HRP20110666T1 - Uporaba 4-ciklopropilmetoksi-n-(3,5-diklor-1-oksidopiridin-4-il)-5-(metoksi)piridin-2-karboksamida u liječenju motoričkih poremećaja povezanih s parkinsonovom bolesti - Google Patents

Uporaba 4-ciklopropilmetoksi-n-(3,5-diklor-1-oksidopiridin-4-il)-5-(metoksi)piridin-2-karboksamida u liječenju motoričkih poremećaja povezanih s parkinsonovom bolesti Download PDF

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Publication number
HRP20110666T1
HRP20110666T1 HR20110666T HRP20110666T HRP20110666T1 HR P20110666 T1 HRP20110666 T1 HR P20110666T1 HR 20110666 T HR20110666 T HR 20110666T HR P20110666 T HRP20110666 T HR P20110666T HR P20110666 T1 HRP20110666 T1 HR P20110666T1
Authority
HR
Croatia
Prior art keywords
oxidopyridin
carboxamide
use according
disorders
cyclopropylmethoxy
Prior art date
Application number
HR20110666T
Other languages
English (en)
Croatian (hr)
Inventor
Delay-Goyet Philippe
Delgorge Claire
Menet Christine
Poughon Gilles
Ravinet-Trillou Christine
Original Assignee
Sanofi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi filed Critical Sanofi
Publication of HRP20110666T1 publication Critical patent/HRP20110666T1/hr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
HR20110666T 2007-04-19 2008-04-16 Uporaba 4-ciklopropilmetoksi-n-(3,5-diklor-1-oksidopiridin-4-il)-5-(metoksi)piridin-2-karboksamida u liječenju motoričkih poremećaja povezanih s parkinsonovom bolesti HRP20110666T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0702853A FR2915100B1 (fr) 2007-04-19 2007-04-19 Utilisation du 4-cyclopropylmethoxy-n-(3,5-dichloro-1-oxydo- pyridin-4-yl)-5-(methoxy)pyridine-2-carboxalide pour le traitement des desordres moteurs lies a la maladie de parkinson
PCT/FR2008/000534 WO2008145841A1 (fr) 2007-04-19 2008-04-16 Utilisation du 4-cyclopropylmethoxy-n-(3,5-dichloro-1 -oxydo- pyridin-4-yl)-5-(methoxy)pyridine-2-carboxamide pour le traitement des desordres moteurs lies a la maladie de parkinson

Publications (1)

Publication Number Publication Date
HRP20110666T1 true HRP20110666T1 (hr) 2011-10-31

Family

ID=38712405

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20110666T HRP20110666T1 (hr) 2007-04-19 2008-04-16 Uporaba 4-ciklopropilmetoksi-n-(3,5-diklor-1-oksidopiridin-4-il)-5-(metoksi)piridin-2-karboksamida u liječenju motoričkih poremećaja povezanih s parkinsonovom bolesti

Country Status (33)

Country Link
US (1) US20100130554A1 (Direct)
EP (1) EP2146714B1 (Direct)
JP (1) JP5386478B2 (Direct)
KR (2) KR101503942B1 (Direct)
CN (1) CN101663035B (Direct)
AR (1) AR066108A1 (Direct)
AT (1) ATE513548T1 (Direct)
AU (1) AU2008257322B2 (Direct)
BR (1) BRPI0810444A2 (Direct)
CA (1) CA2684174C (Direct)
CL (1) CL2008001136A1 (Direct)
CY (1) CY1111840T1 (Direct)
DK (1) DK2146714T3 (Direct)
EA (1) EA019194B1 (Direct)
ES (1) ES2367408T3 (Direct)
FR (1) FR2915100B1 (Direct)
HR (1) HRP20110666T1 (Direct)
IL (1) IL201448A (Direct)
JO (1) JO2678B1 (Direct)
MA (1) MA31367B1 (Direct)
ME (1) ME00935B (Direct)
MX (1) MX2009011284A (Direct)
MY (1) MY148092A (Direct)
NZ (1) NZ580482A (Direct)
PA (1) PA8776801A1 (Direct)
PL (1) PL2146714T3 (Direct)
PT (1) PT2146714E (Direct)
RS (1) RS51869B (Direct)
SI (1) SI2146714T1 (Direct)
TW (1) TWI439269B (Direct)
UY (1) UY31035A1 (Direct)
WO (1) WO2008145841A1 (Direct)
ZA (1) ZA200907251B (Direct)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2621894C2 (ru) * 2012-11-28 2017-06-08 Санофи Способ получения новых кристаллических форм-4(циклопропилметокси)-n-(3, 5-дихлор-1-оксидопиридин-4-ил)-5-метоксипиридин-2-карбоксамида и его кристаллические формы
US9624100B2 (en) 2014-06-12 2017-04-18 Apple Inc. Micro pick up array pivot mount with integrated strain sensing elements
WO2025080415A1 (en) * 2023-10-12 2025-04-17 Alto Neuroscience, Inc. Treatment of neuropsychiatric disorders with tilivapram
WO2025079694A1 (ja) * 2023-10-12 2025-04-17 株式会社 メドレックス 経皮吸収組成物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4193926A (en) * 1974-03-20 1980-03-18 Schering Aktiengesellschaft 4-(Polyalkoxy phenyl)-2-pyrrolidones
EP0711282B1 (en) * 1993-07-28 2002-06-05 Aventis Pharma Limited Compounds as pde iv and tnf inhibitors
US6177077B1 (en) * 1999-02-24 2001-01-23 Edward L. Tobinick TNT inhibitors for the treatment of neurological disorders
EP1244649B1 (en) * 1999-12-23 2005-03-02 Icos Corporation Cyclic amp-specific phosphodiesterase inhibitors
CA2439691A1 (en) * 2001-03-02 2002-09-12 Bristol-Myers Squibb Company Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-amp associated disorders
WO2004005258A1 (en) * 2002-07-02 2004-01-15 Merck Frosst Canada & Co. Di-aryl-substituted-ethane pyridone pde4 inhibitors
DE602004032522D1 (de) * 2003-03-12 2011-06-16 Celgene Corp Mit n-alkylhydroxamsäuren substituierte isoindolylverbindungen und deren pharmazeutische verwendung
CA2611562A1 (en) * 2005-06-10 2006-12-21 Memory Pharmaceuticals Corporation Trisubstituted amines as phosphodiesterase 4 inhibitors
US20070021451A1 (en) * 2005-07-20 2007-01-25 Hamamatsu University School Of Medicine Method for preventing or treating neurologic damage after spinal cord injury

Also Published As

Publication number Publication date
FR2915100A1 (fr) 2008-10-24
ZA200907251B (en) 2011-04-28
US20100130554A1 (en) 2010-05-27
SI2146714T1 (sl) 2011-10-28
BRPI0810444A2 (pt) 2016-05-31
KR20090130059A (ko) 2009-12-17
JO2678B1 (en) 2013-03-03
HK1141725A1 (en) 2010-11-19
PA8776801A1 (es) 2008-11-19
ATE513548T1 (de) 2011-07-15
RS51869B (sr) 2012-02-29
EA019194B1 (ru) 2014-01-30
CL2008001136A1 (es) 2009-01-16
JP5386478B2 (ja) 2014-01-15
EP2146714B1 (fr) 2011-06-22
PL2146714T3 (pl) 2011-10-31
JP2010524906A (ja) 2010-07-22
ME00935B (me) 2012-06-20
TW200911247A (en) 2009-03-16
CA2684174C (fr) 2014-02-25
KR20150004885A (ko) 2015-01-13
TWI439269B (zh) 2014-06-01
MX2009011284A (es) 2009-11-02
WO2008145841A1 (fr) 2008-12-04
CA2684174A1 (fr) 2008-12-04
CY1111840T1 (el) 2015-10-07
AU2008257322B2 (en) 2013-06-13
AU2008257322A1 (en) 2008-12-04
UY31035A1 (es) 2008-11-28
DK2146714T3 (da) 2011-10-10
IL201448A0 (en) 2010-05-31
MA31367B1 (fr) 2010-05-03
CN101663035A (zh) 2010-03-03
IL201448A (en) 2014-08-31
CN101663035B (zh) 2012-06-20
EP2146714A1 (fr) 2010-01-27
ES2367408T3 (es) 2011-11-03
NZ580482A (en) 2011-10-28
PT2146714E (pt) 2011-09-02
FR2915100B1 (fr) 2009-06-05
AR066108A1 (es) 2009-07-22
EA200970970A1 (ru) 2010-02-26
KR101503942B1 (ko) 2015-03-18
MY148092A (en) 2013-02-28

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