ITMI992048A0 - Procedimento stereoselettivo per la preparazione di endo-3-amminoazabi cicloalcani - Google Patents

Procedimento stereoselettivo per la preparazione di endo-3-amminoazabi cicloalcani

Info

Publication number
ITMI992048A0
ITMI992048A0 IT99MI002048A ITMI992048A ITMI992048A0 IT MI992048 A0 ITMI992048 A0 IT MI992048A0 IT 99MI002048 A IT99MI002048 A IT 99MI002048A IT MI992048 A ITMI992048 A IT MI992048A IT MI992048 A0 ITMI992048 A0 IT MI992048A0
Authority
IT
Italy
Prior art keywords
aminoazab
cycloalkanes
endo
preparation
stereoselective procedure
Prior art date
Application number
IT99MI002048A
Other languages
English (en)
Inventor
Marcello Allegretti
Roberto Curti
Maria Candida Cesta
Luca Nicolini
Original Assignee
Dompe Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dompe Spa filed Critical Dompe Spa
Priority to IT1999MI002048A priority Critical patent/IT1313660B1/it
Publication of ITMI992048A0 publication Critical patent/ITMI992048A0/it
Priority to AU73061/00A priority patent/AU7306100A/en
Priority to PCT/IB2000/001360 priority patent/WO2001025236A2/en
Publication of ITMI992048A1 publication Critical patent/ITMI992048A1/it
Application granted granted Critical
Publication of IT1313660B1 publication Critical patent/IT1313660B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
IT1999MI002048A 1999-10-01 1999-10-01 Procedimento stereoselettivo per la preparazione di endo-3-amminoazabicicloalcani. IT1313660B1 (it)

Priority Applications (3)

Application Number Priority Date Filing Date Title
IT1999MI002048A IT1313660B1 (it) 1999-10-01 1999-10-01 Procedimento stereoselettivo per la preparazione di endo-3-amminoazabicicloalcani.
AU73061/00A AU7306100A (en) 1999-10-01 2000-09-26 A stereoselective process for the preparation of endo-3-aminoazabicycloalkanes
PCT/IB2000/001360 WO2001025236A2 (en) 1999-10-01 2000-09-26 A stereoselective process for the preparation of endo-3-aminoazabicycloalkanes

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1999MI002048A IT1313660B1 (it) 1999-10-01 1999-10-01 Procedimento stereoselettivo per la preparazione di endo-3-amminoazabicicloalcani.

Publications (3)

Publication Number Publication Date
ITMI992048A0 true ITMI992048A0 (it) 1999-10-01
ITMI992048A1 ITMI992048A1 (it) 2001-04-01
IT1313660B1 IT1313660B1 (it) 2002-09-09

Family

ID=11383702

Family Applications (1)

Application Number Title Priority Date Filing Date
IT1999MI002048A IT1313660B1 (it) 1999-10-01 1999-10-01 Procedimento stereoselettivo per la preparazione di endo-3-amminoazabicicloalcani.

Country Status (3)

Country Link
AU (1) AU7306100A (it)
IT (1) IT1313660B1 (it)
WO (1) WO2001025236A2 (it)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200533348A (en) 2004-02-18 2005-10-16 Theravance Inc Indazole-carboxamide compounds as 5-ht4 receptor agonists
DE602005016446D1 (de) 2004-11-05 2009-10-15 Theravance Inc 5-HT4-Rezeptoragonistenverbindungen
ATE431824T1 (de) 2004-11-05 2009-06-15 Theravance Inc Chinolinon-carboxamid-verbindungen
ES2347265T3 (es) 2004-12-22 2010-10-27 Theravance, Inc. Compuestos de indazol-carboxamida.
KR20070107807A (ko) 2005-03-02 2007-11-07 세라밴스 인코포레이티드 5-ht4 수용체 아고니스트인 퀴놀리논 화합물
EP1984362B1 (en) 2006-02-16 2011-05-11 Theravance, Inc. Process for preparing intermediates to 5-ht4 receptor agonist compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL59004A0 (en) * 1978-12-30 1980-03-31 Beecham Group Ltd Substituted benzamides their preparation and pharmaceutical compositions containing them
US5625065A (en) * 1994-06-27 1997-04-29 Eli Lilly And Company Stereoselective process for making endo-tropanamine and like compounds
GB9414900D0 (en) * 1994-07-23 1994-09-14 Smithkline Beecham Plc Novel process

Also Published As

Publication number Publication date
IT1313660B1 (it) 2002-09-09
WO2001025236A3 (en) 2002-01-17
AU7306100A (en) 2001-05-10
ITMI992048A1 (it) 2001-04-01
WO2001025236A2 (en) 2001-04-12

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