IL72003A - Beta-lactamase inhibiting 6-(alkoxyaminomethyl)-penicillanic acid 1,1-dioxides and intermediates therefor - Google Patents

Beta-lactamase inhibiting 6-(alkoxyaminomethyl)-penicillanic acid 1,1-dioxides and intermediates therefor

Info

Publication number
IL72003A
IL72003A IL72003A IL7200384A IL72003A IL 72003 A IL72003 A IL 72003A IL 72003 A IL72003 A IL 72003A IL 7200384 A IL7200384 A IL 7200384A IL 72003 A IL72003 A IL 72003A
Authority
IL
Israel
Prior art keywords
beta
dioxides
penicillanic acid
alkoxyaminomethyl
intermediates therefor
Prior art date
Application number
IL72003A
Other languages
English (en)
Other versions
IL72003A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL72003A0 publication Critical patent/IL72003A0/xx
Publication of IL72003A publication Critical patent/IL72003A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
IL72003A 1983-06-06 1984-06-04 Beta-lactamase inhibiting 6-(alkoxyaminomethyl)-penicillanic acid 1,1-dioxides and intermediates therefor IL72003A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/501,475 US4499017A (en) 1983-06-06 1983-06-06 Beta-lactamase inhibiting 6-(alkoxyamino-methyl) penicillanic acid 1,1-dioxide and derivatives

Publications (2)

Publication Number Publication Date
IL72003A0 IL72003A0 (en) 1984-10-31
IL72003A true IL72003A (en) 1988-02-29

Family

ID=23993709

Family Applications (1)

Application Number Title Priority Date Filing Date
IL72003A IL72003A (en) 1983-06-06 1984-06-04 Beta-lactamase inhibiting 6-(alkoxyaminomethyl)-penicillanic acid 1,1-dioxides and intermediates therefor

Country Status (21)

Country Link
US (1) US4499017A (es)
EP (1) EP0128037B1 (es)
JP (1) JPS606693A (es)
KR (1) KR870000312B1 (es)
AT (1) ATE24512T1 (es)
AU (1) AU545467B2 (es)
CA (1) CA1247597A (es)
DE (1) DE3461800D1 (es)
DK (1) DK275884A (es)
ES (1) ES533147A0 (es)
FI (1) FI842255L (es)
GR (1) GR82214B (es)
HU (1) HU193573B (es)
IL (1) IL72003A (es)
NO (1) NO842248L (es)
NZ (1) NZ208381A (es)
PH (2) PH21372A (es)
PL (1) PL144040B1 (es)
PT (1) PT78689A (es)
YU (1) YU97084A (es)
ZA (1) ZA844184B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8928373D0 (en) * 1989-12-15 1990-02-21 Erba Carlo Spa Beta-lactam derivatives
PE20020613A1 (es) * 2000-07-19 2002-08-07 Novartis Ag Sales de (s)-n-(1-carboxi-2-metil-prop-1-il)-n-pentanoil-n-[2'-(1h-tetrazol-5-il)-bifenil-4-ilmetil]-amina como antagonista del receptor at1

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
RO84910B (ro) * 1982-01-11 1984-09-30 Pfizer Inc. Procedeu pentru prepararea unor derivati 1, 1-dioxizi ai acidului 6-aminoalchilpenicilanic

Also Published As

Publication number Publication date
DK275884D0 (da) 1984-06-04
ES8506720A1 (es) 1985-08-01
DE3461800D1 (en) 1987-02-05
HUT35266A (en) 1985-06-28
PL144040B1 (en) 1988-04-30
GR82214B (es) 1984-12-13
ZA844184B (en) 1986-01-29
NO842248L (no) 1984-12-07
JPS606693A (ja) 1985-01-14
IL72003A0 (en) 1984-10-31
YU97084A (en) 1986-10-31
ATE24512T1 (de) 1987-01-15
FI842255A0 (fi) 1984-06-05
DK275884A (da) 1985-01-09
CA1247597A (en) 1988-12-28
KR850000446A (ko) 1985-02-27
PH21372A (en) 1987-10-15
KR870000312B1 (ko) 1987-02-26
AU545467B2 (en) 1985-07-18
PT78689A (en) 1984-07-01
EP0128037B1 (en) 1986-12-30
AU2907684A (en) 1984-12-13
US4499017A (en) 1985-02-12
EP0128037A1 (en) 1984-12-12
ES533147A0 (es) 1985-08-01
FI842255A7 (fi) 1984-12-07
HU193573B (en) 1987-10-28
PL248043A1 (en) 1985-07-30
NZ208381A (en) 1987-05-29
PH22842A (en) 1989-01-19
FI842255L (fi) 1984-12-07

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Legal Events

Date Code Title Description
MM9K Patent not in force due to non-payment of renewal fees