IL41801A0 - New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and their manufacture - Google Patents

New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and their manufacture

Info

Publication number
IL41801A0
IL41801A0 IL41801A IL4180173A IL41801A0 IL 41801 A0 IL41801 A0 IL 41801A0 IL 41801 A IL41801 A IL 41801A IL 4180173 A IL4180173 A IL 4180173A IL 41801 A0 IL41801 A0 IL 41801A0
Authority
IL
Israel
Prior art keywords
carboxylic acid
penam
cephem
manufacture
new derivatives
Prior art date
Application number
IL41801A
Other languages
English (en)
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH425172A external-priority patent/CH560705A5/xx
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of IL41801A0 publication Critical patent/IL41801A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/20—Nitrogen atoms
    • C07D241/22—Benzenesulfonamido pyrazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/36—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1896—Compounds having one or more Si-O-acyl linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL41801A 1972-03-22 1973-03-16 New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and their manufacture IL41801A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH425172A CH560705A5 (sv) 1972-03-22 1972-03-22
CH1291972 1972-09-01
CH1853072 1972-12-20

Publications (1)

Publication Number Publication Date
IL41801A0 true IL41801A0 (en) 1973-05-31

Family

ID=27174774

Family Applications (1)

Application Number Title Priority Date Filing Date
IL41801A IL41801A0 (en) 1972-03-22 1973-03-16 New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and their manufacture

Country Status (13)

Country Link
US (1) US3996208A (sv)
AT (3) ATA863274A (sv)
AU (1) AU5349973A (sv)
CA (1) CA1049501A (sv)
DD (1) DD105617A5 (sv)
ES (1) ES412838A1 (sv)
FR (1) FR2181839B1 (sv)
GB (1) GB1423386A (sv)
HU (1) HU169031B (sv)
IE (1) IE37420B1 (sv)
IL (1) IL41801A0 (sv)
NL (1) NL7304036A (sv)
SE (1) SE7602730L (sv)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4071683A (en) * 1973-10-30 1978-01-31 Bayer Aktiengesellschaft Oxoimidazolidinylthiocarbonyl derivatives of ceph-3-em-4-carboxylic acids
US4086341A (en) * 1974-08-22 1978-04-25 Bayer Aktiengesellschaft Cephalosporin derivatives
DE2855884A1 (de) * 1978-12-23 1980-07-10 Hoechst Ag N-nitroaryl-n'-halogensulfonylharnstoffe, verfahren zu ihrer herstellung und ihre verwendung zur herstellung von nitroarylharnstoffen

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1545644A (fr) * 1966-07-15 1968-11-15 Astra Ab Procédé de fabrication de pénicillines renfermant un groupe amino-sulfonyle
GB1162261A (en) 1966-07-15 1969-08-20 Astra Ab Penicillins
IE32700B1 (en) 1968-02-03 1973-10-31 Beecham Group Ltd Penicillins
US3483188A (en) * 1968-06-13 1969-12-09 Bristol Myers Co 6-(alpha - 3 - allophanamidophenylacetamido) and 6 - (alpha - 3 - allophanamidothienylacetamido)-penicillanic acids
US3481922A (en) * 1968-06-13 1969-12-02 Bristol Myers Co 6-(alpha - 3 - acylthioureidophenylacetamido)-and 6 - (alpha-3-acylthioureidothienylacetamido)-penicillanic acids
US3687949A (en) * 1969-01-21 1972-08-29 Bristol Myers Co Synthetic cephalosporins
US3579501A (en) * 1969-08-22 1971-05-18 Bristol Myers Co 6-(alpha-(3 - guanyl - 1 - ureido)phenyl- or thienyl-acetamido)penicillanic acids

Also Published As

Publication number Publication date
AT326824B (de) 1975-12-29
US3996208A (en) 1976-12-07
HU169031B (sv) 1976-09-28
IE37420B1 (en) 1977-07-20
FR2181839A1 (sv) 1973-12-07
ES412838A1 (es) 1976-05-16
SE7602730L (sv) 1976-02-27
GB1423386A (en) 1976-02-04
AT325765B (de) 1975-11-10
ATA251973A (de) 1975-01-15
DD105617A5 (sv) 1974-05-05
NL7304036A (sv) 1973-09-25
FR2181839B1 (sv) 1976-03-05
CA1049501A (en) 1979-02-27
ATA863274A (de) 1975-03-15
IE37420L (en) 1973-09-22
AU5349973A (en) 1974-09-26

Similar Documents

Publication Publication Date Title
HK86679A (en) Dethiacephalosporanic acid derivatives and their preparation and use
IL43174A0 (en) New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid their manufacture and pharmaceutical compositions containing them
MY7900245A (en) Derivatives of cyclopentaneacetic acid
JPS57112397A (en) Manufacture of novel cephalosporin
IL42510A0 (en) Cephalosporin derivatives and their manufacture
GB1404392A (en) Quinolineacetic acid derivatives and processes for their manufacture
IL47477A (en) 7-acylamino-3-trialzolylthiomethyl 3-cephem-4-carboxylic acid derivatives and their production
ZA732010B (en) New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and processes for their manufacture
IL35312A0 (en) New derivatives of cephalosporin and process of preparation
IL41771A0 (en) Novel octanoic acid derivatives and their production
AU5843573A (en) Derivatives of 9-hydroxy-13-trans-prostenoic acid
IL41801A0 (en) New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and their manufacture
GB1403850A (en) Synthesis of n5-methyltetrahydrohomofolic acid and related reduced derivatives of homofolic acid
IL42712A0 (en) Phosphorus derivatives of triazolin-5-ones and-thiones and their manufacture
AU474986B2 (en) New derivatives of glycyprhetinic acid
ZA737223B (en) New derivatives of peman-3-carboxylic acid and cephem-4-carboxylic acid and processes for their manufacture
ZA731905B (en) New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and processes for their manufacture
JPS54138578A (en) Manufacture of 33oxyy2*33dihydroo1*44benzoxazine derivative
IL42820A0 (en) Novel derivatives of 6-amino-penicillanic acid and their preparation
ZA733099B (en) Preparation of 2-chloroethanephosphonic acid
ZA731818B (en) Derivatives of pyrazole-5-acetic acid and methods of preparing same
IE39538B1 (en) Derivatives of cyclopentanecetic acid
IL41162A (en) Halophenylthioacetamido cephalosporanic acid derivatives and their preparation
CA899863A (en) Derivatives of 7-aminocephalosporanic acid and process for their manufacture
CA899864A (en) Derivatives of 7-aminocephalosporanic acid and process for their manufacture