IN2014CN02315A - - Google Patents

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Publication number
IN2014CN02315A
IN2014CN02315A IN2315CHN2014A IN2014CN02315A IN 2014CN02315 A IN2014CN02315 A IN 2014CN02315A IN 2315CHN2014 A IN2315CHN2014 A IN 2315CHN2014A IN 2014CN02315 A IN2014CN02315 A IN 2014CN02315A
Authority
IN
India
Prior art keywords
proliferation
formula
carcinoma cells
mucoepidermoid carcinoma
imidazoquinolines
Prior art date
Application number
Other languages
English (en)
Inventor
James D Griffin
Lizi Wu
Jie Chen
Original Assignee
Dana Farber Cancer Inst Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dana Farber Cancer Inst Inc filed Critical Dana Farber Cancer Inst Inc
Publication of IN2014CN02315A publication Critical patent/IN2014CN02315A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7088Compounds having three or more nucleosides or nucleotides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IN2315CHN2014 2011-09-30 2012-09-27 IN2014CN02315A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161541758P 2011-09-30 2011-09-30
US201261660377P 2012-06-15 2012-06-15
PCT/US2012/057480 WO2013049300A1 (fr) 2011-09-30 2012-09-27 Procédé de traitement du carcinome mucoépidermoïde

Publications (1)

Publication Number Publication Date
IN2014CN02315A true IN2014CN02315A (fr) 2015-06-19

Family

ID=47016842

Family Applications (1)

Application Number Title Priority Date Filing Date
IN2315CHN2014 IN2014CN02315A (fr) 2011-09-30 2012-09-27

Country Status (12)

Country Link
US (1) US20140243396A1 (fr)
EP (1) EP2760445A1 (fr)
JP (1) JP2014532057A (fr)
KR (1) KR20140069038A (fr)
CN (1) CN103906515A (fr)
AU (1) AU2012316020A1 (fr)
BR (1) BR112014005730A2 (fr)
CA (1) CA2848065A1 (fr)
EA (1) EA201490725A1 (fr)
IN (1) IN2014CN02315A (fr)
MX (1) MX2014003873A (fr)
WO (1) WO2013049300A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016185443A1 (fr) 2015-05-20 2016-11-24 Novartis Ag Combinaison pharmaceutique d'évérolimus et de dactolisib
AU2017363970A1 (en) 2016-11-23 2019-06-20 Novartis Ag Methods of enhancing immune response with everolimus, dactolisib or both
US20200362303A1 (en) * 2017-11-30 2020-11-19 Kyoto University Maintenance-and-amplification method and differentiation induction method for primordial germ cells/primordial germ cell-like cells
WO2019157516A1 (fr) 2018-02-12 2019-08-15 resTORbio, Inc. Polythérapies

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2604629A1 (fr) 2005-04-11 2006-10-19 The Trustees Of Columbia University In The City Of New York Methodes permettant de traiter les troubles cognitifs moderes
GB0510390D0 (en) 2005-05-20 2005-06-29 Novartis Ag Organic compounds
CN101541793A (zh) * 2006-11-20 2009-09-23 诺瓦提斯公司 2-甲基-2-[4-(3-甲基-2-氧代-8-喹啉-3-基-2,3-二氢-咪唑并[4,5-c]喹啉-1-基)-苯基]-丙腈的盐和晶型
WO2009052467A1 (fr) * 2007-10-19 2009-04-23 Board Of Regents Of The University Of Texas System Procédés d'identification d'une résistance à l'inhibiteur de pi-3 kinase
WO2009067397A2 (fr) * 2007-11-19 2009-05-28 Ore Pharmaceuticals Inc. Traitement de tumeurs solides
WO2009155659A1 (fr) * 2008-06-27 2009-12-30 The University Of Queensland Polythérapie
US8476431B2 (en) * 2008-11-03 2013-07-02 Itellikine LLC Benzoxazole kinase inhibitors and methods of use
WO2011133668A2 (fr) * 2010-04-20 2011-10-27 President And Fellows Of Harvard College Méthodes et compositions utilisées pour le traitement du cancer
WO2012068487A1 (fr) * 2010-11-18 2012-05-24 Synta Pharmaceuticals Corp. Présélection de patients pour un traitement thérapeutique fondé sur un état hypoxique, avec des agents sensibles à l'oxygène

Also Published As

Publication number Publication date
US20140243396A1 (en) 2014-08-28
BR112014005730A2 (pt) 2017-03-28
WO2013049300A1 (fr) 2013-04-04
CN103906515A (zh) 2014-07-02
KR20140069038A (ko) 2014-06-09
AU2012316020A1 (en) 2013-05-09
MX2014003873A (es) 2014-05-28
EA201490725A1 (ru) 2014-11-28
CA2848065A1 (fr) 2013-04-04
EP2760445A1 (fr) 2014-08-06
JP2014532057A (ja) 2014-12-04

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