IT1216783B - 8 ALFA ACILAMMINOERGOLINE, THEIR PREPARATION AND THEIR USE AS MEDICATIONS - Google Patents

8 ALFA ACILAMMINOERGOLINE, THEIR PREPARATION AND THEIR USE AS MEDICATIONS

Info

Publication number
IT1216783B
IT1216783B IT8747551A IT4755187A IT1216783B IT 1216783 B IT1216783 B IT 1216783B IT 8747551 A IT8747551 A IT 8747551A IT 4755187 A IT4755187 A IT 4755187A IT 1216783 B IT1216783 B IT 1216783B
Authority
IT
Italy
Prior art keywords
acilamminoergoline
alfa
medications
preparation
alfa acilamminoergoline
Prior art date
Application number
IT8747551A
Other languages
Italian (it)
Other versions
IT8747551A0 (en
Inventor
Ziegler Rene
Baumann Peter
Haefliger Walter
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IT8747551A0 publication Critical patent/IT8747551A0/en
Application granted granted Critical
Publication of IT1216783B publication Critical patent/IT1216783B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/10Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
    • C07D457/12Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
IT8747551A 1986-01-24 1987-01-22 8 ALFA ACILAMMINOERGOLINE, THEIR PREPARATION AND THEIR USE AS MEDICATIONS IT1216783B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3602058 1986-01-24

Publications (2)

Publication Number Publication Date
IT8747551A0 IT8747551A0 (en) 1987-01-22
IT1216783B true IT1216783B (en) 1990-03-14

Family

ID=6292510

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8747551A IT1216783B (en) 1986-01-24 1987-01-22 8 ALFA ACILAMMINOERGOLINE, THEIR PREPARATION AND THEIR USE AS MEDICATIONS

Country Status (18)

Country Link
JP (1) JPS62190184A (en)
KR (1) KR870007175A (en)
AU (1) AU6791487A (en)
BE (1) BE1000039A4 (en)
DK (1) DK35787A (en)
ES (1) ES2003774A6 (en)
FI (1) FI870293A (en)
FR (1) FR2595699A1 (en)
GB (1) GB2185743A (en)
GR (1) GR870093B (en)
HU (1) HUT45248A (en)
IL (1) IL81355A0 (en)
IT (1) IT1216783B (en)
LU (1) LU86743A1 (en)
NL (1) NL8700046A (en)
PT (1) PT84184A (en)
SE (1) SE8700250L (en)
ZA (1) ZA87520B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8714767D0 (en) * 1987-06-24 1987-07-29 Erba Farmitalia Egoline derivatives
DE3587860D1 (en) * 1984-04-09 1994-07-28 Schering Ag 2-Substituted ergoline derivatives, process for their preparation and their use as medicines.
DK338789A (en) * 1988-07-15 1990-01-16 Schering Ag 2-SUBSTITUTED ERGOLINYLURINE DERIVATIVES AND PROCEDURES FOR THE PRODUCTION THEREOF, THEIR USE AS MEDICINES AND INTERMEDIATES FOR THE PRODUCTION THEREOF
DE3915950A1 (en) * 1989-05-12 1990-11-15 Schering Ag 8 (ALPHA) ACYLAMINO ERGOLINE, THEIR PRODUCTION AND USE AS A MEDICINAL PRODUCT
CN103827113A (en) * 2011-06-23 2014-05-28 Map药物公司 Novel fluoroergoline analogs
CA2859173A1 (en) * 2011-12-19 2013-06-27 Map Pharmaceuticals, Inc. Novel iso-ergoline derivatives
US9657020B2 (en) 2015-01-20 2017-05-23 Xoc Pharmaceuticals, Inc. Ergoline compounds and uses thereof
BR112017015510A2 (en) * 2015-01-20 2018-01-30 Xoc Pharmaceuticals Inc compound of formula (i), method of treatment and / or prevention, d2 receptor agonizing method in one individual, d3 receptor antagonizing method in one individual, 5-ht1d receptor agonizing method in one individual, 5-ht1a receptor agonization in one individual, selective 5-ht1d receptor agonizing method instead of 5-ht1b receptor in one individual, 5-ht2c re-receptor selective agonizing method instead of 5-ht2a or 5 receptor -ht2b in one individual, method of 5-ht2c receptor agonization in one individual, method of providing functional antagonist activity at 5-ht2b receptor or 5-ht7 receptor, and, method of providing functional antagonist activity at adrenergic receptors in one individual
WO2018223065A1 (en) 2017-06-01 2018-12-06 Xoc Pharmaceuticals, Inc. Ergoline derivatives for use in medicine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1517971A (en) * 1974-07-19 1978-07-19 Sandoz Ltd 8alpha-substituted ergoline i derivatives
CH615929A5 (en) * 1975-06-02 1980-02-29 Sandoz Ag Process for the preparation of novel ergoline compounds
NL193541C (en) * 1984-01-12 2000-01-04 Novartis Ag Alpha-acylaminoergolines, methods for their preparation, and preparations containing them.

Also Published As

Publication number Publication date
LU86743A1 (en) 1987-09-03
PT84184A (en) 1987-02-01
GR870093B (en) 1987-05-25
AU6791487A (en) 1987-07-30
FR2595699A1 (en) 1987-09-18
JPS62190184A (en) 1987-08-20
DK35787D0 (en) 1987-01-22
HUT45248A (en) 1988-06-28
SE8700250D0 (en) 1987-01-22
NL8700046A (en) 1987-08-17
ZA87520B (en) 1988-09-28
DK35787A (en) 1987-07-25
GB2185743A (en) 1987-07-29
BE1000039A4 (en) 1987-12-15
GB8701274D0 (en) 1987-02-25
IL81355A0 (en) 1987-08-31
ES2003774A6 (en) 1988-11-16
IT8747551A0 (en) 1987-01-22
KR870007175A (en) 1987-08-17
FI870293A0 (en) 1987-01-23
FI870293A (en) 1987-07-25
SE8700250L (en) 1987-07-25

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