IT8249095A0 - DERIVATIVES OF 4-PYRIDILPYRYDAZINONE WITH ANTI-INFLAMMATORY AND ANALGESIC ACTIVITY - Google Patents
DERIVATIVES OF 4-PYRIDILPYRYDAZINONE WITH ANTI-INFLAMMATORY AND ANALGESIC ACTIVITYInfo
- Publication number
- IT8249095A0 IT8249095A0 IT8249095A IT4909582A IT8249095A0 IT 8249095 A0 IT8249095 A0 IT 8249095A0 IT 8249095 A IT8249095 A IT 8249095A IT 4909582 A IT4909582 A IT 4909582A IT 8249095 A0 IT8249095 A0 IT 8249095A0
- Authority
- IT
- Italy
- Prior art keywords
- pyridilpyrydazinone
- inflammatory
- derivatives
- analgesic activity
- analgesic
- Prior art date
Links
- 230000001760 anti-analgesic effect Effects 0.000 title 1
- 230000003110 anti-inflammatory effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US30132881A | 1981-09-11 | 1981-09-11 |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8249095A0 true IT8249095A0 (en) | 1982-09-09 |
IT1149073B IT1149073B (en) | 1986-12-03 |
Family
ID=23162890
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT49095/82A IT1149073B (en) | 1981-09-11 | 1982-09-09 | 4-PYRIDYLPYRIDAZINONE DERIVATIVES EQUIPPED WITH ANTI-INFLAMMATORY AND ANALGESIC ACTIVITY |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0088128A4 (en) |
JP (1) | JPS58501432A (en) |
IL (1) | IL66761A0 (en) |
IT (1) | IT1149073B (en) |
WO (1) | WO1983000863A1 (en) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5622948A (en) * | 1994-12-01 | 1997-04-22 | Syntex (U.S.A.) Inc. | Pyrrole pyridazine and pyridazinone anti-inflammatory agents |
US6004960A (en) * | 1997-03-14 | 1999-12-21 | Merck Frosst Canada, Inc. | Pyridazinones as inhibitors of cyclooxygenase-2 |
CA2283399C (en) * | 1997-03-14 | 2006-02-21 | Merck Frosst Canada & Co. | Pyridazinones as inhibitors of cyclooxygenase-2 |
PT1043317E (en) * | 1997-11-19 | 2009-05-11 | Kowa Co | Pyridazine derivatives and medicaments containing them as active ingredient |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB840522A (en) * | 1957-11-05 | 1960-07-06 | Lepetit Spa | A new analgesic 2-hydroxymethyl-6-phenyl-3-pyridazone |
US3920646A (en) * | 1967-11-02 | 1975-11-18 | Sandoz Ag | 3-Substituted-1-pyridyl-1,4,5,6-tetrahydropyridazines |
US3658814A (en) * | 1970-03-17 | 1972-04-25 | Sandoz Ag | 2-(omega-chloroalkyl)-6-aryl substituted-4 5-dihydropyridazin(2h)-3-one |
CH557820A (en) * | 1970-11-12 | 1975-01-15 | Sandoz Ag | METHOD OF PREPARING NEW 2- (2-HYDROXYALKYL) 4,5-DIHYDRO-PYRIDAZINE (2H) -3-ONES. |
AT333774B (en) * | 1974-09-24 | 1976-12-10 | Chemie Linz Ag | PROCESS FOR THE PREPARATION OF 3-PHENYLPYRIDAZONES |
JPS5419987A (en) * | 1977-07-15 | 1979-02-15 | Yoshitomi Pharmaceut Ind Ltd | Pyridazinone derivative and its preparation |
DE2834624A1 (en) * | 1978-08-08 | 1980-02-28 | Bayer Ag | NEW 1,4-DIHYDROPYRIDAZINE-3-CARBONIC ACID DERIVATIVES, METHOD FOR THE PRODUCTION AND USE THEREOF AS A MEDICINAL PRODUCT |
US4238490A (en) * | 1979-02-12 | 1980-12-09 | Diamond Shamrock Corporation | Antihypertensive pyridazin(2H)-3-ones |
US4298609A (en) * | 1979-08-30 | 1981-11-03 | Sterling Drug Inc. | 4,5-Dihydro-6-(4-pyridinyl)-3-pyridazinol and salts, their preparation and use as blood pressure lowering agents |
-
1982
- 1982-08-18 WO PCT/US1982/001118 patent/WO1983000863A1/en not_active Application Discontinuation
- 1982-08-18 JP JP57503139A patent/JPS58501432A/en active Pending
- 1982-08-18 EP EP19820903161 patent/EP0088128A4/en not_active Withdrawn
- 1982-09-09 IT IT49095/82A patent/IT1149073B/en active
- 1982-09-10 IL IL66761A patent/IL66761A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP0088128A4 (en) | 1984-04-06 |
IT1149073B (en) | 1986-12-03 |
IL66761A0 (en) | 1982-12-31 |
JPS58501432A (en) | 1983-08-25 |
EP0088128A1 (en) | 1983-09-14 |
WO1983000863A1 (en) | 1983-03-17 |
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