IN2014MN02127A - - Google Patents
Info
- Publication number
- IN2014MN02127A IN2014MN02127A IN2127MUN2014A IN2014MN02127A IN 2014MN02127 A IN2014MN02127 A IN 2014MN02127A IN 2127MUN2014 A IN2127MUN2014 A IN 2127MUN2014A IN 2014MN02127 A IN2014MN02127 A IN 2014MN02127A
- Authority
- IN
- India
- Prior art keywords
- compounds
- calcium
- crac
- channel
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN2127MUN2014 IN2014MN02127A (fr) | 2012-05-02 | 2013-05-01 |
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN6KO2012 | 2012-05-02 | ||
IN1474KO2012 | 2012-12-28 | ||
PCT/IB2013/053446 WO2013164773A1 (fr) | 2012-05-02 | 2013-05-01 | Composés substitués de pyrazole en tant que modulateurs de crac |
IN2127MUN2014 IN2014MN02127A (fr) | 2012-05-02 | 2013-05-01 |
Publications (1)
Publication Number | Publication Date |
---|---|
IN2014MN02127A true IN2014MN02127A (fr) | 2015-09-11 |
Family
ID=48428566
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IN2127MUN2014 IN2014MN02127A (fr) | 2012-05-02 | 2013-05-01 |
Country Status (7)
Country | Link |
---|---|
US (2) | US9409898B2 (fr) |
EP (1) | EP2844656A1 (fr) |
AU (1) | AU2013255441B2 (fr) |
CA (1) | CA2871222A1 (fr) |
IN (1) | IN2014MN02127A (fr) |
WO (1) | WO2013164773A1 (fr) |
ZA (1) | ZA201407668B (fr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2015197187A1 (fr) * | 2014-06-24 | 2015-12-30 | Grünenthal GmbH | Carboxamides à base de pyrazolyle v |
WO2015197188A1 (fr) * | 2014-06-24 | 2015-12-30 | Grünenthal GmbH | Carboxamides à base de pyrazolyle utilisables comme inhibiteurs de crac |
US20180161388A1 (en) | 2015-05-18 | 2018-06-14 | Beth Israel Deaconess Medical Center, Inc. | Substance p, mast cell degranulation inhibitors, and peripheral neuropathy |
CA3112907A1 (fr) | 2018-09-14 | 2020-03-19 | Rhizen Pharmaceuticals Ag | Compositions comprenant un inhibiteur de crac et un corticosteroide ainsi que leurs methodes d'utilisation |
CA3121202A1 (fr) | 2018-11-30 | 2020-06-04 | Nuvation Bio Inc. | Composes pyrrole et pyrazole et leurs procedes d'utilisation |
BR112021021028A2 (pt) | 2019-06-06 | 2021-12-14 | Basf Se | Uso dos compostos de fórmula i, compostos da fórmula i, composição e método para combater fungos fitopatogênicos |
CN110604735B (zh) * | 2019-09-18 | 2022-10-25 | 华东师范大学 | 一种治疗肝纤维化、硬皮病的化合物及其应用 |
WO2021063735A1 (fr) | 2019-10-02 | 2021-04-08 | Basf Se | Nouveaux dérivés pyridines bicycliques |
Family Cites Families (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU751139B2 (en) * | 1997-10-13 | 2002-08-08 | Astellas Pharma Inc. | Amide derivative |
CA2327185A1 (fr) * | 1998-04-08 | 1999-10-14 | Abbott Laboratories | Inhibiteurs de type pyrazole de la production de cytokine |
WO1999062885A1 (fr) * | 1998-06-05 | 1999-12-09 | Boehringer Ingelheim Pharmaceuticals, Inc. | 1-(4-aminophenyl) pyrazoles substitues et leur utilisation en tant qu'agents anti-inflammatoires |
EP1653968A4 (fr) | 2003-07-23 | 2006-09-06 | Synta Pharmaceuticals Corp | Procede de modulation de canaux d'ions calcium actives par la liberation d'ions calcium |
EP1809294A4 (fr) | 2004-09-21 | 2008-08-06 | Synta Pharmaceuticals Corp | Composes pour l'inflammation et applications associees aux troubles immuns |
WO2006083477A2 (fr) | 2005-01-07 | 2006-08-10 | Synta Pharmaceuticals Corp. | Composes utilises pour des etats inflammatoires et immunitaires |
JP5221147B2 (ja) | 2005-01-25 | 2013-06-26 | シンタ ファーマシューティカルズ コーポレーション | 炎症及び免疫に関連する用途に用いる化合物 |
BRPI0607308A2 (pt) | 2005-01-25 | 2009-08-25 | Synta Pharmaceuticals Corp | compostos, composições farmacêuticas e usos dos referidos compostos |
JP5430943B2 (ja) | 2006-01-25 | 2014-03-05 | シンタ ファーマシューティカルズ コーポレーション | 炎症及び免疫関連用途のための置換芳香族化合物 |
CA2639913A1 (fr) | 2006-01-25 | 2007-08-02 | Synta Pharmaceutical Corp. | Composes a base de phenyle et de pyridyle pour des utilisations liees aux inflammations ou aux troubles immunitaires |
CA2639927A1 (fr) | 2006-01-25 | 2007-08-02 | Synta Pharmaceuticals Corp. | Composes biaryle substitues destines a des utilisations contre des inflammations et des troubles immunitaires |
JP5430944B2 (ja) | 2006-01-31 | 2014-03-05 | シンタ ファーマシューティカルズ コーポレーション | 炎症および免疫関連用途のためのピリジルフェニル化合物 |
CA2695148A1 (fr) | 2007-08-01 | 2009-02-05 | Synta Pharmaceuticals Corp. | Composes pyridine utilises pour des etats inflammatoires et des troubles immunitaires |
RU2465272C2 (ru) | 2007-09-10 | 2012-10-27 | КалсиМедика, Инк. | Соединения, моделирующие внутриклеточный кальций |
WO2009076454A2 (fr) | 2007-12-12 | 2009-06-18 | Calcimedica, Inc. | Compositions qui modulant le calcium intracellulaire |
AU2009288245B2 (en) | 2008-08-27 | 2012-12-20 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
US8524763B2 (en) | 2008-09-22 | 2013-09-03 | Calcimedica, Inc. | Inhibitors of store operated calcium release |
EP2350006A1 (fr) | 2008-10-01 | 2011-08-03 | Synta Pharmaceuticals Corp. | Composés pour des utilisations liées à une inflammation et au système immunitaire |
EP2477982A4 (fr) | 2009-09-16 | 2013-04-03 | Calcimedica Inc | Composés qui modulent le calcium intracellulaire |
US8377970B2 (en) * | 2009-10-08 | 2013-02-19 | Rhizen Pharmaceuticals Sa | Modulators of calcium release-activated calcium channel |
WO2012022487A1 (fr) | 2010-08-20 | 2012-02-23 | Grünenthal GmbH | Dérivés de carboxamide et d'urée cycliques substitués en tant que ligands du récepteur vanilloïde |
JP5387541B2 (ja) | 2010-10-29 | 2014-01-15 | 住友電装株式会社 | グロメット |
SI2632906T1 (sl) | 2010-10-30 | 2016-08-31 | Lupin Limited | Derivati oksazolina in izooksazolina kot crac modulatorji |
AR083817A1 (es) | 2010-11-10 | 2013-03-27 | Gruenenthal Gmbh | Derivados de carboxamida y urea heteroaromaticos sustituidos como ligandos del receptor vanilloide |
US9604978B2 (en) | 2011-05-03 | 2017-03-28 | Synta Pharmaceuticals Corp. | Compounds for inflammation and immune-related uses |
EP2768810A1 (fr) | 2011-10-19 | 2014-08-27 | Calcimedica, Inc. | Composés qui modulent le calcium intracellulaire |
US9856240B2 (en) | 2011-10-19 | 2018-01-02 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
-
2013
- 2013-05-01 EP EP13722112.3A patent/EP2844656A1/fr not_active Withdrawn
- 2013-05-01 IN IN2127MUN2014 patent/IN2014MN02127A/en unknown
- 2013-05-01 WO PCT/IB2013/053446 patent/WO2013164773A1/fr active Application Filing
- 2013-05-01 US US14/398,161 patent/US9409898B2/en not_active Expired - Fee Related
- 2013-05-01 CA CA 2871222 patent/CA2871222A1/fr not_active Abandoned
- 2013-05-01 AU AU2013255441A patent/AU2013255441B2/en not_active Expired - Fee Related
-
2014
- 2014-10-22 ZA ZA2014/07668A patent/ZA201407668B/en unknown
-
2016
- 2016-06-28 US US15/194,795 patent/US20160304507A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US9409898B2 (en) | 2016-08-09 |
EP2844656A1 (fr) | 2015-03-11 |
AU2013255441B2 (en) | 2017-11-09 |
CA2871222A1 (fr) | 2013-11-07 |
ZA201407668B (en) | 2015-11-25 |
US20150111925A1 (en) | 2015-04-23 |
US20160304507A1 (en) | 2016-10-20 |
AU2013255441A1 (en) | 2014-11-13 |
WO2013164773A1 (fr) | 2013-11-07 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IN2014MN02126A (fr) | ||
IN2014MN02127A (fr) | ||
CO6430427A2 (es) | Derivados de benzofuranilo | |
TN2013000348A1 (en) | Compounds and compositions as trk inhibitors | |
PH12015500551A1 (en) | Tricyclic quinoline and quinoline derivatives | |
GEP20166438B (en) | Imidazopyrrolidinone compounds | |
PH12014502757B1 (en) | Dihydronaphthyridines and related compounds useful as kinase inhibitors for the treatment of proliferative diseases | |
CR20110103A (es) | Heteroarilos sustituidos | |
IN2014CN04907A (fr) | ||
MX2015012478A (es) | Metodos y composiciones para inhibicion de proteinas que contienen bromodominio. | |
MD20140109A2 (ro) | Compuşi ai indolului şi indazolului care activează AMPK | |
IN2012DN00943A (fr) | ||
WO2012170931A3 (fr) | Composés qui modulent le calcium intracellulaire | |
MX337711B (es) | Compuestos que modulan el calcio intracelular. | |
EA201200570A1 (ru) | Соединения и композиции в качестве модуляторов активности gpr119 | |
MY162689A (en) | Oxazoline and isoxazoline derivatives as crac modulators | |
TN2013000346A1 (en) | Asymmetric ureas and medical uses thereof | |
EA026940B9 (ru) | Замещенные хромановые соединения в качестве модуляторов чувствительного к кальцию рецептора | |
WO2012170951A3 (fr) | Composés modulant le calcium intracellulaire | |
TW201613878A (en) | Pyrazine GPR40 agonists for the treatment of type II diabetes | |
AU2011322715A8 (en) | Treatment of MeCP2-associated disorders | |
UY36081A (es) | Compuestos inhibidores de metaloenzima como fungicidas. | |
PH12014501979B1 (en) | Fused bicyclic 2,4-diaminopyrimidine derivative as a dual alk and fak inhibitor | |
IN2015MN00421A (fr) | ||
MX357828B (es) | Composición con factores de crecimiento destinada al tratamiento intranasal de una enfermedad neurodegenerativa u otra patología del sistema nervioso central, y su método de fabricación. |