IL192230A0 - Pharmaceutical formulations of fenofibrate having improved bioavailability - Google Patents

Pharmaceutical formulations of fenofibrate having improved bioavailability

Info

Publication number
IL192230A0
IL192230A0 IL192230A IL19223008A IL192230A0 IL 192230 A0 IL192230 A0 IL 192230A0 IL 192230 A IL192230 A IL 192230A IL 19223008 A IL19223008 A IL 19223008A IL 192230 A0 IL192230 A0 IL 192230A0
Authority
IL
Israel
Prior art keywords
fenofibrate
pharmaceutical formulations
improved bioavailability
bioavailability
improved
Prior art date
Application number
IL192230A
Original Assignee
Teva Pharma
Fleshner Barak Moshe
Lerner Itzhak
Rosenberger Vered
Moldavski Naomi
Drabkin Anna
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharma, Fleshner Barak Moshe, Lerner Itzhak, Rosenberger Vered, Moldavski Naomi, Drabkin Anna filed Critical Teva Pharma
Publication of IL192230A0 publication Critical patent/IL192230A0/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1635Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL192230A 2005-12-28 2008-06-16 Pharmaceutical formulations of fenofibrate having improved bioavailability IL192230A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2005/047346 WO2007075171A1 (en) 2005-12-28 2005-12-28 Pharmaceutical formulations of fenofibrate having improved bioavailability

Publications (1)

Publication Number Publication Date
IL192230A0 true IL192230A0 (en) 2008-12-29

Family

ID=36499668

Family Applications (1)

Application Number Title Priority Date Filing Date
IL192230A IL192230A0 (en) 2005-12-28 2008-06-16 Pharmaceutical formulations of fenofibrate having improved bioavailability

Country Status (7)

Country Link
JP (1) JP2009522258A (en)
CN (1) CN101351191A (en)
BR (1) BRPI0520821A2 (en)
CA (1) CA2634094A1 (en)
IL (1) IL192230A0 (en)
MX (1) MX2008008589A (en)
WO (1) WO2007075171A1 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20120225946A1 (en) * 2009-09-09 2012-09-06 Bernard Charles Sherman Choline fenofibrate delayed release compositions
CN109125283A (en) 2013-03-14 2019-01-04 艾慕恩治疗公司 The preparation of peanut preparation for oral desensitization
KR101850119B1 (en) 2015-11-11 2018-04-20 제이투에이치바이오텍 (주) Novel Fenofibric Acid Prodrugs with Improved Bioavailability
JP2022532547A (en) 2019-05-10 2022-07-15 アイミューン セラピューティクス,インコーポレイテッド Ways to improve the quality of life of patients with peanut allergies
CN112618511A (en) * 2020-12-31 2021-04-09 辰欣药业股份有限公司 Prescription composition of fenofibrate capsule and preparation process thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2627696B1 (en) * 1988-02-26 1991-09-13 Fournier Innovation Synergie NEW GALENIC FORM OF FENOFIBRATE
FR2758459B1 (en) * 1997-01-17 1999-05-07 Pharma Pass FENOFIBRATE PHARMACEUTICAL COMPOSITION HAVING HIGH BIODAVAILABILITY AND PROCESS FOR PREPARING THE SAME
US6368622B2 (en) * 1999-01-29 2002-04-09 Abbott Laboratories Process for preparing solid formulations of lipid regulating agents with enhanced dissolution and absorption
TWI293877B (en) * 2000-09-20 2008-03-01 Rtp Pharma Inc Spray drying process and compositions of fenofibrate
MXPA04009385A (en) * 2002-03-26 2005-01-25 Teva Pharma Drug microparticles.
EP1680091B1 (en) * 2003-10-10 2017-05-31 Veloxis Pharmaceuticals A/S A solid dosage form comprising a fibrate
RU2343905C2 (en) * 2003-10-10 2009-01-20 Лайфсайкл Фарма А/С Solid dosed out forms including fibrat and statin

Also Published As

Publication number Publication date
CN101351191A (en) 2009-01-21
BRPI0520821A2 (en) 2009-06-30
JP2009522258A (en) 2009-06-11
CA2634094A1 (en) 2007-07-05
MX2008008589A (en) 2009-02-25
WO2007075171A1 (en) 2007-07-05

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