IT1096690B - Diammino-benzil-pirimidine solubili - Google Patents

Diammino-benzil-pirimidine solubili

Info

Publication number
IT1096690B
IT1096690B IT25569/78A IT2556978A IT1096690B IT 1096690 B IT1096690 B IT 1096690B IT 25569/78 A IT25569/78 A IT 25569/78A IT 2556978 A IT2556978 A IT 2556978A IT 1096690 B IT1096690 B IT 1096690B
Authority
IT
Italy
Prior art keywords
pyrimidine
benzyl
soluble diamine
diamine
soluble
Prior art date
Application number
IT25569/78A
Other languages
English (en)
Italian (it)
Other versions
IT7825569A0 (it
Original Assignee
Dick Pierre R G
Rombi Max Andre
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dick Pierre R G, Rombi Max Andre filed Critical Dick Pierre R G
Publication of IT7825569A0 publication Critical patent/IT7825569A0/it
Application granted granted Critical
Publication of IT1096690B publication Critical patent/IT1096690B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02Heterocyclic radicals containing only nitrogen as ring hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IT25569/78A 1977-07-11 1978-07-11 Diammino-benzil-pirimidine solubili IT1096690B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7722323A FR2397407A2 (fr) 1977-07-11 1977-07-11 Derives de 2,4-diamino pyrimidines et leur mise en solution en association avec des sulfamides

Publications (2)

Publication Number Publication Date
IT7825569A0 IT7825569A0 (it) 1978-07-11
IT1096690B true IT1096690B (it) 1985-08-26

Family

ID=9193583

Family Applications (1)

Application Number Title Priority Date Filing Date
IT25569/78A IT1096690B (it) 1977-07-11 1978-07-11 Diammino-benzil-pirimidine solubili

Country Status (13)

Country Link
US (1) US4232023A (https=)
JP (1) JPS5448776A (https=)
AT (1) AT362381B (https=)
AU (1) AU3793378A (https=)
BE (1) BE868893A (https=)
DE (1) DE2829820A1 (https=)
FR (1) FR2397407A2 (https=)
GB (1) GB2001965B (https=)
IE (1) IE47232B1 (https=)
IT (1) IT1096690B (https=)
LU (1) LU79949A1 (https=)
NL (1) NL7807440A (https=)
ZA (1) ZA783957B (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2502152A1 (fr) * 1981-03-20 1982-09-24 Panmedica Laboratoires Nouveaux derives solubles n2 substitues de la diamino-2,4-benzyl-5-pyrimidines, leur procede de preparation et medicaments les contenant
US6583148B1 (en) 1999-04-08 2003-06-24 Krenitsky Pharmaceuticals, Inc. Neurotrophic substituted pyrimidines
JP5154728B2 (ja) 2000-07-24 2013-02-27 クレニツキー・ファーマシューティカルズ,インコーポレイテッド 神経栄養活性を有する置換5−アルキニルピリミジン
CA2557372C (en) * 2004-03-05 2013-01-08 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 antagonists
MX2008002731A (es) * 2005-09-01 2008-03-26 Hoffmann La Roche Diaminopirimidinas como moduladores de p2x3 y p3x2/3.
ES2562056T3 (es) * 2005-09-01 2016-03-02 F. Hoffmann-La Roche Ag Diaminopirimidinas como moduladores P2X3 y P2X2/3
EP1924564B1 (en) * 2005-09-01 2016-11-09 F.Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
EP3546452A1 (en) * 2007-10-08 2019-10-02 MMV Medicines for Malaria Venture Antimalarial compounds with flexible side-chains
WO2012121682A2 (en) * 2011-03-10 2012-09-13 National Science And Technology Development Agency Anti-folate antimalarials with dual-binding modes and their preparation

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2287071A (en) * 1938-08-08 1942-06-23 Parke Davis & Co Organic amine derivatives and method of obtaining same
US2374791A (en) * 1942-06-22 1945-05-01 Parke Davis & Co Organic amine derivatives and method of obtaining same
US3111521A (en) * 1962-04-25 1963-11-19 Parke Davis & Co 2-aryl-nu-(polyamino-5-pyrimidinyl)-glycinonitriles
GB1375162A (https=) * 1970-10-22 1974-11-27
BE791627A (fr) * 1971-11-20 1973-05-21 Knapsack Ag Procede pour l'oxydation du monoxyde de carbone et des hydrocarbures

Also Published As

Publication number Publication date
GB2001965A (en) 1979-02-14
FR2397407A2 (fr) 1979-02-09
IE47232B1 (en) 1984-01-25
ATA496978A (de) 1980-10-15
LU79949A1 (fr) 1979-04-09
ZA783957B (en) 1979-09-26
AU3793378A (en) 1980-01-17
US4232023A (en) 1980-11-04
NL7807440A (nl) 1979-01-15
FR2397407B2 (https=) 1980-01-04
BE868893A (fr) 1979-01-11
AT362381B (de) 1981-05-11
JPS5448776A (en) 1979-04-17
IT7825569A0 (it) 1978-07-11
GB2001965B (en) 1982-03-10
DE2829820A1 (de) 1979-02-01
IE781377L (en) 1979-01-11

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