IT8148952A0 - AMIDINATED AMINOGLUCOSIDES PROCEDURE FOR THEIR PREPARATION AND THEIR USE AS MEDICINES - Google Patents

AMIDINATED AMINOGLUCOSIDES PROCEDURE FOR THEIR PREPARATION AND THEIR USE AS MEDICINES

Info

Publication number
IT8148952A0
IT8148952A0 IT8148952A IT4895281A IT8148952A0 IT 8148952 A0 IT8148952 A0 IT 8148952A0 IT 8148952 A IT8148952 A IT 8148952A IT 4895281 A IT4895281 A IT 4895281A IT 8148952 A0 IT8148952 A0 IT 8148952A0
Authority
IT
Italy
Prior art keywords
amidinated
aminoglucosides
medicines
procedure
preparation
Prior art date
Application number
IT8148952A
Other languages
Italian (it)
Other versions
IT1171411B (en
Inventor
Loibner Hans
Streicher Wolfgang
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IT8148952A0 publication Critical patent/IT8148952A0/en
Application granted granted Critical
Publication of IT1171411B publication Critical patent/IT1171411B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • C07H15/236—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2 a saccharide radical being substituted by an alkylamino radical in position 3 and by two substituents different from hydrogen in position 4, e.g. gentamicin complex, sisomicin, verdamycin
IT48952/81A 1980-07-28 1981-07-22 AMMINOGLUCOSIDES AMMIDINATED PROCEDURE FOR THEIR PREPARATION AND USE AS A MEDICATION IT1171411B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH575680 1980-07-28
CH777880 1980-10-17
CH184281 1981-03-18

Publications (2)

Publication Number Publication Date
IT8148952A0 true IT8148952A0 (en) 1981-07-22
IT1171411B IT1171411B (en) 1987-06-10

Family

ID=27173293

Family Applications (1)

Application Number Title Priority Date Filing Date
IT48952/81A IT1171411B (en) 1980-07-28 1981-07-22 AMMINOGLUCOSIDES AMMIDINATED PROCEDURE FOR THEIR PREPARATION AND USE AS A MEDICATION

Country Status (9)

Country Link
EP (1) EP0056408A1 (en)
JP (1) JPS57501084A (en)
CS (1) CS228516B2 (en)
GR (1) GR74312B (en)
IL (1) IL63429A0 (en)
IT (1) IT1171411B (en)
PT (1) PT73428B (en)
WO (1) WO1982000464A1 (en)
YU (1) YU184481A (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2707787T3 (en) 2005-12-02 2019-04-05 Ionis Pharmaceuticals Inc Antibacterial analogs of 4,5-substituted aminoglycoside having multiple substituents
EP2324076B1 (en) 2008-07-31 2017-11-01 3M Innovative Properties Company Fluoropolymer compositions and method of making and using thereof
EP2315802A4 (en) * 2008-07-31 2012-04-18 3M Innovative Properties Co Azide compositions and methods of making and using thereof
WO2010030704A2 (en) 2008-09-10 2010-03-18 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010030690A1 (en) 2008-09-10 2010-03-18 Isis Pharmaceuticals, Inc. Antibacterial 4,6-substituted 6', 6" and 1 modified aminoglycoside analogs
WO2010042851A1 (en) 2008-10-09 2010-04-15 Achaogen, Inc. Antibacterial aminoglycoside analogs
WO2010042850A1 (en) 2008-10-09 2010-04-15 Achaogen, Inc. Antibacterial aminoglycoside analogs
EP2486044A2 (en) 2009-10-09 2012-08-15 Achaogen, Inc. Antibacterial aminoglycoside analogs
AR083879A1 (en) 2010-11-17 2013-03-27 Achaogen Inc ANTIBACTERIAL AMINOGLYCOSID ANALOGS, METHODS OF PREPARATION AND USE AS THERAPEUTIC AGENTS
CN116462721B (en) * 2023-04-18 2024-02-02 江南大学 Antibacterial aminoglycoside derivative

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1087537A (en) * 1975-08-21 1980-10-14 John H. E. J. Martin Antibiotic bm123 and production thereof
JPS5488241A (en) * 1977-12-21 1979-07-13 Kyowa Hakko Kogyo Co Ltd Novel fortimicin a derivative

Also Published As

Publication number Publication date
WO1982000464A1 (en) 1982-02-18
CS228516B2 (en) 1984-05-14
PT73428B (en) 1983-01-13
YU184481A (en) 1983-09-30
PT73428A (en) 1981-08-01
IL63429A0 (en) 1981-10-30
EP0056408A1 (en) 1982-07-28
JPS57501084A (en) 1982-06-24
IT1171411B (en) 1987-06-10
GR74312B (en) 1984-06-22

Similar Documents

Publication Publication Date Title
IT1137272B (en) INTERCOMS AND PROCEDURE FOR THEIR PREPARATION
IT1189229B (en) POLIPEPTEDI, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1194394B (en) CEFEM-DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION
IT1172093B (en) DIBENZAZEPINE THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1167782B (en) KINOXALIN-2-IL-ETHENYL-KETONES AND PROCEDURE FOR THEIR PREPARATION
IT1164076B (en) PHARMACEUTICAL COMPOUNDS WITH ANTI-ULTER ACTION AND PROCEDURE FOR THEIR PREPARATION
IT8048615A0 (en) PYRAZINOBENZODIAZEPINES THEIR PREPARATION AND THEIR USE AS MEDICINES
IT8348232A0 (en) AZEPINOINDOLS, THEIR PREPARATION AND THEIR USE AS MEDICINES
IT8148952A0 (en) AMIDINATED AMINOGLUCOSIDES PROCEDURE FOR THEIR PREPARATION AND THEIR USE AS MEDICINES
IT1108968B (en) ACETYLENPROSTAGLANDINE AND PROCEDURE FOR THEIR PREPARATION
IT1160450B (en) NITROSUREIC COMPOUNDS AND PROCEDURE FOR THEIR PREPARATION
IT1171361B (en) AMINOCYCLOPENTANON-AMIDES AND PROCEDURE FOR THEIR PHARMACEUTICAL PREPARATION AND FORMULATION
IT1107653B (en) IMIDAZO-CHINOLIN-DIONI AND PROCEDURE FOR THEIR PREPARATION
IT1194158B (en) CARBACICLINE, PROCEDURE FOR THEIR PREPARATION AND USE AS MEDICINAL PRODUCTS
IT1165040B (en) ALCOSSIALKILIDENIDRAZINOPIRIDAZIONE AND PROCEDURE FOR THEIR PREPARATION
IT1136556B (en) TIOLI AND THEIR PREPARATION
FI810874L (en) PHARMACEUTICAL PREPARATION
IT8347702A0 (en) ERGOPEPTIDE ALKALOIDS, THEIR PREPARATION AND THEIR USE AS MEDICINES
IT7950162A0 (en) SUBSTITUTED AMINOALKYLGUANIDINES AND PROCEDURE FOR THEIR PREPARATION
IT1104583B (en) 3-DI-N-PROFIL-ACETOXY-BENZO-DIAZEPIN-2-ONI AND PROCEDURE FOR THEIR PREPARATION
IT8147787A0 (en) PIPERAZINE COMPOUNDS: PROCEDURE FOR PREPARING THEM AND THEIR USE
IT1130215B (en) 3-ARILTIO-4-HYDROXYPYRROLIDINE 1-REPLACED AND PROCEDURE FOR THEIR PREPARATION
IT1164412B (en) CIANALCHILPIPERAZINE PROCEDURES FOR THEIR PREPARATION AND USE
IT1143906B (en) TIOCARNITINE PROCEDURE FOR THEIR PREPARATION AND THERAPEUTIC USE
IT1164413B (en) 2-PYRIMIDYLALCAN-SULPHONATES PROCEDURES FOR THEIR PREPARATION AND USE