IL160043A0 - Process for the preparation of indole derivatives - Google Patents
Process for the preparation of indole derivativesInfo
- Publication number
- IL160043A0 IL160043A0 IL16004302A IL16004302A IL160043A0 IL 160043 A0 IL160043 A0 IL 160043A0 IL 16004302 A IL16004302 A IL 16004302A IL 16004302 A IL16004302 A IL 16004302A IL 160043 A0 IL160043 A0 IL 160043A0
- Authority
- IL
- Israel
- Prior art keywords
- preparation
- indole derivatives
- indole
- derivatives
- Prior art date
Links
- 229940054051 antipsychotic indole derivative Drugs 0.000 title 1
- 150000002475 indoles Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D209/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an alkyl or cycloalkyl radical attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
- C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01810817 | 2001-08-22 | ||
| PCT/EP2002/009046 WO2003018555A1 (en) | 2001-08-22 | 2002-08-13 | Process for the preparation of indole derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL160043A0 true IL160043A0 (en) | 2004-06-20 |
Family
ID=8184102
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL16004302A IL160043A0 (en) | 2001-08-22 | 2002-08-13 | Process for the preparation of indole derivatives |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20050032875A1 (ru) |
| EP (1) | EP1423365A1 (ru) |
| JP (1) | JP2005503393A (ru) |
| CN (1) | CN1545502A (ru) |
| CA (1) | CA2455842A1 (ru) |
| IL (1) | IL160043A0 (ru) |
| WO (1) | WO2003018555A1 (ru) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2453505C (en) | 2001-07-13 | 2011-04-19 | Astrazeneca Uk Limited | Preparation of aminopyrimidine compounds |
| EP2335700A1 (en) * | 2001-07-25 | 2011-06-22 | Boehringer Ingelheim (Canada) Ltd. | Hepatitis C virus polymerase inhibitors with a heterobicylic structure |
| GB0218781D0 (en) | 2002-08-13 | 2002-09-18 | Astrazeneca Ab | Chemical process |
| US7098231B2 (en) * | 2003-01-22 | 2006-08-29 | Boehringer Ingelheim International Gmbh | Viral polymerase inhibitors |
| US7223785B2 (en) * | 2003-01-22 | 2007-05-29 | Boehringer Ingelheim International Gmbh | Viral polymerase inhibitors |
| US20060105441A1 (en) * | 2003-03-13 | 2006-05-18 | Reinhold Ohrlein | Process for the preparation of indole derivatives by enzymatic acylation |
| GB0312896D0 (en) | 2003-06-05 | 2003-07-09 | Astrazeneca Ab | Chemical process |
| UY28501A1 (es) | 2003-09-10 | 2005-04-29 | Astrazeneca Uk Ltd | Compuestos químicos |
| US7432380B2 (en) * | 2003-10-16 | 2008-10-07 | Ciba Specialty Chemicals Corp. | Crystalline form of Fluvastatin sodium |
| GB0324791D0 (en) | 2003-10-24 | 2003-11-26 | Astrazeneca Ab | Chemical process |
| ES2431314T3 (es) * | 2004-02-20 | 2013-11-26 | Boehringer Ingelheim International Gmbh | Inhibidores de polimerasa vírica |
| WO2006030304A2 (en) * | 2004-09-17 | 2006-03-23 | Ranbaxy Laboratories Limited | Novel forms of fluvastatin sodium, processes for preparation and pharmaceutical compositions thereof |
| GB0428328D0 (en) * | 2004-12-24 | 2005-02-02 | Astrazeneca Uk Ltd | Chemical process |
| AU2006213769B2 (en) * | 2005-02-11 | 2012-10-04 | Boehringer Ingelheim International Gmbh | Process for preparing 2,3-disubstituted indoles |
| CA2618682C (en) * | 2005-08-12 | 2011-06-21 | Boehringer Ingelheim International Gmbh | Viral polymerase inhibitors |
| MX357470B (es) * | 2011-01-18 | 2018-07-11 | Dsm Sinochem Pharm Nl Bv | Procedimiento para la preparación de estatinas en presencia de base. |
| US10968187B2 (en) * | 2017-07-28 | 2021-04-06 | Lonza Solutions Ag | Method for preparation of alkylated or fluoro, chloro and fluorochloro alkylated compounds by heterogeneous cobalt catalysis |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5354772A (en) * | 1982-11-22 | 1994-10-11 | Sandoz Pharm. Corp. | Indole analogs of mevalonolactone and derivatives thereof |
| US4739073A (en) * | 1983-11-04 | 1988-04-19 | Sandoz Pharmaceuticals Corp. | Intermediates in the synthesis of indole analogs of mevalonolactone and derivatives thereof |
| US4808621A (en) * | 1986-07-07 | 1989-02-28 | Warner-Lambert Company | Trans-6-[2-(N-heteroaryl-3,5-disubstituted)pyrazol-4-yl)-ethyl]- or ethenyl]tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis |
| US5102893A (en) * | 1986-07-07 | 1992-04-07 | Warner-Lambert Company | Trans-6-(2-(n-heteroaryl-3,5-disubstituted)pyrazol-4-yl)-ethyl- or ethenyl)tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis |
| JP2002505663A (ja) * | 1997-04-09 | 2002-02-19 | コモンウエルス サイエンティフィック アンド インダストリアル リサーチ オーガナイゼーション | アリールホウ酸エステル |
| PT1064243E (pt) * | 1998-03-18 | 2003-03-31 | Ciba Sc Holding Ag | Reaccoes de acoplamento com catalisadores de paladio |
| AU2001274049A1 (en) * | 2000-05-26 | 2001-12-11 | Ciba Specialty Chemicals Holding Inc. | Process for the preparation of indole derivatives and intermediates of the process |
-
2002
- 2002-08-13 EP EP02796227A patent/EP1423365A1/en not_active Withdrawn
- 2002-08-13 CN CNA028164350A patent/CN1545502A/zh active Pending
- 2002-08-13 IL IL16004302A patent/IL160043A0/xx unknown
- 2002-08-13 WO PCT/EP2002/009046 patent/WO2003018555A1/en not_active Application Discontinuation
- 2002-08-13 JP JP2003523219A patent/JP2005503393A/ja not_active Withdrawn
- 2002-08-13 CA CA002455842A patent/CA2455842A1/en not_active Abandoned
- 2002-08-13 US US10/487,269 patent/US20050032875A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20050032875A1 (en) | 2005-02-10 |
| EP1423365A1 (en) | 2004-06-02 |
| CN1545502A (zh) | 2004-11-10 |
| JP2005503393A (ja) | 2005-02-03 |
| CA2455842A1 (en) | 2003-03-06 |
| WO2003018555A1 (en) | 2003-03-06 |
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