IT8049233A0 - Composizioni farmaceutiche contenenti composti eterociclici derivati dalla pirazolina ad attivita'anti spasmodica e procedimento per laloro preparazione - Google Patents

Composizioni farmaceutiche contenenti composti eterociclici derivati dalla pirazolina ad attivita'anti spasmodica e procedimento per laloro preparazione

Info

Publication number
IT8049233A0
IT8049233A0 IT8049233A IT4923380A IT8049233A0 IT 8049233 A0 IT8049233 A0 IT 8049233A0 IT 8049233 A IT8049233 A IT 8049233A IT 4923380 A IT4923380 A IT 4923380A IT 8049233 A0 IT8049233 A0 IT 8049233A0
Authority
IT
Italy
Prior art keywords
pyrazolin
procedure
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
IT8049233A
Other languages
English (en)
Other versions
IT1207128B (it
Inventor
Albert Gordon Caldwell
Stanley Richard Challand
Frederick Charles Copp
Clive Vincent Denyer
Kenneth Ernest Eakins
John Michael Graham Walker
Norman Whittaker
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of IT8049233A0 publication Critical patent/IT8049233A0/it
Application granted granted Critical
Publication of IT1207128B publication Critical patent/IT1207128B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT8049233A 1979-07-13 1980-07-11 Composizioni farmaceutiche contenenti composti eterociclici derivati dalla pirazolina ad attivita'anti spasmodica e procedimento per laloro preparazione IT1207128B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US5736279A 1979-07-13 1979-07-13

Publications (2)

Publication Number Publication Date
IT8049233A0 true IT8049233A0 (it) 1980-07-11
IT1207128B IT1207128B (it) 1989-05-17

Family

ID=22010106

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8049233A IT1207128B (it) 1979-07-13 1980-07-11 Composizioni farmaceutiche contenenti composti eterociclici derivati dalla pirazolina ad attivita'anti spasmodica e procedimento per laloro preparazione

Country Status (10)

Country Link
EP (1) EP0022578B1 (it)
JP (1) JPS5632416A (it)
AU (1) AU537499B2 (it)
CA (1) CA1150632A (it)
DE (1) DE3072103D1 (it)
DK (1) DK302880A (it)
IL (1) IL60550A (it)
IT (1) IT1207128B (it)
NZ (1) NZ194328A (it)
ZA (1) ZA804196B (it)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL64555A (en) * 1980-12-16 1986-01-31 Wellcome Found Pharmaceutical compositions containing aryl-pyrazolineamine derivatives,certain such novel derivatives and their preparation
US4465685A (en) * 1980-12-23 1984-08-14 Burroughs Wellcome Co. Antiinflammatory pyrazole thioureas
US4572913A (en) * 1980-12-23 1986-02-25 Burroughs Wellcome Co. Use of 3-(arylmethyleneamino)-1-aryl-2-pyrazolines in the prophylaxis and treatment of inflammation, pain, pyresis, and asthma
US4447442A (en) * 1981-07-13 1984-05-08 American Cyanamid Company 3-Trifluoroacetylamino-1-aryl-2-pyrazolines
EP0070376A1 (en) * 1981-07-13 1983-01-26 American Cyanamid Company Heterocyclic substituted-amino-pyrazolines
US4451479A (en) * 1981-07-13 1984-05-29 American Cyanamid Company Therapeutically active 3-amino-1-halogenated phenyl-2-pyrazolines and their C4 and C5 analogs
US4432991A (en) * 1981-07-13 1984-02-21 American Cyanamid Company Therapeutically active 3-amino-1-phenyl(and substituted phenyl)-2-pyrazolines
US4448783A (en) * 1982-05-17 1984-05-15 Burroughs Wellcome Co. Substituted pyrazoline, and its use in treatment of gastro-intestinal disturbances
EP0119450A1 (en) * 1983-02-11 1984-09-26 The Wellcome Foundation Limited Preparation of aminopyrazolines and intermediates used therein
GB8303782D0 (en) * 1983-02-11 1983-03-16 Wellcome Found Heterocyclic compounds
US4824859A (en) * 1983-05-21 1989-04-25 Fisons Plc. Pyrazoline compounds compositions and use
ATE49198T1 (de) * 1984-05-12 1990-01-15 Fisons Plc Antiinflammatorische 1,n-diarylpyrazol-3-amine, deren zusammensetzungen und verfahren zu deren herstellung.
US4970210A (en) * 1987-07-17 1990-11-13 Abbott Laboratories Triazinone lipoxygenase compounds
NZ739834A (en) 2012-10-02 2018-11-30 Bayer Cropscience Ag Heterocyclic compounds as pesticides
US9108946B2 (en) * 2013-10-17 2015-08-18 Dow Agrosciences Llc Processes for the preparation of pesticidal compounds
WO2016018444A1 (en) * 2014-07-31 2016-02-04 Dow Agrosciences Llc Process for the preparation of 3-(3-chloro-1h-pyrazol-1-yl)pyridine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1324687A (en) * 1970-08-06 1973-07-25 Chinoin Gyogyszer Es Vegyeszet 3-amino-delta2-pyrazoline derivatives and process for the preparation thereof
IT1061812B (it) * 1976-06-25 1983-04-30 Montedison Spa Processo per la preparazione di i fenil 3 ammino pirazoli

Also Published As

Publication number Publication date
IT1207128B (it) 1989-05-17
EP0022578B1 (en) 1988-06-29
IL60550A0 (en) 1980-09-16
NZ194328A (en) 1985-03-20
CA1150632A (en) 1983-07-26
DE3072103D1 (en) 1988-08-04
ZA804196B (en) 1982-02-24
AU6032780A (en) 1981-01-15
AU537499B2 (en) 1984-06-28
JPH0248549B2 (it) 1990-10-25
IL60550A (en) 1984-12-31
EP0022578A1 (en) 1981-01-21
JPS5632416A (en) 1981-04-01
DK302880A (da) 1981-01-14

Similar Documents

Publication Publication Date Title
NZ192615A (en) Substituted phenyl j-substituted piperidinoalkanone derivatives and pharmaceutical compositions
DE3071738D1 (en) 2,3-dihydro-1h-indole derivatives and intermediates therefor, processes for their preparation, pharmaceutical compositions containing these derivatives and their preparation
IT8049233A0 (it) Composizioni farmaceutiche contenenti composti eterociclici derivati dalla pirazolina ad attivita'anti spasmodica e procedimento per laloro preparazione
IT8048394A0 (it) Procedimento per preparare composizioni farmaceutiche attivate
DE3064910D1 (en) 2-oxo-benzothiazoline, benzoxazoline or indoline derivatives, their preparation, and pharmaceutical compositions comprising such derivatives
AR226845A1 (es) Compuestos de eter 2-halo-4-halo o trifluormetil-3'-carbonilo substituido-4'-nitrodifenilico,composicion herbicida que los contiene y procedimientos para prepararlos
AR231987A1 (es) Procedimiento para preparar derivados farmaceuticos de pirrolo-2,1-c 1,4 tiazepin-1,5-diona y compuesto intermediario para uso exclusivo en el mismo
IL59770A (en) Pharmaceutical compositions containing 3-alkoxy-flavone derivatives,some novel compounds of this type and their preparation
IT1205337B (it) Derivati amminometil-benzenici eteroaril-sostituiti ad attivita' regolatrice del ritmo cardiaco e composizioni farmaceutiche che li contengono
SE7714558L (sv) Forening med desinficerande, aktivitet och farmaceutiska kompositioner innehallande denna
DE3062893D1 (en) Fluorinated methyl beta-alanine derivatives, their preparation and pharmaceutical compositions containing them
IT8049163A0 (it) Fenossiammine eterocicliche sostituite procedimento per prepararle e composizioni farmaceutiche che le contengono
IT7850986A0 (it) 5-imminodaunomicina e suoi derivati procedimento per prepararla nonche'composizioni farmaceutiche che la contengono
IT1129933B (it) Derivati tioetilammidici loro composizioni farmaceutiche e procedimento per la loro preparazione
HU177942B (en) Insecticide compositions containing substituted phenyl-carbamoy-2-pyrazoline derivatives and process for preparing the active substances
IL56797A (en) 1-imidazolinyl alkyl urea and amide derivatives,their preparation and pharmaceutical composition containing them
IT1194793B (it) Derivati tiazolidinici ad attivita' farmacologica,procedimento per la loro preparazione e composizioni farmaceutiche contenenti detti derivati
IT1132991B (it) Derivati di prostagliandina e prostaciclina ad attivita'farmacologica
FI803704A7 (fi) Heterosyklinen yhdiste ja sen synteesi, sitä sisältävät farmaseuttiset koostumukset ja yhdisteiden ja koostumukoostumusten käyttö lääketieteessä.
IL60813A0 (en) Heterocyclic compounds, their preparation and pharmaceutical compositions containing them
IT1093504B (it) Procedimento per la preparazione di derivati di cefalosporina,e composti cosi' preparati
IT1120537B (it) Perfezionate composizioni contenenti etomidate dotate di attivita' anestetica e procedimento di preparazione
IT8024152A0 (it) Derivati dell'1,1,2-trifenilpropano e dell'1,1,2-trifenilpropene, procedimento per la loro preparazione e composizioni farmaceutiche contenenti i composti
FI803483L (fi) Makrolidantibiotika foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska kompositioner
BE883215A (fr) Tetrahydro-pyrrolo-(1,2-a) pyrimidines substituees en position 3, leur preparation et compositions pharmaceutique contenant ces composes