JP2000503984A5 - - Google Patents

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Publication number
JP2000503984A5
JP2000503984A5 JP1997526720A JP52672097A JP2000503984A5 JP 2000503984 A5 JP2000503984 A5 JP 2000503984A5 JP 1997526720 A JP1997526720 A JP 1997526720A JP 52672097 A JP52672097 A JP 52672097A JP 2000503984 A5 JP2000503984 A5 JP 2000503984A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP1997526720A
Other languages
English (en)
Japanese (ja)
Other versions
JP2000503984A (ja
Filing date
Publication date
Priority claimed from GBGB9601235.6A external-priority patent/GB9601235D0/en
Priority claimed from AUPO1111A external-priority patent/AUPO111196A0/en
Application filed filed Critical
Priority claimed from PCT/JP1997/000073 external-priority patent/WO1997027190A1/en
Publication of JP2000503984A publication Critical patent/JP2000503984A/ja
Publication of JP2000503984A5 publication Critical patent/JP2000503984A5/ja
Ceased legal-status Critical Current

Links

JP9526720A 1996-01-22 1997-01-17 チアゾリルベンゾフラン誘導体およびその医薬組成物 Ceased JP2000503984A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB9601235.6A GB9601235D0 (en) 1996-01-22 1996-01-22 Novel compounds
AUPO1111A AUPO111196A0 (en) 1996-07-18 1996-07-18 Novel compounds
AU1111 1996-07-18
AU9601235.6 1996-07-18
PCT/JP1997/000073 WO1997027190A1 (en) 1996-01-22 1997-01-17 Thiazolylbenzofuran derivatives and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
JP2000503984A JP2000503984A (ja) 2000-04-04
JP2000503984A5 true JP2000503984A5 (cg-RX-API-DMAC10.html) 2004-11-04

Family

ID=25645218

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9526720A Ceased JP2000503984A (ja) 1996-01-22 1997-01-17 チアゾリルベンゾフラン誘導体およびその医薬組成物

Country Status (12)

Country Link
US (1) US5994378A (cg-RX-API-DMAC10.html)
EP (2) EP1170009B1 (cg-RX-API-DMAC10.html)
JP (1) JP2000503984A (cg-RX-API-DMAC10.html)
KR (1) KR19990076788A (cg-RX-API-DMAC10.html)
CN (1) CN1209809A (cg-RX-API-DMAC10.html)
AT (2) ATE216384T1 (cg-RX-API-DMAC10.html)
CA (1) CA2244189A1 (cg-RX-API-DMAC10.html)
DE (2) DE69728581D1 (cg-RX-API-DMAC10.html)
EA (1) EA199800650A1 (cg-RX-API-DMAC10.html)
ES (1) ES2171878T3 (cg-RX-API-DMAC10.html)
HU (1) HUP9900424A2 (cg-RX-API-DMAC10.html)
WO (1) WO1997027190A1 (cg-RX-API-DMAC10.html)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9919413D0 (en) * 1999-08-18 1999-10-20 Zeneca Ltd Chemical compounds
WO2001032621A1 (en) * 1999-10-29 2001-05-10 Wakunaga Pharmaceutical Co., Ltd. Novel indole derivatives and drugs containing the same as the active ingredient
BR0208956A (pt) * 2001-04-16 2004-07-13 Tanabe Seiyaku Co Abridor de canais de k ativados por cálcio de grande condutância
BRPI0211844B8 (pt) 2001-08-10 2021-05-25 Nippon Chemiphar Co composto de ácido fenóxi-acético ou um de seus sais farmaceuticamente aceitáveis, e, composição farmacêutica
KR100933652B1 (ko) 2001-10-12 2009-12-23 닛뽕 케미파 가부시키가이샤 페록시좀 증식제 응답성 수용체 δ의 활성화제
MX2007000481A (es) * 2004-07-14 2007-03-29 Ptc Therapeutics Inc Metodos para tratar hepatitis c.
US7598397B2 (en) * 2004-10-12 2009-10-06 Decode Genetics Ehf Sulfonamide peri-substituted bicyclics for occlusive artery disease
WO2006046683A1 (en) * 2004-10-25 2006-05-04 Astellas Pharma Inc. Thiazolylbenzofuran derivatives as leukotriene and prostaglandin d2 receptor antagonists
GB2431927B (en) * 2005-11-04 2010-03-17 Amira Pharmaceuticals Inc 5-Lipoxygenase-activating protein (FLAP) inhibitors
US8399666B2 (en) 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
US7977359B2 (en) 2005-11-04 2011-07-12 Amira Pharmaceuticals, Inc. 5-lipdxygenase-activating protein (FLAP) inhibitors
CN101460458A (zh) * 2006-02-15 2009-06-17 阿勒根公司 具有1-磷酸-鞘氨醇(s1p)受体拮抗剂生物活性的带芳基或者杂芳基基团的吲哚-3-羧酸的酰胺、酯、硫代酰胺和硫羟酸酯化合物
AU2007214434B2 (en) * 2006-02-15 2012-06-14 Allergan, Inc. Indole-3-carboxylic acid amide, ester, thioamide and thiol ester compounds bearing aryl or heteroaryl groups having sphingosine-1-phosphate (S1P) receptor antagonist biological activity
NZ572268A (en) 2006-04-18 2011-09-30 Nippon Chemiphar Co Activating agent for peroxisome proliferator activated receptor delta (ppar)
DE102006021733A1 (de) * 2006-05-09 2007-11-22 Bayer Healthcare Ag 3-Tetrazolylindazole und 3-Tetrazolylpyrazolopyridine sowie ihre Verwendung
US7579483B2 (en) * 2006-05-16 2009-08-25 Decode Genetics, Ehf. Process for preparing 7-(acryloyl)indoles
DE102006043443A1 (de) * 2006-09-15 2008-03-27 Bayer Healthcare Ag Neue aza-bicyclische Verbindungen und ihre Verwendung
US8524917B2 (en) 2007-01-11 2013-09-03 Allergan, Inc. 6-substituted indole-3-carboxylic acid amide compounds having sphingosine-1-phosphate (S1P) receptor antagonist biological activity
KR20090101307A (ko) * 2007-01-11 2009-09-24 알러간, 인코포레이티드 스핑고신-1-포스페이트(s1p) 수용체 길항제 생물학적 활성을 갖는 6-치환된 인돌-3-카르복실산 아미드 화합물
JP5474769B2 (ja) 2008-04-15 2014-04-16 日本ケミファ株式会社 ペルオキシソーム増殖剤活性化受容体の活性化剤
US8546431B2 (en) 2008-10-01 2013-10-01 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
DE102008063992A1 (de) 2008-12-19 2010-09-02 Lerner, Zinoviy, Dipl.-Ing. Neue aliphatisch substituierte Pyrazolopyridine und ihre Verwendung
CA2792844C (en) 2010-03-12 2014-12-09 Omeros Corporation Pde10 inhibitors and related compositions and methods
WO2012087833A1 (en) 2010-12-22 2012-06-28 Abbott Laboratories Hepatitis c inhibitors and uses thereof
KR20150119871A (ko) 2013-02-21 2015-10-26 아드베리오 파마 게엠베하 메틸 {4,6-디아미노-2-[1-(2-플루오로벤질)-1H-피라졸로[3,4-b]피리디노-3-일]피리미디노-5-일}메틸 카르바메이트의 형태
NZ630810A (en) 2014-04-28 2016-03-31 Omeros Corp Processes and intermediates for the preparation of a pde10 inhibitor
NZ630803A (en) 2014-04-28 2016-03-31 Omeros Corp Optically active pde10 inhibitor
WO2016033445A1 (en) 2014-08-29 2016-03-03 Chdi Foundation, Inc. Probes for imaging huntingtin protein
US9879002B2 (en) 2015-04-24 2018-01-30 Omeros Corporation PDE10 inhibitors and related compositions and methods
JP2018535969A (ja) 2015-11-04 2018-12-06 オメロス コーポレーション Pde10阻害剤の固体状態形態
AU2018367909B2 (en) 2017-11-17 2022-03-10 Cellix Bio Private Limited Compositions and methods for the treatment of eye disorders

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2600644B2 (ja) * 1991-08-16 1997-04-16 藤沢薬品工業株式会社 チアゾリルベンゾフラン誘導体
JPH07179856A (ja) * 1993-12-21 1995-07-18 Canon Inc 液晶性化合物、これを含有する液晶組成物、該液晶組成物を用いた液晶素子並びにこれらを用いた表示方法、表示装置

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