IT1107551B - PENTAPEPTIDES USEFUL AS MEDICATIONS IN HUMAN AND VETERINARY MEDICINE AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM COEM ACTIVE INGREDIENT - Google Patents

PENTAPEPTIDES USEFUL AS MEDICATIONS IN HUMAN AND VETERINARY MEDICINE AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM COEM ACTIVE INGREDIENT

Info

Publication number
IT1107551B
IT1107551B IT50431/78A IT5043178A IT1107551B IT 1107551 B IT1107551 B IT 1107551B IT 50431/78 A IT50431/78 A IT 50431/78A IT 5043178 A IT5043178 A IT 5043178A IT 1107551 B IT1107551 B IT 1107551B
Authority
IT
Italy
Prior art keywords
coem
medications
human
contain
active ingredient
Prior art date
Application number
IT50431/78A
Other languages
Italian (it)
Other versions
IT7850431A0 (en
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB30909/77A external-priority patent/GB1604644A/en
Priority claimed from GB48980/77A external-priority patent/GB1604850A/en
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of IT7850431A0 publication Critical patent/IT7850431A0/en
Application granted granted Critical
Publication of IT1107551B publication Critical patent/IT1107551B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/675Beta-endorphins
    • C07K14/6755Beta-endorphins with at least 1 amino acid in D-form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/70Enkephalins
    • C07K14/702Enkephalins with at least 1 amino acid in D-form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biophysics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Pulmonology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
IT50431/78A 1977-07-22 1978-07-21 PENTAPEPTIDES USEFUL AS MEDICATIONS IN HUMAN AND VETERINARY MEDICINE AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM COEM ACTIVE INGREDIENT IT1107551B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB30909/77A GB1604644A (en) 1977-07-22 1977-07-22 Biologically active pentapeptide amides
GB48980/77A GB1604850A (en) 1977-11-24 1977-11-24 Biologically active peptides

Publications (2)

Publication Number Publication Date
IT7850431A0 IT7850431A0 (en) 1978-07-21
IT1107551B true IT1107551B (en) 1985-11-25

Family

ID=26260658

Family Applications (1)

Application Number Title Priority Date Filing Date
IT50431/78A IT1107551B (en) 1977-07-22 1978-07-21 PENTAPEPTIDES USEFUL AS MEDICATIONS IN HUMAN AND VETERINARY MEDICINE AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM COEM ACTIVE INGREDIENT

Country Status (4)

Country Link
EP (1) EP0000559B1 (en)
JP (1) JPS5424850A (en)
DE (1) DE2862327D1 (en)
IT (1) IT1107551B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU178001B (en) * 1976-09-16 1982-02-28 Gyogyszekutato Intezet Process for preparing new pentapeptides with morphine-like activity and derivatives thereof
FR2424253A1 (en) * 1978-04-27 1979-11-23 Brun Lab Sa Le NEW DERIVATIVES OF PEPTIDES ANALOGUES OF ENKEPHALINS, THEIR METHOD OF PREPARATION AND THEIR THERAPEUTIC APPLICATION
NL8005121A (en) * 1979-09-20 1981-03-24 Erba Farmitalia ORGANICALLY ACTIVE PEPTIDES.
BR8208035A (en) * 1981-12-28 1983-11-22 Beckman Instruments Inc SYNTHETIC PEPTIDEOS HAVING HORMONE RELEASE ACTIVITY FROM PITUITARY GROWTH
EP0085963B1 (en) * 1982-02-05 1987-01-21 The Wellcome Foundation Limited Pharmaceutical compounds, preparation, use and intermediates therefor and their preparation

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL51332A (en) * 1976-01-26 1980-09-16 Wellcome Found Peptides having a morphine-like effect, their preparation and pharmalceutical compositions containing them
NZ183712A (en) * 1976-04-08 1979-10-25 Ici Ltd Polypeptide analogues of enkephalins, and pharmaceutical compositions
FR2359817A1 (en) * 1976-07-27 1978-02-24 Reckitt & Colmann Prod Ltd Peptide cpds. contg. tyrosine, glycine, phenylalanine and d-amino acid - local anaesthetics, smooth muscle relaxants, adrenergic neutron blockers, beta-stimulants etc.
HU178001B (en) * 1976-09-16 1982-02-28 Gyogyszekutato Intezet Process for preparing new pentapeptides with morphine-like activity and derivatives thereof
US4259234A (en) * 1976-09-27 1981-03-31 Eli Lilly And Company Analgesic compounds

Also Published As

Publication number Publication date
EP0000559A1 (en) 1979-02-07
DE2862327D1 (en) 1983-11-10
JPS5424850A (en) 1979-02-24
IT7850431A0 (en) 1978-07-21
EP0000559B1 (en) 1983-10-05

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