IT7950555A0 - Derivati adenosinici e procedimento per la loro preparazione - Google Patents

Derivati adenosinici e procedimento per la loro preparazione

Info

Publication number
IT7950555A0
IT7950555A0 IT7950555A IT5055579A IT7950555A0 IT 7950555 A0 IT7950555 A0 IT 7950555A0 IT 7950555 A IT7950555 A IT 7950555A IT 5055579 A IT5055579 A IT 5055579A IT 7950555 A0 IT7950555 A0 IT 7950555A0
Authority
IT
Italy
Prior art keywords
procedure
preparation
adenosine derivatives
adenosine
derivatives
Prior art date
Application number
IT7950555A
Other languages
English (en)
Other versions
IT1164735B (it
Inventor
Gerald Wolberg
Thomas Paul Zimmerman
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of IT7950555A0 publication Critical patent/IT7950555A0/it
Application granted granted Critical
Publication of IT1164735B publication Critical patent/IT1164735B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/052Imidazole radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
IT50555/79A 1978-10-13 1979-10-12 Derivati adenosinici e procedimento per la loro preparazione IT1164735B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7840447 1978-10-13

Publications (2)

Publication Number Publication Date
IT7950555A0 true IT7950555A0 (it) 1979-10-12
IT1164735B IT1164735B (it) 1987-04-15

Family

ID=10500310

Family Applications (1)

Application Number Title Priority Date Filing Date
IT50555/79A IT1164735B (it) 1978-10-13 1979-10-12 Derivati adenosinici e procedimento per la loro preparazione

Country Status (6)

Country Link
US (1) US4309419A (it)
EP (1) EP0010668B1 (it)
JP (1) JPS5555199A (it)
DE (1) DE2967570D1 (it)
DK (1) DK431879A (it)
IT (1) IT1164735B (it)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0038569B1 (en) * 1980-04-23 1985-01-30 The Wellcome Foundation Limited Deazapurine nucleosides, formulations and preparation thereof
GB2074858B (en) * 1980-04-23 1985-03-20 Wellcome Found Compositions containing 3-deazaaden-osine
US4481197A (en) * 1980-04-25 1984-11-06 Burroughs Wellcome Co. Anti-inflammatory deoxyribosides
US4322411A (en) * 1980-04-25 1982-03-30 Burroughs Wellcome Co. Anti-inflammatory nucleosides
US4388308A (en) * 1980-06-09 1983-06-14 G.D. Searle & Co. N6 -[(2-Hydroxypropyl)aryl]adenosines
US4680285A (en) * 1980-12-15 1987-07-14 Viratek, Inc. Treatment of malignant tumors with 2-(β-D-ribofuranosylthiazole-4-carboxamide related compounds
US4386093A (en) * 1981-09-16 1983-05-31 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services (±)3-Deazaaristeromycin and uses
US4780452A (en) * 1986-09-08 1988-10-25 Burroughs Wellcome Co. F-substituted-3-β-D-ribofuranosyl-3H-imidazo[4,5-b]pyridines and pharmaceutical compositions thereof
US4931431A (en) * 1986-09-15 1990-06-05 Livingston William S Arthritis treatment with hypoxanthine
US4853373A (en) * 1986-09-15 1989-08-01 Livingston William S Therapeutic treatment for arthritic condition
US4918060A (en) * 1987-09-04 1990-04-17 The Johns Hopkins University Method of treating myasthenia gravis and related diseases
US4880784A (en) * 1987-12-21 1989-11-14 Brigham Young University Antiviral methods utilizing ribofuranosylthiazolo[4,5-d]pyrimdine derivatives
US5308837A (en) * 1990-08-22 1994-05-03 Merrell Dow Pharmaceuticals Inc. 5'-amine substituted adenosine analogs as immunosuppressants
US5137876A (en) * 1990-10-12 1992-08-11 Merck & Co., Inc. Nucleoside antiviral and anti-inflammatory compounds and compositions and methods for using same
US5747474A (en) * 1996-07-29 1998-05-05 Immune Modulation, Inc. Immunosuppression by administration of N6,N6 -disubstituted cAMP's, analogues thereof, and related nucleosides
ES2270614T3 (es) 1998-09-03 2007-04-01 Kerckhoff-Klinik Gesellschaft Mit Beschrankter Haftung 3-desazaadenosina utilizada en la prevencion de la ateroesclerosis y la vasculopatia de los injertos.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3919193A (en) * 1973-07-06 1975-11-11 Icn Pharmaceuticals 3-Deazaguanosine and derivatives thereof
US4148888A (en) * 1978-03-13 1979-04-10 The United States Of America As Represented By The Department Of Health, Education And Welfare 3-Deazaadenosine as an inhibitor of adenosylhomocysteine hydrolase with antiviral activity

Also Published As

Publication number Publication date
US4309419A (en) 1982-01-05
EP0010668A1 (en) 1980-05-14
IT1164735B (it) 1987-04-15
JPS5555199A (en) 1980-04-22
DE2967570D1 (en) 1986-03-06
JPH0134970B2 (it) 1989-07-21
EP0010668B1 (en) 1986-01-22
DK431879A (da) 1980-04-14

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