chain, it represents that a 5- to 8-membered ring may be formed together with the nitrogen atom to be bonded. At this time, the alkylene chain may contain one oxygen atom or sulfur atom, and C _1- It may be optionally substituted by C ₄ alkyl group or a C ₁ -C ₄ alkoxy group,
R ¹⁹ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₆ alkynyl, -CHO, C ₁ ~C ₆ alkyl carbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenyl (C ₁ ~C ₄₎ alkoxycarbonyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkoxycarbonyl, phenoxycarbonyl, phenoxycarbonyl substituted by (Z) _p1 , Phenylcarbonyl, phenylcarbonyl substituted by (Z) _p1 , phenyl or phenyl substituted by (Z) _p1 ,
R ²⁰ represents a hydrogen atom, C ₁ -C ₆ alkyl, -CHO, C ₁ -C ₆ alkylcarbonyl, a C ₁ -C ₆ haloalkylcarbonyl or C ₁ -C ₆ alkoxycarbonyl,
R ²¹ is cyano, C _{3 to} C ₈ cycloalkyl, C _{3 to} C ₈ halocycloalkyl, —OH, —OR ⁸ , —SH, —S (O) _r R ⁸ , —N (R ¹⁰ ) R ⁹ , -N (R ¹⁰ ) CHO, -N (R ¹⁰ ) C (O) R ⁹ , -N (R ¹⁰ ) C (O) OR ⁹ , -N (R ¹⁰ ) C (O) SR ⁹ , -N (R ¹⁰ ) C (S) OR ⁹ , -N (R ¹⁰ ) C (S) SR ⁹ , -N (R ¹⁰ ) S (O) ₂ R ⁹ , -C (O) OR ⁹ , -C (O ) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , phenyl, (Z) represents phenyl, L or M substituted by _p1 ;
R ²² represents C ₁ -C ₆ alkyl or C ₁ -C ₆ haloalkyl,
R ²³ is a halogen atom, cyano, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, hydroxy (C ₁ -C ₆ ) alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkoxycarbonyl (C ₁ ~C ₄₎ represents alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ alkoxycarbonyl, phenyl substituted by phenyl or _{(Z) p1, q1, q2} , q3 or q4 When each represents an integer of 2 or more, each R ²³ may be the same as or different from each other;
R ²⁴ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, -CHO, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ haloalkylcarbonyl, phenyl (C ₁ ~C ₄₎ alkylcarbonyl (Z) phenyl (C ₁ -C ₄ ) alkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenyl (C ₁ -C ₄ ) alkoxycarbonyl, substituted by _p1 (Z ) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkoxycarbonyl, C ₁ -C ₆ alkylthiocarbonyl, C ₁ -C ₆ alkoxythiocarbonyl, C ₁ -C ₆ alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl, C ₁ -C ₆ alkylamino thiocarbonyl, di (C ₁ -C ₆ alkyl) aminothiocarbonyl, phenylcarbonyl, (Z) phenylcarbonyl substituted by _p1, C ₁ -C ₆ alkyl sulfonyl Represents C ₁ -C ₆ haloalkylsulfonyl, phenylsulfonyl, and (Z) phenylsulfonyl substituted by _{p1, -P (O) (OR} 22) 2 or ^{-P (S) (OR 22)} 2,
R ²⁵ is a halogen atom, cyano, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino, -CHO, C ₁ -C ₆ alkyl carbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ ^{haloalkoxycarbonyl, -CH = NOR 11, -C (} R 9) = NOR 11, phenyl, the (Z) _p1 Represents substituted phenyl, L or M;
R ²⁶ is a hydrogen atom, C ₁ -C ₈ alkyl, optionally substituted by R ³³ (C ₁ ~C ₈₎ alkyl, C ₃ -C ₈ cycloalkyl, optionally substituted by R ³³ (C ₃ -C ₈₎ cycloalkyl, C ₃ -C ₈ alkenyl, optionally substituted by R ³³ (C ₃ ~C ₈₎ alkenyl, optionally substituted by C ₃ -C ₈ alkynyl, R ³³ (C ₃ ~ C ₈ ) alkynyl, -CHO, -C (O) R ²⁹ , -C (O) OR ²⁹ , -C (O) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) R ²⁹ , -C (O) C (O) OR ²⁹ , -C (S) R ²⁹ , -C (S) OR ²⁹ , -C (S) SR ²⁹ , -C (S) NHR ³⁰ , -C (S) N (R ³⁰ ) R ²⁹ , -S (O) ₂ R ²⁹ , -S (O) ₂ N (R ³⁰ ) R ²⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , phenyl, (Z) represents phenyl, L or M substituted by _p1 ;
R ²⁷ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ cycloalkyl or C ₁ -C ₆ alkoxy, or R ²⁶ and R ²⁷ together by now it forms a C ₂ -C ₅ alkylene chain, represents that may form a 3-6 membered ring together with the nitrogen atom to which they are attached this case the alkylene chain may contain one oxygen atom or a sulfur atom But often, and halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ alkoxy group, a phenyl group or (Z) _p1 may be substituted by a phenyl group substituted by,
R ²⁸ is, C ₁ -C ₈ alkyl, optionally substituted by R ³³ (C ₁ ~C ₈₎ alkyl, optionally substituted by C ₃ -C ₈ cycloalkyl, R ³³ (C ₃ ~C ₈ ) cycloalkyl, optionally substituted by C ₃ -C _{8 ^{alkenyl, R 33 (C 3 ~C 8}} ) alkenyl, optionally substituted by C ₃ -C _{8 ^{alkynyl, R 33 (C 3 ~C 8}} ) alkynyl, -SH, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, phenylthio substituted by _{(Z) p1, -CHO, -C} (O) R 29, -C (O) OR 29 , -C (O) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) R ²⁹ , -C (O) C (O ) OR ²⁹ , -C (S) R ²⁹ , -C (S) OR ²⁹ , -C (S) SR ²⁹ , -C (S) NHR ³⁰ , -C (S) N (R ³⁰ ) R ²⁹ ,- P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , phenyl, phenyl substituted by (Z ¹ ) _p1 , L-18, L-21, L-25, L-30 ~ Represents L-35, L-45, L-48, L-49 or M;
R ²⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ haloalkoxy (C _{1 ~C 4)} alkyl, C ₁ -C ₆ alkylthio (C _{1 ~C 4)} alkyl, C ₁ -C ₆ haloalkylthio (C _{1 ~C 4)} alkyl, C ₁ -C ₆ alkylsulfonyl (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ haloalkylsulfonyl (C ₁ ~C ₄₎ alkyl, cyano (C ₁ -C ₆₎ alkyl, C ₁ -C ₆ alkylcarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₆ haloalkylcarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₆ alkoxycarbonyl (C ₁ -C ₄₎ alkyl, di (C ₁ -C ₆ alkyl) aminocarbonyl (C ₁ -C ₄₎ alkyl, tri (C ₁ -C ₄ alkyl) silyl (C ₁ -C ₄₎ alkyl, phenyl (C ₁ -C ₄₎ alkyl, phenyl substituted by _{(Z) p1 (C 1 ~C} 4 ) alkyl, L- (C ₁ C ₄₎ alkyl, M- (C ₁ ~C ₄₎ alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₂ -C ₆ alkenyl, C ₂ -C ₆ haloalkenyl, C ₂ -C ₆ alkynyl, C ₂ -C ₆ haloalkynyl, represents phenyl, phenyl, L or M, which is substituted by (Z) _p1,
R ³⁰ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl or phenyl substituted by (Z) _{p 1} , or R ²⁹ and R ³⁰ together represent C By forming a _{2 to} C ₅ alkylene chain, it represents that a 3 to 6 membered ring may be formed together with the nitrogen atom to be bonded. At this time, this alkylene chain contains one oxygen atom, sulfur atom or nitrogen atom. But often, and halogen atom, C ₁ -C ₆ alkyl group, C ₁ -C ₆ alkoxy group, a formyl group, C ₁ -C ₆ alkylcarbonyl group, C ₁ -C ₆ alkoxycarbonyl group, a phenyl group or (Z) optionally substituted by a phenyl group substituted by _p1 ,
R ³¹ is hydrogen atom, C ₁ -C ₈ alkyl, (C ₁ -C ₈ ) alkyl optionally substituted by R ³³ , C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ alkenyl, optional by R ³³ substituted a (C ₃ ~C ₈₎ alkenyl, optionally substituted by C ₃ -C ₈ alkynyl, or R ³³ (C ₃ ~C ₈₎ alkynyl,
R ³² is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkoxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ haloalkoxy (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkylthio (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ haloalkylthio (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkylsulfonyl (C _{1 ~C 4)} alkyl, C ₁ -C ₆ haloalkylsulfonyl (C _{1 ~C 4)} alkyl, phenyl (C _{1 ~C 4)} alkyl, phenyl substituted by (Z) _p1 (C ₁ ~C ₄₎ represents alkyl, phenyl substituted by phenyl or (Z) _p1,
R ³³ is a halogen atom, cyano, nitro, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, —OH, —OR ³⁴ , —SH, —S (O) _r R ³⁴ , —NHR ³⁵ , -N (R ³⁵ ) R ³⁴ , -CHO, -C (O) R ²⁹ , -C (O) OR ²⁹ , -C (O) SR ²⁹ , -C (O) NHR ³⁰ , -C (O) N (R ³⁰ ) R ²⁹ , -C (O) C (O) OR ²⁹ , -CH = NOR ¹¹ , -C (R ⁹ ) = NOR ¹¹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² ,- P (O) (OR ²² ) ₂ , -P (S) (OR ²² ) ₂ , -P (phenyl) ₂ , -P (O) (phenyl) ₂ , phenyl, phenyl substituted by (Z) _p1 , L or M represents
R ³⁴ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylthio (C ₁ -C ₄ ) alkyl, phenyl ( C ₁ -C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₈ cycloalkenyl, C ₃ -C ₈ halocycloalkyl cycloalkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, -CHO, C ₁ ~C ₆ alkyl carbonyl , C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, C ₁ -C ₆ alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl, phenylcarbonyl, (Z) phenylcarbonyl substituted by _p1, C _{1 ~C 6} alkylaminothiocarbonyl It represents di (C ₁ -C ₆ alkyl) aminothiocarbonyl, phenyl, phenyl, L or M, which is substituted by (Z) _p1,
R ³⁵ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, C ₁ -C ₆ alkylcarbonyl , C ₁ -C ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, phenoxycarbonyl, phenoxycarbonyl substituted by (Z) _p1, phenylcarbonyl, substituted by (Z) _p1 phenylcarbonyl, C ₁ -C ₆ alkylsulfonyl and, C ₁ -C ₆ haloalkylsulfonyl, phenyl, phenyl substituted by (Z) _p1, or represents L or M, or the R ³⁴ and R ³⁵ together form by now it forms a C ₂ -C ₅ alkylene chain, represents that may form a 3-6 membered ring together with the nitrogen atom to which they are attached this case the alkylene chain may contain one oxygen atom or a sulfur atom so May, be substituted and the halogen atom or a methyl group,
m represents an integer of 0 to 4,
n represents an integer of 0 to 4,
p1 represents an integer of 1 to 5,
p2 represents an integer of 0 to 4,
p3 represents an integer of 0 to 3,
p4 represents an integer of 0 to 2,
p5 represents an integer of 0 or 1,
q1 represents an integer of 0 to 3,
q2 represents an integer of 0 to 5,
q3 represents an integer of 0 to 7,
q4 represents an integer of 0 to 9,
r represents an integer of 0 to 2;
t represents an integer of 0 or 1. ]
The substituted benzanilide compound or its salt represented by these. W ¹ and W ² represent an oxygen atom,
X is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl or C ₁ -C ₆ represents haloalkylsulfonyl, and when m represents 2 or 3, each X may be the same as or different from each other;
Further, when two Xs are adjacent to each other, the two adjacent Xs form —OCH ₂ O— or —OCH ₂ CH ₂ O— to form a 5-membered ring or 6-membered together with the carbon atom to which each is bonded. may form a ring, this time, the hydrogen atoms bonded to each carbon atom forming the ring is optionally substituted by halogen atom, C ₁ -C ₄ alkyl or C ₁ -C ₄ haloalkyl group Well,
Y is a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, hydroxy (C ₁ ~C ₆₎ alkyl, C ₁ -C ₃ alkoxy (C ₁ ~C ₃₎ alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ represents haloalkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, a C ₁ -C ₆ alkylamino or di (C ₁ -C ₆ alkyl) amino, n is 2 or 3 may be the same as or different from each other,
R ¹ is C ₁ -C ₈ alkyl, (C ₁ -C ₈ ) alkyl optionally substituted by R ¹⁶ , C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ alkenyl, C ₃ -C ₈ alkynyl, C ₁ -C ₈ -alkoxy, a M-4, M-5, M-8, M-9, M-13~M-19, M-21 or M-22,
R ² and R ³ are each independently a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl. , C ₁ -C ₄ alkylsulfonyl (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z ) represents phenylthio substituted by _p1 or —SN (R ¹⁸ ) R ¹⁷ , or R ² together with R ¹ forms a C ₂ -C ₆ alkylene chain, together with the nitrogen atom to which it is attached. Represents that a 3- to 7-membered ring may be formed, in which case this alkylene chain may contain one oxygen or sulfur atom,
R ⁴ is optionally substituted by C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, R ²¹ (C ₁ ~C ₆₎ represents haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, C ₃ -C ₆ haloalkenyl, C ₃ -C ₆ haloalkynyl, phenyl substituted by phenyl or (Z) _p1,
R ⁵ is cyano, optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ alkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ ^{alkynyl, -C (O) OR 9,} - C (O) SR ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) OR ⁹ , -C (S) SR ⁹ , -C (S) NHR ^{10, -C (S) N (} R 10) R 9, phenyl, (Z) phenyl substituted by _p1, (Z) phenoxyphenyl phenyl substituted by _p1, pyridyloxy phenyl substituted by (Z) _p1, L-1 ~ L-4, L-8 ~ L-13, L-15 ~ L-23, L-25 ~ L-35, L-37, L-38, L-40, L-43 ~ L- 58, M-4, M-5, M-8, M-9, M-14 to M-18 or M-19, or C ₂ to C together with Y present in the adjacent position by forming a ₃ alkylene chain, condensed with a benzene ring 5 Membered indicates that may form a ring, this time the alkylene chain an oxygen atom, may contain one sulfur atom or a nitrogen atom, optionally substituted and the halogen atom or a C ₁ -C ₆ haloalkyl group You can,
R ⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl , cyano (C ₁ ~C ₆₎ alkyl, phenyl (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ substituted by (Z) _p1 alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ haloalkenyl, phenyl (C ₃ -C ₆₎ alkenyl, (Z) phenyl substituted by _p1 (C ₃ -C ₆₎ alkenyl, C ₃ -C ₆ alkynyl, C ₃ -C ₆ haloalkynyl, phenyl (C ₃ -C ₆ ) alkynyl, phenyl (C ₃ -C ₆ ) alkynyl substituted by (Z) _p1 , -S (O) ₂ R ⁹ , -C (O) R ⁹ , -C (O) NHR ¹⁰ , -C (O) N (R ¹⁰ ) R ⁹ , -C (S) NHR ¹⁰ , -C (S) N (R ¹⁰ ) R ⁹ , -Si (R ¹³ ) (R ¹⁴ ) R ¹² , -P ( O) (OR ²² ) ₂ or -P (S) (OR ²² ) ₂
Z is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkylthio (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylthio (C ₁ ~ C ₃₎ alkyl, C ₁ -C ₃ alkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ alkylsulfonyl (C ₁ -C ₃ ) alkyl, C ₁ -C ₃ haloalkylsulfonyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₃ haloalkoxy (C ₁ -C ₃₎ haloalkoxy , C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, -C (O) NH ₂ or - Represents C (S) NH _2, and when p1, p2, p3 or p4 represents an integer of 2 or more, each Z may be the same as or different from each other;
Further, when _two Zs are adjacent, the two adjacent Zs are -CF ₂ CF ₂ O-, -CF ₂ OCF _2- , -OCF ₂ O-, -OCF ₂ CHFO-, -OCF ₂ CF ₂ By forming O- or -CH = CHCH = CH-, a 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each of two Zs is bonded,
R ⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₆ cycloalkyl (C ₁ -C ₄ ) alkyl, phenyl (C ₁ -C ₄ ) alkyl, (Z) substituted by _p1 phenyl (C ₁ ~C ₄₎ represents alkyl, C ₃ -C ₈ cycloalkyl, C ₃ -C ₈ halocycloalkyl, phenyl substituted by phenyl or (Z) _p1,
R ¹⁰ represents a hydrogen atom or C ₁ -C ₆ alkyl, or R ⁹ and R ¹⁰ together form a C ₄ -C ₅ alkylene chain to form a 5-membered atom together with the nitrogen atom to which it is attached. Represents that a ring or a 6-membered ring may be formed, in which case the alkylene chain may contain one oxygen atom or sulfur atom,
R ¹² represents C ₁ -C ₆ alkyl, phenyl or phenyl substituted by (Z) _{p 1}
R ¹³ and R ¹⁴ each independently represent C ₁ -C ₆ alkyl;
R ¹⁵ is, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, phenyl (C ₁ ~C ₄₎ alkyl, phenyl (C ₁ ~C ₄₎ substituted by (Z) _p1 alkyl, phenyl or (Z ) represents phenyl substituted by _p1 ,
R ¹⁶ is a halogen atom, cyano, C ₃ -C ₆ cycloalkyl, -OR ²⁶ , -N (R ²⁷ ) R ²⁶ , -S (O) _r R ²⁸ , -SO ₂ N (R ³⁰ ) R ²⁹ , C ₁ -C ₆ alkoxycarbonyl, -C (O) N (R 30) R 29, -C (R 32) = NOH, -C (R 32) = NOR 31, -Si (R 13) (R 14) R ^{12 represents} phenyl, phenyl substituted by (Z) _p1 , L-1, L-2, L-3, L-4, L-45, L-46, L-47 or M;
R ¹⁷ represents C ₁ -C ₆ alkyl, C ₁ -C ₆ alkoxycarbonyl (C ₁ -C ₄ ) alkyl or C ₁ -C ₆ alkoxycarbonyl,
R ¹⁸ represents C ₁ -C ₆ alkyl, or R ¹⁷ and R ¹⁸ together form a C ₄ -C ₅ alkylene chain to form a 5-membered ring or 6 together with the nitrogen atom to which R ¹⁸ is bonded. The alkylene chain may contain one oxygen atom or one sulfur atom, and may be optionally substituted with a methyl group or a methoxy group,
R ²¹ is cyano, C ₃ -C ₆ cycloalkyl, C ₃ -C ₆ halocycloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z) phenoxy substituted by _{p 1} , C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, phenylthio, (Z) phenylthio substituted by _p1, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl , C ₁ -C ₆ haloalkylsulfonyl, phenylsulfonyl, phenylsulfonyl substituted by _{(Z) p1, C 1 ~C} 6 alkyl amino, di (C ₁ -C ₆ alkyl) amino, phenylamino, by (Z) _p1 substituted phenylamino, C ₁ -C ₆ alkoxycarbonyl, phenyl, (Z) phenyl substituted by _{p1, L-1~L-5,} L-8~L-24, L-36, L-39, Represents L-45 to L-52 or L-53,
R ²² represents C ₁ -C ₆ alkyl;
R ²³ represents C ₁ -C ₄ alkyl, and when q1, q2, q3 or q4 represents an integer of 2 or more, each R ²³ may be the same as or different from each other;
R ²⁴ represents -CHO, C ₁ -C ₆ alkylcarbonyl, a C ₁ -C ₆ alkoxycarbonyl or C ₁ -C ₆ alkylsulfonyl,
R ²⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl , phenyl (C ₁ ~C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₃ -C ₆ cycloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, -C (O) N (R 30) R 29, C 1 ~C 6 alkyl sulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl, phenylsulfonyl, (Z ) phenylsulfonyl substituted by _p1, di (C ₁ -C ₆ alkyl) phosphoryl, di (C ₁ -C ₆ alkyl) thiophosphoryl, tri (C ₁ -C ₄ alkyl) silyl, by phenyl or (Z) _p1 Represents substituted phenyl,
R ²⁷ represents a hydrogen atom or a C ₁ -C ₆ alkyl,
R ²⁸ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, hydroxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio ( C ₁ -C ₄₎ alkyl, C ₁ -C ₄ alkylcarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₄ alkoxycarbonyl (C ₁ -C ₄₎ alkyl, C ₁ -C ₄ alkylaminocarbonyl (C ₁ -C ₄₎ alkyl, di (C ₁ -C ₄ alkyl) aminocarbonyl (C ₁ -C ₄₎ alkyl, tri (C ₁ -C ₄ alkyl) silyl (C ₁ -C ₄₎ alkyl, phenyl (C ₁ -C ₄₎ alkyl, (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ alkenyl, C ₃ -C ₆ alkynyl, C ₁ -C ₆ alkylthio, phenyl, (Z) _represents phenyl, L-21, L-35, L-45 or L-48 substituted by _p1 ,
R ²⁹ is C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl, phenyl (C ₁ -C ₄ ) alkyl. It is replaced by (Z) phenyl substituted by _p1 (C ₁ ~C ₄₎ alkyl, C ₃ -C ₆ cycloalkyl, C ₃ -C ₆ alkenyl, C ₂ -C ₆ alkynyl, phenyl or (Z) _p1 Represents phenyl,
R ³⁰ represents a hydrogen atom or C _{1 to} C ₆ alkyl, or R ²⁹ and R ³⁰ together form a C _{2 to} C ₅ alkylene chain to form a 3- Represents that a 6-membered ring may be formed, in which case the alkylene chain may contain one oxygen or sulfur atom,
R ³¹ is, C ₁ -C ₆ alkyl, phenyl (C ₁ ~C ₄₎ phenyl substituted by alkyl or _{(Z) p1 (C 1 ~C} 4) alkyl,
R ³² represents a hydrogen atom or C ₁ -C ₆ alkyl,
m represents an integer of 0 to 3,
n represents an integer of 0 to 3,
The substituted benzanilide compound or a salt thereof according to claim 1, wherein q2, q3 and q4 each independently represents an integer of 0 to 2. X is a halogen atom, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl or C ₁ -C ₆ haloalkylsulfonyl, m represents 2 Each X may be the same or different from each other,
Y is a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy or C ₁ -C ₆ alkylthio, when n is 2, each Y is identical to each other May be different from each other,
R ¹ represents C ₁ -C ₈ alkyl, (C ₁ -C ₈ ) alkyl, C ₃ -C ₈ alkenyl or C ₃ -C ₈ alkynyl optionally substituted by R ¹⁶ ,
R ² represents a hydrogen atom or C ₁ -C ₆ alkyl,
R ³ represents a hydrogen atom,
R ⁴ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ -C ₃ ) haloalkyl, C ₁ -C ₃ alkylthio (C ₁ -C ₃ ) haloalkyl, C ₃ -C ₆ cycloalkyl or C ₃ -C ₆ halocycloalkyl,
R ⁵ is optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, optionally substituted by R ²¹ (C ₂ ~ C ₆₎ alkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ alkynyl, C ₁ -C ₆ alkoxycarbonyl, phenyl, phenyl substituted by (Z) _p1, substituted by (Z) _p1 Phenoxyphenyl, pyridyloxyphenyl substituted by (Z) _p1 , L-1 to L-4, L-8 to L-13, L-15 to L-23, L-45 to L-52 or L-53 or it represents, or indicates that by forming a C ₂ -C ₃ alkylene chain together with Y being present on the adjacent positions, may form a 5- or 6-membered ring fused with a benzene ring, In this case, the alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and may be optionally substituted with a halogen atom. ,
R ⁶ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylcarbonyl or tri (C ₁ -C ₄ alkyl) silyl;
R ¹⁶ is -OR ²⁶ , -N (R ²⁷ ) R ²⁶ , -S (O) _r R ²⁸ , -SO ₂ N (R ³⁰ ) R ²⁹ , -C (R ³² ) = NOH or -C (R ³² ) = NOR ³¹
R ²¹ is, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z) _p1 phenoxy substituted by, phenylthio, phenylthio substituted by (Z) _p1, phenylsulfonyl, (Z) _p1 phenylsulfonyl substituted by, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino, phenylamino, (Z) phenylamino substituted by _p1, C ₁ -C ₆ alkoxycarbonyl, phenyl, (Z) represents phenyl substituted by _p1 , L-1 to L-5, L-8 to L-24, L-36, L-39, L-45 to L-52 or L-53;
R ²⁶ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ alkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ alkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl or represents C ₁ -C ₆ alkylsulfonyl,
R ²⁸ represents C ₁ -C ₆ alkyl,
R ²⁹ represents C ₁ -C ₆ alkyl;
R ³⁰ represents a hydrogen atom or C ₁ -C ₆ alkyl,
R ³¹ represents C ₁ -C ₆ alkyl;
R ³² represents a hydrogen atom,
m represents an integer of 0 to 2,
The substituted benzanilide compound or a salt thereof according to claim 2, wherein n represents an integer of 0 to 2. X represents a halogen atom, nitro, C ₁ -C ₄ alkyl, C ₁ -C ₄ haloalkyl, C ₁ -C ₄ alkylthio, a C ₁ -C ₄ alkylsulfinyl or C ₁ -C ₄ alkylsulfonyl, m is 2 Each X may be the same as or different from each other;
Y represents a halogen atom or a C ₁ -C ₄ alkyl, when n is 2, each Y may be the even or different from each other the same as each other,
R ¹ is C ₁ -C ₈ alkyl, C ₁ -C ₄ alkylthio (C ₁ -C ₄ ) alkyl, C ₁ -C ₄ alkylsulfinyl (C ₁ -C ₄ ) alkyl or C ₁ -C ₄ alkylsulfonyl ( C ₁ -C ₄₎ alkyl,
R ² represents a hydrogen atom,
R ⁴ represents C ₁ -C ₆ alkyl or C ₁ -C ₆ haloalkyl,
R ⁵ is phenyl, (Z) phenyl substituted by _p1, (Z) phenoxyphenyl phenyl substituted by _p1, (Z) pyridyloxy phenyl substituted by _{p1, L-1~L-4,} L-8 ~ L-13, L-15 ~ L-23, L-45 ~ L-52 or L-53,
The substituted benzanilide compound or a salt thereof according to claim 3, wherein R ⁶ represents a hydrogen atom. General formula (2) or general formula (3):

[Wherein Y ¹ represents a hydrogen atom, a halogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₆ alkoxy or C ₁ -C ₆ alkylthio,
Y ² and Y ³ each independently represent a hydrogen atom, or, together with R ⁵ , form a C ₂ -C ₃ alkylene chain to form a 5- to 6-membered ring condensed with a benzene ring. The alkylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and may be optionally substituted with a halogen atom,
R ⁴ is C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkoxy (C ₁ -C ₃ ) haloalkyl, C ₁ -C ₃ alkylthio (C ₁ -C ₃ ) haloalkyl, C ₃ -C ₆ cycloalkyl or C ₃ -C ₆ halocycloalkyl,
R ⁵ is optionally substituted by R ²¹ (C ₁ ~C ₆₎ alkyl, optionally substituted by R ²¹ (C ₁ ~C ₆₎ haloalkyl, optionally substituted by R ²¹ (C ₂ ~ C ₆₎ alkenyl, optionally substituted by R ²¹ (C ₂ ~C ₆₎ alkynyl, C ₁ -C ₆ alkoxycarbonyl, phenyl, phenyl substituted by (Z) _p1, substituted by (Z) _p1 Phenoxyphenyl, pyridyloxyphenyl substituted by (Z) _p1 , L-1 to L-4, L-8 to L-13, L-15 to L-23, L-45 to L-52 or L-53 Represents
R ⁶ represents a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₄ alkoxy (C ₁ -C ₄ ) alkyl, C ₁ -C ₆ alkylcarbonyl or tri (C ₁ -C ₄ alkyl) silyl;
R ²¹ is, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, phenoxy, (Z) _p1 phenoxy substituted by, phenylthio, phenylthio substituted by (Z) _p1, phenylsulfonyl, (Z) _p1 phenylsulfonyl substituted by, C ₁ -C ₆ alkylamino, di (C ₁ -C ₆ alkyl) amino, phenylamino, (Z) phenylamino substituted by _p1, C ₁ -C ₆ alkoxycarbonyl, phenyl, (Z) represents phenyl substituted by _p1 , L-1 to L-5, L-8 to L-24, L-36, L-39, L-45 to L-52 or L-53;
L-1 to L-5, L-8 to L-24, L-36, L-39, L-45 to L-52 or L-53 each represents the following aromatic heterocycle:

Z is a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₁ -C ₃ alkylthio (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylthio (C ₁ ~ C ₃₎ alkyl, C ₁ -C ₃ alkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ haloalkylsulfinyl (C ₁ ~C ₃₎ alkyl, C ₁ -C ₃ alkylsulfonyl (C ₁ -C ₃ ) alkyl, C ₁ -C ₃ haloalkylsulfonyl (C ₁ -C ₃₎ alkyl, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₃ haloalkoxy (C ₁ -C ₃₎ haloalkoxy , C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C ₁ -C ₆ haloalkylsulfinyl, C ₁ -C ₆ alkylsulfonyl, C ₁ -C ₆ haloalkylsulfonyl, -C (O) NH ₂ or - Represents C (S) NH _2, and when p1, p2, p3 or p4 represents an integer of 2 or more, each Z may be the same as or different from each other;
Further, when _two Zs are adjacent, the two adjacent Zs are -CF ₂ CF ₂ O-, -CF ₂ OCF _2- , -OCF ₂ O-, -OCF ₂ CHFO-, -OCF ₂ CF ₂ By forming O- or -CH = CHCH = CH-, a 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each of two Zs is bonded,
R ¹⁵ represents C ₁ -C ₆ alkyl, phenyl or phenyl substituted by (Z) _p1 ,
p1 represents an integer of 1 to 5,
p2 represents an integer of 0 to 4,
p3 represents an integer of 0 to 3,
p4 represents an integer of 0 to 2,
p5 represents an integer of 0 or 1,
r represents an integer of 0 to 2;
t represents an integer of 0 or 1. ]
N-substituted phenyl-3-nitrophthalimide or substituted aniline represented by the formula:   A pest control agent comprising one or more selected from the substituted benzanilide compound according to any one of claims 1 to 4 and a salt thereof as an active ingredient.   An agrochemical comprising one or more selected from the substituted benzanilide compound according to any one of claims 1 to 4 and a salt thereof as an active ingredient.   An insecticide or acaricide containing one or more selected from the substituted benzanilide compound according to any one of claims 1 to 4 and a salt thereof as an active ingredient.