IL307918A - Methods for producing cyclic compounds comprising n-substituted amino acid residues - Google Patents

Methods for producing cyclic compounds comprising n-substituted amino acid residues

Info

Publication number
IL307918A
IL307918A IL307918A IL30791823A IL307918A IL 307918 A IL307918 A IL 307918A IL 307918 A IL307918 A IL 307918A IL 30791823 A IL30791823 A IL 30791823A IL 307918 A IL307918 A IL 307918A
Authority
IL
Israel
Prior art keywords
methods
amino acid
acid residues
substituted amino
cyclic compounds
Prior art date
Application number
IL307918A
Other languages
Hebrew (he)
Inventor
Hou Zengye
SETO Kentarou
Tanaka Kota
Aoki Masahide
SAKON Aya
Original Assignee
Chugai Pharmaceutical Co Ltd
Hou Zengye
SETO Kentarou
Tanaka Kota
Aoki Masahide
SAKON Aya
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Pharmaceutical Co Ltd, Hou Zengye, SETO Kentarou, Tanaka Kota, Aoki Masahide, SAKON Aya filed Critical Chugai Pharmaceutical Co Ltd
Priority claimed from PCT/JP2022/019606 external-priority patent/WO2022234864A1/en
Publication of IL307918A publication Critical patent/IL307918A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/1072General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups
    • C07K1/1075General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups by covalent attachment of amino acids or peptide residues
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/113General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides without change of the primary structure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/14Extraction; Separation; Purification
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64Cyclic peptides containing only normal peptide links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL307918A 2021-05-07 2022-05-06 Methods for producing cyclic compounds comprising n-substituted amino acid residues IL307918A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2021079014 2021-05-07
JP2021188473 2021-11-19
PCT/JP2022/019606 WO2022234864A1 (en) 2021-05-07 2022-05-06 Method for producing cyclic compound containing n-substituted amino acid residue

Publications (1)

Publication Number Publication Date
IL307918A true IL307918A (en) 2023-12-01

Family

ID=83887084

Family Applications (1)

Application Number Title Priority Date Filing Date
IL307918A IL307918A (en) 2021-05-07 2022-05-06 Methods for producing cyclic compounds comprising n-substituted amino acid residues

Country Status (6)

Country Link
JP (2) JP7165289B1 (en)
KR (2) KR102569348B1 (en)
AU (1) AU2022269959A1 (en)
CA (1) CA3219081A1 (en)
IL (1) IL307918A (en)
MX (1) MX2023013098A (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106928086B (en) 2015-12-31 2019-05-31 深圳翰宇药业股份有限公司 A kind of preparation method of long-chain compound

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUE054006T2 (en) 2011-12-28 2021-08-30 Chugai Pharmaceutical Co Ltd Peptide-compound cyclization method
US11542299B2 (en) * 2017-06-09 2023-01-03 Chugai Seiyaku Kabushiki Kaisha Method for synthesizing peptide containing N-substituted amino acid
EP3725796A4 (en) * 2017-12-15 2021-09-15 Chugai Seiyaku Kabushiki Kaisha Method for producing peptide, and method for processing bases
JPWO2020111238A1 (en) 2018-11-30 2021-10-21 中外製薬株式会社 Deprotection method for peptide compounds or amide compounds, resin removal method for solid-phase reaction, and method for producing peptide compounds.

Also Published As

Publication number Publication date
MX2023013098A (en) 2023-11-16
JP2022186851A (en) 2022-12-15
AU2022269959A1 (en) 2023-11-16
JPWO2022234864A1 (en) 2022-11-10
KR102569348B1 (en) 2023-08-21
KR20230169072A (en) 2023-12-15
KR20230003614A (en) 2023-01-06
JP7165289B1 (en) 2022-11-02
CA3219081A1 (en) 2022-11-10

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