IL57599A - Indole derivatives,their preparation and pharmaceutical compositions comprising them - Google Patents

Indole derivatives,their preparation and pharmaceutical compositions comprising them

Info

Publication number
IL57599A
IL57599A IL57599A IL5759979A IL57599A IL 57599 A IL57599 A IL 57599A IL 57599 A IL57599 A IL 57599A IL 5759979 A IL5759979 A IL 5759979A IL 57599 A IL57599 A IL 57599A
Authority
IL
Israel
Prior art keywords
preparation
pharmaceutical compositions
indole derivatives
indole
derivatives
Prior art date
Application number
IL57599A
Other languages
English (en)
Other versions
IL57599A0 (en
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19782827874 external-priority patent/DE2827874A1/de
Priority claimed from DE19792910367 external-priority patent/DE2910367A1/de
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of IL57599A0 publication Critical patent/IL57599A0/xx
Publication of IL57599A publication Critical patent/IL57599A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL57599A 1978-06-24 1979-06-20 Indole derivatives,their preparation and pharmaceutical compositions comprising them IL57599A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19782827874 DE2827874A1 (de) 1978-06-24 1978-06-24 Indolalkylamine und verfahren zu ihrer herstellung
DE19792910367 DE2910367A1 (de) 1979-03-16 1979-03-16 Indolalkylamine, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung

Publications (2)

Publication Number Publication Date
IL57599A0 IL57599A0 (en) 1979-10-31
IL57599A true IL57599A (en) 1983-03-31

Family

ID=25774808

Family Applications (1)

Application Number Title Priority Date Filing Date
IL57599A IL57599A (en) 1978-06-24 1979-06-20 Indole derivatives,their preparation and pharmaceutical compositions comprising them

Country Status (9)

Country Link
US (1) US4251538A (xx)
EP (1) EP0007399B1 (xx)
AU (1) AU525995B2 (xx)
CA (1) CA1133484A (xx)
DE (1) DE2961867D1 (xx)
ES (1) ES481715A1 (xx)
HU (1) HU180873B (xx)
IL (1) IL57599A (xx)
YU (1) YU42650B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3301758A1 (de) * 1983-01-20 1984-07-26 Merck Patent Gmbh, 6100 Darmstadt Indolderivate
DE3308668A1 (de) * 1983-03-11 1984-09-13 Merck Patent Gmbh, 6100 Darmstadt Indolderivate
DE3342632A1 (de) * 1983-11-25 1985-06-05 Merck Patent Gmbh, 6100 Darmstadt Indolderivate
US5256673A (en) * 1983-11-25 1993-10-26 Merck Patent Gesellschaft Mit Beschrankter Haftung Indole-3-yl-A-tetrahydropyridyl or piperidyl compounds
US4914114A (en) * 1984-05-28 1990-04-03 Merck Patent Gesellschaft Mit Breschrankter Haftung 3-[4-(4-phenyl-1,2,3,6-tetrahydro-1-pyridyl)butyl]-5-hydroxy-indole methanesulfonate having sedating and anti-parkinsonism properties
DE3419935A1 (de) * 1984-05-28 1985-11-28 Merck Patent Gmbh, 6100 Darmstadt Verwendung von hydroxyindolderivaten bei der senkung des blutdrucks
DE3604949A1 (de) * 1986-02-17 1987-08-20 Merck Patent Gmbh Hydroxyindolester
WO1988001998A1 (en) * 1986-09-16 1988-03-24 MERCK Patent Gesellschaft mit beschränkter Haftung Hydroxylindol derivatives
US5643784A (en) * 1990-12-04 1997-07-01 H, Lundbeck A/S Indan derivatives
NZ243065A (en) * 1991-06-13 1995-07-26 Lundbeck & Co As H Piperidine derivatives and pharmaceutical compositions
WO1998022110A1 (en) * 1996-11-20 1998-05-28 Virginia Tech Intellectual Properties, Inc. Prodrugs for the selective inhibition of monoamine oxidase-b
DE19725664A1 (de) * 1997-06-18 1998-12-24 Merck Patent Gmbh 3-Benzylpiperidine

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3155668A (en) * 1960-04-11 1964-11-03 Sterling Drug Inc 1-[3-, 2-, and 1-indolyl)-lower-alkyl]-tertiary amines and intermediates therefor
US3238215A (en) 1963-10-17 1966-03-01 Sterling Drug Inc 1-[(3-, 2-, and 1-indolyl)-lower-alkyl-, lower-alkenyl-, and lower-alkynyl]piperidines
US3217011A (en) 1965-05-07 1965-11-09 Sterling Drug Inc 1-(indolyglyoxalyl)-piperidines
GB1189064A (en) * 1967-05-01 1970-04-22 Sterling Drug Inc Indole Derivatives
US3487091A (en) * 1967-12-18 1969-12-30 American Home Prod 1-(benzyl- or substituted-benzyl)-3-(2-substituted-ethyl) indoles
DE2060816C3 (de) 1970-12-10 1980-09-04 Merck Patent Gmbh, 6100 Darmstadt 4-Phenylpiperidinderivate Verfahren zu ihrer Herstellung und pharmazeutische Zubereitungen enthaltend diese Verbindungen
GB1374414A (en) * 1972-06-12 1974-11-20 Sterling Drug Inc 1-acyl-3-amino-alkyl-indoles and their preparation

Also Published As

Publication number Publication date
EP0007399A1 (de) 1980-02-06
HU180873B (en) 1983-04-29
CA1133484A (en) 1982-10-12
IL57599A0 (en) 1979-10-31
YU144379A (en) 1983-02-28
EP0007399B1 (de) 1982-01-20
DE2961867D1 (en) 1982-03-04
YU42650B (en) 1988-10-31
AU525995B2 (en) 1982-12-09
AU4830279A (en) 1980-01-03
ES481715A1 (es) 1980-02-16
US4251538A (en) 1981-02-17

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Legal Events

Date Code Title Description
KB Patent renewed