IL304513A - שיטה להכנת צורה מועשרת אננטיומרית של 3-(2-כלורותיאזול-5-איל)-8-מתיל-7-אוקסו-6-פניל-3,2-דיהידרותיאזולו[2,3-a]פירימידין-4-איום-5-אולט - Google Patents
שיטה להכנת צורה מועשרת אננטיומרית של 3-(2-כלורותיאזול-5-איל)-8-מתיל-7-אוקסו-6-פניל-3,2-דיהידרותיאזולו[2,3-a]פירימידין-4-איום-5-אולטInfo
- Publication number
- IL304513A IL304513A IL304513A IL30451323A IL304513A IL 304513 A IL304513 A IL 304513A IL 304513 A IL304513 A IL 304513A IL 30451323 A IL30451323 A IL 30451323A IL 304513 A IL304513 A IL 304513A
- Authority
- IL
- Israel
- Prior art keywords
- dihydrothiazolo
- chlorothiazol
- olate
- ium
- pyrimidin
- Prior art date
Links
- YGDKLOWGWUOTRD-UHFFFAOYSA-N 3-(2-chloro-1,3-thiazol-5-yl)-8-methyl-5-oxo-6-phenyl-2,3-dihydro-[1,3]thiazolo[3,2-a]pyrimidin-8-ium-7-olate Chemical compound ClC=1SC(=CN=1)C1CSC=2N1C(=C(C([N+]=2C)=O)C1=CC=CC=C1)[O-] YGDKLOWGWUOTRD-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Catalysts (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP21153036.5A EP4032893A1 (en) | 2021-01-22 | 2021-01-22 | Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate |
| PCT/EP2022/051362 WO2022157321A1 (en) | 2021-01-22 | 2022-01-21 | Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL304513A true IL304513A (he) | 2023-09-01 |
Family
ID=74215738
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL304513A IL304513A (he) | 2021-01-22 | 2023-07-17 | שיטה להכנת צורה מועשרת אננטיומרית של 3-(2-כלורותיאזול-5-איל)-8-מתיל-7-אוקסו-6-פניל-3,2-דיהידרותיאזולו[2,3-a]פירימידין-4-איום-5-אולט |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US12559507B2 (he) |
| EP (2) | EP4032893A1 (he) |
| JP (1) | JP7840970B2 (he) |
| KR (1) | KR20230135109A (he) |
| CN (1) | CN116917291A (he) |
| AU (1) | AU2022210826C1 (he) |
| CA (1) | CA3205579A1 (he) |
| IL (1) | IL304513A (he) |
| MX (1) | MX2023008617A (he) |
| TW (1) | TW202246280A (he) |
| WO (1) | WO2022157321A1 (he) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP4063362A1 (en) * | 2021-03-25 | 2022-09-28 | Basf Se | Method for preparing enantiomerically enriched 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one by hydrogenation of the 2-oxo derivative in the presence of a chiral transition metal catalyst |
| WO2025223938A1 (en) * | 2024-04-26 | 2025-10-30 | Basf Se | Method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2- hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one |
| WO2025252510A1 (en) * | 2024-06-04 | 2025-12-11 | Basf Se | Method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR096022A1 (es) | 2013-04-11 | 2015-12-02 | Basf Se | Compuestos de pirimidinio sustituido, útiles para combatir plagas de animales |
| CN116076518A (zh) | 2017-03-31 | 2023-05-09 | 巴斯夫欧洲公司 | 用于防除动物害虫的嘧啶鎓化合物及其混合物 |
| CA3058083A1 (en) | 2017-04-27 | 2018-11-01 | Basf Se | Process for preparing optically active 2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium compounds |
| AR111671A1 (es) | 2017-05-03 | 2019-08-07 | Basf Se | Proceso para la preparación de compuestos de pirimidinio que contienen s |
| CN109970731B (zh) * | 2017-12-27 | 2020-05-29 | 湖南化工研究院有限公司 | 杀虫活性的1,3-二氮杂环并吡啶季胺盐化合物及其制备方法与应用 |
| EP4032878A1 (en) | 2021-01-22 | 2022-07-27 | Basf Se | Method for preparing 2-[2-(2-chlorothiazol-5-yl)-2-oxo-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one |
-
2021
- 2021-01-22 EP EP21153036.5A patent/EP4032893A1/en not_active Withdrawn
-
2022
- 2022-01-21 EP EP22702214.2A patent/EP4281461B1/en active Active
- 2022-01-21 TW TW111102686A patent/TW202246280A/zh unknown
- 2022-01-21 US US18/272,884 patent/US12559507B2/en active Active
- 2022-01-21 AU AU2022210826A patent/AU2022210826C1/en active Active
- 2022-01-21 KR KR1020237027986A patent/KR20230135109A/ko active Pending
- 2022-01-21 CA CA3205579A patent/CA3205579A1/en active Pending
- 2022-01-21 JP JP2023544051A patent/JP7840970B2/ja active Active
- 2022-01-21 MX MX2023008617A patent/MX2023008617A/es unknown
- 2022-01-21 CN CN202280011141.6A patent/CN116917291A/zh active Pending
- 2022-01-21 WO PCT/EP2022/051362 patent/WO2022157321A1/en not_active Ceased
-
2023
- 2023-07-17 IL IL304513A patent/IL304513A/he unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA3205579A1 (en) | 2022-07-28 |
| US12559507B2 (en) | 2026-02-24 |
| EP4281461B1 (en) | 2026-01-21 |
| WO2022157321A1 (en) | 2022-07-28 |
| CN116917291A (zh) | 2023-10-20 |
| JP2024504688A (ja) | 2024-02-01 |
| EP4032893A1 (en) | 2022-07-27 |
| KR20230135109A (ko) | 2023-09-22 |
| US20230416273A1 (en) | 2023-12-28 |
| AU2022210826B2 (en) | 2025-12-04 |
| AU2022210826C1 (en) | 2026-04-23 |
| EP4281461A1 (en) | 2023-11-29 |
| AU2022210826A9 (en) | 2025-03-20 |
| TW202246280A (zh) | 2022-12-01 |
| AU2022210826A1 (en) | 2023-08-03 |
| EP4281461C0 (en) | 2026-01-21 |
| MX2023008617A (es) | 2023-08-07 |
| JP7840970B2 (ja) | 2026-04-06 |
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