IL130971A0 - Gemcitabine derivatives - Google Patents

Gemcitabine derivatives

Info

Publication number
IL130971A0
IL130971A0 IL13097198A IL13097198A IL130971A0 IL 130971 A0 IL130971 A0 IL 130971A0 IL 13097198 A IL13097198 A IL 13097198A IL 13097198 A IL13097198 A IL 13097198A IL 130971 A0 IL130971 A0 IL 130971A0
Authority
IL
Israel
Prior art keywords
gemcitabine derivatives
gemcitabine
derivatives
Prior art date
Application number
IL13097198A
Original Assignee
Norsk Hydro As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Norsk Hydro As filed Critical Norsk Hydro As
Priority claimed from PCT/NO1998/000020 external-priority patent/WO1998032762A1/en
Publication of IL130971A0 publication Critical patent/IL130971A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
IL13097198A 1997-01-24 1998-01-23 Gemcitabine derivatives IL130971A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9701427A GB2321454A (en) 1997-01-24 1997-01-24 Gemcitabine esters and amides
PCT/NO1998/000020 WO1998032762A1 (en) 1997-01-24 1998-01-23 Gemcitabine derivatives

Publications (1)

Publication Number Publication Date
IL130971A0 true IL130971A0 (en) 2001-01-28

Family

ID=10806509

Family Applications (1)

Application Number Title Priority Date Filing Date
IL13097198A IL130971A0 (en) 1997-01-24 1998-01-23 Gemcitabine derivatives

Country Status (7)

Country Link
CZ (1) CZ293245B6 (en)
ES (1) ES2196528T3 (en)
GB (1) GB2321454A (en)
IL (1) IL130971A0 (en)
RU (1) RU2194711C2 (en)
TW (1) TW458981B (en)
ZA (1) ZA98576B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0420722D0 (en) * 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
BRPI0519117A2 (en) * 2004-12-17 2008-12-23 Lilly Co Eli compound, pharmaceutical composition, method for treating susceptible neoplasms in a mammal, and use of a compound
WO2009128805A1 (en) * 2008-04-17 2009-10-22 The Johns Hopkins University On01910. na enhances chemotherapeutic agent activity in drug-resistant tumors
JP6420247B2 (en) 2012-11-13 2018-11-07 ボーイエン セラピューティクス,インコーポレイティド Gemcitabine prodrug and use thereof
CN110713502A (en) * 2019-11-29 2020-01-21 南京科技职业学院 Synthesis method of gemcitabine impurity

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA891076B (en) * 1988-02-16 1990-10-31 Lilly Co Eli 2',3'-dideoxy-2',2'-difluoronucleosides
YU43193A (en) * 1992-06-22 1997-01-08 Eli Lilly And Company 2'-DEOXY-2 ', 2'-DIFLUORO (4-SUBSTITUTED) PYRIMIDINE NUCLEOSIDS OF ANTIVIRUS AND ANTICANCEROGENIC ACTIVITY AND INTERMEDIATES

Also Published As

Publication number Publication date
GB9701427D0 (en) 1997-03-12
CZ293245B6 (en) 2004-03-17
GB2321454A (en) 1998-07-29
TW458981B (en) 2001-10-11
CZ247999A3 (en) 1999-12-15
ZA98576B (en) 1998-07-23
RU2194711C2 (en) 2002-12-20
ES2196528T3 (en) 2003-12-16

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees