IT1216783B - 8 ALFA ACILAMMINOERGOLINE, THEIR PREPARATION AND THEIR USE AS MEDICATIONS - Google Patents
8 ALFA ACILAMMINOERGOLINE, THEIR PREPARATION AND THEIR USE AS MEDICATIONSInfo
- Publication number
- IT1216783B IT1216783B IT8747551A IT4755187A IT1216783B IT 1216783 B IT1216783 B IT 1216783B IT 8747551 A IT8747551 A IT 8747551A IT 4755187 A IT4755187 A IT 4755187A IT 1216783 B IT1216783 B IT 1216783B
- Authority
- IT
- Italy
- Prior art keywords
- acilamminoergoline
- alfa
- medications
- preparation
- alfa acilamminoergoline
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
- C07D457/10—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
- C07D457/12—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3602058 | 1986-01-24 |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8747551A0 IT8747551A0 (en) | 1987-01-22 |
IT1216783B true IT1216783B (en) | 1990-03-14 |
Family
ID=6292510
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT8747551A IT1216783B (en) | 1986-01-24 | 1987-01-22 | 8 ALFA ACILAMMINOERGOLINE, THEIR PREPARATION AND THEIR USE AS MEDICATIONS |
Country Status (18)
Country | Link |
---|---|
JP (1) | JPS62190184A (en) |
KR (1) | KR870007175A (en) |
AU (1) | AU6791487A (en) |
BE (1) | BE1000039A4 (en) |
DK (1) | DK35787A (en) |
ES (1) | ES2003774A6 (en) |
FI (1) | FI870293A (en) |
FR (1) | FR2595699A1 (en) |
GB (1) | GB2185743A (en) |
GR (1) | GR870093B (en) |
HU (1) | HUT45248A (en) |
IL (1) | IL81355A0 (en) |
IT (1) | IT1216783B (en) |
LU (1) | LU86743A1 (en) |
NL (1) | NL8700046A (en) |
PT (1) | PT84184A (en) |
SE (1) | SE8700250L (en) |
ZA (1) | ZA87520B (en) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8714767D0 (en) * | 1987-06-24 | 1987-07-29 | Erba Farmitalia | Egoline derivatives |
DE3587860D1 (en) * | 1984-04-09 | 1994-07-28 | Schering Ag | 2-Substituted ergoline derivatives, process for their preparation and their use as medicines. |
DK338789A (en) * | 1988-07-15 | 1990-01-16 | Schering Ag | 2-SUBSTITUTED ERGOLINYLURINE DERIVATIVES AND PROCEDURES FOR THE PRODUCTION THEREOF, THEIR USE AS MEDICINES AND INTERMEDIATES FOR THE PRODUCTION THEREOF |
DE3915950A1 (en) * | 1989-05-12 | 1990-11-15 | Schering Ag | 8 (ALPHA) ACYLAMINO ERGOLINE, THEIR PRODUCTION AND USE AS A MEDICINAL PRODUCT |
CN103827113A (en) * | 2011-06-23 | 2014-05-28 | Map药物公司 | Novel fluoroergoline analogs |
CA2859173A1 (en) * | 2011-12-19 | 2013-06-27 | Map Pharmaceuticals, Inc. | Novel iso-ergoline derivatives |
US9657020B2 (en) | 2015-01-20 | 2017-05-23 | Xoc Pharmaceuticals, Inc. | Ergoline compounds and uses thereof |
BR112017015510A2 (en) * | 2015-01-20 | 2018-01-30 | Xoc Pharmaceuticals Inc | compound of formula (i), method of treatment and / or prevention, d2 receptor agonizing method in one individual, d3 receptor antagonizing method in one individual, 5-ht1d receptor agonizing method in one individual, 5-ht1a receptor agonization in one individual, selective 5-ht1d receptor agonizing method instead of 5-ht1b receptor in one individual, 5-ht2c re-receptor selective agonizing method instead of 5-ht2a or 5 receptor -ht2b in one individual, method of 5-ht2c receptor agonization in one individual, method of providing functional antagonist activity at 5-ht2b receptor or 5-ht7 receptor, and, method of providing functional antagonist activity at adrenergic receptors in one individual |
WO2018223065A1 (en) | 2017-06-01 | 2018-12-06 | Xoc Pharmaceuticals, Inc. | Ergoline derivatives for use in medicine |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1517971A (en) * | 1974-07-19 | 1978-07-19 | Sandoz Ltd | 8alpha-substituted ergoline i derivatives |
CH615929A5 (en) * | 1975-06-02 | 1980-02-29 | Sandoz Ag | Process for the preparation of novel ergoline compounds |
NL193541C (en) * | 1984-01-12 | 2000-01-04 | Novartis Ag | Alpha-acylaminoergolines, methods for their preparation, and preparations containing them. |
-
1987
- 1987-01-12 HU HU8792A patent/HUT45248A/en unknown
- 1987-01-12 NL NL8700046A patent/NL8700046A/en not_active Application Discontinuation
- 1987-01-21 GB GB08701274A patent/GB2185743A/en not_active Withdrawn
- 1987-01-22 PT PT84184A patent/PT84184A/en unknown
- 1987-01-22 DK DK035787A patent/DK35787A/en not_active Application Discontinuation
- 1987-01-22 IL IL81355A patent/IL81355A0/en unknown
- 1987-01-22 AU AU67914/87A patent/AU6791487A/en not_active Abandoned
- 1987-01-22 SE SE8700250A patent/SE8700250L/en not_active Application Discontinuation
- 1987-01-22 FR FR8700834A patent/FR2595699A1/en active Pending
- 1987-01-22 GR GR870093A patent/GR870093B/en unknown
- 1987-01-22 IT IT8747551A patent/IT1216783B/en active
- 1987-01-22 ES ES8700163A patent/ES2003774A6/en not_active Expired
- 1987-01-22 LU LU86743A patent/LU86743A1/en unknown
- 1987-01-22 KR KR870000556A patent/KR870007175A/en not_active Application Discontinuation
- 1987-01-23 JP JP62015028A patent/JPS62190184A/en active Pending
- 1987-01-23 FI FI870293A patent/FI870293A/en not_active IP Right Cessation
- 1987-01-23 BE BE8700046A patent/BE1000039A4/en not_active IP Right Cessation
- 1987-01-23 ZA ZA87520A patent/ZA87520B/en unknown
Also Published As
Publication number | Publication date |
---|---|
LU86743A1 (en) | 1987-09-03 |
PT84184A (en) | 1987-02-01 |
GR870093B (en) | 1987-05-25 |
AU6791487A (en) | 1987-07-30 |
FR2595699A1 (en) | 1987-09-18 |
JPS62190184A (en) | 1987-08-20 |
DK35787D0 (en) | 1987-01-22 |
HUT45248A (en) | 1988-06-28 |
SE8700250D0 (en) | 1987-01-22 |
NL8700046A (en) | 1987-08-17 |
ZA87520B (en) | 1988-09-28 |
DK35787A (en) | 1987-07-25 |
GB2185743A (en) | 1987-07-29 |
BE1000039A4 (en) | 1987-12-15 |
GB8701274D0 (en) | 1987-02-25 |
IL81355A0 (en) | 1987-08-31 |
ES2003774A6 (en) | 1988-11-16 |
IT8747551A0 (en) | 1987-01-22 |
KR870007175A (en) | 1987-08-17 |
FI870293A0 (en) | 1987-01-23 |
FI870293A (en) | 1987-07-25 |
SE8700250L (en) | 1987-07-25 |
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