IT1097762B - Procedimento per la n-protezione selettiva di amminoglicos idi e prodotti intermedi amminoglicosidi selettivamente protetti cosi' ottenuti - Google Patents
Procedimento per la n-protezione selettiva di amminoglicos idi e prodotti intermedi amminoglicosidi selettivamente protetti cosi' ottenutiInfo
- Publication number
- IT1097762B IT1097762B IT26293/78A IT2629378A IT1097762B IT 1097762 B IT1097762 B IT 1097762B IT 26293/78 A IT26293/78 A IT 26293/78A IT 2629378 A IT2629378 A IT 2629378A IT 1097762 B IT1097762 B IT 1097762B
- Authority
- IT
- Italy
- Prior art keywords
- amminoglicosides
- amminoglicos
- ides
- selective
- procedure
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/822,118 US4282350A (en) | 1977-08-05 | 1977-08-05 | Selective 3"-N-acylation of 1,3"-di-N-unprotected-poly-N-protected-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols |
Publications (2)
Publication Number | Publication Date |
---|---|
IT7826293A0 IT7826293A0 (it) | 1978-07-28 |
IT1097762B true IT1097762B (it) | 1985-08-31 |
Family
ID=25235190
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT26293/78A IT1097762B (it) | 1977-08-05 | 1978-07-28 | Procedimento per la n-protezione selettiva di amminoglicos idi e prodotti intermedi amminoglicosidi selettivamente protetti cosi' ottenuti |
Country Status (10)
Country | Link |
---|---|
US (1) | US4282350A (it) |
EP (1) | EP0000800B1 (it) |
JP (1) | JPS5430134A (it) |
DE (1) | DE2860297D1 (it) |
DK (1) | DK341078A (it) |
FI (1) | FI782369A (it) |
GR (1) | GR72425B (it) |
HU (1) | HU180095B (it) |
IT (1) | IT1097762B (it) |
PT (1) | PT68372A (it) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2840907A1 (de) * | 1978-09-20 | 1980-04-03 | Bayer Ag | Selektiv geschuetzte 4,6-di-o-(aminoglykosyl)-1,3-diaminocyclitole |
JPS6383351U (it) * | 1986-11-20 | 1988-06-01 | ||
JPS63225393A (ja) * | 1988-02-09 | 1988-09-20 | Microbial Chem Res Found | 1位以外のアミノ基が選択的に保護されたアミノグリコシド抗生物質保護誘導体 |
JPH027892U (it) * | 1989-06-14 | 1990-01-18 | ||
TWI425947B (zh) | 2007-11-21 | 2014-02-11 | Achaogen Inc | 抗菌性胺基糖苷類似物 |
WO2010132757A2 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
WO2010132768A1 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial derivatives of sisomicin |
WO2010132760A1 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial derivatives of tobramycin |
WO2010132759A1 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial derivatives of dibekacin |
WO2010132765A2 (en) | 2009-05-15 | 2010-11-18 | Achaogen, Inc. | Antibacterial aminoglycoside analogs |
DE202013011690U1 (de) | 2013-04-05 | 2014-02-26 | Isabellenhütte Heusler Gmbh & Co. Kg | Messwiderstand |
CN106866756A (zh) * | 2017-01-10 | 2017-06-20 | 苏利制药科技江阴有限公司 | 一种合成1‑n‑乙基西索米星的方法 |
CN113960183A (zh) * | 2020-12-28 | 2022-01-21 | 常州方圆制药有限公司 | 依替米星中间体中乙酰化杂质的检测方法 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5644076B2 (it) * | 1973-07-12 | 1981-10-16 | ||
CH606076A5 (it) * | 1973-08-06 | 1978-10-13 | Scherico Ltd | |
US4063015A (en) * | 1973-08-27 | 1977-12-13 | Schering Corporation | Garamine and derivatives thereof |
JPS5512039B2 (it) * | 1974-03-22 | 1980-03-29 | ||
US4044123A (en) * | 1975-05-02 | 1977-08-23 | Schering Corporation | 6'-N-alkyl-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols, methods for their use as antibacterial agents and compositions useful therefor |
US4066752A (en) * | 1976-06-21 | 1978-01-03 | Schering Corporation | 1-Desamino-1-hydroxy and 1-desamino-1-epi-hydroxy-4,6-di-o-(aminoglycosyl)-1,3-diaminocyclitols; 1-desamino-1-oxo-4,6-di-o-(aminoglycosyl)-1,3-diaminocyclitols, intermediates and use as antibacterial agents |
DE2712160A1 (de) * | 1977-03-19 | 1978-09-28 | Bayer Ag | Pseudotrisaccharide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
-
1977
- 1977-08-05 US US05/822,118 patent/US4282350A/en not_active Expired - Lifetime
-
1978
- 1978-07-28 IT IT26293/78A patent/IT1097762B/it active
- 1978-07-31 EP EP78200121A patent/EP0000800B1/en not_active Expired
- 1978-07-31 DE DE7878200121T patent/DE2860297D1/de not_active Expired
- 1978-08-01 JP JP9408178A patent/JPS5430134A/ja active Pending
- 1978-08-01 DK DK341078A patent/DK341078A/da not_active Application Discontinuation
- 1978-08-01 GR GR56905A patent/GR72425B/el unknown
- 1978-08-01 FI FI782369A patent/FI782369A/fi not_active Application Discontinuation
- 1978-08-01 PT PT68372A patent/PT68372A/pt unknown
- 1978-08-04 HU HU78SCHE655A patent/HU180095B/hu unknown
Also Published As
Publication number | Publication date |
---|---|
US4282350A (en) | 1981-08-04 |
EP0000800A1 (en) | 1979-02-21 |
IT7826293A0 (it) | 1978-07-28 |
DK341078A (da) | 1979-02-06 |
EP0000800B1 (en) | 1980-12-10 |
GR72425B (it) | 1983-11-04 |
HU180095B (en) | 1983-01-28 |
DE2860297D1 (en) | 1981-02-19 |
PT68372A (en) | 1978-09-01 |
FI782369A (fi) | 1979-02-06 |
JPS5430134A (en) | 1979-03-06 |
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