AU2001274049A1 - Process for the preparation of indole derivatives and intermediates of the process - Google Patents
Process for the preparation of indole derivatives and intermediates of the processInfo
- Publication number
- AU2001274049A1 AU2001274049A1 AU2001274049A AU7404901A AU2001274049A1 AU 2001274049 A1 AU2001274049 A1 AU 2001274049A1 AU 2001274049 A AU2001274049 A AU 2001274049A AU 7404901 A AU7404901 A AU 7404901A AU 2001274049 A1 AU2001274049 A1 AU 2001274049A1
- Authority
- AU
- Australia
- Prior art keywords
- intermediates
- preparation
- indole derivatives
- indole
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D209/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an alkyl or cycloalkyl radical attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP00810460 | 2000-05-26 | ||
EP00810460 | 2000-05-26 | ||
PCT/EP2001/005667 WO2001092223A1 (en) | 2000-05-26 | 2001-05-17 | Process for the preparation of indole derivatives and intermediates of the process |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001274049A1 true AU2001274049A1 (en) | 2001-12-11 |
Family
ID=8174725
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001274049A Abandoned AU2001274049A1 (en) | 2000-05-26 | 2001-05-17 | Process for the preparation of indole derivatives and intermediates of the process |
Country Status (9)
Country | Link |
---|---|
US (2) | US6743926B2 (en) |
EP (1) | EP1284964A1 (en) |
JP (1) | JP2003535077A (en) |
CN (1) | CN1217930C (en) |
AR (1) | AR036000A1 (en) |
AU (1) | AU2001274049A1 (en) |
CA (1) | CA2407862A1 (en) |
IL (1) | IL152580A0 (en) |
WO (1) | WO2001092223A1 (en) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001092223A1 (en) * | 2000-05-26 | 2001-12-06 | Ciba Specialty Chemicals Holding Inc. | Process for the preparation of indole derivatives and intermediates of the process |
PT1404642E (en) * | 2001-07-06 | 2010-03-29 | Basf Se | Process for the preparatiom of 7-amino syn 3,5-dihydroxy heptanoic acid derivatives, intermediates thereof and methods for their preparation |
CN1545502A (en) * | 2001-08-22 | 2004-11-10 | �������⻯ѧƷ�ع�����˾ | Process for the preparation of indole derivatives |
GB0204129D0 (en) | 2002-02-21 | 2002-04-10 | Novartis Ag | Process for the manufacture of organic compounds |
EP1515717B8 (en) * | 2002-06-13 | 2009-12-16 | Novartis AG | Calcium salts of indole derived statins |
WO2004009527A1 (en) * | 2002-07-19 | 2004-01-29 | Aryx Therapeutics | Materials and methods for treating hypercholesterolemia |
US20060105441A1 (en) * | 2003-03-13 | 2006-05-18 | Reinhold Ohrlein | Process for the preparation of indole derivatives by enzymatic acylation |
JP4269902B2 (en) | 2003-08-27 | 2009-05-27 | 住友化学株式会社 | Method for producing aromatic unsaturated compound |
US7432380B2 (en) * | 2003-10-16 | 2008-10-07 | Ciba Specialty Chemicals Corp. | Crystalline form of Fluvastatin sodium |
WO2006030304A2 (en) * | 2004-09-17 | 2006-03-23 | Ranbaxy Laboratories Limited | Novel forms of fluvastatin sodium, processes for preparation and pharmaceutical compositions thereof |
WO2006085338A2 (en) * | 2005-02-11 | 2006-08-17 | Jubilant Organosys Limited | Novel polymorphic forms of fluvastatin sodium and process for preparing the same |
CN1978428B (en) * | 2005-12-05 | 2012-07-04 | 四川抗菌素工业研究所有限公司 | Method for preparing (3R, %S)-Fluvastatin |
DE602006006899D1 (en) | 2006-04-20 | 2009-07-02 | Italiana Sint Spa | Process for the preparation of fluvastatin sodium |
CN104250222A (en) * | 2013-06-27 | 2014-12-31 | 上海朴颐化学科技有限公司 | Improvement method of preparation technology of tert-butyl (E)-7-[3'-(4''-fluorophenyl)-1'-methylethyl-indol-2'-yl)-3-oxo-5-hydroxy-6-heptenoate |
CN103342721B (en) * | 2013-07-15 | 2016-04-13 | 凯莱英医药集团(天津)股份有限公司 | A kind of method preparing fluvastatin key intermediate |
JP6649263B2 (en) * | 2014-10-10 | 2020-02-19 | 株式会社エーピーアイ コーポレーション | Method for purifying statins |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU570021B2 (en) | 1982-11-22 | 1988-03-03 | Novartis Ag | Analogs of mevalolactone |
US4739073A (en) * | 1983-11-04 | 1988-04-19 | Sandoz Pharmaceuticals Corp. | Intermediates in the synthesis of indole analogs of mevalonolactone and derivatives thereof |
US4571428A (en) * | 1983-07-08 | 1986-02-18 | Sandoz, Inc. | 6-Substituted-4-hydroxy-tetrahydropyran-2-ones |
US4650890A (en) * | 1984-04-03 | 1987-03-17 | Sandoz Corp. | Preparation of olefinic compounds and intermediates thereof |
US4677211A (en) * | 1984-06-29 | 1987-06-30 | Sandoz Pharmaceuticals Corp. | Preparation of lactones |
US4870199A (en) * | 1986-04-30 | 1989-09-26 | Sandoz Pharm. Corp. | Processes for the synthesis of diprotected R[R*,S*]-3,5-dihydroxy-6-oxohexanoate esters |
JPS6322056A (en) * | 1986-04-30 | 1988-01-29 | サンド・アクチエンゲゼルシヤフト | Manufacture of olefinic compound |
EP0363934B1 (en) * | 1988-10-13 | 1993-12-29 | Sandoz Ag | Process for the preparation of 7-substituted-hept-6-enoic and -heptanoic acids and derivatives thereof |
DK181190D0 (en) | 1990-07-30 | 1990-07-30 | Lundbeck & Co As H | 3-ARYL-INDOL OR 3-ARYL-INDAZOL DERIVATIVES |
HU9203780D0 (en) * | 1991-12-12 | 1993-03-29 | Sandoz Ag | Stabilized pharmaceutical products of hmg-coa reductase inhibitor and method for producing them |
CA2321791A1 (en) | 1998-03-18 | 1999-09-23 | Ciba Specialty Chemicals Holding Inc. | Coupling reactions with palladium catalysts |
WO2001092223A1 (en) * | 2000-05-26 | 2001-12-06 | Ciba Specialty Chemicals Holding Inc. | Process for the preparation of indole derivatives and intermediates of the process |
-
2001
- 2001-05-17 WO PCT/EP2001/005667 patent/WO2001092223A1/en not_active Application Discontinuation
- 2001-05-17 EP EP01940495A patent/EP1284964A1/en not_active Withdrawn
- 2001-05-17 IL IL15258001A patent/IL152580A0/en unknown
- 2001-05-17 CA CA002407862A patent/CA2407862A1/en not_active Abandoned
- 2001-05-17 JP JP2002500838A patent/JP2003535077A/en active Pending
- 2001-05-17 US US10/296,106 patent/US6743926B2/en not_active Expired - Fee Related
- 2001-05-17 AU AU2001274049A patent/AU2001274049A1/en not_active Abandoned
- 2001-05-17 CN CN01810202.6A patent/CN1217930C/en not_active Expired - Fee Related
- 2001-05-24 AR ARP010102482A patent/AR036000A1/en not_active Application Discontinuation
-
2004
- 2004-03-18 US US10/803,705 patent/US20040176614A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US20040176614A1 (en) | 2004-09-09 |
WO2001092223A1 (en) | 2001-12-06 |
EP1284964A1 (en) | 2003-02-26 |
CN1217930C (en) | 2005-09-07 |
CA2407862A1 (en) | 2001-12-06 |
US20030166946A1 (en) | 2003-09-04 |
CN1430604A (en) | 2003-07-16 |
JP2003535077A (en) | 2003-11-25 |
AR036000A1 (en) | 2004-08-04 |
IL152580A0 (en) | 2003-05-29 |
US6743926B2 (en) | 2004-06-01 |
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