IT1096690B - Diammino-benzil-pirimidine solubili - Google Patents

Diammino-benzil-pirimidine solubili

Info

Publication number
IT1096690B
IT1096690B IT25569/78A IT2556978A IT1096690B IT 1096690 B IT1096690 B IT 1096690B IT 25569/78 A IT25569/78 A IT 25569/78A IT 2556978 A IT2556978 A IT 2556978A IT 1096690 B IT1096690 B IT 1096690B
Authority
IT
Italy
Prior art keywords
pyrimidine
benzyl
soluble diamine
diamine
soluble
Prior art date
Application number
IT25569/78A
Other languages
English (en)
Italian (it)
Other versions
IT7825569A0 (it
Original Assignee
Dick Pierre R G
Rombi Max Andre
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dick Pierre R G, Rombi Max Andre filed Critical Dick Pierre R G
Publication of IT7825569A0 publication Critical patent/IT7825569A0/it
Application granted granted Critical
Publication of IT1096690B publication Critical patent/IT1096690B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02Heterocyclic radicals containing only nitrogen as ring hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IT25569/78A 1977-07-11 1978-07-11 Diammino-benzil-pirimidine solubili IT1096690B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7722323A FR2397407A2 (fr) 1977-07-11 1977-07-11 Derives de 2,4-diamino pyrimidines et leur mise en solution en association avec des sulfamides

Publications (2)

Publication Number Publication Date
IT7825569A0 IT7825569A0 (it) 1978-07-11
IT1096690B true IT1096690B (it) 1985-08-26

Family

ID=9193583

Family Applications (1)

Application Number Title Priority Date Filing Date
IT25569/78A IT1096690B (it) 1977-07-11 1978-07-11 Diammino-benzil-pirimidine solubili

Country Status (13)

Country Link
US (1) US4232023A (OSRAM)
JP (1) JPS5448776A (OSRAM)
AT (1) AT362381B (OSRAM)
AU (1) AU3793378A (OSRAM)
BE (1) BE868893A (OSRAM)
DE (1) DE2829820A1 (OSRAM)
FR (1) FR2397407A2 (OSRAM)
GB (1) GB2001965B (OSRAM)
IE (1) IE47232B1 (OSRAM)
IT (1) IT1096690B (OSRAM)
LU (1) LU79949A1 (OSRAM)
NL (1) NL7807440A (OSRAM)
ZA (1) ZA783957B (OSRAM)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2502152A1 (fr) * 1981-03-20 1982-09-24 Panmedica Laboratoires Nouveaux derives solubles n2 substitues de la diamino-2,4-benzyl-5-pyrimidines, leur procede de preparation et medicaments les contenant
US6583148B1 (en) 1999-04-08 2003-06-24 Krenitsky Pharmaceuticals, Inc. Neurotrophic substituted pyrimidines
JP5154728B2 (ja) 2000-07-24 2013-02-27 クレニツキー・ファーマシューティカルズ,インコーポレイテッド 神経栄養活性を有する置換5−アルキニルピリミジン
CA2557372C (en) * 2004-03-05 2013-01-08 F. Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 antagonists
MX2008002731A (es) * 2005-09-01 2008-03-26 Hoffmann La Roche Diaminopirimidinas como moduladores de p2x3 y p3x2/3.
ES2562056T3 (es) * 2005-09-01 2016-03-02 F. Hoffmann-La Roche Ag Diaminopirimidinas como moduladores P2X3 y P2X2/3
EP1924564B1 (en) * 2005-09-01 2016-11-09 F.Hoffmann-La Roche Ag Diaminopyrimidines as p2x3 and p2x2/3 modulators
EP3546452A1 (en) * 2007-10-08 2019-10-02 MMV Medicines for Malaria Venture Antimalarial compounds with flexible side-chains
WO2012121682A2 (en) * 2011-03-10 2012-09-13 National Science And Technology Development Agency Anti-folate antimalarials with dual-binding modes and their preparation

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2287071A (en) * 1938-08-08 1942-06-23 Parke Davis & Co Organic amine derivatives and method of obtaining same
US2374791A (en) * 1942-06-22 1945-05-01 Parke Davis & Co Organic amine derivatives and method of obtaining same
US3111521A (en) * 1962-04-25 1963-11-19 Parke Davis & Co 2-aryl-nu-(polyamino-5-pyrimidinyl)-glycinonitriles
GB1375162A (OSRAM) * 1970-10-22 1974-11-27
BE791627A (fr) * 1971-11-20 1973-05-21 Knapsack Ag Procede pour l'oxydation du monoxyde de carbone et des hydrocarbures

Also Published As

Publication number Publication date
GB2001965A (en) 1979-02-14
FR2397407A2 (fr) 1979-02-09
IE47232B1 (en) 1984-01-25
ATA496978A (de) 1980-10-15
LU79949A1 (fr) 1979-04-09
ZA783957B (en) 1979-09-26
AU3793378A (en) 1980-01-17
US4232023A (en) 1980-11-04
NL7807440A (nl) 1979-01-15
FR2397407B2 (OSRAM) 1980-01-04
BE868893A (fr) 1979-01-11
AT362381B (de) 1981-05-11
JPS5448776A (en) 1979-04-17
IT7825569A0 (it) 1978-07-11
GB2001965B (en) 1982-03-10
DE2829820A1 (de) 1979-02-01
IE781377L (en) 1979-01-11

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