IL78700A - (7-(3-acylamino)-phenyl)pyrazolo(1,5-a)-pyrimidines,their preparation and pharmaceutical compositions containing them - Google Patents

(7-(3-acylamino)-phenyl)pyrazolo(1,5-a)-pyrimidines,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL78700A
IL78700A IL78700A IL7870086A IL78700A IL 78700 A IL78700 A IL 78700A IL 78700 A IL78700 A IL 78700A IL 7870086 A IL7870086 A IL 7870086A IL 78700 A IL78700 A IL 78700A
Authority
IL
Israel
Prior art keywords
alkyl
pyrimidines
pyrazolo
acylamino
phenyl
Prior art date
Application number
IL78700A
Other versions
IL78700A0 (en
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/732,986 external-priority patent/US4626538A/en
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of IL78700A0 publication Critical patent/IL78700A0/en
Publication of IL78700A publication Critical patent/IL78700A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • G—PHYSICS
    • G11—INFORMATION STORAGE
    • G11B—INFORMATION STORAGE BASED ON RELATIVE MOVEMENT BETWEEN RECORD CARRIER AND TRANSDUCER
    • G11B5/00—Recording by magnetisation or demagnetisation of a record carrier; Reproducing by magnetic means; Record carriers therefor
    • G11B5/48—Disposition or mounting of heads or head supports relative to record carriers ; arrangements of heads, e.g. for scanning the record carrier to increase the relative speed
    • G11B5/58—Disposition or mounting of heads or head supports relative to record carriers ; arrangements of heads, e.g. for scanning the record carrier to increase the relative speed with provision for moving the head for the purpose of maintaining alignment of the head relative to the record carrier during transducing operation, e.g. to compensate for surface irregularities of the latter or for track following
    • G11B5/584—Disposition or mounting of heads or head supports relative to record carriers ; arrangements of heads, e.g. for scanning the record carrier to increase the relative speed with provision for moving the head for the purpose of maintaining alignment of the head relative to the record carrier during transducing operation, e.g. to compensate for surface irregularities of the latter or for track following for track following on tapes
    • G11B5/588—Disposition or mounting of heads or head supports relative to record carriers ; arrangements of heads, e.g. for scanning the record carrier to increase the relative speed with provision for moving the head for the purpose of maintaining alignment of the head relative to the record carrier during transducing operation, e.g. to compensate for surface irregularities of the latter or for track following for track following on tapes by controlling the position of the rotating heads
    • G—PHYSICS
    • G11—INFORMATION STORAGE
    • G11B—INFORMATION STORAGE BASED ON RELATIVE MOVEMENT BETWEEN RECORD CARRIER AND TRANSDUCER
    • G11B15/00—Driving, starting or stopping record carriers of filamentary or web form; Driving both such record carriers and heads; Guiding such record carriers or containers therefor; Control thereof; Control of operating function
    • G11B15/18—Driving; Starting; Stopping; Arrangements for control or regulation thereof
    • G11B15/1808—Driving of both record carrier and head
    • G11B15/1816—Programmed access in sequence to indexed parts of operating tapes cooperating with rotating heads
    • G—PHYSICS
    • G11—INFORMATION STORAGE
    • G11B—INFORMATION STORAGE BASED ON RELATIVE MOVEMENT BETWEEN RECORD CARRIER AND TRANSDUCER
    • G11B15/00—Driving, starting or stopping record carriers of filamentary or web form; Driving both such record carriers and heads; Guiding such record carriers or containers therefor; Control thereof; Control of operating function
    • G11B15/18—Driving; Starting; Stopping; Arrangements for control or regulation thereof
    • G11B15/1808—Driving of both record carrier and head
    • G11B15/1825—Driving of both record carrier and head driving or moving the head in a direction which cuts across the direction of travel of the tape, e.g. for helicoïdal scanning
    • G11B15/1833—Driving of both record carrier and head driving or moving the head in a direction which cuts across the direction of travel of the tape, e.g. for helicoïdal scanning with head driven in a plane, cyclically around an axis, e.g. on headwheel
    • G—PHYSICS
    • G11—INFORMATION STORAGE
    • G11B—INFORMATION STORAGE BASED ON RELATIVE MOVEMENT BETWEEN RECORD CARRIER AND TRANSDUCER
    • G11B15/00—Driving, starting or stopping record carriers of filamentary or web form; Driving both such record carriers and heads; Guiding such record carriers or containers therefor; Control thereof; Control of operating function
    • G11B15/18—Driving; Starting; Stopping; Arrangements for control or regulation thereof
    • G11B15/1808—Driving of both record carrier and head
    • G11B15/1875—Driving of both record carrier and head adaptations for special effects or editing
    • G—PHYSICS
    • G11—INFORMATION STORAGE
    • G11B—INFORMATION STORAGE BASED ON RELATIVE MOVEMENT BETWEEN RECORD CARRIER AND TRANSDUCER
    • G11B5/00—Recording by magnetisation or demagnetisation of a record carrier; Reproducing by magnetic means; Record carriers therefor
    • G11B5/008—Recording on, or reproducing or erasing from, magnetic tapes, sheets, e.g. cards, or wires
    • G11B5/00813—Recording on, or reproducing or erasing from, magnetic tapes, sheets, e.g. cards, or wires magnetic tapes
    • G11B5/00817—Recording on, or reproducing or erasing from, magnetic tapes, sheets, e.g. cards, or wires magnetic tapes on longitudinal tracks only, e.g. for serpentine format recording
    • G11B5/00839—Recording on, or reproducing or erasing from, magnetic tapes, sheets, e.g. cards, or wires magnetic tapes on longitudinal tracks only, e.g. for serpentine format recording using cyclically driven heads providing segmented tracks

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Signal Processing (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROCEDURE FOR PREPARING PYRAZOLE (1,5-A) PYRIMIDINES. IT INCLUDES: A) REACTING (II) WITH DIMETHYLFORMAMIDE DIMETHYLACETHOLE AT REFLUX, TO OBTAIN A (A); B) TREAT A (A) WITH SODIUM HYDRIDE IN DIMETHYLFORMAMIDE, TO GENERATE AN ANION; C) MAKE THE ANION REACT WITH FORMULA ALKYL HALIDE (R5X), TO GIVE A (III) AND D) TREAT (III) WITH (IV) IN GLACIAL ACETIC ACID AND REFLUX, TO OBTAIN A (I). BEING: (A), N- (3- (3-DIMETILAMINO) -1-OXO-2-PROPENIL) FENIL) ALCANAMIDA; R1, H, HAL OR CIANO; R2, H OR C 1 TO 4 ALKYL; R3, (V); R5, H, C 1A 6 ALKYL AND OTHERS; R6, ALKYL, C 1 TO 6, CYCLOALKYL FROM C 3 TO 6 AND OTHERS AND X, BR O I. ARE USED AS ANSIOLYTICS AND ANTISEPTICS. *FORMULA* (Machine-translation by Google Translate, not legally binding)
IL78700A 1985-05-13 1986-05-06 (7-(3-acylamino)-phenyl)pyrazolo(1,5-a)-pyrimidines,their preparation and pharmaceutical compositions containing them IL78700A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/732,986 US4626538A (en) 1983-06-23 1985-05-13 [7-(3-disubstituted amino)phenyl]pyrazolo[1,5-a]pyrimidines

Publications (2)

Publication Number Publication Date
IL78700A0 IL78700A0 (en) 1986-08-31
IL78700A true IL78700A (en) 1989-06-30

Family

ID=24945743

Family Applications (1)

Application Number Title Priority Date Filing Date
IL78700A IL78700A (en) 1985-05-13 1986-05-06 (7-(3-acylamino)-phenyl)pyrazolo(1,5-a)-pyrimidines,their preparation and pharmaceutical compositions containing them

Country Status (16)

Country Link
JP (1) JPH0784468B2 (en)
KR (1) KR900001887B1 (en)
AT (1) ATE97414T1 (en)
AU (1) AU587617B2 (en)
CA (1) CA1270825A (en)
DE (2) DE19975048I2 (en)
DK (1) DK170534B1 (en)
ES (1) ES8900165A1 (en)
FI (1) FI83324C (en)
HK (1) HK127795A (en)
IE (1) IE61755B1 (en)
IL (1) IL78700A (en)
NZ (1) NZ216052A (en)
PH (1) PH24037A (en)
SG (1) SG30590G (en)
ZA (1) ZA863499B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE269082T1 (en) * 1999-09-02 2004-07-15 Neurocrine Biosciences Inc POLYMORPHS OF N-METHYL-N-(3-(2-THIENYLCARBONYL)-PYRAZOLE(1,5-A)PYRIMIDINE-7-YL PHENYL)ACETAMIDE AND COMPOSITIONS AND METHODS RELATED
DE10004790B4 (en) * 2000-02-01 2004-09-09 Lts Lohmann Therapie-Systeme Ag Method for producing sewn or embroidered three-dimensional textile structure utilized for e.g. table cloth, involves connecting points on lattice structure with threads to form thread arrangement under which lattice structure is not visible
ES2222813B1 (en) * 2003-07-24 2005-12-16 Ferrer Internacional, S.A. N- (3- (3-SUBSTITUTES-PIRAZOLO (1,5-A) PIRIMIDIN-7-IL) -PENYL) -SULPHONAMIDS AND RELATED COMPOSITIONS AND METHODS

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4178449A (en) * 1978-04-17 1979-12-11 American Cyanamid Company Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines
NZ208554A (en) * 1983-06-23 1987-06-30 American Cyanamid Co (aryl and heteroaryl)-(7-(aryl and heteroaryl)-pyrazolo (1,5-a) pyrimidin-3-yl)-methanone derivatives and pharmaceutical compositions

Also Published As

Publication number Publication date
FI83324C (en) 1991-06-25
PH24037A (en) 1990-02-09
CA1270825A (en) 1990-06-26
FI83324B (en) 1991-03-15
NZ216052A (en) 1989-04-26
HK127795A (en) 1995-08-18
DK218286A (en) 1986-11-14
JPS61260083A (en) 1986-11-18
ES8900165A1 (en) 1989-03-01
KR900001887B1 (en) 1990-03-26
SG30590G (en) 1995-09-18
AU587617B2 (en) 1989-08-24
DE19975048I2 (en) 2001-06-13
ES554887A0 (en) 1989-03-01
FI861973A0 (en) 1986-05-12
KR860009017A (en) 1986-12-19
IL78700A0 (en) 1986-08-31
DE3689294T2 (en) 1994-06-09
AU5736086A (en) 1986-11-20
IE61755B1 (en) 1994-11-30
DK170534B1 (en) 1995-10-16
FI861973A (en) 1986-11-14
ATE97414T1 (en) 1993-12-15
ZA863499B (en) 1987-11-12
IE861247L (en) 1986-11-13
JPH0784468B2 (en) 1995-09-13
DK218286D0 (en) 1986-05-12
DE3689294D1 (en) 1993-12-23

Similar Documents

Publication Publication Date Title
MY109731A (en) Process for preparing aryl piperazinyl-heterocyclic compounds.
MX9702658A (en) New carboxylic acid derivatives, their preparation and their use.
ES8607252A1 (en) Redox indicators.
NZ233735A (en) Heterocyclic substituted aminophenol derivatives
CA2095587A1 (en) Process for preparing aryl piperazinyl-hetero-cyclic compounds
AU641952B2 (en) Substituted N-(imidazolyl)alkyl alanine derivatives
ES2001703A6 (en) Imidazolinyl derivatives, process for their preparation and agents with herbicidal activity containing them.
ES8704917A1 (en) 1-Piperazine carboxamide derivatives, their preparation and their use in pharmaceutical compositions.
ES8304919A1 (en) Dichloroamino acid derivatives useful as potent germicidal and fungicidal agents.
IL78700A (en) (7-(3-acylamino)-phenyl)pyrazolo(1,5-a)-pyrimidines,their preparation and pharmaceutical compositions containing them
IE850185L (en) Benzopyrans
EP0074130A3 (en) New imidazole compounds, process for the preparation thereof and pharmaceutical compositions containing them
ES8501607A1 (en) Five-membered nitrogen-containing heterocycles, process for their preparation and their use as pesticides.
IE56917B1 (en) N-sulphenylated hydantoins,a process for their preparation and their use as microbicides
ES8605247A1 (en) Substituted arylsulfonyl guanidines.
ES8506310A1 (en) Aminocyclic N-oxide derivatives, process for their preparation and their therapeutical use.
EP0008950A3 (en) Pyrimido(1,6-a)indole derivatives and intermediates therefor, processes for their preparation, pharmaceutical compositions containing the derivatives and their use
ES8705454A1 (en) Imidazoalkylcarboxylic-acid derivatives, process for their preparation and their use in the preparation of pharmaceutically active compounds.
ES8703855A1 (en) Sulfonyl-guanidinotriazine derivatives.
PT78364A (en) Process for preparing iminosulphonamides from pharmaceutic preparation wich contain these compounds and its therapeutical utilization
ES8407047A1 (en) Carboline derivatives.
IL57273A0 (en) Substituted phenylpropyl halides,their preparation and their use in the production of fungicidal morpholines and piperidines
CH609344A5 (en) Process for the preparation of novel 1-(5-nitrothiazol-2-yl)imidazole derivatives
ES2009463A6 (en) New 2-propanol derivatives, their preparation and their application as medicaments
ES486648A1 (en) 3,4-Dioxo-1,2,5-thiadiazolidine-1-oxides (I), their preparation, their use as fungicides, antifungal compositions containing the compounds (I) and the preparation of these compositions.

Legal Events

Date Code Title Description
KB Patent renewed
KB Patent renewed
KB Patent renewed
EXP Patent expired