IT1157211B - Preparati a base di n/6-acilderivati di 3'-deossi-adenosina e loro impiego come intensificatori di effetto antitumorale - Google Patents
Preparati a base di n/6-acilderivati di 3'-deossi-adenosina e loro impiego come intensificatori di effetto antitumoraleInfo
- Publication number
- IT1157211B IT1157211B IT48651/82A IT4865182A IT1157211B IT 1157211 B IT1157211 B IT 1157211B IT 48651/82 A IT48651/82 A IT 48651/82A IT 4865182 A IT4865182 A IT 4865182A IT 1157211 B IT1157211 B IT 1157211B
- Authority
- IT
- Italy
- Prior art keywords
- intensifiers
- deoxy
- adenosine
- acyl derivatives
- preparations based
- Prior art date
Links
- 230000000259 anti-tumor effect Effects 0.000 title 1
- OFEZSBMBBKLLBJ-BAJZRUMYSA-N cordycepin Chemical class C1=NC=2C(N)=NC=NC=2N1[C@@H]1O[C@H](CO)C[C@H]1O OFEZSBMBBKLLBJ-BAJZRUMYSA-N 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP56094676A JPS57209225A (en) | 1981-06-18 | 1981-06-18 | Antitumor activity intensifier |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT8248651A0 IT8248651A0 (it) | 1982-06-16 |
| IT1157211B true IT1157211B (it) | 1987-02-11 |
Family
ID=14116819
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT48651/82A IT1157211B (it) | 1981-06-18 | 1982-06-16 | Preparati a base di n/6-acilderivati di 3'-deossi-adenosina e loro impiego come intensificatori di effetto antitumorale |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP0068268B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JPS57209225A (cg-RX-API-DMAC7.html) |
| AU (1) | AU552409B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA1164346A (cg-RX-API-DMAC7.html) |
| DE (1) | DE3263372D1 (cg-RX-API-DMAC7.html) |
| IT (1) | IT1157211B (cg-RX-API-DMAC7.html) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5679648A (en) * | 1994-11-30 | 1997-10-21 | The University Hospital | Methods for the treatment and prevention of fungal infections by administration of 3'-deoxypurine nucleosides |
| US6174873B1 (en) * | 1998-11-04 | 2001-01-16 | Supergen, Inc. | Oral administration of adenosine analogs |
| CN101574362B (zh) * | 2009-06-03 | 2012-05-23 | 西南大学 | N-烷酰基虫草素在制备治疗肿瘤疾病的药物中的应用 |
| CN103254195B (zh) * | 2013-03-26 | 2016-08-03 | 内蒙古医科大学 | 7-氨基-四氮唑[1,5-a]并嘧啶-5-醇(化合物II)及其合成路线 |
| CN113413385A (zh) * | 2014-02-07 | 2021-09-21 | 纽罗克里生物科学有限公司 | 包含抗精神病药物和vmat2抑制剂的药物组合物及其用途 |
| HRP20240304T1 (hr) | 2015-10-30 | 2024-05-10 | Neurocrine Biosciences, Inc. | Soli valbenazin dihidroklorida i njihovi polimorfi |
| LT3394057T (lt) | 2015-12-23 | 2022-06-27 | Neurocrine Biosciences, Inc. | Sintezės būdas, skirtas pagaminti (s)-(2r,3r,11br)-3-izobutil-9,10-dimetoksi-2,3,4,6,7,11b-heksahidro-1h-pirido[2,1-a]izochinolin-2-ilo 2-amino-3-metilbutanoato di(4-metilbenzensulfonatą) |
| KR20190108146A (ko) | 2017-01-27 | 2019-09-23 | 뉴로크린 바이오사이언시즈 인코퍼레이티드 | 특정 vmat2 억제제의 투여 방법 |
| IL309802A (en) | 2017-09-21 | 2024-02-01 | Neurocrine Biosciences Inc | High dose valbenazine formulation and related preparations, methods and kits |
| KR20250070134A (ko) | 2017-10-10 | 2025-05-20 | 뉴로크린 바이오사이언시즈 인코퍼레이티드 | 특정 vmat2 억제제의 투여 방법 |
| JP2021502959A (ja) | 2017-10-10 | 2021-02-04 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | 特定のvmat2インヒビターを投与するための方法 |
| JOP20200336A1 (ar) | 2018-08-15 | 2020-12-22 | Neurocrine Biosciences Inc | طرق إعطاء مثبطات vmat2 معينة |
| US10940141B1 (en) | 2019-08-23 | 2021-03-09 | Neurocrine Biosciences, Inc. | Methods for the administration of certain VMAT2 inhibitors |
| CN113563401A (zh) * | 2021-07-14 | 2021-10-29 | 河南牧业经济学院 | 一种新型虫草素烷酰胺衍生物及其制备方法和应用 |
-
1981
- 1981-06-18 JP JP56094676A patent/JPS57209225A/ja active Granted
-
1982
- 1982-06-14 DE DE8282105194T patent/DE3263372D1/de not_active Expired
- 1982-06-14 EP EP82105194A patent/EP0068268B1/en not_active Expired
- 1982-06-16 IT IT48651/82A patent/IT1157211B/it active
- 1982-06-18 AU AU85007/82A patent/AU552409B2/en not_active Ceased
- 1982-06-18 CA CA000405511A patent/CA1164346A/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| CA1164346A (en) | 1984-03-27 |
| JPS57209225A (en) | 1982-12-22 |
| AU8500782A (en) | 1982-12-23 |
| EP0068268B1 (en) | 1985-05-02 |
| DE3263372D1 (en) | 1985-06-05 |
| AU552409B2 (en) | 1986-05-29 |
| JPS637164B2 (cg-RX-API-DMAC7.html) | 1988-02-15 |
| IT8248651A0 (it) | 1982-06-16 |
| EP0068268A1 (en) | 1983-01-05 |
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