IL88163A - Method for the preparation of anilopiperidine derivatives - Google Patents

Method for the preparation of anilopiperidine derivatives

Info

Publication number
IL88163A
IL88163A IL88163A IL8816388A IL88163A IL 88163 A IL88163 A IL 88163A IL 88163 A IL88163 A IL 88163A IL 8816388 A IL8816388 A IL 8816388A IL 88163 A IL88163 A IL 88163A
Authority
IL
Israel
Prior art keywords
anilopiperidine
derivatives
preparation
anilopiperidine derivatives
Prior art date
Application number
IL88163A
Other languages
English (en)
Other versions
IL88163A0 (en
Original Assignee
Boc Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boc Inc filed Critical Boc Inc
Publication of IL88163A0 publication Critical patent/IL88163A0/xx
Publication of IL88163A publication Critical patent/IL88163A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
IL88163A 1987-11-02 1988-10-25 Method for the preparation of anilopiperidine derivatives IL88163A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/115,276 US4849521A (en) 1987-11-02 1987-11-02 Stereoselective preparation of 3-substituted-4-piperidine compounds and derivatives

Publications (2)

Publication Number Publication Date
IL88163A0 IL88163A0 (en) 1989-06-30
IL88163A true IL88163A (en) 1993-01-31

Family

ID=22360323

Family Applications (1)

Application Number Title Priority Date Filing Date
IL88163A IL88163A (en) 1987-11-02 1988-10-25 Method for the preparation of anilopiperidine derivatives

Country Status (12)

Country Link
US (1) US4849521A (fi)
EP (1) EP0389551A1 (fi)
JP (1) JPH02504393A (fi)
CN (1) CN1033273A (fi)
AU (1) AU2802389A (fi)
DK (1) DK108190D0 (fi)
ES (1) ES2009100A6 (fi)
FI (1) FI902082A0 (fi)
GR (1) GR880100742A (fi)
IL (1) IL88163A (fi)
NZ (1) NZ226715A (fi)
WO (1) WO1989004300A1 (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5223540A (en) * 1987-10-22 1993-06-29 Massachusetts Institute Of Technology Method for treating the premenstrual or late luteal phase syndrome
US7361666B2 (en) 1999-05-25 2008-04-22 Sepracor, Inc. Heterocyclic analgesic compounds and methods of use thereof
US6677332B1 (en) 1999-05-25 2004-01-13 Sepracor, Inc. Heterocyclic analgesic compounds and methods of use thereof
US6635661B2 (en) 2000-05-25 2003-10-21 Sepracor Inc. Heterocyclic analgesic compounds and methods of use thereof
WO2005080394A1 (en) * 2004-02-24 2005-09-01 Bioaxone Therapeutique Inc. 4-substituted piperidine derivatives
US10106525B2 (en) 2015-01-26 2018-10-23 BioAxone BioSciences, Inc. Rho kinase inhibitor BA-1049 (R) and active metabolites thereof
US10149856B2 (en) 2015-01-26 2018-12-11 BioAxone BioSciences, Inc. Treatment of cerebral cavernous malformations and cerebral aneurysms with rho kinase inhibitors
US10857157B2 (en) 2015-01-26 2020-12-08 BioAxone BioSciences, Inc. Treatment of cerebral cavernous malformations and cerebral aneurysms with rho kinase inhibitors
US11198680B2 (en) 2016-12-21 2021-12-14 BioAxone BioSciences, Inc. Rho kinase inhibitor BA-1049 (R) and active metabolites thereof
WO2019014322A1 (en) * 2017-07-11 2019-01-17 BioAxone BioSciences, Inc. KINASE INHIBITORS FOR THE TREATMENT OF DISEASES

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE623427A (fi) * 1961-10-10
US3161637A (en) * 1961-10-10 1964-12-15 Res Lab Dr C Janssen N V 1-(gamma-aroyl-propyl)-4-(nu-arylcarbonyl amino) piperidines and related compounds
US3907813A (en) * 1973-09-11 1975-09-23 Janssen Pharmaceutica Nv Stereoisomeric forms of 4-anilino-3-methyl piperidines
US3907811A (en) * 1973-09-11 1975-09-23 Janssen Pharmaceutica Nv Stereoisomeric forms of 4-anilido-3-methyl-piperidine-1-carboxylates
US3998834A (en) * 1975-03-14 1976-12-21 Janssen Pharmaceutica N.V. N-(4-piperidinyl)-n-phenylamides and -carbamates
US4196210A (en) * 1975-09-23 1980-04-01 Janssen Pharmaceutica N.V. N-Aryl-N-(1-L-4-piperidinyl)-arylacetamides
US4496732A (en) * 1983-03-14 1985-01-29 Hoechst-Roussel Pharmaceuticals Inc. Stereoselective reduction of 2- or 3-substituted 4-piperidones with sodium borohydride
US4584303A (en) * 1984-04-09 1986-04-22 The Boc Group, Inc. N-aryl-N-(4-piperidinyl)amides and pharmaceutical compositions and method employing such compounds

Also Published As

Publication number Publication date
EP0389551A1 (en) 1990-10-03
WO1989004300A1 (en) 1989-05-18
NZ226715A (en) 1990-10-26
DK108190A (da) 1990-05-01
US4849521A (en) 1989-07-18
CN1033273A (zh) 1989-06-07
IL88163A0 (en) 1989-06-30
ES2009100A6 (es) 1989-08-16
GR880100742A (el) 1994-03-31
FI902082A0 (fi) 1990-04-25
AU2802389A (en) 1989-06-01
DK108190D0 (da) 1990-05-01
JPH02504393A (ja) 1990-12-13

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