HUP0102902A3 - Cyclic somatostatin analogs, process for production thereof and their use - Google Patents
Cyclic somatostatin analogs, process for production thereof and their useInfo
- Publication number
- HUP0102902A3 HUP0102902A3 HU0102902A HUP0102902A HUP0102902A3 HU P0102902 A3 HUP0102902 A3 HU P0102902A3 HU 0102902 A HU0102902 A HU 0102902A HU P0102902 A HUP0102902 A HU P0102902A HU P0102902 A3 HUP0102902 A3 HU P0102902A3
- Authority
- HU
- Hungary
- Prior art keywords
- production
- somatostatin analogs
- cyclic somatostatin
- cyclic
- analogs
- Prior art date
Links
- NHXLMOGPVYXJNR-ATOGVRKGSA-N somatostatin Chemical class C([C@H]1C(=O)N[C@H](C(N[C@@H](CO)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N1)[C@@H](C)O)NC(=O)CNC(=O)[C@H](C)N)C(O)=O)=O)[C@H](O)C)C1=CC=CC=C1 NHXLMOGPVYXJNR-ATOGVRKGSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8950398P | 1998-06-16 | 1998-06-16 | |
| US9818198A | 1998-06-16 | 1998-06-16 | |
| PCT/US1999/013304 WO1999065942A1 (en) | 1998-06-16 | 1999-06-11 | Cyclic somatostatin analogs |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUP0102902A2 HUP0102902A2 (hu) | 2002-01-28 |
| HUP0102902A3 true HUP0102902A3 (en) | 2002-02-28 |
Family
ID=26780645
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0102902A HUP0102902A3 (en) | 1998-06-16 | 1999-06-11 | Cyclic somatostatin analogs, process for production thereof and their use |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP1086131A1 (hu) |
| JP (1) | JP2002518409A (hu) |
| CN (1) | CN1200000C (hu) |
| AR (1) | AR021161A1 (hu) |
| AU (1) | AU745493B2 (hu) |
| CA (1) | CA2335184A1 (hu) |
| HU (1) | HUP0102902A3 (hu) |
| NO (1) | NO20006320L (hu) |
| PL (1) | PL345037A1 (hu) |
| RU (1) | RU2242481C2 (hu) |
| TW (3) | TWI242441B (hu) |
| WO (1) | WO1999065942A1 (hu) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL139835A (en) | 1998-06-12 | 2005-11-20 | Sod Conseils Rech Applic | Imidazolyl derivatives and their use as somatostatin receptor ligands |
| FR2796945B1 (fr) * | 1999-07-30 | 2002-06-28 | Sod Conseils Rech Applic | Nouveaux derives d'hydantoines, de thiohydantoines, de pyrimidinediones et de thioxopyrimidinones, leurs procedes de preparation et leur application a titre de medicaments |
| IL154222A0 (en) * | 2000-08-01 | 2003-07-31 | Sod Conseils Rech Applic | Imidazolyl derivatives |
| WO2004071448A2 (en) * | 2003-02-12 | 2004-08-26 | Transtech Pharma Inc. | Substituted azole derivatives as inhibitors of protein tyrosine phosphatases |
| WO2006063465A1 (en) * | 2004-12-15 | 2006-06-22 | Diamedica Inc. | Treatment of insulin resistance by modulating somatostatin using somatostatin receptor antagonists |
| CN101341129B (zh) * | 2005-12-14 | 2011-12-14 | 布里斯托尔-迈尔斯斯奎布公司 | 作为因子xia抑制剂的芳基丙酰胺，芳基丙烯酰胺，芳基丙炔酰胺，或芳基甲基脲类似物 |
| JP5225098B2 (ja) | 2005-12-14 | 2013-07-03 | ブリストル−マイヤーズ スクイブ カンパニー | 第ＸＩａ因子インヒビターとしてのアリールプロピオンアミド、アリールアクリルアミド、アリールプロピンアミド、またはアリールメチルウレアアナログ |
| AU2009296267B2 (en) | 2008-09-26 | 2013-10-31 | Ambrx, Inc. | Non-natural amino acid replication-dependent microorganisms and vaccines |
| EP2168983A1 (fr) | 2008-09-30 | 2010-03-31 | Ipsen Pharma | Nouveaux composés octapeptidiques et leur utilisation thérapeutique |
| EP2351743A4 (en) * | 2008-10-27 | 2012-05-09 | Takeda Pharmaceutical | BICYCLIC CONNECTION |
| AU2017217271C1 (en) * | 2016-02-09 | 2021-08-05 | Cdrd Ventures Inc. | Somatostatin receptor antagonist compounds and methods of using the same |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5770687A (en) * | 1995-06-07 | 1998-06-23 | Peptor Limited | Comformationally constrained backbone cyclized somatostatin analogs |
| US6673927B2 (en) * | 1996-02-16 | 2004-01-06 | Societe De Conseils De Recherches Et D'applications Scientifiques, S.A.S. | Farnesyl transferase inhibitors |
-
1999
- 1999-06-11 WO PCT/US1999/013304 patent/WO1999065942A1/en active IP Right Grant
- 1999-06-11 RU RU2001101530/04A patent/RU2242481C2/ru not_active IP Right Cessation
- 1999-06-11 AU AU48223/99A patent/AU745493B2/en not_active Ceased
- 1999-06-11 CN CNB998075027A patent/CN1200000C/zh not_active Expired - Fee Related
- 1999-06-11 JP JP2000554767A patent/JP2002518409A/ja active Pending
- 1999-06-11 PL PL99345037A patent/PL345037A1/xx not_active Application Discontinuation
- 1999-06-11 EP EP99931793A patent/EP1086131A1/en not_active Withdrawn
- 1999-06-11 CA CA002335184A patent/CA2335184A1/en not_active Abandoned
- 1999-06-11 HU HU0102902A patent/HUP0102902A3/hu unknown
- 1999-06-15 AR ARP990102857A patent/AR021161A1/es unknown
- 1999-06-15 TW TW091115003A patent/TWI242441B/zh active
- 1999-06-15 TW TW093100348A patent/TWI242442B/zh active
- 1999-06-15 TW TW088110016A patent/TW527361B/zh not_active IP Right Cessation
-
2000
- 2000-12-12 NO NO20006320A patent/NO20006320L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| TW527361B (en) | 2003-04-11 |
| TWI242441B (en) | 2005-11-01 |
| NO20006320L (no) | 2001-02-12 |
| WO1999065942A8 (en) | 2000-02-17 |
| NO20006320D0 (no) | 2000-12-12 |
| HUP0102902A2 (hu) | 2002-01-28 |
| AU4822399A (en) | 2000-01-05 |
| EP1086131A1 (en) | 2001-03-28 |
| WO1999065942A1 (en) | 1999-12-23 |
| TW200410986A (en) | 2004-07-01 |
| AU745493B2 (en) | 2002-03-21 |
| PL345037A1 (en) | 2001-11-19 |
| TWI242442B (en) | 2005-11-01 |
| JP2002518409A (ja) | 2002-06-25 |
| CN1305496A (zh) | 2001-07-25 |
| CN1200000C (zh) | 2005-05-04 |
| AR021161A1 (es) | 2002-07-03 |
| CA2335184A1 (en) | 1999-12-23 |
| RU2242481C2 (ru) | 2004-12-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD9A | Lapse of provisional protection due to non-payment of fees |