ECSP056252A - PIRAZOLOPIRIMIDINAS - Google Patents
PIRAZOLOPIRIMIDINASInfo
- Publication number
- ECSP056252A ECSP056252A ECSP056252A ECSP056252A EC SP056252 A ECSP056252 A EC SP056252A EC SP056252 A ECSP056252 A EC SP056252A EC SP056252 A ECSP056252 A EC SP056252A
- Authority
- EC
- Ecuador
- Prior art keywords
- xii
- products
- obtaining
- procedures
- pirazolopirimidinas
- Prior art date
Links
Abstract
Nuevas pirazolopirimidinas de la fórmula (I) (I)en la queR1, R2, R3, R4, X y Hal tienen los significados anteriormente indicados,varios procedimientos para la obtención de estos productos y su empleo para la lucha contra los microorganismos indeseados. Nuevos productos intermedios de las fórmulas (II), (X), (XII-a) y (XII-b) (II) (X) (XII-a)y (XII-b)así como procedimientos para la obtención de estos productos.New pyrazolopyrimidines of the formula (I) (I) in which R1, R2, R3, R4, X and Hal have the meanings indicated above, various procedures for obtaining these products and their use for the fight against unwanted microorganisms. New intermediate products of the formulas (II), (X), (XII-a) and (XII-b) (II) (X) (XII-a) and (XII-b) as well as procedures for obtaining these products.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10328996 | 2003-06-27 | ||
DE10339360A DE10339360A1 (en) | 2003-06-27 | 2003-08-27 | New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood |
DE2003157570 DE10357570A1 (en) | 2003-12-10 | 2003-12-10 | New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP056252A true ECSP056252A (en) | 2006-04-19 |
Family
ID=40506494
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSP056252 ECSP056252A (en) | 2003-06-27 | 2005-12-26 | PIRAZOLOPIRIMIDINAS |
Country Status (3)
Country | Link |
---|---|
EA (1) | EA009517B1 (en) |
EC (1) | ECSP056252A (en) |
IL (1) | IL172592A0 (en) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP5503655B2 (en) | 2008-09-22 | 2014-05-28 | アレイ バイオファーマ、インコーポレイテッド | Substituted imidazo [1,2B] pyridazine compounds as TRK kinase inhibitors |
SI2350071T1 (en) | 2008-10-22 | 2014-05-30 | Array Biopharma, Inc. | SUBSTITUTED PYRAZOLOŠ1,5-aĆPYRIMIDINE COMPOUNDS AS TRK KINASE INHIBITORS |
AR077468A1 (en) | 2009-07-09 | 2011-08-31 | Array Biopharma Inc | PIRAZOLO COMPOUNDS (1,5-A) PYRIMIDINE SUBSTITUTED AS TRK-QUINASA INHIBITORS |
PT2775842T (en) * | 2011-08-17 | 2017-11-15 | Adama Makhteshim Ltd | 1-substituted-5-fluoro-3,6-dihydro-6-imino-2(1h)-pyrimidinone derivatives as fungicidal agents for use in plant protection |
MX351460B (en) * | 2011-10-06 | 2017-10-16 | Bayer Ip Gmbh | Heterocyclylpyri(mi)dinylpyrazole. |
RU2616293C2 (en) * | 2011-10-06 | 2017-04-14 | Байер Интеллектуэль Проперти Гмбх | Geterocyclilpyridinylpyrazols as fungicidal agents |
HUE047711T2 (en) * | 2012-12-28 | 2020-05-28 | Adama Makhteshim Ltd | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives |
US9642368B2 (en) * | 2012-12-31 | 2017-05-09 | Adama Makhteshim Ltd. | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides |
CN113354649A (en) | 2014-11-16 | 2021-09-07 | 阵列生物制药公司 | Novel crystal form |
US10724102B2 (en) | 2015-10-26 | 2020-07-28 | Loxo Oncology, Inc. | Point mutations in TRK inhibitor-resistant cancer and methods relating to the same |
US10045991B2 (en) | 2016-04-04 | 2018-08-14 | Loxo Oncology, Inc. | Methods of treating pediatric cancers |
CU20180125A7 (en) | 2016-04-04 | 2019-05-03 | Loxo Oncology Inc | LIQUID FORMULATIONS OF (S) -N- (5 - ((R) -2- (2,5-DIFLUOROPHENYL) -PIRROLIDIN-1-IL) -PIRAZOLO [1,5-ALPIRIMIDIN-3-IL) -3 HYDROXIPIRROLIDINE- 1-CARBOXAMIDE |
PL3442974T3 (en) | 2016-04-15 | 2023-12-04 | Elanco Animal Health Gmbh | Pyrazolopyrimidine derivatives |
AU2017268371B2 (en) | 2016-05-18 | 2020-11-19 | Array Biopharma Inc. | Preparation of (S)-N-(5-((R)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)pyrazolo(1,5-A)pyrimidin-3-y l)-3-hydroxypyrrolidine-1-carboxamide |
JOP20190092A1 (en) | 2016-10-26 | 2019-04-25 | Array Biopharma Inc | PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF |
JOP20190213A1 (en) | 2017-03-16 | 2019-09-16 | Array Biopharma Inc | Macrocyclic compounds as ros1 kinase inhibitors |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4908056A (en) * | 1986-04-25 | 1990-03-13 | E. I. Du Pont De Nemours And Company | Heterocyclic acyl sulfonamides |
-
2004
- 2004-06-18 EA EA200600021A patent/EA009517B1/en not_active IP Right Cessation
-
2005
- 2005-12-15 IL IL172592A patent/IL172592A0/en unknown
- 2005-12-26 EC ECSP056252 patent/ECSP056252A/en unknown
Also Published As
Publication number | Publication date |
---|---|
EA009517B1 (en) | 2008-02-28 |
IL172592A0 (en) | 2006-04-10 |
EA200600021A1 (en) | 2006-06-30 |
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