GT200600048A - PIRROLES REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING AND USE PROCESS. - Google Patents
PIRROLES REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING AND USE PROCESS.Info
- Publication number
- GT200600048A GT200600048A GT200600048A GT200600048A GT200600048A GT 200600048 A GT200600048 A GT 200600048A GT 200600048 A GT200600048 A GT 200600048A GT 200600048 A GT200600048 A GT 200600048A GT 200600048 A GT200600048 A GT 200600048A
- Authority
- GT
- Guatemala
- Prior art keywords
- compositions
- replaced
- contain
- pirroles
- manufacturing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyrrole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
PIRROLES SUSTITUIDOS, COMPOSICIONES QUE LOS CONTIENEN, PROCESO DE FABRICACIÓN Y UTILIZACIÓN. LA PRESENTE INVENCIÓN SE REFIERE PARTICULARMENTE A LA PREPARACIÓN DE PIRROLES SUSTITUIDOS, A LAS COMPOSICIONES QUE LOS CONTIENEN, A SU PROCESO DE PREPARACIÓN, Y A SU UTILIZACIÓN COMO MEDICAMENTO, EN PARTICULAR COMO AGENTES ANTICANCERÍGENOS.PIRROLES REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING AND USE PROCESS. THE PRESENT INVENTION REFERS IN PARTICULARLY TO THE PREPARATION OF REPLACED PIRROLS, TO THE COMPOSITIONS THAT CONTAIN THEM, TO THEIR PREPARATION PROCESS, AND TO ITS USE AS A MEDICINAL PRODUCT, IN PARTICULAR AS ANTI-BANKER AGENTS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0501354A FR2881742B1 (en) | 2005-02-10 | 2005-02-10 | SUBSTITUTED PYRROLES, COMPOSITIONS CONTAINING SAME, METHOD OF MANUFACTURE AND USE |
Publications (1)
Publication Number | Publication Date |
---|---|
GT200600048A true GT200600048A (en) | 2006-07-03 |
Family
ID=35478244
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT200600048A GT200600048A (en) | 2005-02-10 | 2006-02-08 | PIRROLES REPLACED, COMPOSITIONS THAT CONTAIN THEM, MANUFACTURING AND USE PROCESS. |
Country Status (36)
Country | Link |
---|---|
US (1) | US7592365B2 (en) |
EP (1) | EP1851198B1 (en) |
JP (1) | JP2008530061A (en) |
KR (1) | KR20070101317A (en) |
CN (1) | CN101115716A (en) |
AR (1) | AR052571A1 (en) |
AT (1) | ATE419234T1 (en) |
AU (1) | AU2006212106A1 (en) |
BR (1) | BRPI0606955A2 (en) |
CA (1) | CA2596822A1 (en) |
CR (1) | CR9231A (en) |
CY (1) | CY1108916T1 (en) |
DE (1) | DE602006004566D1 (en) |
DK (1) | DK1851198T3 (en) |
DO (1) | DOP2006000028A (en) |
EA (1) | EA013060B1 (en) |
ES (1) | ES2319926T3 (en) |
FR (1) | FR2881742B1 (en) |
GT (1) | GT200600048A (en) |
HR (1) | HRP20090158T1 (en) |
IL (1) | IL184488A0 (en) |
MA (1) | MA29248B1 (en) |
MX (1) | MX2007008789A (en) |
MY (1) | MY142082A (en) |
NO (1) | NO20074528L (en) |
PA (1) | PA8661601A1 (en) |
PE (1) | PE20061086A1 (en) |
PL (1) | PL1851198T3 (en) |
PT (1) | PT1851198E (en) |
RS (1) | RS50806B (en) |
SI (1) | SI1851198T1 (en) |
TN (1) | TNSN07241A1 (en) |
TW (1) | TW200640858A (en) |
UY (1) | UY29371A1 (en) |
WO (1) | WO2006084996A1 (en) |
ZA (1) | ZA200706157B (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2881426B1 (en) | 2005-02-03 | 2007-03-30 | Aventis Pharma Sa | SUBSTITUTED PYROLLES AND IMIDAZOLES, COMPOSITIONS CONTAINING THE SAME, PROCESS FOR FRABRICATION AND USE |
US7951941B2 (en) * | 2006-10-23 | 2011-05-31 | Lexicon Pharmaceuticals, Inc. | Process for preparing 5-alkyl-7H-pyrrolo[2,3-d] pyrimindine-2-ols |
TW201111385A (en) | 2009-08-27 | 2011-04-01 | Biocryst Pharm Inc | Heterocyclic compounds as janus kinase inhibitors |
US20120244141A1 (en) | 2010-09-28 | 2012-09-27 | Boehringer Ingelheim International Gmbh | Stratification of cancer patients for susceptibility to therapy with PTK2 inhibitors |
WO2020034988A1 (en) * | 2018-08-14 | 2020-02-20 | 江苏豪森药业集团有限公司 | Salt of apoptosis signal-regulating kinase 1 inhibitor and crystal form thereof |
WO2020113094A1 (en) | 2018-11-30 | 2020-06-04 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0107901D0 (en) * | 2001-03-29 | 2001-05-23 | Cyclacel Ltd | Anti-cancer compounds |
ES2307780T3 (en) * | 2001-09-21 | 2008-12-01 | Smithkline Beecham Corporation | CHEMICAL COMPOUNDS. |
JP2006515828A (en) | 2001-09-27 | 2006-06-08 | スミスクライン・ビーチャム・コーポレイション | Chemical compound |
US20040138269A1 (en) * | 2002-10-11 | 2004-07-15 | Sugen, Inc. | Substituted pyrroles as kinase inhibitors |
GB0229581D0 (en) * | 2002-12-19 | 2003-01-22 | Cyclacel Ltd | Use |
JP4808154B2 (en) * | 2003-03-13 | 2011-11-02 | バーテックス ファーマシューティカルズ インコーポレイテッド | Compositions useful as protein kinase inhibitors |
DE10354060A1 (en) * | 2003-11-19 | 2005-06-02 | Merck Patent Gmbh | pyrrole |
US7183285B2 (en) * | 2004-04-29 | 2007-02-27 | Pharmix Corp. | Compositions and treatments for inhibiting kinase and/or HMG-CoA reductase |
FR2881426B1 (en) | 2005-02-03 | 2007-03-30 | Aventis Pharma Sa | SUBSTITUTED PYROLLES AND IMIDAZOLES, COMPOSITIONS CONTAINING THE SAME, PROCESS FOR FRABRICATION AND USE |
-
2005
- 2005-02-10 FR FR0501354A patent/FR2881742B1/en not_active Expired - Fee Related
-
2006
- 2006-02-02 PE PE2006000135A patent/PE20061086A1/en not_active Application Discontinuation
- 2006-02-02 PA PA20068661601A patent/PA8661601A1/en unknown
- 2006-02-02 DO DO2006000028A patent/DOP2006000028A/en unknown
- 2006-02-03 MY MYPI20060441A patent/MY142082A/en unknown
- 2006-02-08 DE DE602006004566T patent/DE602006004566D1/en active Active
- 2006-02-08 ZA ZA200706157A patent/ZA200706157B/en unknown
- 2006-02-08 PT PT06709274T patent/PT1851198E/en unknown
- 2006-02-08 EP EP06709274A patent/EP1851198B1/en active Active
- 2006-02-08 GT GT200600048A patent/GT200600048A/en unknown
- 2006-02-08 AT AT06709274T patent/ATE419234T1/en active
- 2006-02-08 SI SI200630232T patent/SI1851198T1/en unknown
- 2006-02-08 AU AU2006212106A patent/AU2006212106A1/en not_active Withdrawn
- 2006-02-08 PL PL06709274T patent/PL1851198T3/en unknown
- 2006-02-08 EA EA200701688A patent/EA013060B1/en not_active IP Right Cessation
- 2006-02-08 ES ES06709274T patent/ES2319926T3/en active Active
- 2006-02-08 JP JP2007554598A patent/JP2008530061A/en active Pending
- 2006-02-08 RS RSP-2009/0128A patent/RS50806B/en unknown
- 2006-02-08 MX MX2007008789A patent/MX2007008789A/en active IP Right Grant
- 2006-02-08 AR ARP060100452A patent/AR052571A1/en unknown
- 2006-02-08 DK DK06709274T patent/DK1851198T3/en active
- 2006-02-08 BR BRPI0606955-0A patent/BRPI0606955A2/en not_active IP Right Cessation
- 2006-02-08 CA CA002596822A patent/CA2596822A1/en not_active Abandoned
- 2006-02-08 CN CNA2006800044573A patent/CN101115716A/en active Pending
- 2006-02-08 WO PCT/FR2006/000286 patent/WO2006084996A1/en active Application Filing
- 2006-02-08 KR KR1020077018321A patent/KR20070101317A/en not_active Application Discontinuation
- 2006-02-09 TW TW095104288A patent/TW200640858A/en unknown
- 2006-02-10 UY UY29371A patent/UY29371A1/en unknown
-
2007
- 2007-06-26 TN TNP2007000241A patent/TNSN07241A1/en unknown
- 2007-07-06 CR CR9231A patent/CR9231A/en not_active Application Discontinuation
- 2007-07-08 IL IL184488A patent/IL184488A0/en unknown
- 2007-08-01 US US11/832,208 patent/US7592365B2/en not_active Expired - Fee Related
- 2007-08-13 MA MA30134A patent/MA29248B1/en unknown
- 2007-09-06 NO NO20074528A patent/NO20074528L/en not_active Application Discontinuation
-
2009
- 2009-03-17 HR HR20090158T patent/HRP20090158T1/en unknown
- 2009-03-23 CY CY20091100344T patent/CY1108916T1/en unknown
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