IL172592A0 - Pyrazolopyrimidines - Google Patents
PyrazolopyrimidinesInfo
- Publication number
- IL172592A0 IL172592A0 IL172592A IL17259205A IL172592A0 IL 172592 A0 IL172592 A0 IL 172592A0 IL 172592 A IL172592 A IL 172592A IL 17259205 A IL17259205 A IL 17259205A IL 172592 A0 IL172592 A0 IL 172592A0
- Authority
- IL
- Israel
- Prior art keywords
- pyrazolopyrimidines
- Prior art date
Links
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10328996 | 2003-06-27 | ||
DE10339360A DE10339360A1 (en) | 2003-06-27 | 2003-08-27 | New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood |
DE2003157570 DE10357570A1 (en) | 2003-12-10 | 2003-12-10 | New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood |
PCT/EP2004/006609 WO2005000851A1 (en) | 2003-06-27 | 2004-06-18 | Pyrazolopyrimidines |
Publications (1)
Publication Number | Publication Date |
---|---|
IL172592A0 true IL172592A0 (en) | 2006-04-10 |
Family
ID=40506494
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL172592A IL172592A0 (en) | 2003-06-27 | 2005-12-15 | Pyrazolopyrimidines |
Country Status (3)
Country | Link |
---|---|
EA (1) | EA009517B1 (en) |
EC (1) | ECSP056252A (en) |
IL (1) | IL172592A0 (en) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010033941A1 (en) | 2008-09-22 | 2010-03-25 | Array Biopharma Inc. | Substituted imidazo[1,2b]pyridazine compounds as trk kinase inhibitors |
UY32192A (en) * | 2008-10-22 | 2011-05-31 | Array Biopharma Inc | PIRAZOLO COMPOUNDS [1,5-a] PIRIMIDINE REPLACED AS TRK CINASA INHIBITORS |
AR077468A1 (en) | 2009-07-09 | 2011-08-31 | Array Biopharma Inc | PIRAZOLO COMPOUNDS (1,5-A) PYRIMIDINE SUBSTITUTED AS TRK-QUINASA INHIBITORS |
PT2775842T (en) * | 2011-08-17 | 2017-11-15 | Adama Makhteshim Ltd | 1-substituted-5-fluoro-3,6-dihydro-6-imino-2(1h)-pyrimidinone derivatives as fungicidal agents for use in plant protection |
UA114490C2 (en) * | 2011-10-06 | 2017-06-26 | Байєр Інтеллектуал Проперті Гмбх | Heterocyclylpyri(mi)dinylpyrazole as fungicidals |
DK2763993T3 (en) * | 2011-10-06 | 2017-07-24 | Bayer Ip Gmbh | HETEROCYCLYLPYRI (MI) DINYLPYRAZOL |
UA115462C2 (en) * | 2012-12-28 | 2017-11-10 | Адама Махтешім Лтд. | -(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives |
AU2013370494B2 (en) * | 2012-12-31 | 2017-08-17 | Adama Makhteshim Ltd. | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides |
KR102649887B1 (en) | 2014-11-16 | 2024-03-22 | 어레이 바이오파마 인크. | Crystalline form of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide hydrogen sulfate |
TN2018000138A1 (en) | 2015-10-26 | 2019-10-04 | Array Biopharma Inc | Point mutations in trk inhibitor-resistant cancer and methods relating to the same |
MX2018012163A (en) | 2016-04-04 | 2019-07-08 | Loxo Oncology Inc | Liquid formulations of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrro lidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine- 1-carboxamide. |
US10045991B2 (en) | 2016-04-04 | 2018-08-14 | Loxo Oncology, Inc. | Methods of treating pediatric cancers |
MX2018012544A (en) * | 2016-04-15 | 2019-01-31 | Bayer Animal Health Gmbh | Pyrazolopyrimidine derivatives. |
JP7443057B2 (en) | 2016-05-18 | 2024-03-05 | ロクソ オンコロジー, インコーポレイテッド | (S)-N-(5-((R)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine -1-Preparation of carboxamide |
JOP20190092A1 (en) | 2016-10-26 | 2019-04-25 | Array Biopharma Inc | PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF |
JOP20190213A1 (en) | 2017-03-16 | 2019-09-16 | Array Biopharma Inc | Macrocyclic compounds as ros1 kinase inhibitors |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4908056A (en) * | 1986-04-25 | 1990-03-13 | E. I. Du Pont De Nemours And Company | Heterocyclic acyl sulfonamides |
-
2004
- 2004-06-18 EA EA200600021A patent/EA009517B1/en not_active IP Right Cessation
-
2005
- 2005-12-15 IL IL172592A patent/IL172592A0/en unknown
- 2005-12-26 EC ECSP056252 patent/ECSP056252A/en unknown
Also Published As
Publication number | Publication date |
---|---|
EA200600021A1 (en) | 2006-06-30 |
EA009517B1 (en) | 2008-02-28 |
ECSP056252A (en) | 2006-04-19 |
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