JP2004529177A - 高眼圧症および緑内障の処置方法 - Google Patents
高眼圧症および緑内障の処置方法 Download PDFInfo
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- JP2004529177A JP2004529177A JP2002589015A JP2002589015A JP2004529177A JP 2004529177 A JP2004529177 A JP 2004529177A JP 2002589015 A JP2002589015 A JP 2002589015A JP 2002589015 A JP2002589015 A JP 2002589015A JP 2004529177 A JP2004529177 A JP 2004529177A
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- prostaglandin compound
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- XXUPXHKCPIKWLR-JHUOEJJVSA-N isopropyl unoprostone Chemical compound CCCCCCCC(=O)CC[C@H]1[C@H](O)C[C@H](O)[C@@H]1C\C=C/CCCC(=O)OC(C)C XXUPXHKCPIKWLR-JHUOEJJVSA-N 0.000 description 1
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- HNQIVZYLYMDVSB-UHFFFAOYSA-N methanesulfonimidic acid Chemical compound CS(N)(=O)=O HNQIVZYLYMDVSB-UHFFFAOYSA-N 0.000 description 1
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- MGJXBDMLVWIYOQ-UHFFFAOYSA-N methylazanide Chemical compound [NH-]C MGJXBDMLVWIYOQ-UHFFFAOYSA-N 0.000 description 1
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- XAEFZNCEHLXOMS-UHFFFAOYSA-M potassium benzoate Chemical compound [K+].[O-]C(=O)C1=CC=CC=C1 XAEFZNCEHLXOMS-UHFFFAOYSA-M 0.000 description 1
- 239000000843 powder Substances 0.000 description 1
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- MFDFERRIHVXMIY-UHFFFAOYSA-N procaine Chemical class CCN(CC)CCOC(=O)C1=CC=C(N)C=C1 MFDFERRIHVXMIY-UHFFFAOYSA-N 0.000 description 1
- 235000010409 propane-1,2-diol alginate Nutrition 0.000 description 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 description 1
- GMVPRGQOIOIIMI-DWKJAMRDSA-N prostaglandin E1 Chemical compound CCCCC[C@H](O)\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(O)=O GMVPRGQOIOIIMI-DWKJAMRDSA-N 0.000 description 1
- DZUXGQBLFALXCR-CDIPTNKSSA-N prostaglandin F1alpha Chemical compound CCCCC[C@H](O)\C=C\[C@H]1[C@H](O)C[C@H](O)[C@@H]1CCCCCCC(O)=O DZUXGQBLFALXCR-CDIPTNKSSA-N 0.000 description 1
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- YWIVKILSMZOHHF-QJZPQSOGSA-N sodium;(2s,3s,4s,5r,6r)-6-[(2s,3r,4r,5s,6r)-3-acetamido-2-[(2s,3s,4r,5r,6r)-6-[(2r,3r,4r,5s,6r)-3-acetamido-2,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-2-carboxy-4,5-dihydroxyoxan-3-yl]oxy-5-hydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-3,4,5-trihydroxyoxane-2- Chemical compound [Na+].CC(=O)N[C@H]1[C@H](O)O[C@H](CO)[C@@H](O)[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@H](O[C@H]2[C@@H]([C@@H](O[C@H]3[C@@H]([C@@H](O)[C@H](O)[C@H](O3)C(O)=O)O)[C@H](O)[C@@H](CO)O2)NC(C)=O)[C@@H](C(O)=O)O1 YWIVKILSMZOHHF-QJZPQSOGSA-N 0.000 description 1
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Images
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
- A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Ophthalmology & Optometry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29035501P | 2001-05-14 | 2001-05-14 | |
| PCT/JP2002/004600 WO2002092098A1 (en) | 2001-05-14 | 2002-05-13 | Method for treating ocular hypertension and glaucoma |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004529177A true JP2004529177A (ja) | 2004-09-24 |
| JP2004529177A5 JP2004529177A5 (enExample) | 2005-12-22 |
Family
ID=23115609
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002589015A Pending JP2004529177A (ja) | 2001-05-14 | 2002-05-13 | 高眼圧症および緑内障の処置方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20050014837A1 (enExample) |
| EP (1) | EP1390035A1 (enExample) |
| JP (1) | JP2004529177A (enExample) |
| KR (1) | KR20040008174A (enExample) |
| CN (1) | CN1525861A (enExample) |
| BR (1) | BR0209601A (enExample) |
| CA (1) | CA2444627A1 (enExample) |
| MX (1) | MXPA03010363A (enExample) |
| NO (1) | NO20035043D0 (enExample) |
| WO (1) | WO2002092098A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2003082257A2 (en) * | 2002-03-28 | 2003-10-09 | Sucampo Ag | Method for treating ocular hypertension and glaucoma |
| US8580851B2 (en) | 2002-08-21 | 2013-11-12 | Sucampo Ag | Ophthalmic solution |
| AR043161A1 (es) * | 2003-02-14 | 2005-07-20 | Sucampo Pharmaceuticals Inc | Composicion oftalmica para tratar hipertension ocular y glaucoma |
| ES2431640T3 (es) * | 2003-08-21 | 2013-11-27 | Sucampo Ag | Composición oftálmica que comprende éster isopropílico de unoprostona y un agente de viscosidad |
| US10206813B2 (en) | 2009-05-18 | 2019-02-19 | Dose Medical Corporation | Implants with controlled drug delivery features and methods of using same |
| US12478503B2 (en) | 2009-05-18 | 2025-11-25 | Glaukos Corporation | Implants with controlled drug delivery features and methods of using same |
| ES2911174T3 (es) | 2010-07-29 | 2022-05-18 | Allergan Inc | Soluciones de bimatoprost y timolol sin conservantes |
| US9061034B2 (en) | 2010-07-29 | 2015-06-23 | Allergan, Inc. | Preservative free bimatoprost and timolol solutions |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5212200A (en) * | 1987-09-18 | 1993-05-18 | R-Tech Ueno, Ltd. | Ocular hypotensive agents |
| US5208256A (en) * | 1990-05-22 | 1993-05-04 | R-Tech Ueno, Ltd. | Treatment of ocular hypertension with a synergistic combination for ocular administration |
| ATE207360T1 (de) * | 1992-03-19 | 2001-11-15 | R Tech Ueno Ltd | Behandlung von augenhochdruck mit betablockern und prostansäurederivaten |
| TW420611B (en) * | 1995-03-10 | 2001-02-01 | R Tech Ueno Ltd | Pharmaceutical composition containing prostanoic acid compounds for the treatment of optic nerve disorder |
| WO2000038689A1 (en) * | 1998-12-25 | 2000-07-06 | Sucampo, A.G. | Drug compositions for the treatment of ocular hypertension or glaucoma |
| US6458836B1 (en) * | 2000-03-16 | 2002-10-01 | Sucampo, A.G. | Treatment of ocular hypertension and glaucoma |
-
2002
- 2002-05-13 KR KR10-2003-7014707A patent/KR20040008174A/ko not_active Withdrawn
- 2002-05-13 CA CA002444627A patent/CA2444627A1/en not_active Abandoned
- 2002-05-13 EP EP02724768A patent/EP1390035A1/en not_active Withdrawn
- 2002-05-13 WO PCT/JP2002/004600 patent/WO2002092098A1/en not_active Ceased
- 2002-05-13 JP JP2002589015A patent/JP2004529177A/ja active Pending
- 2002-05-13 BR BR0209601-3A patent/BR0209601A/pt not_active IP Right Cessation
- 2002-05-13 MX MXPA03010363A patent/MXPA03010363A/es unknown
- 2002-05-13 US US10/477,359 patent/US20050014837A1/en not_active Abandoned
- 2002-05-13 CN CNA028137566A patent/CN1525861A/zh active Pending
-
2003
- 2003-11-13 NO NO20035043A patent/NO20035043D0/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20040008174A (ko) | 2004-01-28 |
| NO20035043D0 (no) | 2003-11-13 |
| WO2002092098A1 (en) | 2002-11-21 |
| BR0209601A (pt) | 2004-03-23 |
| US20050014837A1 (en) | 2005-01-20 |
| EP1390035A1 (en) | 2004-02-25 |
| MXPA03010363A (es) | 2004-03-16 |
| CA2444627A1 (en) | 2002-11-21 |
| CN1525861A (zh) | 2004-09-01 |
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