IT1149073B - Derivati di 4-piridilpiridazinone dotati di attivita' antiinfiammatoria ed analgesica - Google Patents

Derivati di 4-piridilpiridazinone dotati di attivita' antiinfiammatoria ed analgesica

Info

Publication number
IT1149073B
IT1149073B IT49095/82A IT4909582A IT1149073B IT 1149073 B IT1149073 B IT 1149073B IT 49095/82 A IT49095/82 A IT 49095/82A IT 4909582 A IT4909582 A IT 4909582A IT 1149073 B IT1149073 B IT 1149073B
Authority
IT
Italy
Prior art keywords
pyridylpyridazinone
inflammatory
analgesic activity
derivatives
derivatives equipped
Prior art date
Application number
IT49095/82A
Other languages
English (en)
Other versions
IT8249095A0 (it
Inventor
Larry J Powers
Original Assignee
Diamond Shamrock Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Diamond Shamrock Corp filed Critical Diamond Shamrock Corp
Publication of IT8249095A0 publication Critical patent/IT8249095A0/it
Application granted granted Critical
Publication of IT1149073B publication Critical patent/IT1149073B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT49095/82A 1981-09-11 1982-09-09 Derivati di 4-piridilpiridazinone dotati di attivita' antiinfiammatoria ed analgesica IT1149073B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30132881A 1981-09-11 1981-09-11

Publications (2)

Publication Number Publication Date
IT8249095A0 IT8249095A0 (it) 1982-09-09
IT1149073B true IT1149073B (it) 1986-12-03

Family

ID=23162890

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49095/82A IT1149073B (it) 1981-09-11 1982-09-09 Derivati di 4-piridilpiridazinone dotati di attivita' antiinfiammatoria ed analgesica

Country Status (5)

Country Link
EP (1) EP0088128A4 (it)
JP (1) JPS58501432A (it)
IL (1) IL66761A0 (it)
IT (1) IT1149073B (it)
WO (1) WO1983000863A1 (it)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5622948A (en) * 1994-12-01 1997-04-22 Syntex (U.S.A.) Inc. Pyrrole pyridazine and pyridazinone anti-inflammatory agents
ATE271547T1 (de) * 1997-03-14 2004-08-15 Merck Frosst Canada Inc Pyridazinone als inhibitoren von cyclooxygenase-2
US6004960A (en) * 1997-03-14 1999-12-21 Merck Frosst Canada, Inc. Pyridazinones as inhibitors of cyclooxygenase-2
EP2017266A1 (en) * 1997-11-19 2009-01-21 Kowa Co., Ltd. Pyridazine derivatives and medicines containing the same as effective ingredients

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB840522A (en) * 1957-11-05 1960-07-06 Lepetit Spa A new analgesic 2-hydroxymethyl-6-phenyl-3-pyridazone
US3920646A (en) * 1967-11-02 1975-11-18 Sandoz Ag 3-Substituted-1-pyridyl-1,4,5,6-tetrahydropyridazines
US3658814A (en) * 1970-03-17 1972-04-25 Sandoz Ag 2-(omega-chloroalkyl)-6-aryl substituted-4 5-dihydropyridazin(2h)-3-one
CH557819A (de) * 1970-11-12 1975-01-15 Sandoz Ag Verfahren zur herstellung von neuen 2-(2-hydroxyalkyl)4,5-dihydro-pyridazin(2h)-3-onen.
AT333774B (de) * 1974-09-24 1976-12-10 Chemie Linz Ag Verfahren zur herstellung von 3-phenylpyridazonen
JPS5419987A (en) * 1977-07-15 1979-02-15 Yoshitomi Pharmaceut Ind Ltd Pyridazinone derivative and its preparation
DE2834624A1 (de) * 1978-08-08 1980-02-28 Bayer Ag Neue 1,4-dihydropyridazin-3-carbonsaeurederivate, verfahren zu ihrer herstellung und verwendung als arzneimittel
US4238490A (en) * 1979-02-12 1980-12-09 Diamond Shamrock Corporation Antihypertensive pyridazin(2H)-3-ones
US4298609A (en) * 1979-08-30 1981-11-03 Sterling Drug Inc. 4,5-Dihydro-6-(4-pyridinyl)-3-pyridazinol and salts, their preparation and use as blood pressure lowering agents

Also Published As

Publication number Publication date
EP0088128A4 (en) 1984-04-06
EP0088128A1 (en) 1983-09-14
JPS58501432A (ja) 1983-08-25
IT8249095A0 (it) 1982-09-09
WO1983000863A1 (en) 1983-03-17
IL66761A0 (en) 1982-12-31

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