HU196064B - Process for production of 1,3,4-tiadiasole-derivatives and medical preparatives containing such compositions - Google Patents

Process for production of 1,3,4-tiadiasole-derivatives and medical preparatives containing such compositions Download PDF

Info

Publication number
HU196064B
HU196064B HU854098A HU409885A HU196064B HU 196064 B HU196064 B HU 196064B HU 854098 A HU854098 A HU 854098A HU 409885 A HU409885 A HU 409885A HU 196064 B HU196064 B HU 196064B
Authority
HU
Hungary
Prior art keywords
formula
compound
thiadiazole
phenoxy
alkyl
Prior art date
Application number
HU854098A
Other languages
English (en)
Hungarian (hu)
Other versions
HUT44525A (en
Inventor
Helmut Schickaneder
Rolf Herter
Kurt Wegner
Istvan Szelenyi
Stefan Postius
Hennig K Ahrens
Walter Schunack
Original Assignee
Heumann Ludwig & Co Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Heumann Ludwig & Co Gmbh filed Critical Heumann Ludwig & Co Gmbh
Publication of HUT44525A publication Critical patent/HUT44525A/hu
Publication of HU196064B publication Critical patent/HU196064B/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/121,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/1251,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • C07D285/135Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU854098A 1985-04-12 1985-10-24 Process for production of 1,3,4-tiadiasole-derivatives and medical preparatives containing such compositions HU196064B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19853513184 DE3513184A1 (de) 1985-04-12 1985-04-12 1,3,4-thiadiazolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (2)

Publication Number Publication Date
HUT44525A HUT44525A (en) 1988-03-28
HU196064B true HU196064B (en) 1988-09-28

Family

ID=6267864

Family Applications (1)

Application Number Title Priority Date Filing Date
HU854098A HU196064B (en) 1985-04-12 1985-10-24 Process for production of 1,3,4-tiadiasole-derivatives and medical preparatives containing such compositions

Country Status (14)

Country Link
US (1) US4738960A (US08080257-20111220-C00005.png)
EP (1) EP0197189A3 (US08080257-20111220-C00005.png)
JP (1) JPS61238782A (US08080257-20111220-C00005.png)
KR (1) KR860008172A (US08080257-20111220-C00005.png)
AU (1) AU578766B2 (US08080257-20111220-C00005.png)
DE (1) DE3513184A1 (US08080257-20111220-C00005.png)
DK (1) DK501385A (US08080257-20111220-C00005.png)
ES (1) ES8700245A1 (US08080257-20111220-C00005.png)
GR (1) GR852573B (US08080257-20111220-C00005.png)
HU (1) HU196064B (US08080257-20111220-C00005.png)
IL (1) IL77097A0 (US08080257-20111220-C00005.png)
NZ (1) NZ214231A (US08080257-20111220-C00005.png)
PT (1) PT81409B (US08080257-20111220-C00005.png)
ZA (1) ZA858841B (US08080257-20111220-C00005.png)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR228941A1 (es) * 1978-04-26 1983-05-13 Glaxo Group Ltd Procedimiento para preparar nuevos derivados de 3,5-diamino-1,2,4-triazol que son activos contra receptores histaminicos
JPS60255756A (ja) * 1984-06-01 1985-12-17 Ikeda Mohandou:Kk アミノアルキルフエノキシ誘導体
CA1275097A (en) * 1984-10-02 1990-10-09 Fujio Nohara Pyridyloxy derivatives
EP4196793A1 (en) 2020-08-11 2023-06-21 Université de Strasbourg H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3118126A1 (de) * 1981-05-07 1982-12-02 Bayer Ag, 5090 Leverkusen Sulfenamide zur verwendung in arzneimitteln
US4600779A (en) * 1982-03-29 1986-07-15 Bristol-Myers Company Substituted 3,4-diamino-1,2,5-thiadiazoles having histamine H2 -receptor antagonist activity
US4578471A (en) * 1982-03-29 1986-03-25 Bristol-Myers Company Substituted amino alkyl pyridyl ethanediimidamides
US4440933A (en) * 1983-03-16 1984-04-03 Bristol-Myers Company Process for preparing 1,2,5-thiadiazoles
JPS59196879A (ja) * 1983-04-08 1984-11-08 Wakamoto Pharmaceut Co Ltd 新規な1,3,4−チアジアゾ−ル誘導体
JPS6067474A (ja) * 1983-09-24 1985-04-17 Wakamoto Pharmaceut Co Ltd 新規な1,3,4−チアジアゾ−ル誘導体及びそれを有効成分とする抗潰瘍剤
DE3341750A1 (de) * 1983-11-18 1985-05-30 Ludwig Heumann & Co GmbH, 8500 Nürnberg 1,2,4-triazolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
JPS60255756A (ja) * 1984-06-01 1985-12-17 Ikeda Mohandou:Kk アミノアルキルフエノキシ誘導体
DE3441086A1 (de) * 1984-11-09 1986-05-15 Ludwig Heumann & Co GmbH, 8500 Nürnberg 3,4-diazolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
DK501385A (da) 1986-10-13
US4738960A (en) 1988-04-19
HUT44525A (en) 1988-03-28
PT81409B (de) 1987-04-13
GR852573B (US08080257-20111220-C00005.png) 1986-08-13
JPS61238782A (ja) 1986-10-24
ES8700245A1 (es) 1986-10-16
ES549378A0 (es) 1986-10-16
AU5024185A (en) 1986-10-16
AU578766B2 (en) 1988-11-03
PT81409A (de) 1985-11-01
EP0197189A3 (de) 1987-05-27
NZ214231A (en) 1988-07-28
DK501385D0 (da) 1985-10-31
KR860008172A (ko) 1986-11-12
EP0197189A2 (de) 1986-10-15
ZA858841B (en) 1986-07-30
IL77097A0 (en) 1986-04-29
DE3513184A1 (de) 1986-10-16

Similar Documents

Publication Publication Date Title
EP0040696B1 (en) Aminothiadiazoles as gastric secretion inhibitors
EP0684945B1 (en) Pyrazole- or isoxazole-substituted alkyl amide acat inhibitors
KR860001818B1 (ko) 2-아미노-5-하이드록시-4-메틸 피리미딘 유도체의 제조 방법
CA1190224A (en) Derivatives of 1,2-diamino-cyclobutene-3,4-dione as potent histamine h.sub.2-antagonists
RU2348620C2 (ru) Производные тиазола в качестве модуляторов каннабиноидного рецептора
EP0161841B1 (en) 2-(n-substituteguanidino)-4-hetero-arylthiazole antiulcer agents
CA2168443A1 (en) Piperazine derivatives as .alpha.1a-adrenergic receptor antagonists
US4200578A (en) Thiazole derivatives
CS241072B2 (en) Method of 3-/(amino or subst,amino/)-4-/(subst.amino/)-1,2,5-thiadizoles production
US5100910A (en) Aryl substituted tetrazole derivatives, and application thereof in therapeutics
US4840967A (en) Carbamate or urea derivatives, their preparation and pharmaceutical compositions comprising them
HU196064B (en) Process for production of 1,3,4-tiadiasole-derivatives and medical preparatives containing such compositions
US4968808A (en) Process for the preparation of nitroethene derivatives
US4158013A (en) N-Cyano-N'-alkynyl-N"-2-mercaptoethylguanidines
US4378357A (en) Novel heterocyclic compounds
JPS6044307B2 (ja) 新規のo−アルキル化オキシムおよび医薬としてのその用途
EP0073971B1 (en) Thiadiazole oxides as gastric antisecretory agents
EP0081955B1 (en) Benzo-fused heterocyclic compounds
US4727081A (en) 3,4-Diazole derivatives and pharmaceutical preparations containing these compounds
EP0185368B1 (en) Aminobenzamide derivatives
HU202506B (en) Process for producing benzoxazolone derivatives
US4975462A (en) Antiarthritic α-arylcarbamoyl cyanoacetic acid derivatives
HU188742B (en) Process for producing substituted 3,4-diamni-1,2,5-thiadiazoles and pharmaceutical compositions of hystamine-h2-receptor antagonistic aczivity containing them as active agents
CA1322755C (en) Acetamide compounds
US4590192A (en) Benzisothiazoles, their pharmaceutical compositions, and method of use

Legal Events

Date Code Title Description
HU90 Patent valid on 900628
HMM4 Cancellation of final prot. due to non-payment of fee