IT8322998A0 - Esteri 3-acilammino-2-osso-1-azetidinilici di acidi fosfonici, acido fosforico e esteri dell'acido fosforico ad attivita'antimicrobica. - Google Patents

Esteri 3-acilammino-2-osso-1-azetidinilici di acidi fosfonici, acido fosforico e esteri dell'acido fosforico ad attivita'antimicrobica.

Info

Publication number
IT8322998A0
IT8322998A0 IT8322998A IT2299883A IT8322998A0 IT 8322998 A0 IT8322998 A0 IT 8322998A0 IT 8322998 A IT8322998 A IT 8322998A IT 2299883 A IT2299883 A IT 2299883A IT 8322998 A0 IT8322998 A0 IT 8322998A0
Authority
IT
Italy
Prior art keywords
esters
phosphoric acid
azetidinylic
acylamino
oxo
Prior art date
Application number
IT8322998A
Other languages
English (en)
Other versions
IT1169846B (it
Inventor
William A Slusarchyk
Tamara Dejneka
William H Koster
Eric M Gordon
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of IT8322998A0 publication Critical patent/IT8322998A0/it
Application granted granted Critical
Publication of IT1169846B publication Critical patent/IT1169846B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/568Four-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT22998/83A 1982-09-27 1983-09-26 Esteri 3-acilammino-2-osso-1-azetidinilici di acidi fosfonici, acido fosforico e esteri dell'acido fosforico ad attivita'antimicrobica IT1169846B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/424,132 US4681937A (en) 1982-09-27 1982-09-27 3-acylamino-2-oxo-1-azetidinyl esters of phosphonic acids, phosphoric acid and phosphoric acid esters

Publications (2)

Publication Number Publication Date
IT8322998A0 true IT8322998A0 (it) 1983-09-26
IT1169846B IT1169846B (it) 1987-06-03

Family

ID=23681576

Family Applications (1)

Application Number Title Priority Date Filing Date
IT22998/83A IT1169846B (it) 1982-09-27 1983-09-26 Esteri 3-acilammino-2-osso-1-azetidinilici di acidi fosfonici, acido fosforico e esteri dell'acido fosforico ad attivita'antimicrobica

Country Status (7)

Country Link
US (1) US4681937A (it)
JP (1) JPS5978199A (it)
CA (1) CA1268763C (it)
DE (1) DE3334984A1 (it)
FR (1) FR2533569A1 (it)
GB (1) GB2127411B (it)
IT (1) IT1169846B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985004876A1 (en) * 1984-04-24 1985-11-07 Takeda Chemical Industries, Ltd. 2-azetidinone derivatives and process for their preparation
CN103435650B (zh) * 2012-12-28 2015-12-02 南京海融医药科技有限公司 单环β-内酰胺类化合物、制备方法及其制药用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS604811B2 (ja) * 1976-07-28 1985-02-06 塩野義製薬株式会社 メチルケトンのハロゲン化
NZ205240A (en) * 1980-02-07 1984-07-31 Squibb & Sons Inc Sulphonamide derivatives,being starting materials for producing beta-lactams
US4337197A (en) * 1980-10-31 1982-06-29 E. R. Squibb & Sons, Inc. O-sulfated β-lactam hydroxamic acids and intermediates
WO1982001873A1 (en) * 1980-12-05 1982-06-10 Takeda Chemical Industries Ltd 1-sulfo-2-oxoazetidine derivatives and process for their preparation
MX7096E (es) * 1980-12-05 1987-06-19 Takeda Chemical Industries Ltd Metodo para preparacion de derivados de 2-oxoazetidina

Also Published As

Publication number Publication date
DE3334984A1 (de) 1984-03-29
JPS5978199A (ja) 1984-05-04
CA1262134A (en) 1989-10-03
IT1169846B (it) 1987-06-03
GB2127411A (en) 1984-04-11
US4681937A (en) 1987-07-21
GB2127411B (en) 1986-04-03
GB8323276D0 (en) 1983-10-05
FR2533569A1 (fr) 1984-03-30
CA1268763C (en) 1990-05-08
FR2533569B1 (it) 1985-04-19

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