JP2004525982A5 - - Google Patents
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- Publication number
- JP2004525982A5 JP2004525982A5 JP2002583414A JP2002583414A JP2004525982A5 JP 2004525982 A5 JP2004525982 A5 JP 2004525982A5 JP 2002583414 A JP2002583414 A JP 2002583414A JP 2002583414 A JP2002583414 A JP 2002583414A JP 2004525982 A5 JP2004525982 A5 JP 2004525982A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- hydrogen
- ring system
- alkyl
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 claims description 8
- 125000005843 halogen group Chemical group 0.000 claims description 7
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims description 6
- 229910052739 hydrogen Inorganic materials 0.000 claims description 6
- 239000001257 hydrogen Substances 0.000 claims description 6
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 claims description 5
- 125000003282 alkyl amino group Chemical group 0.000 claims description 4
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims description 4
- 150000001875 compounds Chemical class 0.000 claims description 3
- 150000003839 salts Chemical class 0.000 claims description 3
- 239000012453 solvate Substances 0.000 claims description 3
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 2
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims description 2
- 125000004122 cyclic group Chemical group 0.000 claims 4
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 2
- 125000003118 aryl group Chemical group 0.000 claims 2
- 229920006395 saturated elastomer Polymers 0.000 claims 2
- 150000001204 N-oxides Chemical class 0.000 claims 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 1
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- 229910052757 nitrogen Inorganic materials 0.000 claims 1
- 125000004433 nitrogen atom Chemical group N* 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 239000001301 oxygen Substances 0.000 claims 1
- 125000004434 sulfur atom Chemical group 0.000 claims 1
- 238000000034 method Methods 0.000 description 8
- 239000000126 substance Substances 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0105361A FR2823749B1 (fr) | 2001-04-20 | 2001-04-20 | Phenyl- et pyridyl-piperidines, procede pour leur preparation et compositions pharmaceutiques les contenant |
| PCT/FR2002/001342 WO2002085887A1 (fr) | 2001-04-20 | 2002-04-19 | Phenyl- et pyridyl-piperidines avec une activite du tnf |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2004525982A JP2004525982A (ja) | 2004-08-26 |
| JP2004525982A5 true JP2004525982A5 (enExample) | 2009-06-18 |
| JP4324381B2 JP4324381B2 (ja) | 2009-09-02 |
Family
ID=8862517
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002583414A Expired - Fee Related JP4324381B2 (ja) | 2001-04-20 | 2002-04-19 | Ｔｎｆ活性を有するフェニル−およびピリジル−ピペリジン類 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US7326720B2 (enExample) |
| EP (1) | EP1383761B1 (enExample) |
| JP (1) | JP4324381B2 (enExample) |
| AT (1) | ATE500241T1 (enExample) |
| DE (1) | DE60239324D1 (enExample) |
| FR (1) | FR2823749B1 (enExample) |
| WO (1) | WO2002085887A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2831166B1 (fr) * | 2001-10-18 | 2004-02-27 | Sanofi Synthelabo | Aralkyl-tetrahydro-pyridines, leur preparation et compositions pharmaceutiques les contenant |
| FR2883285B1 (fr) * | 2005-03-17 | 2007-05-18 | Sanofi Aventis Sa | Sel besylate de la 7-(2-(4-(3-trifluoromethyl-phenyl) -1,2,3,6-tetrahudro-pyrid-1-yl)ethyl) isoquinoleine, sa preparation et son utilisation en therapeutique |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PH17194A (en) | 1980-03-06 | 1984-06-19 | Otsuka Pharma Co Ltd | Novel carbostyril derivatives,and pharmaceutical composition containing the same |
-
2001
- 2001-04-20 FR FR0105361A patent/FR2823749B1/fr not_active Expired - Fee Related
-
2002
- 2002-04-19 AT AT02727675T patent/ATE500241T1/de not_active IP Right Cessation
- 2002-04-19 EP EP02727675A patent/EP1383761B1/fr not_active Expired - Lifetime
- 2002-04-19 JP JP2002583414A patent/JP4324381B2/ja not_active Expired - Fee Related
- 2002-04-19 DE DE60239324T patent/DE60239324D1/de not_active Expired - Lifetime
- 2002-04-19 WO PCT/FR2002/001342 patent/WO2002085887A1/fr not_active Ceased
- 2002-04-19 US US10/475,272 patent/US7326720B2/en not_active Expired - Fee Related
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