IT1254134B - Oligonucleotidi antisenso chimicamente modificati. - Google Patents

Oligonucleotidi antisenso chimicamente modificati.

Info

Publication number
IT1254134B
IT1254134B ITRM920025A ITRM920025A IT1254134B IT 1254134 B IT1254134 B IT 1254134B IT RM920025 A ITRM920025 A IT RM920025A IT RM920025 A ITRM920025 A IT RM920025A IT 1254134 B IT1254134 B IT 1254134B
Authority
IT
Italy
Prior art keywords
chemically modified
antisense oligonucleotides
modified antisense
residues
hydrogen
Prior art date
Application number
ITRM920025A
Other languages
English (en)
Inventor
Adolfo Iribarren
Original Assignee
Angeletti P Ist Richerche Bio
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Angeletti P Ist Richerche Bio filed Critical Angeletti P Ist Richerche Bio
Priority to ITRM920025A priority Critical patent/IT1254134B/it
Publication of ITRM920025A0 publication Critical patent/ITRM920025A0/it
Publication of ITRM920025A1 publication Critical patent/ITRM920025A1/it
Application granted granted Critical
Publication of IT1254134B publication Critical patent/IT1254134B/it

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Abstract

Oligonucleotidi antisenso chimicamente modificati, caratterizzati dal fatto di avere la seguente formula generale (1): (FORMULA I) in cui n è un numero intero da 0 a 200;R1-5 rappresenta una serie di sostituenti, per conferire alla sostituzione una struttura simmetrica nel suo insieme, scelti indipendentemente l'uno dall'altro dal gruppo comprendente idrogeno, eteroatomi, residui con eteroatomi, e residui idrocarbile;R rappresenta idrogeno, sostituenti con eteroatomi oppure residui idrocarbile; e B rappresenta un residuo eterociclico a uno o più anelli, e caratterizzati dal fatto che nella loro molecola sono presenti gruppi fosfato non-ionici e non-chirali.
ITRM920025A 1992-01-16 1992-01-16 Oligonucleotidi antisenso chimicamente modificati. IT1254134B (it)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ITRM920025A IT1254134B (it) 1992-01-16 1992-01-16 Oligonucleotidi antisenso chimicamente modificati.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITRM920025A IT1254134B (it) 1992-01-16 1992-01-16 Oligonucleotidi antisenso chimicamente modificati.

Publications (3)

Publication Number Publication Date
ITRM920025A0 ITRM920025A0 (it) 1992-01-16
ITRM920025A1 ITRM920025A1 (it) 1993-07-16
IT1254134B true IT1254134B (it) 1995-09-08

Family

ID=11400569

Family Applications (1)

Application Number Title Priority Date Filing Date
ITRM920025A IT1254134B (it) 1992-01-16 1992-01-16 Oligonucleotidi antisenso chimicamente modificati.

Country Status (1)

Country Link
IT (1) IT1254134B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL293592A (en) 2019-12-06 2022-08-01 Vertex Pharma Transduced tetrahydrofurans as sodium channel modulators
AU2022284886A1 (en) 2021-06-04 2023-11-30 Vertex Pharmaceuticals Incorporated N-(hydroxyalkyl (hetero)aryl) tetrahydrofuran carboxamides as modulators of sodium channels

Also Published As

Publication number Publication date
ITRM920025A1 (it) 1993-07-16
ITRM920025A0 (it) 1992-01-16

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Effective date: 19950126