IN2014MU00197A - - Google Patents

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Publication number
IN2014MU00197A
IN2014MU00197A IN197MU2014A IN2014MU00197A IN 2014MU00197 A IN2014MU00197 A IN 2014MU00197A IN 197MU2014 A IN197MU2014 A IN 197MU2014A IN 2014MU00197 A IN2014MU00197 A IN 2014MU00197A
Authority
IN
India
Prior art keywords
preparation
apixaban
intermediate formula
discloses
present
Prior art date
Application number
Other languages
English (en)
Inventor
Sharadchandra Pradhan Nitin
Ulhas Sonavane Sachin
Ghangadhar Patil Dayaghan
Sakharam Pujari Uttam
Bhausaheb Pagire Ravindra
Original Assignee
Wanbury Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wanbury Ltd filed Critical Wanbury Ltd
Priority to PCT/IN2015/000007 priority Critical patent/WO2015111073A2/en
Priority to US15/113,430 priority patent/US20170008886A1/en
Priority to EP15723309.9A priority patent/EP3097100A2/en
Priority to IN197MU2014 priority patent/IN2014MU00197A/en
Publication of IN2014MU00197A publication Critical patent/IN2014MU00197A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
IN197MU2014 2014-01-21 2015-01-06 IN2014MU00197A (zh)

Priority Applications (4)

Application Number Priority Date Filing Date Title
PCT/IN2015/000007 WO2015111073A2 (en) 2014-01-21 2015-01-06 A process for the preparation of apixaban and its intermediates
US15/113,430 US20170008886A1 (en) 2014-01-21 2015-01-06 A process for the preparation of apixaban and its intermediates
EP15723309.9A EP3097100A2 (en) 2014-01-21 2015-01-06 A process for the preparation of apixaban and its intermediates
IN197MU2014 IN2014MU00197A (zh) 2014-01-21 2015-01-06

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN197MU2014 IN2014MU00197A (zh) 2014-01-21 2015-01-06

Publications (1)

Publication Number Publication Date
IN2014MU00197A true IN2014MU00197A (zh) 2015-08-28

Family

ID=53189106

Family Applications (1)

Application Number Title Priority Date Filing Date
IN197MU2014 IN2014MU00197A (zh) 2014-01-21 2015-01-06

Country Status (4)

Country Link
US (1) US20170008886A1 (zh)
EP (1) EP3097100A2 (zh)
IN (1) IN2014MU00197A (zh)
WO (1) WO2015111073A2 (zh)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113504317A (zh) * 2021-06-22 2021-10-15 哈尔滨珍宝制药有限公司 阿哌沙班中基因毒性杂质的检测方法和应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI331526B (en) 2001-09-21 2010-10-11 Bristol Myers Squibb Pharma Co Lactam-containing compounds and derivatives thereof as factor xa inhibitors
TW200738672A (en) 2001-12-10 2007-10-16 Bristol Myers Squibb Co Intermediated for the preparation of 4,5-dihydro-pyrazolo [3,4-c] pyrid-2-ones
US20100130543A1 (en) 2008-09-15 2010-05-27 Auspex Pharmaceuticals, Inc. Pyrazole carboxamide inhibitors of factor xa
TW201039822A (en) * 2009-02-06 2010-11-16 Taisho Pharmaceutical Co Ltd Dihydroquinolinone derivatives
JP2014516072A (ja) 2011-06-10 2014-07-07 ディフアルマ フランチス ソシエタ ア レスポンサビリタ リミタータ アピキサバン製造方法
CZ304846B6 (cs) * 2012-11-13 2014-12-03 Zentiva, K.S. Způsob přípravy APIXABANU
US9718779B2 (en) * 2013-01-09 2017-08-01 Msn Laboratories Limited Intermediate and polymorphs of 1-(4-methoxypheny1)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetra hydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide and process thereof

Also Published As

Publication number Publication date
EP3097100A2 (en) 2016-11-30
US20170008886A1 (en) 2017-01-12
WO2015111073A2 (en) 2015-07-30
WO2015111073A3 (en) 2015-11-12

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