JP2004248675A5 - - Google Patents

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Publication number
JP2004248675A5
JP2004248675A5 JP2004087151A JP2004087151A JP2004248675A5 JP 2004248675 A5 JP2004248675 A5 JP 2004248675A5 JP 2004087151 A JP2004087151 A JP 2004087151A JP 2004087151 A JP2004087151 A JP 2004087151A JP 2004248675 A5 JP2004248675 A5 JP 2004248675A5
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JP
Japan
Prior art keywords
substrate
enzyme
mutant
orthogonal
accepts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2004087151A
Other languages
English (en)
Japanese (ja)
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JP2004248675A (ja
Filing date
Publication date
Application filed filed Critical
Publication of JP2004248675A publication Critical patent/JP2004248675A/ja
Publication of JP2004248675A5 publication Critical patent/JP2004248675A5/ja
Withdrawn legal-status Critical Current

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JP2004087151A 1997-02-07 2004-03-24 変性ヌクレオチド三燐酸基質を利用できる組み換えタンパクキナーゼ Withdrawn JP2004248675A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79752297A 1997-02-07 1997-02-07
US4672797P 1997-05-16 1997-05-16

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP53499998A Division JP3784076B2 (ja) 1997-02-07 1998-02-09 変性ヌクレオチド三燐酸基質を利用できる組み換えタンパクキナーゼ

Publications (2)

Publication Number Publication Date
JP2004248675A JP2004248675A (ja) 2004-09-09
JP2004248675A5 true JP2004248675A5 (cg-RX-API-DMAC7.html) 2005-07-28

Family

ID=26724237

Family Applications (2)

Application Number Title Priority Date Filing Date
JP53499998A Expired - Fee Related JP3784076B2 (ja) 1997-02-07 1998-02-09 変性ヌクレオチド三燐酸基質を利用できる組み換えタンパクキナーゼ
JP2004087151A Withdrawn JP2004248675A (ja) 1997-02-07 2004-03-24 変性ヌクレオチド三燐酸基質を利用できる組み換えタンパクキナーゼ

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP53499998A Expired - Fee Related JP3784076B2 (ja) 1997-02-07 1998-02-09 変性ヌクレオチド三燐酸基質を利用できる組み換えタンパクキナーゼ

Country Status (8)

Country Link
US (5) US6390821B1 (cg-RX-API-DMAC7.html)
EP (1) EP1017823B1 (cg-RX-API-DMAC7.html)
JP (2) JP3784076B2 (cg-RX-API-DMAC7.html)
AT (1) ATE271130T1 (cg-RX-API-DMAC7.html)
AU (1) AU755062B2 (cg-RX-API-DMAC7.html)
CA (1) CA2279846C (cg-RX-API-DMAC7.html)
DE (1) DE69825066T2 (cg-RX-API-DMAC7.html)
WO (1) WO1998035048A2 (cg-RX-API-DMAC7.html)

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US7429596B2 (en) * 2003-06-20 2008-09-30 The Regents Of The University Of California 1H-pyrrolo [2,3-D] pyrimidine derivatives and methods of use thereof
EP1656379B1 (en) * 2003-08-15 2007-01-10 Merck & Co., Inc. 4-cycloalkylaminopyrazolo pyrimidine nmda/nr2b antagonists
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WO2009046448A1 (en) * 2007-10-04 2009-04-09 Intellikine, Inc. Chemical entities and therapeutic uses thereof
US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
CN104926815B (zh) 2008-01-04 2017-11-03 英特利凯恩有限责任公司 某些化学实体、组合物和方法
US8065217B2 (en) * 2008-02-12 2011-11-22 Bids Trading, L.P. Real-time portfolio balancing and/or optimization system and method
WO2009114874A2 (en) 2008-03-14 2009-09-17 Intellikine, Inc. Benzothiazole kinase inhibitors and methods of use
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WO2010006086A2 (en) 2008-07-08 2010-01-14 Intellikine, Inc. Kinase inhibitors and methods of use
WO2010006072A2 (en) 2008-07-08 2010-01-14 The Regents Of The University Of California Mtor modulators and uses thereof
EP2346508B1 (en) 2008-09-26 2016-08-24 Intellikine, LLC Heterocyclic kinase inhibitors
JP5819195B2 (ja) 2008-10-16 2015-11-18 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア 融合環ヘテロアリールキナーゼ阻害剤
US8476282B2 (en) 2008-11-03 2013-07-02 Intellikine Llc Benzoxazole kinase inhibitors and methods of use
JP5789252B2 (ja) 2009-05-07 2015-10-07 インテリカイン, エルエルシー 複素環式化合物およびその使用
AU2010284254B2 (en) 2009-08-17 2015-09-17 Intellikine, Llc Heterocyclic compounds and uses thereof
US8980899B2 (en) 2009-10-16 2015-03-17 The Regents Of The University Of California Methods of inhibiting Ire1
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AR084824A1 (es) 2011-01-10 2013-06-26 Intellikine Inc Procesos para preparar isoquinolinonas y formas solidas de isoquinolinonas
TWI592411B (zh) 2011-02-23 2017-07-21 英特爾立秦有限責任公司 激酶抑制劑之組合及其用途
CA2842190A1 (en) 2011-07-19 2013-01-24 Infinity Pharmaceuticals Inc. Heterocyclic compounds and uses thereof
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EP2751112B1 (en) 2011-09-02 2019-10-09 The Regents of The University of California Substituted pyrazolo[3,4-d]pyrimidines and uses thereof
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US9708348B2 (en) 2014-10-03 2017-07-18 Infinity Pharmaceuticals, Inc. Trisubstituted bicyclic heterocyclic compounds with kinase activities and uses thereof
CN114230571B (zh) 2015-09-14 2025-07-08 无限药品股份有限公司 异喹啉酮的固体形式、其制备方法、包含其的组合物及其使用方法
US10759806B2 (en) 2016-03-17 2020-09-01 Infinity Pharmaceuticals, Inc. Isotopologues of isoquinolinone and quinazolinone compounds and uses thereof as PI3K kinase inhibitors
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US6100254A (en) 1997-10-10 2000-08-08 Board Of Regents, The University Of Texas System Inhibitors of protein tyrosine kinases
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US6610483B1 (en) 1999-07-23 2003-08-26 Princeton University Methods for identifying cellular responses attributable to signaling molecule inhibition and inhibitors thereof

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