HU9200432D0 - Chemical process - Google Patents
Chemical processInfo
- Publication number
- HU9200432D0 HU9200432D0 HU9200432A HU9200432A HU9200432D0 HU 9200432 D0 HU9200432 D0 HU 9200432D0 HU 9200432 A HU9200432 A HU 9200432A HU 9200432 A HU9200432 A HU 9200432A HU 9200432 D0 HU9200432 D0 HU 9200432D0
- Authority
- HU
- Hungary
- Prior art keywords
- chemical process
- chemical
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU9200432A HUT64064A (en) | 1992-02-13 | 1992-02-13 | Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient |
MX9300779A MX9300779A (es) | 1992-02-13 | 1993-02-12 | 3-(1h-tetrazol-5-y1)-4h-pyrido[1,2-a]pirimidina-4-onas composiciones farmaceuticas que las contienen y su preparacion de las mismas |
SI19939300075A SI9300075A (en) | 1992-02-13 | 1993-02-12 | 3-(1h-tetrazol-5-yl)-4h-pyrido(1,2a)pyrimidin-4-ones, pharmaceutical preparations comprising the same and process pro their preparing |
IL104706A IL104706A0 (en) | 1992-02-13 | 1993-02-12 | 3-(1h-tetrazol-5-yl)-4h-pyrido(1,2-a)pyrimidine-4-ones and process for the preparation thereof |
AU35737/93A AU3573793A (en) | 1992-02-13 | 1993-02-12 | 3-(1H-tetrazol-5-yl)-4H-pyrido(1,2-a)pyrimidine-4-ones pharmaceutical compositions containing the same and the preparation thereof |
PCT/HU1993/000009 WO1993016076A1 (en) | 1992-02-13 | 1993-02-12 | 3-(1h^_-tetrazol-5-yl)-4h^_-pyrido[1,2-a^_]pyrimidine-4-ones, pharmaceutical compositions containing the same and the preparation thereof |
CN93102959.7A CN1080289A (zh) | 1992-02-13 | 1993-02-13 | 3-(1H-四唑-5-基)-4H-吡啶并[1,2-a]嘧啶-4-酮,含有该化合物的药物组合物及其制备 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU9200432A HUT64064A (en) | 1992-02-13 | 1992-02-13 | Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient |
Publications (2)
Publication Number | Publication Date |
---|---|
HU9200432D0 true HU9200432D0 (en) | 1992-04-28 |
HUT64064A HUT64064A (en) | 1993-11-29 |
Family
ID=10981335
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU9200432A HUT64064A (en) | 1992-02-13 | 1992-02-13 | Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient |
Country Status (7)
Country | Link |
---|---|
CN (1) | CN1080289A (hu) |
AU (1) | AU3573793A (hu) |
HU (1) | HUT64064A (hu) |
IL (1) | IL104706A0 (hu) |
MX (1) | MX9300779A (hu) |
SI (1) | SI9300075A (hu) |
WO (1) | WO1993016076A1 (hu) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HU209793B (en) * | 1990-09-25 | 1994-11-28 | Chinoin Gyogyszer Es Vegyeszet | Process for the production of pyrido[1,2-a]pyrimidine-derivatives and pharmaceutical compositions containing the same |
ITMI20011764A1 (it) * | 2001-08-10 | 2003-02-10 | Dinamite Dipharma Spa | Metodo per l'ottenimento del pemirolast ad elevata purezza |
ES2440217T3 (es) * | 2002-10-04 | 2014-01-28 | Prana Biotechnology Limited | Compuestos neurológicamente activos |
WO2007093184A2 (en) * | 2006-02-13 | 2007-08-23 | Astion Pharma A/S | Treatment of mmp-mediated dermatological diseases with pemirolast |
EP1818058A3 (en) * | 2006-02-13 | 2007-11-07 | Astion Pharma A/S | Treatment of mmp-mediated dermatological diseases with pemirolast |
ES2486715T3 (es) | 2009-06-29 | 2014-08-19 | Incyte Corporation | Pirimidinonas como inhibidores de PI3K |
US8759359B2 (en) | 2009-12-18 | 2014-06-24 | Incyte Corporation | Substituted heteroaryl fused derivatives as PI3K inhibitors |
CA2796311A1 (en) | 2010-04-14 | 2011-10-20 | Incyte Corporation | Fused derivatives as pi3k.delta. inhibitors |
US9062055B2 (en) | 2010-06-21 | 2015-06-23 | Incyte Corporation | Fused pyrrole derivatives as PI3K inhibitors |
ES2764848T3 (es) | 2010-12-20 | 2020-06-04 | Incyte Holdings Corp | N-(1-(fenilo sustituido)etilo)-9H-purina-6-aminas como inhibidores de PI3K |
US9108984B2 (en) | 2011-03-14 | 2015-08-18 | Incyte Corporation | Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors |
US9126948B2 (en) | 2011-03-25 | 2015-09-08 | Incyte Holdings Corporation | Pyrimidine-4,6-diamine derivatives as PI3K inhibitors |
EP2751109B1 (en) | 2011-09-02 | 2016-11-30 | Incyte Holdings Corporation | Heterocyclylamines as pi3k inhibitors |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
EP3262046B1 (en) | 2015-02-27 | 2020-11-04 | Incyte Corporation | Salts of pi3k inhibitor and processes for their preparation |
WO2016183060A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
WO2016183063A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Crystalline forms of a pi3k inhibitor |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2044796C (en) * | 1990-06-21 | 2001-10-16 | Atsunori Sano | Process for producing pyrido[1,2-a] pyrimidine derivative |
-
1992
- 1992-02-13 HU HU9200432A patent/HUT64064A/hu unknown
-
1993
- 1993-02-12 WO PCT/HU1993/000009 patent/WO1993016076A1/en active Application Filing
- 1993-02-12 MX MX9300779A patent/MX9300779A/es unknown
- 1993-02-12 IL IL104706A patent/IL104706A0/xx unknown
- 1993-02-12 AU AU35737/93A patent/AU3573793A/en not_active Withdrawn
- 1993-02-12 SI SI19939300075A patent/SI9300075A/sl unknown
- 1993-02-13 CN CN93102959.7A patent/CN1080289A/zh active Pending
Also Published As
Publication number | Publication date |
---|---|
IL104706A0 (en) | 1993-06-10 |
MX9300779A (es) | 1993-09-30 |
WO1993016076A1 (en) | 1993-08-19 |
AU3573793A (en) | 1993-09-03 |
HUT64064A (en) | 1993-11-29 |
CN1080289A (zh) | 1994-01-05 |
SI9300075A (en) | 1993-09-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
DFA9 | Temporary protection cancelled due to abandonment | ||
DFC4 | Cancellation of temporary protection due to refusal |