GT201500169A - THERAPEUTICALLY ACTIVE DERIVATIVES OF PIRAZOL-PYRIMIDINE - Google Patents

THERAPEUTICALLY ACTIVE DERIVATIVES OF PIRAZOL-PYRIMIDINE

Info

Publication number
GT201500169A
GT201500169A GT201500169A GT201500169A GT201500169A GT 201500169 A GT201500169 A GT 201500169A GT 201500169 A GT201500169 A GT 201500169A GT 201500169 A GT201500169 A GT 201500169A GT 201500169 A GT201500169 A GT 201500169A
Authority
GT
Guatemala
Prior art keywords
pyrimidine
pirazol
therapeutically active
active derivatives
human
Prior art date
Application number
GT201500169A
Other languages
Spanish (es)
Inventor
James Ford Daniel
Jeremy Franklin Richard
Ramrao Ghawalkar Anant
Huang Qiuya
Thomas Reuberson James
Vanderhoydonck Bart
Tracey Horsley Helen
Original Assignee
Ucb Biopharma Sprl
Katholieke Univ Leuven K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ucb Biopharma Sprl, Katholieke Univ Leuven K filed Critical Ucb Biopharma Sprl
Publication of GT201500169A publication Critical patent/GT201500169A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

UNA SERIE DE DERIVADOS DE PIRAZOL [3,4-D] PIRIMIDINA QUE SON SUSTITUIDOS EN LA POSICIÓN 4 POR UNA FRACCIÓN DIAZA MONOCÍCLICA, BICÍCLICA O ESPIROCÍCLICA, SON BENEFICIOSOS EN EL TRATAMIENTO Y/O PREVENCIÓN DE VARIAS DOLENCIAS HUMANAS, INCLUYENDO DESÓRDENES INFLAMATORIOS, AUTOINMUNES Y ONCOLÓGICOS; ENFERMEDADES VIRALES Y MALARIA; Y RECHAZO DE TRANSPLANTE DE ÓRGANOS Y CÉLULAS.A SERIES OF DERIVATIVES OF PIRAZOLE [3,4-D] PYRIMIDINE WHICH ARE REPLACED IN POSITION 4 BY A MONOCYCLIC, BICYCLIC OR SPIROCYCLIC DIAZA FRACTION, ARE BENEFICIAL IN THE TREATMENT AND / OR PREVENTION OF SEVERAL SELF-INFRINGED HUMAN INJURIES, INCLUDING INFLUENTIOUS HUMAN INCIDENTS AND ONCOLOGICALS; VIRAL DISEASES AND MALARIA; AND REJECTION OF TRANSPLANTATION OF ORGANS AND CELLS.

GT201500169A 2012-12-20 2015-06-19 THERAPEUTICALLY ACTIVE DERIVATIVES OF PIRAZOL-PYRIMIDINE GT201500169A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB1223021.5A GB201223021D0 (en) 2012-12-20 2012-12-20 Therapeutic agents

Publications (1)

Publication Number Publication Date
GT201500169A true GT201500169A (en) 2019-08-30

Family

ID=47682284

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201500169A GT201500169A (en) 2012-12-20 2015-06-19 THERAPEUTICALLY ACTIVE DERIVATIVES OF PIRAZOL-PYRIMIDINE

Country Status (4)

Country Link
EC (1) ECSP15031293A (en)
GB (1) GB201223021D0 (en)
GT (1) GT201500169A (en)
MA (1) MA38279B1 (en)

Also Published As

Publication number Publication date
ECSP15031293A (en) 2018-07-31
MA38279B1 (en) 2018-10-31
MA38279A1 (en) 2018-02-28
GB201223021D0 (en) 2013-02-06

Similar Documents

Publication Publication Date Title
UY36171A (en) BICYCLIC HETEROAROMATIC DERIVATIVES FUSED AS QUINASE INHIBITORS
CR20150379A (en) DERIVATIVES OF PIRAZOLO-PYRIMIDINE THERAPEUTICALLY ACTIVE
ECSP14013224A (en) SUBSTITUTED RINGED PYRIMIDINES AND USE OF THE SAME
PE20151157A1 (en) SUSTAINED RELEASE RUXOLITINIB DOSAGE FORMS
CL2016001629A1 (en) Tricyclic compounds as anticancer agents
CY1119840T1 (en) CYCLICALLY SUBSTITUTED SOURCES AND USE OF THESE
CO7081142A2 (en) Methods of treating retinal degeneration diseases
CU23874B1 (en) 4-ARIL-1,4-DIHIDRO-1,6-SUBSTITUTED NAFTIRIDINAMIDS AND THEIR USE
BR112012016866A2 (en) Thiazolo [5,4-d] pyrimidines and their use as agrochemicals.
ECSP12011692A (en) DERIVATIVES OF OXAZINE AND ITS USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS
CL2014002342A1 (en) Combined antibody therapy against human csf-1r and its uses.
BR112012020863A2 (en) rifaximin forms and uses thereof
ECSP12011716A (en) (HETEROARILMETIL) SUBSTITUTED THIOHYDANTOINS AS ANTI-CANCER DRUGS
CR20160454A (en) CHROMENE AND 1.1 a, 2.7b — TETRAHYDROCICLOPROPA [C] CHROME PIRIDOPIRAZINADIONAS NOVEDOSAS
PE20142457A1 (en) HETEROCICLIC COMPOUNDS AND THEIR USES
EP2601967A4 (en) Drug and method for the prophylaxis of hiv infection and for the prophylaxis and treatment of diseases caused by or associated with hiv, including aids
BR112016029632A2 (en) fused bicyclic heteroaromatic derivatives as kinase inhibitors
CL2017001454A1 (en) Methods for preparing compositions containing alkaloids and uses thereof
GT201500169A (en) THERAPEUTICALLY ACTIVE DERIVATIVES OF PIRAZOL-PYRIMIDINE
PE20150869A1 (en) TRIS- (HETERO) ARIL-PIRAZOLES AND ITS USE
WO2014025749A3 (en) Small molecule inhibitors of viral protein interactions with human t-rna
AR125919A2 (en) SUSTAINED-RELEASE RUXOLITINIB DOSAGE FORMS
ECSP15025357A (en) SUSTAINED RELEASE RUXOLITINIB DOSAGE FORMS
UA114825C2 (en) Therapeutically active pyrazolo-pyrimidine derivatives
CR20120083A (en) DERIVATIVES OF OXAZINE AND ITS USE IN THE TREATMENT OF NEUROLOGICAL DISORDERS