IT8421705A0 - Sostanze anti-ulcera ad attivita'citoprotettiva. - Google Patents

Sostanze anti-ulcera ad attivita'citoprotettiva.

Info

Publication number
IT8421705A0
IT8421705A0 IT8421705A IT2170584A IT8421705A0 IT 8421705 A0 IT8421705 A0 IT 8421705A0 IT 8421705 A IT8421705 A IT 8421705A IT 2170584 A IT2170584 A IT 2170584A IT 8421705 A0 IT8421705 A0 IT 8421705A0
Authority
IT
Italy
Prior art keywords
cytoprotective activity
ulcer
substances
ulcer substances
cytoprotective
Prior art date
Application number
IT8421705A
Other languages
English (en)
Other versions
IT1207046B (it
Inventor
Peter Frederick Juby
Thomas William Hudyma
Douglas G Colton
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of IT8421705A0 publication Critical patent/IT8421705A0/it
Application granted granted Critical
Publication of IT1207046B publication Critical patent/IT1207046B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IT8421705A 1983-07-22 1984-07-02 Sostanze anti-ulcera ad attivita'citoprotettiva. IT1207046B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/516,026 US4457932A (en) 1983-07-22 1983-07-22 Anti-ulcer agents

Publications (2)

Publication Number Publication Date
IT8421705A0 true IT8421705A0 (it) 1984-07-02
IT1207046B IT1207046B (it) 1989-05-17

Family

ID=24053806

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8421705A IT1207046B (it) 1983-07-22 1984-07-02 Sostanze anti-ulcera ad attivita'citoprotettiva.

Country Status (7)

Country Link
US (1) US4457932A (it)
BE (1) BE900082A (it)
CA (1) CA1227428A (it)
DE (1) DE3424324A1 (it)
IT (1) IT1207046B (it)
PT (1) PT78834B (it)
ZA (1) ZA845044B (it)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1283411C (en) * 1985-09-25 1991-04-23 Masami Doteuchi 9-(substituted thio)-4h-pyrido[1,2-a]-pyrimidin-4-one derivatives
US5547943A (en) * 1986-04-30 1996-08-20 Chugai Seiyaku Kabushiki Kaisha Sucralfate preparation
JP2504788B2 (ja) * 1987-11-10 1996-06-05 東京田辺製薬株式会社 9−メチル−3−(1H−テトラゾ―ル−5−イル)−4H−ピリド[1,2−a]ピリミジン−4−オンカリウム塩の水性製剤
JP2668259B2 (ja) * 1988-02-18 1997-10-27 塩野義製薬株式会社 複素環化合物および抗潰瘍剤
HU209793B (en) * 1990-09-25 1994-11-28 Chinoin Gyogyszer Es Vegyeszet Process for the production of pyrido[1,2-a]pyrimidine-derivatives and pharmaceutical compositions containing the same
US5527802A (en) * 1992-10-01 1996-06-18 Bristol-Myers Squibb Company New uses of 3-tetrazolo -5,6,7,8- substituted-pyrido (1,2-a) pyrimidin-4-ones
US7226624B2 (en) * 2002-07-24 2007-06-05 Rabinowitz Israel N Synergistic compositions from yeast-modified aqueous extracts from almond hulls
EP1818058A3 (en) * 2006-02-13 2007-11-07 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
WO2007093184A2 (en) * 2006-02-13 2007-08-23 Astion Pharma A/S Treatment of mmp-mediated dermatological diseases with pemirolast
US20070225301A1 (en) * 2006-02-13 2007-09-27 Astion Inflammation Aps Treatment of acne and other diseases

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3072485A (en) * 1960-08-24 1963-01-08 Eastman Kodak Co Optically sensitized azido polymers for photomechanical resist compositions
CH538494A (de) * 1966-11-02 1973-06-30 Chinoin Gyogyszer Es Vegyeszet Verfahren zur Herstellung neuer Homopyrimidazol-Derivate
US4152448A (en) * 1972-02-15 1979-05-01 Fisons Limited Method and composition for the treatment of a condition of the gastro intestinal tract
US3960847A (en) * 1972-04-17 1976-06-01 E. R. Squibb & Sons, Inc. 9-Substituted-4-oxopyrido(1,2-α)pyrimidine-3-carboxylic acids and derivatives thereof
US3855216A (en) * 1973-05-29 1974-12-17 Warner Lambert Co Substituted pyrano(3,2-c)(1,2)benzothiazine 6,6-dioxides
US3862141A (en) * 1973-08-23 1975-01-21 Warner Lambert Co 1-substituted 1,2,3,4-tetrahydroxanthen-9-ones
US3929787A (en) * 1974-04-22 1975-12-30 Squibb & Sons Inc 6,7,8,9-Tetrahydro-pyrido(1,2-a)pyrimidin-4-ones
US4014881A (en) * 1975-07-10 1977-03-29 Pfizer Inc. 1-Oxo-1H-6-piperidinopyrimido[1,2-a]quinoline-2-carboxylic acids and esters
US4041163A (en) * 1976-03-29 1977-08-09 Pfizer Inc. N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents
US4141979A (en) * 1976-12-23 1979-02-27 Pfizer Inc. Tetrazolo[a]quinazol-5-ones antiallergy and antiulcer agents
US4122274A (en) * 1977-05-25 1978-10-24 Bristol-Myers Company 3-Tetrazolo-5,6,7,8-substituted-pyrido[1,2-a]pyrimidin-4-ones
US4105766A (en) * 1977-08-19 1978-08-08 Sterling Drug Inc. 4,5-Dihydro-5-oxopyrazolo[1,5-a]quinazoline-3-carboxylic acid derivatives
US4105764A (en) * 1977-08-19 1978-08-08 Sterling Drug Inc. 4,5-Dihydro-5-oxopyrazolo[1,5-A]quinazoline-3-carboxamides
US4209620A (en) * 1978-06-19 1980-06-24 Bristol-Myers Company Substituted 3-(1H-tetrazol-5-yl)-4H-pyrido[1,2-a]pyrimidin-4-one derivatives having antiallergy activity
US4215216A (en) * 1979-04-18 1980-07-29 American Home Products Corporation 7,8-Dihydro-2,5,8-trisubstituted-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives
IL59802A (en) * 1979-05-08 1983-07-31 Erba Farmitalia Substituted pyrido(1,2-a)pyrimidine carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
DK151811C (da) * 1979-11-23 1988-06-06 Pfizer Analogifremgangsmaade til fremstilling af n-(5-tetrazolyl)-1-oxo-1h-thiazolooe3,2-aaa-pyrimidin-2-carboxamider eller farmaceutisk acceptable kationsalte deraf samt 1-oxo-1h-thiazolooe3,2-aaapyrimidin-2-carboxylsyrer til anvendelse som udgangsmaterialer ved fremgangsmaaden

Also Published As

Publication number Publication date
ZA845044B (en) 1985-03-27
US4457932A (en) 1984-07-03
DE3424324A1 (de) 1985-01-31
BE900082A (fr) 1985-01-03
DE3424324C2 (it) 1993-07-01
PT78834B (en) 1986-10-21
IT1207046B (it) 1989-05-17
PT78834A (en) 1984-08-01
CA1227428A (en) 1987-09-29

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Legal Events

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970730