HK1036617B - 用作藥物化合物的naalad酶抑制劑和組合物 - Google Patents

用作藥物化合物的naalad酶抑制劑和組合物 Download PDF

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Publication number
HK1036617B
HK1036617B HK01107357.1A HK01107357A HK1036617B HK 1036617 B HK1036617 B HK 1036617B HK 01107357 A HK01107357 A HK 01107357A HK 1036617 B HK1036617 B HK 1036617B
Authority
HK
Hong Kong
Prior art keywords
formula
compound
moiety
pentanedioic acid
acid
Prior art date
Application number
HK01107357.1A
Other languages
German (de)
English (en)
French (fr)
Other versions
HK1036617A1 (zh
Inventor
F. Jackson Paul
M. Maclin Keith
Wang Eric
S. Slusher Barbara
S. Lapidus Rena
Majer Pavel
Original Assignee
Eisai Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/110,262 external-priority patent/US6395718B1/en
Priority claimed from US09/228,391 external-priority patent/US6265609B1/en
Application filed by Eisai Inc. filed Critical Eisai Inc.
Priority claimed from PCT/US1999/015128 external-priority patent/WO2000001668A2/en
Publication of HK1036617A1 publication Critical patent/HK1036617A1/zh
Publication of HK1036617B publication Critical patent/HK1036617B/zh

Links

HK01107357.1A 1998-07-06 1999-07-02 用作藥物化合物的naalad酶抑制劑和組合物 HK1036617B (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US11018698A 1998-07-06 1998-07-06
US09/110,262 US6395718B1 (en) 1998-07-06 1998-07-06 Pharmaceutical compositions and methods of inhibiting angiogenesis using naaladase inhibitors
US09/110,186 1998-07-06
US09/110,262 1998-07-06
US09/228,391 US6265609B1 (en) 1998-07-06 1999-01-12 Thio-substituted pentanedioic acid derivatives
US09/228,391 1999-01-12
PCT/US1999/015128 WO2000001668A2 (en) 1998-07-06 1999-07-02 Naaladase inhibitors useful as pharmaceutical compounds and compositions

Publications (2)

Publication Number Publication Date
HK1036617A1 HK1036617A1 (zh) 2002-01-11
HK1036617B true HK1036617B (zh) 2006-02-03

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