ITMI992048A0 - Procedimento stereoselettivo per la preparazione di endo-3-amminoazabi cicloalcani - Google Patents
Procedimento stereoselettivo per la preparazione di endo-3-amminoazabi cicloalcaniInfo
- Publication number
- ITMI992048A0 ITMI992048A0 IT99MI002048A ITMI992048A ITMI992048A0 IT MI992048 A0 ITMI992048 A0 IT MI992048A0 IT 99MI002048 A IT99MI002048 A IT 99MI002048A IT MI992048 A ITMI992048 A IT MI992048A IT MI992048 A0 ITMI992048 A0 IT MI992048A0
- Authority
- IT
- Italy
- Prior art keywords
- aminoazab
- cycloalkanes
- endo
- preparation
- stereoselective procedure
- Prior art date
Links
- 150000001924 cycloalkanes Chemical class 0.000 title 1
- 230000000707 stereoselective effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1999MI002048A IT1313660B1 (it) | 1999-10-01 | 1999-10-01 | Procedimento stereoselettivo per la preparazione di endo-3-amminoazabicicloalcani. |
AU73061/00A AU7306100A (en) | 1999-10-01 | 2000-09-26 | A stereoselective process for the preparation of endo-3-aminoazabicycloalkanes |
PCT/IB2000/001360 WO2001025236A2 (en) | 1999-10-01 | 2000-09-26 | A stereoselective process for the preparation of endo-3-aminoazabicycloalkanes |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1999MI002048A IT1313660B1 (it) | 1999-10-01 | 1999-10-01 | Procedimento stereoselettivo per la preparazione di endo-3-amminoazabicicloalcani. |
Publications (3)
Publication Number | Publication Date |
---|---|
ITMI992048A0 true ITMI992048A0 (it) | 1999-10-01 |
ITMI992048A1 ITMI992048A1 (it) | 2001-04-01 |
IT1313660B1 IT1313660B1 (it) | 2002-09-09 |
Family
ID=11383702
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT1999MI002048A IT1313660B1 (it) | 1999-10-01 | 1999-10-01 | Procedimento stereoselettivo per la preparazione di endo-3-amminoazabicicloalcani. |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU7306100A (it) |
IT (1) | IT1313660B1 (it) |
WO (1) | WO2001025236A2 (it) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200533348A (en) | 2004-02-18 | 2005-10-16 | Theravance Inc | Indazole-carboxamide compounds as 5-ht4 receptor agonists |
DE602005016446D1 (de) | 2004-11-05 | 2009-10-15 | Theravance Inc | 5-HT4-Rezeptoragonistenverbindungen |
ATE431824T1 (de) | 2004-11-05 | 2009-06-15 | Theravance Inc | Chinolinon-carboxamid-verbindungen |
ES2347265T3 (es) | 2004-12-22 | 2010-10-27 | Theravance, Inc. | Compuestos de indazol-carboxamida. |
KR20070107807A (ko) | 2005-03-02 | 2007-11-07 | 세라밴스 인코포레이티드 | 5-ht4 수용체 아고니스트인 퀴놀리논 화합물 |
EP1984362B1 (en) | 2006-02-16 | 2011-05-11 | Theravance, Inc. | Process for preparing intermediates to 5-ht4 receptor agonist compounds |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL59004A0 (en) * | 1978-12-30 | 1980-03-31 | Beecham Group Ltd | Substituted benzamides their preparation and pharmaceutical compositions containing them |
US5625065A (en) * | 1994-06-27 | 1997-04-29 | Eli Lilly And Company | Stereoselective process for making endo-tropanamine and like compounds |
GB9414900D0 (en) * | 1994-07-23 | 1994-09-14 | Smithkline Beecham Plc | Novel process |
-
1999
- 1999-10-01 IT IT1999MI002048A patent/IT1313660B1/it active
-
2000
- 2000-09-26 WO PCT/IB2000/001360 patent/WO2001025236A2/en active Search and Examination
- 2000-09-26 AU AU73061/00A patent/AU7306100A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
IT1313660B1 (it) | 2002-09-09 |
WO2001025236A3 (en) | 2002-01-17 |
AU7306100A (en) | 2001-05-10 |
ITMI992048A1 (it) | 2001-04-01 |
WO2001025236A2 (en) | 2001-04-12 |
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