IL173036A0 - Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors - Google Patents

Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors

Info

Publication number
IL173036A0
IL173036A0 IL173036A IL17303606A IL173036A0 IL 173036 A0 IL173036 A0 IL 173036A0 IL 173036 A IL173036 A IL 173036A IL 17303606 A IL17303606 A IL 17303606A IL 173036 A0 IL173036 A0 IL 173036A0
Authority
IL
Israel
Prior art keywords
quinoline
affinity
quinazoline derivatives
type receptors
receptors
Prior art date
Application number
IL173036A
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of IL173036A0 publication Critical patent/IL173036A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C04CEMENTS; CONCRETE; ARTIFICIAL STONE; CERAMICS; REFRACTORIES
    • C04BLIME, MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS; REFRACTORIES; TREATMENT OF NATURAL STONE
    • C04B35/00Shaped ceramic products characterised by their composition; Ceramics compositions; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/622Forming processes; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/626Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
    • C04B35/632Organic additives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Manufacturing & Machinery (AREA)
  • Ceramic Engineering (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Inorganic Chemistry (AREA)
  • Psychiatry (AREA)
  • Materials Engineering (AREA)
  • Structural Engineering (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL173036A 2003-07-18 2006-01-09 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors IL173036A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0316915.8A GB0316915D0 (en) 2003-07-18 2003-07-18 Compounds
PCT/EP2004/008000 WO2005014552A1 (en) 2003-07-18 2004-07-15 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors

Publications (1)

Publication Number Publication Date
IL173036A0 true IL173036A0 (en) 2006-06-11

Family

ID=27764115

Family Applications (1)

Application Number Title Priority Date Filing Date
IL173036A IL173036A0 (en) 2003-07-18 2006-01-09 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors

Country Status (29)

Country Link
US (5) US7279481B2 (en)
EP (3) EP1876174B1 (en)
JP (1) JP2006528146A (en)
KR (1) KR20060041242A (en)
CN (1) CN100441571C (en)
AR (1) AR046394A1 (en)
AT (2) ATE448205T1 (en)
AU (1) AU2004263268B2 (en)
BR (1) BRPI0412695A (en)
CA (1) CA2532452A1 (en)
CY (1) CY1107974T1 (en)
DE (2) DE602004012564T2 (en)
DK (1) DK1646613T3 (en)
ES (2) ES2302543T3 (en)
GB (1) GB0316915D0 (en)
HK (1) HK1089438A1 (en)
HR (1) HRP20080226T3 (en)
IL (1) IL173036A0 (en)
IS (1) IS2744B (en)
MA (1) MA27926A1 (en)
MX (1) MXPA06000716A (en)
NO (1) NO20060774L (en)
NZ (1) NZ544586A (en)
PL (1) PL1646613T3 (en)
PT (1) PT1646613E (en)
RU (1) RU2402533C2 (en)
SI (1) SI1646613T1 (en)
TW (1) TW200521115A (en)
WO (1) WO2005014552A1 (en)

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EA034677B1 (en) 2015-11-20 2020-03-05 4Д Фарма Рисёрч Лимитед Compositions for treating or preventing cancer comprising enterococcus gallinarum strain
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EP3638271B1 (en) 2017-06-14 2020-10-14 4D Pharma Research Limited Compositions comprising bacterial strains
HUE052258T2 (en) 2017-06-14 2021-04-28 4D Pharma Res Ltd Compositions comprising a bacterial strain of the genus megasphaera and uses thereof
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Also Published As

Publication number Publication date
PT1646613E (en) 2008-06-19
MA27926A1 (en) 2006-06-01
HK1089438A1 (en) 2006-12-01
US20060229312A1 (en) 2006-10-12
NO20060774L (en) 2006-04-06
US7279481B2 (en) 2007-10-09
EP2145622A1 (en) 2010-01-20
DK1646613T3 (en) 2008-07-14
CY1107974T1 (en) 2013-09-04
HRP20080226T3 (en) 2008-06-30
DE602004024141D1 (en) 2009-12-24
US20080280919A1 (en) 2008-11-13
WO2005014552A1 (en) 2005-02-17
MXPA06000716A (en) 2006-03-30
US20100204273A1 (en) 2010-08-12
US7732600B2 (en) 2010-06-08
US20070167423A1 (en) 2007-07-19
US7592346B2 (en) 2009-09-22
CN100441571C (en) 2008-12-10
CA2532452A1 (en) 2005-02-17
EP1646613A1 (en) 2006-04-19
EP1646613B1 (en) 2008-03-19
SI1646613T1 (en) 2008-08-31
AU2004263268B2 (en) 2010-12-16
KR20060041242A (en) 2006-05-11
PL1646613T3 (en) 2008-08-29
EP1876174B1 (en) 2009-11-11
IS8304A (en) 2006-02-15
US20090312546A1 (en) 2009-12-17
RU2402533C2 (en) 2010-10-27
CN1852896A (en) 2006-10-25
ES2336148T3 (en) 2010-04-08
ATE448205T1 (en) 2009-11-15
TW200521115A (en) 2005-07-01
DE602004012564D1 (en) 2008-04-30
US7459456B2 (en) 2008-12-02
RU2006104993A (en) 2006-08-10
BRPI0412695A (en) 2006-10-03
JP2006528146A (en) 2006-12-14
ATE389637T1 (en) 2008-04-15
AR046394A1 (en) 2005-12-07
EP1876174A1 (en) 2008-01-09
IS2744B (en) 2011-08-15
NZ544586A (en) 2009-05-31
AU2004263268A1 (en) 2005-02-17
ES2302543T3 (en) 2008-07-16
GB0316915D0 (en) 2003-08-20
DE602004012564T2 (en) 2009-04-30

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